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Found 98 with Last Name = 'damour' and Initial = 'd'
LigandPNGBDBM50280830(3-{2-[4-(5-Fluoro-1H-indol-3-ylmethyl)-piperidin-1...)
Affinity DataIC50:  0.5nMAssay Description:Compound was evaluated for inhibition of 5-HT uptake by measuring its ability to inhibit [3H]paroxetine binding to rat cortical membranesMore data for this Ligand-Target Pair
In DepthDetails Article
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50283917(1-(1,1-Diphenyl-silolan-3-yl)-4-(4-fluoro-phenyl)-...)
Affinity DataIC50:  0.900nMAssay Description:In vitro binding affinity towards serotonin 5-HT2A receptor in rat cortical membranes using [3H]ketanserin as radioligandMore data for this Ligand-Target Pair
In DepthDetails Article
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50283931(1-(1,1-Diphenyl-silolan-3-yl)-4-phenyl-piperazine ...)
Affinity DataIC50:  1nMAssay Description:In vitro binding affinity towards serotonin 5-HT2A receptor in rat cortical membranes using [3H]ketanserin as radioligandMore data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50280826(2-{2-[4-(5-Fluoro-1H-indol-3-ylmethyl)-piperidin-1...)
Affinity DataIC50:  1nMAssay Description:Compound was evaluated for inhibition of 5-HT uptake by measuring its ability to inhibit [3H]paroxetine binding to rat cortical membranesMore data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50280822(4-{2-[4-(5-Fluoro-1H-indol-3-ylmethyl)-piperidin-1...)
Affinity DataIC50:  1.10nMAssay Description:Compound was evaluated for inhibition of 5-HT uptake by measuring its ability to inhibit [3H]paroxetine binding to rat cortical membranesMore data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50047098(1-{2-[4-(5-Fluoro-1H-indol-3-ylmethyl)-piperidin-1...)
Affinity DataIC50:  1.20nMAssay Description:Compound was evaluated for inhibition of 5-HT uptake by measuring its ability to inhibit [3H]paroxetine binding to rat cortical membranesMore data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50280819(1-{2-[4-(5-Fluoro-1H-indol-3-ylmethyl)-piperidin-1...)
Affinity DataIC50:  1.5nMAssay Description:Compound was evaluated for inhibition of 5-HT uptake by measuring its ability to inhibit [3H]paroxetine binding to rat cortical membranesMore data for this Ligand-Target Pair
In DepthDetails Article
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50001775((ritanserin)6-(2-{4-[Bis-(4-fluoro-phenyl)-methyle...)
Affinity DataIC50:  1.70nMAssay Description:In vitro binding affinity towards serotonin 5-HT2A receptor in rat cortical membranes using [3H]ketanserin as radioligandMore data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50280831(2-{2-[4-(5-Fluoro-1H-indol-3-ylmethyl)-piperidin-1...)
Affinity DataIC50:  1.80nMAssay Description:Compound was evaluated for inhibition of 5-HT uptake by measuring its ability to inhibit [3H]paroxetine binding to rat cortical membranesMore data for this Ligand-Target Pair
In DepthDetails Article
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50283920(1-[1,1-Bis-(4-fluoro-phenyl)-silolan-3-yl]-4-pheny...)
Affinity DataIC50:  2nMAssay Description:In vitro binding affinity towards serotonin 5-HT2A receptor in rat cortical membranes using [3H]ketanserin as radioligandMore data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50280817(2-{2-[4-(5-Fluoro-1H-indol-3-ylmethyl)-piperidin-1...)
Affinity DataIC50:  2.10nMAssay Description:Compound was evaluated for inhibition of 5-HT uptake by measuring its ability to inhibit [3H]paroxetine binding to rat cortical membranesMore data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50280828(3-{2-[4-(5-Fluoro-1H-indol-3-ylmethyl)-piperidin-1...)
Affinity DataIC50:  2.60nMAssay Description:Compound was evaluated for inhibition of 5-HT uptake by measuring its ability to inhibit [3H]paroxetine binding to rat cortical membranesMore data for this Ligand-Target Pair
In DepthDetails Article
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50283920(1-[1,1-Bis-(4-fluoro-phenyl)-silolan-3-yl]-4-pheny...)
Affinity DataIC50:  3nMAssay Description:In vitro binding affinity towards serotonin 5-HT2A receptor in rat cortical membranes using [3H]ketanserin as radioligandMore data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50280824(1-{2-[4-(5-Fluoro-1H-indol-3-ylmethyl)-piperidin-1...)
Affinity DataIC50:  3.10nMAssay Description:Compound was evaluated for inhibition of 5-HT uptake by measuring its ability to inhibit [3H]paroxetine binding to rat cortical membranesMore data for this Ligand-Target Pair
In DepthDetails Article
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50283928(1-(1,1-Diphenyl-silolan-3-yl)-4-(3-fluoro-phenyl)-...)
Affinity DataIC50:  3.40nMAssay Description:In vitro binding affinity towards serotonin 5-HT2A receptor in rat cortical membranes using [3H]ketanserin as radioligandMore data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50280823(1-{2-[4-(5-Fluoro-1H-indol-3-ylmethyl)-piperidin-1...)
Affinity DataIC50:  3.70nMAssay Description:Compound was evaluated for inhibition of 5-HT uptake by measuring its ability to inhibit [3H]paroxetine binding to rat cortical membranesMore data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50280832(2-{2-[4-(5-Fluoro-1H-indol-3-ylmethyl)-piperidin-1...)
Affinity DataIC50:  3.80nMAssay Description:Compound was evaluated for inhibition of 5-HT uptake by measuring its ability to inhibit [3H]paroxetine binding to rat cortical membranesMore data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50280827(1'-{2-[4-(5-fluoro-1H-3-indolylmethyl)hexahydro-1-...)
Affinity DataIC50:  4nMAssay Description:Compound was evaluated for inhibition of 5-HT uptake by measuring its ability to inhibit [3H]paroxetine binding to rat cortical membranesMore data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50280829(2-{2-[4-(5-Fluoro-1H-indol-3-ylmethyl)-piperidin-1...)
Affinity DataIC50:  5.40nMAssay Description:Compound was evaluated for inhibition of 5-HT uptake by measuring its ability to inhibit [3H]paroxetine binding to rat cortical membranesMore data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50280825(1-{2-[4-(5-Fluoro-1H-indol-3-ylmethyl)-piperidin-1...)
Affinity DataIC50:  5.90nMAssay Description:Compound was evaluated for inhibition of 5-HT uptake by measuring its ability to inhibit [3H]paroxetine binding to rat cortical membranesMore data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50280815(CHEMBL56377 | N-{2-[4-(5-Fluoro-1H-indol-3-ylmethy...)
Affinity DataIC50:  6nMAssay Description:Compound was evaluated for inhibition of 5-HT uptake by measuring its ability to inhibit [3H]paroxetine binding to rat cortical membranesMore data for this Ligand-Target Pair
In DepthDetails Article
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50283929(1-(1,1-Diphenyl-silolan-3-yl)-4-p-tolyl-piperazine...)
Affinity DataIC50:  10nMAssay Description:In vitro binding affinity towards serotonin 5-HT2A receptor in rat cortical membranes using [3H]ketanserin as radioligandMore data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50280818(1-{2-[4-(5-Fluoro-1H-indol-3-ylmethyl)-piperidin-1...)
Affinity DataIC50:  12nMAssay Description:Compound was evaluated for inhibition of 5-HT uptake by measuring its ability to inhibit [3H]paroxetine binding to rat cortical membranesMore data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50280821(2-{2-[4-(5-Fluoro-1H-indol-3-ylmethyl)-piperidin-1...)
Affinity DataIC50:  14nMAssay Description:Compound was evaluated for inhibition of 5-HT uptake by measuring its ability to inhibit [3H]paroxetine binding to rat cortical membranesMore data for this Ligand-Target Pair
In DepthDetails Article
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50283921(1-(1,1-Diphenyl-silolan-3-yl)-4-(4-fluoro-phenyl)-...)
Affinity DataIC50:  14nMAssay Description:In vitro binding affinity towards serotonin 5-HT2A receptor in rat cortical membranes using [3H]ketanserin as radioligandMore data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM30130(CHEMBL1201082 | CHEMBL41 | Fluoxetin | Fluoxetine ...)
Affinity DataIC50:  15nMAssay Description:Compound was evaluated for inhibition of 5-HT uptake by measuring its ability to inhibit [3H]paroxetine binding to rat cortical membranesMore data for this Ligand-Target Pair
In DepthDetails Article
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50283919(1-[1,1-Bis-(4-fluoro-phenyl)-silolan-3-yl]-4-(4-fl...)
Affinity DataIC50:  18nMAssay Description:In vitro binding affinity towards serotonin 5-HT2A receptor in rat cortical membranes using [3H]ketanserin as radioligandMore data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50280820(1-{2-[4-(5-Fluoro-1H-indol-3-ylmethyl)-piperidin-1...)
Affinity DataIC50:  23nMAssay Description:Compound was evaluated for inhibition of 5-HT uptake by measuring its ability to inhibit [3H]paroxetine binding to rat cortical membranesMore data for this Ligand-Target Pair
In DepthDetails Article
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50283924(1-(4-Chloro-phenyl)-4-(1,1-diphenyl-silolan-3-yl)-...)
Affinity DataIC50:  25nMAssay Description:In vitro binding affinity towards serotonin 5-HT2A receptor in rat cortical membranes using [3H]ketanserin as radioligandMore data for this Ligand-Target Pair
In DepthDetails Article
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50283918(1-[1-(4-Fluoro-phenyl)-1-phenyl-silolan-3-yl]-4-ph...)
Affinity DataIC50:  27nMAssay Description:In vitro binding affinity towards serotonin 5-HT2A receptor in rat cortical membranes using [3H]ketanserin as radioligandMore data for this Ligand-Target Pair
In DepthDetails Article
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50283918(1-[1-(4-Fluoro-phenyl)-1-phenyl-silolan-3-yl]-4-ph...)
Affinity DataIC50:  27nMAssay Description:In vitro binding affinity towards serotonin 5-HT2A receptor in rat cortical membranes using [3H]ketanserin as radioligandMore data for this Ligand-Target Pair
In DepthDetails Article
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50283923(1-(1,1-Diphenyl-silolan-3-yl)-4-pyridin-2-yl-piper...)
Affinity DataIC50:  29nMAssay Description:In vitro binding affinity towards serotonin 5-HT2A receptor in rat cortical membranes using [3H]ketanserin as radioligandMore data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50280816(CHEMBL293729 | N-{2-[4-(5-Fluoro-1H-indol-3-ylmeth...)
Affinity DataIC50:  30nMAssay Description:Compound was evaluated for inhibition of 5-HT uptake by measuring its ability to inhibit [3H]paroxetine binding to rat cortical membranesMore data for this Ligand-Target Pair
In DepthDetails Article
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50283926(1-(1,1-Diphenyl-silolan-3-yl)-4-m-tolyl-piperazine...)
Affinity DataIC50:  33nMAssay Description:In vitro binding affinity towards serotonin 5-HT2A receptor in rat cortical membranes using [3H]ketanserin as radioligandMore data for this Ligand-Target Pair
In DepthDetails Article
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50283925(4-[4-(1,1-Diphenyl-silolan-3-yl)-piperazin-1-yl]-p...)
Affinity DataIC50:  46nMAssay Description:In vitro binding affinity towards serotonin 5-HT2A receptor in rat cortical membranes using [3H]ketanserin as radioligandMore data for this Ligand-Target Pair
In DepthDetails Article
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50283927(1-(1,1-Diphenyl-silolan-3-yl)-4-phenyl-piperidine ...)
Affinity DataIC50:  53nMAssay Description:In vitro binding affinity towards serotonin 5-HT2A receptor in rat cortical membranes using [3H]ketanserin as radioligandMore data for this Ligand-Target Pair
In DepthDetails Article
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50283930(2-[4-(1,1-Diphenyl-silolan-3-yl)-piperazin-1-yl]-p...)
Affinity DataIC50:  80nMAssay Description:In vitro binding affinity towards serotonin 5-HT2A receptor in rat cortical membranes using [3H]ketanserin as radioligandMore data for this Ligand-Target Pair
In DepthDetails Article
TargetD(2) dopamine receptor(Mus musculus (Mouse))
TBA

Curated by ChEMBL
LigandPNGBDBM50280818(1-{2-[4-(5-Fluoro-1H-indol-3-ylmethyl)-piperidin-1...)
Affinity DataIC50: >100nMAssay Description:Tested for its binding affinity against Dopamine receptor D2; showed no appreciable affinity at concentration specifiedMore data for this Ligand-Target Pair
In DepthDetails Article
TargetD(2) dopamine receptor(Mus musculus (Mouse))
TBA

Curated by ChEMBL
LigandPNGBDBM50280826(2-{2-[4-(5-Fluoro-1H-indol-3-ylmethyl)-piperidin-1...)
Affinity DataIC50: >100nMAssay Description:Tested for its binding affinity against Dopamine receptor D2; showed no appreciable affinity at concentration specifiedMore data for this Ligand-Target Pair
In DepthDetails Article
TargetD(2) dopamine receptor(Mus musculus (Mouse))
TBA

Curated by ChEMBL
LigandPNGBDBM50280827(1'-{2-[4-(5-fluoro-1H-3-indolylmethyl)hexahydro-1-...)
Affinity DataIC50: >100nMAssay Description:Tested for its binding affinity against Dopamine receptor D2; showed no appreciable affinity at concentration specifiedMore data for this Ligand-Target Pair
In DepthDetails Article
TargetD(2) dopamine receptor(Mus musculus (Mouse))
TBA

Curated by ChEMBL
LigandPNGBDBM50280824(1-{2-[4-(5-Fluoro-1H-indol-3-ylmethyl)-piperidin-1...)
Affinity DataIC50: >100nMAssay Description:Tested for its binding affinity against Dopamine receptor D2; showed no appreciable affinity at concentration specifiedMore data for this Ligand-Target Pair
In DepthDetails Article
TargetD(2) dopamine receptor(Mus musculus (Mouse))
TBA

Curated by ChEMBL
LigandPNGBDBM50280820(1-{2-[4-(5-Fluoro-1H-indol-3-ylmethyl)-piperidin-1...)
Affinity DataIC50: >100nMAssay Description:Tested for its binding affinity against Dopamine receptor D2; showed no appreciable affinity at concentration specifiedMore data for this Ligand-Target Pair
In DepthDetails Article
TargetD(2) dopamine receptor(Mus musculus (Mouse))
TBA

Curated by ChEMBL
LigandPNGBDBM50280828(3-{2-[4-(5-Fluoro-1H-indol-3-ylmethyl)-piperidin-1...)
Affinity DataIC50: >100nMAssay Description:Tested for its binding affinity against Dopamine receptor D2; showed no appreciable affinity at concentration specifiedMore data for this Ligand-Target Pair
In DepthDetails Article
TargetD(2) dopamine receptor(Mus musculus (Mouse))
TBA

Curated by ChEMBL
LigandPNGBDBM50280822(4-{2-[4-(5-Fluoro-1H-indol-3-ylmethyl)-piperidin-1...)
Affinity DataIC50: >100nMAssay Description:Tested for its binding affinity against Dopamine receptor D2; showed no appreciable affinity at concentration specifiedMore data for this Ligand-Target Pair
In DepthDetails Article
TargetD(2) dopamine receptor(Mus musculus (Mouse))
TBA

Curated by ChEMBL
LigandPNGBDBM50280832(2-{2-[4-(5-Fluoro-1H-indol-3-ylmethyl)-piperidin-1...)
Affinity DataIC50: >100nMAssay Description:Tested for its binding affinity against Dopamine receptor D2; showed no appreciable affinity at concentration specifiedMore data for this Ligand-Target Pair
In DepthDetails Article
TargetD(2) dopamine receptor(Mus musculus (Mouse))
TBA

Curated by ChEMBL
LigandPNGBDBM50280823(1-{2-[4-(5-Fluoro-1H-indol-3-ylmethyl)-piperidin-1...)
Affinity DataIC50: >100nMAssay Description:Tested for its binding affinity against Dopamine receptor D2; showed no appreciable affinity at concentration specifiedMore data for this Ligand-Target Pair
In DepthDetails Article
TargetD(2) dopamine receptor(Mus musculus (Mouse))
TBA

Curated by ChEMBL
LigandPNGBDBM50280821(2-{2-[4-(5-Fluoro-1H-indol-3-ylmethyl)-piperidin-1...)
Affinity DataIC50: >100nMAssay Description:Tested for its binding affinity against Dopamine receptor D2; showed no appreciable affinity at concentration specifiedMore data for this Ligand-Target Pair
In DepthDetails Article
TargetD(2) dopamine receptor(Mus musculus (Mouse))
TBA

Curated by ChEMBL
LigandPNGBDBM50280819(1-{2-[4-(5-Fluoro-1H-indol-3-ylmethyl)-piperidin-1...)
Affinity DataIC50: >100nMAssay Description:Tested for its binding affinity against Dopamine receptor D2; showed no appreciable affinity at concentration specifiedMore data for this Ligand-Target Pair
In DepthDetails Article
TargetD(2) dopamine receptor(Mus musculus (Mouse))
TBA

Curated by ChEMBL
LigandPNGBDBM50280816(CHEMBL293729 | N-{2-[4-(5-Fluoro-1H-indol-3-ylmeth...)
Affinity DataIC50: >100nMAssay Description:Tested for its binding affinity against Dopamine receptor D2; showed no appreciable affinity at concentration specifiedMore data for this Ligand-Target Pair
In DepthDetails Article
TargetD(2) dopamine receptor(Mus musculus (Mouse))
TBA

Curated by ChEMBL
LigandPNGBDBM50280831(2-{2-[4-(5-Fluoro-1H-indol-3-ylmethyl)-piperidin-1...)
Affinity DataIC50: >100nMAssay Description:Tested for its binding affinity against Dopamine receptor D2; showed no appreciable affinity at concentration specifiedMore data for this Ligand-Target Pair
In DepthDetails Article
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