Affinity DataKi: 0.200nMAssay Description:Displacement of [3H]-spiperone from human dopamine D3 receptor expressed in CHO cell membranesMore data for this Ligand-Target Pair
Affinity DataKi: 0.400nMAssay Description:Displacement of [3H]spiperone from human dopamine D2S receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 0.5nMAssay Description:Antagonist activity at D3 receptor (unknown origin)More data for this Ligand-Target Pair
Affinity DataKi: 0.5nMAssay Description:Displacement of [3H]-spiperone from human dopamine D3 receptor expressed in CHO cell membranesMore data for this Ligand-Target Pair
Affinity DataKi: 0.550nMAssay Description:Displacement of [3H]spiperone from human dopamine D2S receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 0.590nMAssay Description:Displacement of [3H]spiperone from human dopamine D2S receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 0.600nMAssay Description:Antagonist activity at D3 receptor (unknown origin)More data for this Ligand-Target Pair
Affinity DataKi: 0.600nMAssay Description:Displacement of [3H]spiperone from human dopamine D2S receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 0.670nMAssay Description:Displacement of [3H]-spiperone from human dopamine D3 receptor expressed in CHO cell membranesMore data for this Ligand-Target Pair
Affinity DataKi: 0.700nMAssay Description:Displacement of [3H]-spiperone from human dopamine D3 receptor expressed in CHO cell membranesMore data for this Ligand-Target Pair
Affinity DataKi: 0.730nMAssay Description:Displacement of [3H]-spiperone from human dopamine D3 receptor expressed in CHO cell membranesMore data for this Ligand-Target Pair
Affinity DataKi: 0.760nMAssay Description:Displacement of [3H]spiperone from human dopamine D2S receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 0.800nMAssay Description:Displacement of [3H]spiperone from human dopamine D2S receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 0.900nMAssay Description:Displacement of [3H]-spiperone from human dopamine D3 receptor expressed in CHO cell membranesMore data for this Ligand-Target Pair
Affinity DataKi: 1nMAssay Description:Displacement of [3H]spiperone from human dopamine D2S receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 1nMAssay Description:Displacement of [3H]spiperone from human dopamine D2S receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 1nMAssay Description:Antagonist activity at D3 receptor (unknown origin)More data for this Ligand-Target Pair
Affinity DataKi: 1nMAssay Description:Antagonist activity at D3 receptor (unknown origin)More data for this Ligand-Target Pair
Affinity DataKi: 1.10nMAssay Description:Displacement of [3H]-spiperone from human dopamine D3 receptor expressed in CHO cell membranesMore data for this Ligand-Target Pair
Affinity DataKi: 1.10nMAssay Description:Displacement of [3H]spiperone from human dopamine D2S receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 1.10nMAssay Description:Displacement of [3H]-spiperone from human dopamine D3 receptor expressed in CHO cell membranesMore data for this Ligand-Target Pair
Affinity DataKi: 1.20nMAssay Description:Displacement of [3H]-spiperone from human dopamine D3 receptor expressed in CHO cell membranesMore data for this Ligand-Target Pair
Affinity DataKi: 1.30nMAssay Description:Displacement of [3H]-spiperone from human dopamine D3 receptor expressed in CHO cell membranesMore data for this Ligand-Target Pair
Affinity DataKi: 1.30nMAssay Description:Displacement of [3H]-spiperone from human dopamine D3 receptor expressed in CHO cell membranesMore data for this Ligand-Target Pair
Affinity DataKi: 1.30nMAssay Description:Displacement of [3H]-spiperone from human dopamine D3 receptor expressed in CHO cell membranesMore data for this Ligand-Target Pair
Affinity DataKi: 1.5nMAssay Description:Displacement of [3H]spiperone from human dopamine D2S receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 1.60nMAssay Description:Displacement of [3H]spiperone from human dopamine D2S receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 1.60nMAssay Description:Displacement of [3H]-spiperone from human dopamine D3 receptor expressed in CHO cell membranesMore data for this Ligand-Target Pair
Affinity DataKi: 1.60nMAssay Description:Binding affinity to histamine H4 receptor (unknown origin)More data for this Ligand-Target Pair
Affinity DataKi: 1.70nMAssay Description:Compound was evaluated for inhibition of recombinant human neprilysin(NEP).More data for this Ligand-Target Pair
Affinity DataKi: 1.80nMAssay Description:Displacement of [3H]-spiperone from human dopamine D3 receptor expressed in CHO cell membranesMore data for this Ligand-Target Pair
Affinity DataKi: 2nMAssay Description:Displacement of [3H]-spiperone from human dopamine D3 receptor expressed in CHO cell membranesMore data for this Ligand-Target Pair
Affinity DataKi: 2.20nMAssay Description:Compound was evaluated for inhibition of recombinant human neprilysin(NEP).More data for this Ligand-Target Pair
Affinity DataKi: 2.5nMAssay Description:Displacement of [3H]spiperone from human dopamine D2S receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 2.70nMAssay Description:Antagonist activity at H4 receptor in human SH-SY5Y cells assessed as inhibition of imetit-induced GTPgamma[35S] binding after 30 mins by microbeta s...More data for this Ligand-Target Pair
Affinity DataKi: 2.70nMAssay Description:Antagonist activity at human H4 receptor assessed as inhibition of imetit-induced GTPgamma[35S] binding after 30 mins by microbeta scintillation coun...More data for this Ligand-Target Pair
Affinity DataKi: 2.80nMAssay Description:Antagonist activity at D3 receptor (unknown origin)More data for this Ligand-Target Pair
Affinity DataKi: 3nMAssay Description:Antagonist activity at H4 receptor in human SH-SY5Y cells assessed as inhibition of imetit-induced GTPgamma[35S] binding after 30 mins by microbeta s...More data for this Ligand-Target Pair
Affinity DataKi: 3nMAssay Description:Antagonist activity at human H4 receptor expressed in CHO cells co-expressing Galphai2 assessed as inhibition of imetit-induced GTPgamma[35S] binding...More data for this Ligand-Target Pair
Affinity DataKi: 3.10nMAssay Description:Antagonist activity at D3 receptor (unknown origin)More data for this Ligand-Target Pair
Affinity DataKi: 3.10nMAssay Description:Displacement of [3H]spiperone from human dopamine D2S receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 3.5nMAssay Description:Displacement of [3H]-spiperone from human dopamine D3 receptor expressed in CHO cell membranesMore data for this Ligand-Target Pair
Affinity DataKi: 3.90nMAssay Description:Displacement of [3H]-spiperone from human dopamine D3 receptor expressed in CHO cell membranesMore data for this Ligand-Target Pair
Affinity DataKi: 4nMAssay Description:Antagonist activity at H4 receptor in human SH-SY5Y cells assessed as inhibition of imetit-induced GTPgamma[35S] binding after 30 mins by microbeta s...More data for this Ligand-Target Pair
Affinity DataKi: 4nMAssay Description:Antagonist activity at H4 receptor in human SH-SY5Y cells assessed as inhibition of imetit-induced GTPgamma[35S] binding after 30 mins by microbeta s...More data for this Ligand-Target Pair
Affinity DataKi: 4.70nMAssay Description:Compound was evaluated for inhibition of recombinant human neprilysin(NEP).More data for this Ligand-Target Pair
Affinity DataKi: 4.70nMAssay Description:Displacement of [3H]-spiperone from human dopamine D3 receptor expressed in CHO cell membranesMore data for this Ligand-Target Pair
Affinity DataKi: 4.80nMAssay Description:Antagonist activity at H3 receptor (unknown origin)More data for this Ligand-Target Pair
Affinity DataKi: 4.90nMAssay Description:Compound was evaluated for inhibition of recombinant human neprilysin(NEP).More data for this Ligand-Target Pair
Affinity DataKi: 5nMAssay Description:Displacement of [3H]-prazosin from human ADRA1A receptorMore data for this Ligand-Target Pair