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Found 841 with Last Name = 'connolly' and Initial = 'c'
Target5-hydroxytryptamine receptor 3A(Homo sapiens (Human))
University Of Bern

Curated by ChEMBL
LigandPNGBDBM50363283(CHEMBL1945711)
Affinity DataKi:  0.900nMAssay Description:Displacement of [3H]granisetron from human 5HT3A expressed in HEK293 cells after 1 hr by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 3A(Homo sapiens (Human))
University Of Bern

Curated by ChEMBL
LigandPNGBDBM50363287(CHEMBL1945830)
Affinity DataKi:  1.10nMAssay Description:Displacement of [3H]granisetron from human 5HT3A expressed in HEK293 cells after 1 hr by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 3A(Homo sapiens (Human))
University Of Bern

Curated by ChEMBL
LigandPNGBDBM50363291(CHEMBL1945835)
Affinity DataKi:  1.20nMAssay Description:Displacement of [3H]granisetron from human 5HT3A expressed in HEK293 cells after 1 hr by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 3A(Homo sapiens (Human))
University Of Bern

Curated by ChEMBL
LigandPNGBDBM50000483((BRL 43694)1-Methyl-1H-indazole-3-carboxylic acid ...)
Affinity DataKi:  1.45nMAssay Description:Displacement of [3H]granisetron from human 5HT3A expressed in HEK293 cells after 1 hr by scintillation countingMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 3A(Homo sapiens (Human))
University Of Bern

Curated by ChEMBL
LigandPNGBDBM50363285(CHEMBL1945713)
Affinity DataKi:  1.60nMAssay Description:Displacement of [3H]granisetron from human 5HT3A expressed in HEK293 cells after 1 hr by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 3A(Homo sapiens (Human))
University Of Bern

Curated by ChEMBL
LigandPNGBDBM50363292(CHEMBL1945836)
Affinity DataKi:  1.60nMAssay Description:Displacement of [3H]granisetron from human 5HT3A expressed in HEK293 cells after 1 hr by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 3A(Homo sapiens (Human))
University Of Bern

Curated by ChEMBL
LigandPNGBDBM50363293(CHEMBL1945837)
Affinity DataKi:  1.90nMAssay Description:Displacement of [3H]granisetron from human 5HT3A expressed in HEK293 cells after 1 hr by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 3A(Homo sapiens (Human))
University Of Bern

Curated by ChEMBL
LigandPNGBDBM50363286(CHEMBL1945714)
Affinity DataKi:  7.30nMAssay Description:Displacement of [3H]granisetron from human 5HT3A expressed in HEK293 cells after 1 hr by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 3A(Homo sapiens (Human))
University Of Bern

Curated by ChEMBL
LigandPNGBDBM50363290(CHEMBL1945834)
Affinity DataKi:  8.70nMAssay Description:Displacement of [3H]granisetron from human 5HT3A expressed in HEK293 cells after 1 hr by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFibroblast growth factor receptor 1(Homo sapiens (Human))
Parke-Davis Pharmaceutical Research

Curated by PDSP Ki Database
LigandPNGBDBM3443(1-[2-amino-6-(3,5-dimethoxyphenyl)pyrido[2,3-d]pyr...)
Affinity DataKi:  45.2nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
Target5-hydroxytryptamine receptor 3A(Homo sapiens (Human))
University Of Bern

Curated by ChEMBL
LigandPNGBDBM50363288(CHEMBL1945832)
Affinity DataKi:  142nMAssay Description:Displacement of [3H]granisetron from human 5HT3A expressed in HEK293 cells after 1 hr by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 3A(Homo sapiens (Human))
University Of Bern

Curated by ChEMBL
LigandPNGBDBM50363294(CHEMBL1945838)
Affinity DataKi:  157nMAssay Description:Displacement of [3H]granisetron from human 5HT3A expressed in HEK293 cells after 1 hr by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 3A(Homo sapiens (Human))
University Of Bern

Curated by ChEMBL
LigandPNGBDBM50363284(CHEMBL1945712)
Affinity DataKi:  199nMAssay Description:Displacement of [3H]granisetron from human 5HT3A expressed in HEK293 cells after 1 hr by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 3A(Homo sapiens (Human))
University Of Bern

Curated by ChEMBL
LigandPNGBDBM50363296(CHEMBL1946302)
Affinity DataKi:  208nMAssay Description:Displacement of [3H]granisetron from human 5HT3A expressed in HEK293 cells after 1 hr by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 3A(Homo sapiens (Human))
University Of Bern

Curated by ChEMBL
LigandPNGBDBM50363295(CHEMBL1946154)
Affinity DataKi:  1.30E+3nMAssay Description:Displacement of [3H]granisetron from human 5HT3A expressed in HEK293 cells after 1 hr by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 3A(Homo sapiens (Human))
University Of Bern

Curated by ChEMBL
LigandPNGBDBM50363289(CHEMBL1945833)
Affinity DataKi:  6.30E+3nMAssay Description:Displacement of [3H]granisetron from human 5HT3A expressed in HEK293 cells after 1 hr by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50030815(CHEMBL404594)
Affinity DataIC50:  0.100nMAssay Description:Binding affinity for rat brain Angiotensin II receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRenin(Homo sapiens (Human))
Parke-Davis Pharmaceutical Research Division Of Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50006848(CHEMBL88091 | N-[2-(2-Amino-thiazol-4-yl)-1-(1-cyc...)
Affinity DataIC50:  0.160nMAssay Description:In vitro inhibition of monkey renin.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRenin(Homo sapiens (Human))
Parke-Davis Pharmaceutical Research Division Of Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50006850(CHEMBL313063 | N-[1-(1-Cyclohexylmethyl-2,3-dihydr...)
Affinity DataIC50:  0.200nMAssay Description:In vitro inhibition of monkey renin.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRenin(Homo sapiens (Human))
Parke-Davis Pharmaceutical Research Division Of Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50006858(CHEMBL315380 | N-[1-(1-Cyclohexylmethyl-2,3-dihydr...)
Affinity DataIC50:  0.230nMAssay Description:In vitro inhibition of monkey renin.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRenin(Homo sapiens (Human))
Parke-Davis Pharmaceutical Research Division Of Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50006854(CHEMBL88069 | N-[2-(2-Amino-thiazol-4-yl)-1-(1-cyc...)
Affinity DataIC50:  0.270nMAssay Description:In vitro inhibition of monkey renin.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRenin(Homo sapiens (Human))
Parke-Davis Pharmaceutical Research Division Of Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50006853(CHEMBL315211 | N-(1-Cyclohexylmethyl-2,3-dihydroxy...)
Affinity DataIC50:  0.280nMAssay Description:In vitro inhibition of monkey renin.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRenin(Homo sapiens (Human))
Parke-Davis Pharmaceutical Research Division Of Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50006845(CHEMBL316208 | N-[2-(2-Amino-thiazol-4-yl)-1-(1-cy...)
Affinity DataIC50:  0.350nMAssay Description:In vitro inhibition of monkey renin.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50030815(CHEMBL404594)
Affinity DataIC50:  0.350nMAssay Description:Binding affinity against Angiotensin II receptor, from rat adrenal glandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRenin(Homo sapiens (Human))
Parke-Davis Pharmaceutical Research Division Of Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50006844((S)-N-[(S)-2-(2-Amino-thiazol-4-yl)-1-((1S,2R,3S)-...)
Affinity DataIC50:  0.360nMAssay Description:In vitro inhibition of monkey renin.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRenin(Homo sapiens (Human))
Parke-Davis Pharmaceutical Research Division Of Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50006844((S)-N-[(S)-2-(2-Amino-thiazol-4-yl)-1-((1S,2R,3S)-...)
Affinity DataIC50:  0.370nMAssay Description:Compound was evaluated for inhibition of plasma renin activity in monkeyMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor A/B(RAT)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50230906(CHEMBL308261)
Affinity DataIC50:  0.410nMAssay Description:Inhibitory concentration against binding of [125I]angiotensin II to rat liver expressing Angiotensin II receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRenin(Homo sapiens (Human))
Parke-Davis Pharmaceutical Research Division Of Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50006851(CHEMBL263531 | N-[1-(1-Cyclohexylmethyl-2,3-dihydr...)
Affinity DataIC50:  0.480nMAssay Description:In vitro inhibition of monkey renin.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRenin(Homo sapiens (Human))
Parke-Davis Pharmaceutical Research Division Of Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50009873(6-Acetylamino-2-[2-(morpholine-4-sulfonylamino)-3-...)
Affinity DataIC50:  0.5nMAssay Description:Inhibitory activity against monkey plasma renin.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRenin(Homo sapiens (Human))
Parke-Davis Pharmaceutical Research Division Of Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50006856(4-{3-(2-Amino-thiazol-4-yl)-2-[2-(morpholine-4-sul...)
Affinity DataIC50:  0.5nMAssay Description:In vitro inhibition of monkey renin.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRenin(Homo sapiens (Human))
Parke-Davis Pharmaceutical Research Division Of Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50006846(4-{3-(2-Amino-thiazol-4-yl)-2-[2-(morpholine-4-sul...)
Affinity DataIC50:  0.540nMAssay Description:In vitro inhibition of monkey renin.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRenin(Homo sapiens (Human))
Parke-Davis Pharmaceutical Research Division Of Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50006844((S)-N-[(S)-2-(2-Amino-thiazol-4-yl)-1-((1S,2R,3S)-...)
Affinity DataIC50:  0.570nMAssay Description:Compound was evaluated for inhibition of plasma renin activity in humanMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor A/B(RAT)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50230919(CHEMBL307844 | CI-996)
Affinity DataIC50:  0.580nMAssay Description:Inhibitory concentration against binding of [125I]angiotensin II to rat liver expressing Angiotensin II receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRenin(Homo sapiens (Human))
Parke-Davis Pharmaceutical Research Division Of Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50006843(CHEMBL314066 | N-[(2-Amino-thiazol-4-yl)-(1-cycloh...)
Affinity DataIC50:  0.581nMAssay Description:In vitro inhibition of monkey renin.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRenin(Homo sapiens (Human))
Parke-Davis Pharmaceutical Research Division Of Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50006849(4-{3-(2-Amino-thiazol-4-yl)-2-[2-(morpholine-4-sul...)
Affinity DataIC50:  0.590nMAssay Description:In vitro inhibition of monkey renin.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRenin(Homo sapiens (Human))
Parke-Davis Pharmaceutical Research Division Of Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50006202(3-Amino-N-[1-[1-(1-cyclohexylmethyl-2,3-dihydroxy-...)
Affinity DataIC50:  0.760nMAssay Description:In vitro inhibition of monkey renin.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor A/B(RAT)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50230891(CHEMBL76166)
Affinity DataIC50:  0.800nMAssay Description:Inhibitory concentration against binding of [125I]angiotensin II to rat liver expressing Angiotensin II receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor A/B(RAT)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50230883(CHEMBL309089)
Affinity DataIC50:  0.820nMAssay Description:Inhibitory concentration against binding of [125I]angiotensin II to rat liver expressing Angiotensin II receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRenin(Homo sapiens (Human))
Parke-Davis Pharmaceutical Research Division Of Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM17941((2S,4S,5S)-5-[(2S)-2-[(2S)-2-benzyl-3-[(2-methylpr...)
Affinity DataIC50:  0.830nMAssay Description:In vitro inhibition of monkey renin.More data for this Ligand-Target Pair
TargetType-1 angiotensin II receptor A/B(RAT)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50230915(CHEMBL76169)
Affinity DataIC50:  0.900nMAssay Description:Inhibitory concentration against binding of [125I]angiotensin II to rat liver expressing Angiotensin II receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRenin(Homo sapiens (Human))
Parke-Davis Pharmaceutical Research Division Of Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50006860(CHEMBL85672 | {1-[2-(2-Amino-thiazol-4-yl)-1-(1-cy...)
Affinity DataIC50:  0.910nMAssay Description:In vitro inhibition of monkey renin.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, NMDA 1(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50215294(2-(N-(6-chloro-7-methyl-2,3-dioxo-1,2,3,4-tetrahyd...)
Affinity DataIC50:  1nMAssay Description:Antagonist activity at human NMDA NR1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor A/B(RAT)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50230887(CHEMBL306259)
Affinity DataIC50:  1nMAssay Description:Inhibitory concentration against binding of [125I]angiotensin II to rat liver expressing Angiotensin II receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor A/B(RAT)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50230912(CHEMBL72922)
Affinity DataIC50:  1.20nMAssay Description:Inhibitory concentration against binding of [125I]angiotensin II to rat liver expressing Angiotensin II receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50228195(Angiotensin Ii | CHEBI:2719)
Affinity DataIC50:  1.30nMAssay Description:Binding affinity against Angiotensin II receptor, from rat adrenal glandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor A/B(RAT)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50230886(CHEMBL307455)
Affinity DataIC50:  1.40nMAssay Description:Inhibitory concentration against binding of [125I]angiotensin II to rat liver expressing Angiotensin II receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor A/B(RAT)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50230910(CHEMBL306066)
Affinity DataIC50:  1.60nMAssay Description:Inhibitory concentration against binding of [125I]angiotensin II to rat liver expressing Angiotensin II receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50228894(CHEMBL312754)
Affinity DataIC50:  1.60nMAssay Description:Binding affinity against Angiotensin II receptor, from rat adrenal glandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor A/B(RAT)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50230882(CARBOXYLIC ACID METABOLITE | CHEBI:74125 | E-3174)
Affinity DataIC50:  1.60nMAssay Description:Inhibitory concentration against binding of [125I]angiotensin II to rat liver expressing Angiotensin II receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor A/B(RAT)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50230882(CARBOXYLIC ACID METABOLITE | CHEBI:74125 | E-3174)
Affinity DataIC50:  1.60nMAssay Description:Tested for inhibitory concentration against AT1 receptor binding affinity in rat liverMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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