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Found 42 with Last Name = 'clanton' and Initial = 'dj'
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Aids Drug Screening And Development Laboratory

Curated by ChEMBL
LigandPNGBDBM50073270(CHEMBL333781 | {2-[(1S,3S,4S)-1-Benzyl-3-hydroxy-5...)
Affinity DataKi:  0.0100nMAssay Description:Inhibitory activity against HIV proteaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Aids Drug Screening And Development Laboratory

Curated by ChEMBL
LigandPNGBDBM50073266(CHEMBL119898 | {2-[(1S,3S,4S)-1-Benzyl-4-((2S,3S)-...)
Affinity DataKi:  0.0200nMAssay Description:Inhibitory activity against HIV proteaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Aids Drug Screening And Development Laboratory

Curated by ChEMBL
LigandPNGBDBM50073253(CHEMBL278935 | {2-[(1S,3S,4S)-1-Benzyl-3-hydroxy-5...)
Affinity DataKi:  0.0300nMAssay Description:Inhibitory activity against HIV proteaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Aids Drug Screening And Development Laboratory

Curated by ChEMBL
LigandPNGBDBM50073250(CHEMBL333420 | {2-[(1S,3S,4S)-1-Benzyl-4-((R)-2-et...)
Affinity DataKi:  0.0300nMAssay Description:Inhibitory activity against HIV proteaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Aids Drug Screening And Development Laboratory

Curated by ChEMBL
LigandPNGBDBM50073269((2-{(1S,3S,4S)-1-Benzyl-3-hydroxy-5-phenyl-4-[(R)-...)
Affinity DataKi:  0.0400nMAssay Description:Inhibitory activity against HIV proteaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Aids Drug Screening And Development Laboratory

Curated by ChEMBL
LigandPNGBDBM50073252(CHEMBL324157 | {2-[(1S,3S,4S)-1-Benzyl-3-hydroxy-4...)
Affinity DataKi:  0.0600nMAssay Description:Inhibitory activity against HIV proteaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Aids Drug Screening And Development Laboratory

Curated by ChEMBL
LigandPNGBDBM50073254(Anthranilamide derivative | CHEMBL408110)
Affinity DataKi:  0.0600nMAssay Description:Tested for inhibition of HIV protease using fluorogenic substrateMore data for this Ligand-Target Pair
In DepthDetails Article
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Aids Drug Screening And Development Laboratory

Curated by ChEMBL
LigandPNGBDBM50073265((2-{(1S,2S,3R,4S)-1-Benzyl-2,3-dihydroxy-5-phenyl-...)
Affinity DataKi:  0.0700nMAssay Description:Inhibitory activity against HIV proteaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Aids Drug Screening And Development Laboratory

Curated by ChEMBL
LigandPNGBDBM50285701(Anthranilamide derivative | CHEMBL313767)
Affinity DataKi:  0.0700nMAssay Description:Tested for inhibition of HIV protease using fluorogenic substrateMore data for this Ligand-Target Pair
In DepthDetails Article
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Aids Drug Screening And Development Laboratory

Curated by ChEMBL
LigandPNGBDBM50073254(Anthranilamide derivative | CHEMBL408110)
Affinity DataKi:  0.0700nMAssay Description:Inhibitory activity against HIV proteaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Aids Drug Screening And Development Laboratory

Curated by ChEMBL
LigandPNGBDBM50073268(CHEMBL331294 | {2-[(1S,2S,3R,4S)-1-Benzyl-2,3-dihy...)
Affinity DataKi:  0.0900nMAssay Description:Inhibitory activity against HIV proteaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Aids Drug Screening And Development Laboratory

Curated by ChEMBL
LigandPNGBDBM50073263(CHEMBL117629 | {2-[(1S,3S,4S)-4-(3-Amino-2-methyl-...)
Affinity DataKi:  0.120nMAssay Description:Inhibitory activity against HIV proteaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Aids Drug Screening And Development Laboratory

Curated by ChEMBL
LigandPNGBDBM50073244(CHEMBL332825 | [2-((1S,3S,4S)-1-Benzyl-4-tert-buto...)
Affinity DataKi:  0.130nMAssay Description:Inhibitory activity against HIV proteaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Aids Drug Screening And Development Laboratory

Curated by ChEMBL
LigandPNGBDBM50073262(CHEMBL333290 | [2-((1S,2S,3R,4S)-1-Benzyl-4-tert-b...)
Affinity DataKi:  0.130nMAssay Description:Inhibitory activity against HIV proteaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Aids Drug Screening And Development Laboratory

Curated by ChEMBL
LigandPNGBDBM50285698(Anthranilamide derivative | CHEMBL315500)
Affinity DataKi:  0.260nMAssay Description:Tested for inhibition of HIV protease using fluorogenic substrateMore data for this Ligand-Target Pair
In DepthDetails Article
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Aids Drug Screening And Development Laboratory

Curated by ChEMBL
LigandPNGBDBM50073248(CHEMBL119745 | {2-[(1S,3S,4S)-1-Benzyl-3-hydroxy-4...)
Affinity DataKi:  0.270nMAssay Description:Inhibitory activity against HIV proteaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Aids Drug Screening And Development Laboratory

Curated by ChEMBL
LigandPNGBDBM50073249(CHEMBL331199 | {2-[(1S,3S,4S)-4-(3-Amino-benzoylam...)
Affinity DataKi:  0.400nMAssay Description:Inhibitory activity against HIV proteaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Aids Drug Screening And Development Laboratory

Curated by ChEMBL
LigandPNGBDBM50073243((2-{(1S,2S,3R,4S)-1-Benzyl-2,3-dihydroxy-4-[(isoxa...)
Affinity DataKi:  0.400nMAssay Description:Inhibitory activity against HIV proteaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Aids Drug Screening And Development Laboratory

Curated by ChEMBL
LigandPNGBDBM50073259(CHEMBL333407 | [2-((1S,2R,3S,4S)-1-Benzyl-4-tert-b...)
Affinity DataKi:  0.450nMAssay Description:Inhibitory activity against HIV proteaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Aids Drug Screening And Development Laboratory

Curated by ChEMBL
LigandPNGBDBM50285700(Anthranilamide derivative | CHEMBL315742)
Affinity DataKi:  0.450nMAssay Description:Tested for inhibition of HIV protease using fluorogenic substrateMore data for this Ligand-Target Pair
In DepthDetails Article
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Aids Drug Screening And Development Laboratory

Curated by ChEMBL
LigandPNGBDBM50073261(CHEMBL116482 | {2-[(1S,2S,3R,4S)-1-Benzyl-2,3-dihy...)
Affinity DataKi:  0.5nMAssay Description:Inhibitory activity against HIV proteaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Aids Drug Screening And Development Laboratory

Curated by ChEMBL
LigandPNGBDBM50073251(CHEMBL118396 | {2-[(1S,3S,4S)-1-Benzyl-3-hydroxy-5...)
Affinity DataKi:  0.620nMAssay Description:Inhibitory activity against HIV proteaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Aids Drug Screening And Development Laboratory

Curated by ChEMBL
LigandPNGBDBM50073247(CHEMBL118513 | {2-[(1S,2S,4S)-1-Benzyl-2-hydroxy-4...)
Affinity DataKi:  0.680nMAssay Description:Inhibitory activity against HIV proteaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Aids Drug Screening And Development Laboratory

Curated by ChEMBL
LigandPNGBDBM50073256(CHEMBL122006 | [2-((1S,2S,4S)-1-Benzyl-4-tert-buto...)
Affinity DataKi:  0.850nMAssay Description:Inhibitory activity against HIV proteaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Aids Drug Screening And Development Laboratory

Curated by ChEMBL
LigandPNGBDBM50073246(CHEMBL333392 | {2-[(1S,3S,4S)-1-Benzyl-3-hydroxy-4...)
Affinity DataKi:  0.850nMAssay Description:Inhibitory activity against HIV proteaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Aids Drug Screening And Development Laboratory

Curated by ChEMBL
LigandPNGBDBM50073267((2-{(1S,3S,4S)-1-Benzyl-3-hydroxy-4-[(isoxazole-5-...)
Affinity DataKi:  1.20nMAssay Description:Inhibitory activity against HIV proteaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Aids Drug Screening And Development Laboratory

Curated by ChEMBL
LigandPNGBDBM50285703(Anthranilamide derivative | CHEMBL315928)
Affinity DataKi:  1.20nMAssay Description:Tested for inhibition of HIV protease using fluorogenic substrateMore data for this Ligand-Target Pair
In DepthDetails Article
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Aids Drug Screening And Development Laboratory

Curated by ChEMBL
LigandPNGBDBM50285696(Anthranilamide derivative | CHEMBL85640)
Affinity DataKi:  1.20nMAssay Description:Tested for inhibition of HIV protease using fluorogenic substrateMore data for this Ligand-Target Pair
In DepthDetails Article
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Aids Drug Screening And Development Laboratory

Curated by ChEMBL
LigandPNGBDBM50073264(CHEMBL118531 | {2-[(1S,3S,4S)-4-(4-Amino-benzoylam...)
Affinity DataKi:  1.5nMAssay Description:Inhibitory activity against HIV proteaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Aids Drug Screening And Development Laboratory

Curated by ChEMBL
LigandPNGBDBM50073257(CHEMBL325499 | {2-[(1S,2R,3S,4S)-1-Benzyl-2,3-dihy...)
Affinity DataKi:  1.70nMAssay Description:Inhibitory activity against HIV proteaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Aids Drug Screening And Development Laboratory

Curated by ChEMBL
LigandPNGBDBM50285691(Anthranilamide derivative | CHEMBL264622)
Affinity DataKi:  2.40nMAssay Description:Tested for inhibition of HIV protease using fluorogenic substrateMore data for this Ligand-Target Pair
In DepthDetails Article
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Aids Drug Screening And Development Laboratory

Curated by ChEMBL
LigandPNGBDBM50285695(Anthranilamide derivative | CHEMBL86263)
Affinity DataKi:  3nMAssay Description:Tested for inhibition of HIV protease using fluorogenic substrateMore data for this Ligand-Target Pair
In DepthDetails Article
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Aids Drug Screening And Development Laboratory

Curated by ChEMBL
LigandPNGBDBM50073255((2-{(1S,3S,4S)-1-Benzyl-3-hydroxy-5-phenyl-4-[(thi...)
Affinity DataKi:  4.70nMAssay Description:Inhibitory activity against HIV proteaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Aids Drug Screening And Development Laboratory

Curated by ChEMBL
LigandPNGBDBM50073258(CHEMBL118221 | {2-[(1S,2R,3S,4S)-4-(4-Amino-benzoy...)
Affinity DataKi:  6.60nMAssay Description:Inhibitory activity against HIV proteaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Aids Drug Screening And Development Laboratory

Curated by ChEMBL
LigandPNGBDBM50073245(CHEMBL118362 | {2-[(1S,2S,4S)-1-Benzyl-2-hydroxy-4...)
Affinity DataKi:  8.60nMAssay Description:Inhibitory activity against HIV proteaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Aids Drug Screening And Development Laboratory

Curated by ChEMBL
LigandPNGBDBM50285699(Anthranilamide derivative | CHEMBL87879)
Affinity DataKi:  12nMAssay Description:Tested for inhibition of HIV protease using fluorogenic substrateMore data for this Ligand-Target Pair
In DepthDetails Article
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Aids Drug Screening And Development Laboratory

Curated by ChEMBL
LigandPNGBDBM50285690(Anthranilamide derivative | CHEMBL87309)
Affinity DataKi:  20nMAssay Description:Tested for inhibition of HIV protease using fluorogenic substrateMore data for this Ligand-Target Pair
In DepthDetails Article
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Aids Drug Screening And Development Laboratory

Curated by ChEMBL
LigandPNGBDBM50285702(Anthranilamide derivative | CHEMBL314408)
Affinity DataKi:  20nMAssay Description:Tested for inhibition of HIV protease using fluorogenic substrateMore data for this Ligand-Target Pair
In DepthDetails Article
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Aids Drug Screening And Development Laboratory

Curated by ChEMBL
LigandPNGBDBM50285692(1N-[1-benzyl-2,3-dihydroxy-4-(2-methylcarboxamidop...)
Affinity DataKi:  41nMAssay Description:Tested for inhibition of HIV protease using fluorogenic substrateMore data for this Ligand-Target Pair
In DepthDetails Article
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Aids Drug Screening And Development Laboratory

Curated by ChEMBL
LigandPNGBDBM50285693(Anthranilamide derivative | CHEMBL84884)
Affinity DataKi:  91nMAssay Description:Tested for inhibition of HIV protease using fluorogenic substrateMore data for this Ligand-Target Pair
In DepthDetails Article
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Aids Drug Screening And Development Laboratory

Curated by ChEMBL
LigandPNGBDBM50285697(Anthranilamide derivative | CHEMBL313254)
Affinity DataKi: >1.00E+4nMAssay Description:Tested for inhibition of HIV protease using fluorogenic substrateMore data for this Ligand-Target Pair
In DepthDetails Article
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Aids Drug Screening And Development Laboratory

Curated by ChEMBL
LigandPNGBDBM50285694(Anthranilamide derivative | CHEMBL314004)
Affinity DataKi: >1.00E+4nMAssay Description:Tested for inhibition of HIV protease using fluorogenic substrateMore data for this Ligand-Target Pair
In DepthDetails Article