Affinity DataKi: 0.900nMAssay Description:Displacement of [3H]granisetron from human 5HT3A expressed in HEK293 cells after 1 hr by scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 1.10nMAssay Description:Displacement of [3H]granisetron from human 5HT3A expressed in HEK293 cells after 1 hr by scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 1.20nMAssay Description:Displacement of [3H]granisetron from human 5HT3A expressed in HEK293 cells after 1 hr by scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 1.45nMAssay Description:Displacement of [3H]granisetron from human 5HT3A expressed in HEK293 cells after 1 hr by scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 1.60nMAssay Description:Displacement of [3H]granisetron from human 5HT3A expressed in HEK293 cells after 1 hr by scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 1.60nMAssay Description:Displacement of [3H]granisetron from human 5HT3A expressed in HEK293 cells after 1 hr by scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 1.90nMAssay Description:Displacement of [3H]granisetron from human 5HT3A expressed in HEK293 cells after 1 hr by scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 7.30nMAssay Description:Displacement of [3H]granisetron from human 5HT3A expressed in HEK293 cells after 1 hr by scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 8.70nMAssay Description:Displacement of [3H]granisetron from human 5HT3A expressed in HEK293 cells after 1 hr by scintillation countingMore data for this Ligand-Target Pair
TargetFibroblast growth factor receptor 1(Homo sapiens (Human))
Parke-Davis Pharmaceutical Research
Curated by PDSP Ki Database
Parke-Davis Pharmaceutical Research
Curated by PDSP Ki Database
Affinity DataKi: 142nMAssay Description:Displacement of [3H]granisetron from human 5HT3A expressed in HEK293 cells after 1 hr by scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 157nMAssay Description:Displacement of [3H]granisetron from human 5HT3A expressed in HEK293 cells after 1 hr by scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 199nMAssay Description:Displacement of [3H]granisetron from human 5HT3A expressed in HEK293 cells after 1 hr by scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 208nMAssay Description:Displacement of [3H]granisetron from human 5HT3A expressed in HEK293 cells after 1 hr by scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 1.30E+3nMAssay Description:Displacement of [3H]granisetron from human 5HT3A expressed in HEK293 cells after 1 hr by scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 6.30E+3nMAssay Description:Displacement of [3H]granisetron from human 5HT3A expressed in HEK293 cells after 1 hr by scintillation countingMore data for this Ligand-Target Pair
TargetType-1 angiotensin II receptor A/Type-1 angiotensin II receptor B/Type-2 angiotensin II receptor(RAT)
Warner-Lambert
Curated by ChEMBL
Warner-Lambert
Curated by ChEMBL
Affinity DataIC50: 0.100nMAssay Description:Binding affinity for rat brain Angiotensin II receptorMore data for this Ligand-Target Pair
TargetRenin(Homo sapiens (Human))
Parke-Davis Pharmaceutical Research Division Of Warner-Lambert
Curated by ChEMBL
Parke-Davis Pharmaceutical Research Division Of Warner-Lambert
Curated by ChEMBL
Affinity DataIC50: 0.160nMAssay Description:In vitro inhibition of monkey renin.More data for this Ligand-Target Pair
TargetRenin(Homo sapiens (Human))
Parke-Davis Pharmaceutical Research Division Of Warner-Lambert
Curated by ChEMBL
Parke-Davis Pharmaceutical Research Division Of Warner-Lambert
Curated by ChEMBL
Affinity DataIC50: 0.200nMAssay Description:In vitro inhibition of monkey renin.More data for this Ligand-Target Pair
TargetRenin(Homo sapiens (Human))
Parke-Davis Pharmaceutical Research Division Of Warner-Lambert
Curated by ChEMBL
Parke-Davis Pharmaceutical Research Division Of Warner-Lambert
Curated by ChEMBL
Affinity DataIC50: 0.230nMAssay Description:In vitro inhibition of monkey renin.More data for this Ligand-Target Pair
TargetRenin(Homo sapiens (Human))
Parke-Davis Pharmaceutical Research Division Of Warner-Lambert
Curated by ChEMBL
Parke-Davis Pharmaceutical Research Division Of Warner-Lambert
Curated by ChEMBL
Affinity DataIC50: 0.270nMAssay Description:In vitro inhibition of monkey renin.More data for this Ligand-Target Pair
TargetRenin(Homo sapiens (Human))
Parke-Davis Pharmaceutical Research Division Of Warner-Lambert
Curated by ChEMBL
Parke-Davis Pharmaceutical Research Division Of Warner-Lambert
Curated by ChEMBL
Affinity DataIC50: 0.280nMAssay Description:In vitro inhibition of monkey renin.More data for this Ligand-Target Pair
TargetRenin(Homo sapiens (Human))
Parke-Davis Pharmaceutical Research Division Of Warner-Lambert
Curated by ChEMBL
Parke-Davis Pharmaceutical Research Division Of Warner-Lambert
Curated by ChEMBL
Affinity DataIC50: 0.350nMAssay Description:In vitro inhibition of monkey renin.More data for this Ligand-Target Pair
TargetType-1 angiotensin II receptor A/Type-1 angiotensin II receptor B/Type-2 angiotensin II receptor(RAT)
Warner-Lambert
Curated by ChEMBL
Warner-Lambert
Curated by ChEMBL
Affinity DataIC50: 0.350nMAssay Description:Binding affinity against Angiotensin II receptor, from rat adrenal glandMore data for this Ligand-Target Pair
TargetRenin(Homo sapiens (Human))
Parke-Davis Pharmaceutical Research Division Of Warner-Lambert
Curated by ChEMBL
Parke-Davis Pharmaceutical Research Division Of Warner-Lambert
Curated by ChEMBL
Affinity DataIC50: 0.360nMAssay Description:In vitro inhibition of monkey renin.More data for this Ligand-Target Pair
TargetRenin(Homo sapiens (Human))
Parke-Davis Pharmaceutical Research Division Of Warner-Lambert
Curated by ChEMBL
Parke-Davis Pharmaceutical Research Division Of Warner-Lambert
Curated by ChEMBL
Affinity DataIC50: 0.370nMAssay Description:Compound was evaluated for inhibition of plasma renin activity in monkeyMore data for this Ligand-Target Pair
Affinity DataIC50: 0.410nMAssay Description:Inhibitory concentration against binding of [125I]angiotensin II to rat liver expressing Angiotensin II receptorMore data for this Ligand-Target Pair
TargetRenin(Homo sapiens (Human))
Parke-Davis Pharmaceutical Research Division Of Warner-Lambert
Curated by ChEMBL
Parke-Davis Pharmaceutical Research Division Of Warner-Lambert
Curated by ChEMBL
Affinity DataIC50: 0.480nMAssay Description:In vitro inhibition of monkey renin.More data for this Ligand-Target Pair
TargetRenin(Homo sapiens (Human))
Parke-Davis Pharmaceutical Research Division Of Warner-Lambert
Curated by ChEMBL
Parke-Davis Pharmaceutical Research Division Of Warner-Lambert
Curated by ChEMBL
Affinity DataIC50: 0.5nMAssay Description:Inhibitory activity against monkey plasma renin.More data for this Ligand-Target Pair
TargetRenin(Homo sapiens (Human))
Parke-Davis Pharmaceutical Research Division Of Warner-Lambert
Curated by ChEMBL
Parke-Davis Pharmaceutical Research Division Of Warner-Lambert
Curated by ChEMBL
Affinity DataIC50: 0.5nMAssay Description:In vitro inhibition of monkey renin.More data for this Ligand-Target Pair
TargetRenin(Homo sapiens (Human))
Parke-Davis Pharmaceutical Research Division Of Warner-Lambert
Curated by ChEMBL
Parke-Davis Pharmaceutical Research Division Of Warner-Lambert
Curated by ChEMBL
Affinity DataIC50: 0.540nMAssay Description:In vitro inhibition of monkey renin.More data for this Ligand-Target Pair
TargetRenin(Homo sapiens (Human))
Parke-Davis Pharmaceutical Research Division Of Warner-Lambert
Curated by ChEMBL
Parke-Davis Pharmaceutical Research Division Of Warner-Lambert
Curated by ChEMBL
Affinity DataIC50: 0.570nMAssay Description:Compound was evaluated for inhibition of plasma renin activity in humanMore data for this Ligand-Target Pair
Affinity DataIC50: 0.580nMAssay Description:Inhibitory concentration against binding of [125I]angiotensin II to rat liver expressing Angiotensin II receptorMore data for this Ligand-Target Pair
TargetRenin(Homo sapiens (Human))
Parke-Davis Pharmaceutical Research Division Of Warner-Lambert
Curated by ChEMBL
Parke-Davis Pharmaceutical Research Division Of Warner-Lambert
Curated by ChEMBL
Affinity DataIC50: 0.581nMAssay Description:In vitro inhibition of monkey renin.More data for this Ligand-Target Pair
TargetRenin(Homo sapiens (Human))
Parke-Davis Pharmaceutical Research Division Of Warner-Lambert
Curated by ChEMBL
Parke-Davis Pharmaceutical Research Division Of Warner-Lambert
Curated by ChEMBL
Affinity DataIC50: 0.590nMAssay Description:In vitro inhibition of monkey renin.More data for this Ligand-Target Pair
TargetRenin(Homo sapiens (Human))
Parke-Davis Pharmaceutical Research Division Of Warner-Lambert
Curated by ChEMBL
Parke-Davis Pharmaceutical Research Division Of Warner-Lambert
Curated by ChEMBL
Affinity DataIC50: 0.760nMAssay Description:In vitro inhibition of monkey renin.More data for this Ligand-Target Pair
Affinity DataIC50: 0.800nMAssay Description:Inhibitory concentration against binding of [125I]angiotensin II to rat liver expressing Angiotensin II receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 0.820nMAssay Description:Inhibitory concentration against binding of [125I]angiotensin II to rat liver expressing Angiotensin II receptorMore data for this Ligand-Target Pair
TargetRenin(Homo sapiens (Human))
Parke-Davis Pharmaceutical Research Division Of Warner-Lambert
Curated by ChEMBL
Parke-Davis Pharmaceutical Research Division Of Warner-Lambert
Curated by ChEMBL
Affinity DataIC50: 0.830nMAssay Description:In vitro inhibition of monkey renin.More data for this Ligand-Target Pair
Affinity DataIC50: 0.900nMAssay Description:Inhibitory concentration against binding of [125I]angiotensin II to rat liver expressing Angiotensin II receptorMore data for this Ligand-Target Pair
TargetRenin(Homo sapiens (Human))
Parke-Davis Pharmaceutical Research Division Of Warner-Lambert
Curated by ChEMBL
Parke-Davis Pharmaceutical Research Division Of Warner-Lambert
Curated by ChEMBL
Affinity DataIC50: 0.910nMAssay Description:In vitro inhibition of monkey renin.More data for this Ligand-Target Pair
Affinity DataIC50: 1nMAssay Description:Antagonist activity at human NMDA NR1 receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 1nMAssay Description:Inhibitory concentration against binding of [125I]angiotensin II to rat liver expressing Angiotensin II receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 1.20nMAssay Description:Inhibitory concentration against binding of [125I]angiotensin II to rat liver expressing Angiotensin II receptorMore data for this Ligand-Target Pair
TargetType-1 angiotensin II receptor A/Type-1 angiotensin II receptor B/Type-2 angiotensin II receptor(RAT)
Warner-Lambert
Curated by ChEMBL
Warner-Lambert
Curated by ChEMBL
Affinity DataIC50: 1.30nMAssay Description:Binding affinity against Angiotensin II receptor, from rat adrenal glandMore data for this Ligand-Target Pair
Affinity DataIC50: 1.40nMAssay Description:Inhibitory concentration against binding of [125I]angiotensin II to rat liver expressing Angiotensin II receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 1.60nMAssay Description:Inhibitory concentration against binding of [125I]angiotensin II to rat liver expressing Angiotensin II receptorMore data for this Ligand-Target Pair
TargetType-1 angiotensin II receptor A/Type-1 angiotensin II receptor B/Type-2 angiotensin II receptor(RAT)
Warner-Lambert
Curated by ChEMBL
Warner-Lambert
Curated by ChEMBL
Affinity DataIC50: 1.60nMAssay Description:Binding affinity against Angiotensin II receptor, from rat adrenal glandMore data for this Ligand-Target Pair
Affinity DataIC50: 1.60nMAssay Description:Inhibitory concentration against binding of [125I]angiotensin II to rat liver expressing Angiotensin II receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 1.60nMAssay Description:Tested for inhibitory concentration against AT1 receptor binding affinity in rat liverMore data for this Ligand-Target Pair