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Found 564 with Last Name = 'diller' and Initial = 'dj'
TargetToxin B(Peptoclostridium difficile)
Genesis Biotechnology Group

Curated by ChEMBL
LigandPNGBDBM50454459(CHEMBL4215036)
Affinity DataIC50:  1nMAssay Description:Inhibition of C-terminal 6-His tagged recombinant Clostridium difficile toxin B catalytic fragment (Met1 to Leu543 residues) assessed as reduction in...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase JAK3(Homo sapiens (Human))
Ligand Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50311657(1-(9-(8-fluorochroman-4-yl)-8-oxo-8,9-dihydro-7H-p...)
Affinity DataIC50:  1nMAssay Description:Inhibition of human JAK3 (508-1124) by time resolved fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetToxin B(Peptoclostridium difficile)
Genesis Biotechnology Group

Curated by ChEMBL
LigandPNGBDBM50454500(CHEMBL4212258)
Affinity DataIC50:  3nMAssay Description:Inhibition of C-terminal 6-His tagged recombinant Clostridium difficile toxin B catalytic fragment (Met1 to Leu543 residues) assessed as reduction in...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetToxin B(Peptoclostridium difficile)
Genesis Biotechnology Group

Curated by ChEMBL
LigandPNGBDBM50454498(CHEMBL4215657)
Affinity DataIC50:  3nMAssay Description:Inhibition of C-terminal 6-His tagged recombinant Clostridium difficile toxin B catalytic fragment (Met1 to Leu543 residues) assessed as reduction in...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase JAK3(Homo sapiens (Human))
Ligand Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50311656(2-(6-fluoro-1H-benzo[d]imidazol-1-yl)-9-(8-fluoroc...)
Affinity DataIC50:  3nMAssay Description:Inhibition of human JAK3 (508-1124) by time resolved fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase JAK2(Homo sapiens (Human))
Ligand Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50311657(1-(9-(8-fluorochroman-4-yl)-8-oxo-8,9-dihydro-7H-p...)
Affinity DataIC50:  5nMAssay Description:Inhibition of human JAK2 (532-1132) by time resolved fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase JAK3(Homo sapiens (Human))
Ligand Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50311644(1-(9-(2,6-difluorobenzyl)-8-oxo-8,9-dihydro-7H-pur...)
Affinity DataIC50:  6nMAssay Description:Inhibition of human JAK3 (508-1124) by time resolved fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetToxin B(Peptoclostridium difficile)
Genesis Biotechnology Group

Curated by ChEMBL
LigandPNGBDBM50454497(CHEMBL4214079)
Affinity DataIC50:  7nMAssay Description:Inhibition of C-terminal 6-His tagged recombinant Clostridium difficile toxin B catalytic fragment (Met1 to Leu543 residues) assessed as reduction in...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase JAK3(Homo sapiens (Human))
Ligand Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50311640(1-(8-oxo-9-(tetrahydro-2H-pyran-4-yl)-8,9-dihydro-...)
Affinity DataIC50:  7nMAssay Description:Inhibition of human JAK3 (508-1124) by time resolved fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetToxin B(Peptoclostridium difficile)
Genesis Biotechnology Group

Curated by ChEMBL
LigandPNGBDBM50454486(CHEMBL4203819)
Affinity DataIC50:  9nMAssay Description:Inhibition of C-terminal 6-His tagged recombinant Clostridium difficile toxin B catalytic fragment (Met1 to Leu543 residues) assessed as reduction in...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase JAK3(Homo sapiens (Human))
Ligand Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50311639(2-(6-chloro-1H-benzo[d]imidazol-1-yl)-9-(tetrahydr...)
Affinity DataIC50:  14nMAssay Description:Inhibition of human JAK3 (508-1124) by time resolved fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase JAK3(Homo sapiens (Human))
Ligand Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50311655(2-(6-chloro-1H-benzo[d]imidazol-1-yl)-9-(8-fluoroc...)
Affinity DataIC50:  15nMAssay Description:Inhibition of human JAK3 (508-1124) by time resolved fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase JAK3(Homo sapiens (Human))
Ligand Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50311642(1-(9-(2,3-difluorobenzyl)-8-oxo-8,9-dihydro-7H-pur...)
Affinity DataIC50:  17nMAssay Description:Inhibition of human JAK3 (508-1124) by time resolved fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetToxin B(Peptoclostridium difficile)
Genesis Biotechnology Group

Curated by ChEMBL
LigandPNGBDBM50454504(CHEMBL4210388)
Affinity DataIC50:  18nMAssay Description:Inhibition of C-terminal 6-His tagged recombinant Clostridium difficile toxin B catalytic fragment (Met1 to Leu543 residues) assessed as reduction in...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase JAK2(Homo sapiens (Human))
Ligand Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50311656(2-(6-fluoro-1H-benzo[d]imidazol-1-yl)-9-(8-fluoroc...)
Affinity DataIC50:  26nMAssay Description:Inhibition of human JAK2 (532-1132) by time resolved fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase JAK3(Homo sapiens (Human))
Ligand Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50311653((R)-2-(1H-benzo[d]imidazol-1-yl)-9-(8-fluorochroma...)
Affinity DataIC50:  28nMAssay Description:Inhibition of human JAK3 (508-1124) by time resolved fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase JAK3(Homo sapiens (Human))
Ligand Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50311648((+/-)-2-(1H-benzo[d]imidazol-1-yl)-9-(6-fluorochro...)
Affinity DataIC50:  28nMAssay Description:Inhibition of human JAK3 (508-1124) by time resolved fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase JAK2(Homo sapiens (Human))
Ligand Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50311644(1-(9-(2,6-difluorobenzyl)-8-oxo-8,9-dihydro-7H-pur...)
Affinity DataIC50:  28nMAssay Description:Inhibition of human JAK2 (532-1132) by time resolved fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase JAK3(Homo sapiens (Human))
Ligand Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50311651((+/-)-2-(1H-benzo[d]imidazol-1-yl)-9-(8-fluorochro...)
Affinity DataIC50:  30nMAssay Description:Inhibition of human JAK3 (508-1124) by time resolved fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon receptor(Homo sapiens (Human))
Pharmacopeia

Curated by ChEMBL
LigandPNGBDBM50075780(4-[5-(4-Chloro-phenyl)-3-isopropyl-1H-pyrrol-2-yl]...)
Affinity DataIC50:  32nMAssay Description:Antagonist activity against glucagon receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase JAK3(Homo sapiens (Human))
Ligand Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50311638(2-(6-fluoro-1H-benzo[d]imidazol-1-yl)-9-(tetrahydr...)
Affinity DataIC50:  38nMAssay Description:Inhibition of human JAK3 (508-1124) by time resolved fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetToxin B(Peptoclostridium difficile)
Genesis Biotechnology Group

Curated by ChEMBL
LigandPNGBDBM50454503(CHEMBL4211420)
Affinity DataIC50:  42nMAssay Description:Inhibition of C-terminal 6-His tagged recombinant Clostridium difficile toxin B catalytic fragment (Met1 to Leu543 residues) assessed as reduction in...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetToxin B(Peptoclostridium difficile)
Genesis Biotechnology Group

Curated by ChEMBL
LigandPNGBDBM50454498(CHEMBL4215657)
Affinity DataIC50:  43nMAssay Description:Inhibition of Clostridium difficile toxin B transfected in CHO cells assessed as reduction in caspase 3/7 activation pre-incubated for 1 hr before Tc...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase JAK3(Homo sapiens (Human))
Ligand Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50311647((+/-)-2-(1H-benzo[d]imidazol-1-yl)-9-(5-fluorochro...)
Affinity DataIC50:  48nMAssay Description:Inhibition of human JAK3 (508-1124) by time resolved fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetToxin B(Peptoclostridium difficile)
Genesis Biotechnology Group

Curated by ChEMBL
LigandPNGBDBM50454502(CHEMBL4209041)
Affinity DataIC50:  50nMAssay Description:Inhibition of C-terminal 6-His tagged recombinant Clostridium difficile toxin B catalytic fragment (Met1 to Leu543 residues) assessed as reduction in...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetLuciferin 4-monooxygenase(Photinus pyralis)
National Human Genome Research Institute

Curated by ChEMBL
LigandPNGBDBM50478348(CHEMBL406835)
Affinity DataIC50:  50nMAssay Description:Inhibition of Photinus pyralis luciferaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase JAK2(Homo sapiens (Human))
Ligand Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50311655(2-(6-chloro-1H-benzo[d]imidazol-1-yl)-9-(8-fluoroc...)
Affinity DataIC50:  56nMAssay Description:Inhibition of human JAK2 (532-1132) by time resolved fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLuciferin 4-monooxygenase(Photinus pyralis)
National Human Genome Research Institute

Curated by ChEMBL
LigandPNGBDBM50478348(CHEMBL406835)
Affinity DataIC50:  60nMAssay Description:Inhibition of Photinus pyralis luciferase by Steady-Glo reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase JAK3(Homo sapiens (Human))
Ligand Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50311637(9-(tetrahydro-2H-pyran-4-yl)-2-(6-(trifluoromethyl...)
Affinity DataIC50:  68nMAssay Description:Inhibition of human JAK3 (508-1124) by time resolved fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase JAK3(Homo sapiens (Human))
Ligand Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50311643(9-(2,6-difluorobenzyl)-2-(6-fluoro-1H-benzo[d]imid...)
Affinity DataIC50:  70nMAssay Description:Inhibition of human JAK3 (508-1124) by time resolved fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetToxin B(Peptoclostridium difficile)
Genesis Biotechnology Group

Curated by ChEMBL
LigandPNGBDBM50454501(CHEMBL4214697)
Affinity DataIC50:  78nMAssay Description:Inhibition of C-terminal 6-His tagged recombinant Clostridium difficile toxin B catalytic fragment (Met1 to Leu543 residues) assessed as reduction in...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetLuciferin 4-monooxygenase(Photinus pyralis)
National Human Genome Research Institute

Curated by ChEMBL
LigandPNGBDBM50238208(2,4-dimethoxy-N-(5-methylpyridin-2-yl)benzamide | ...)
Affinity DataIC50:  80nMAssay Description:Inhibition of Photinus pyralis luciferaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLuciferin 4-monooxygenase(Photinus pyralis)
National Human Genome Research Institute

Curated by ChEMBL
LigandPNGBDBM50478343(CHEMBL258888 | CID 2260658)
Affinity DataIC50:  80nMAssay Description:Inhibition of Photinus pyralis luciferase by BrightGlo reporter gene assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetLuciferin 4-monooxygenase(Photinus pyralis)
National Human Genome Research Institute

Curated by ChEMBL
LigandPNGBDBM50478343(CHEMBL258888 | CID 2260658)
Affinity DataIC50:  80nMAssay Description:Inhibition of Photinus pyralis luciferaseMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase JAK2(Homo sapiens (Human))
Ligand Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50311648((+/-)-2-(1H-benzo[d]imidazol-1-yl)-9-(6-fluorochro...)
Affinity DataIC50:  83nMAssay Description:Inhibition of human JAK2 (532-1132) by time resolved fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Pharmacopeia

Curated by ChEMBL
LigandPNGBDBM50075782(4-[4-(4-Fluoro-phenyl)-5-pyridin-4-yl-1H-pyrrol-2-...)
Affinity DataIC50:  90nMAssay Description:Inhibitiory activity against Mitogen-activated protein kinase 14, p38-alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLuciferin 4-monooxygenase(Photinus pyralis)
National Human Genome Research Institute

Curated by ChEMBL
LigandPNGBDBM50478348(CHEMBL406835)
Affinity DataIC50:  90nMAssay Description:Inhibition of Photinus pyralis luciferase by BrightGlo reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase JAK3(Homo sapiens (Human))
Ligand Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50311646((+/-)-2-(1H-benzo[d]imidazol-1-yl)-9-(chroman-4-yl...)
Affinity DataIC50:  95nMAssay Description:Inhibition of human JAK3 (508-1124) by time resolved fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase JAK2(Homo sapiens (Human))
Ligand Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50311650((+/-)-2-(1H-benzo[d]imidazol-1-yl)-9-(7-fluorochro...)
Affinity DataIC50:  95nMAssay Description:Inhibition of human JAK2 (532-1132) by time resolved fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase JAK2(Homo sapiens (Human))
Ligand Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50311647((+/-)-2-(1H-benzo[d]imidazol-1-yl)-9-(5-fluorochro...)
Affinity DataIC50:  97nMAssay Description:Inhibition of human JAK2 (532-1132) by time resolved fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLuciferin 4-monooxygenase(Photinus pyralis)
National Human Genome Research Institute

Curated by ChEMBL
LigandPNGBDBM39025(2-[5-(2-naphthyl)-1,2,4-oxadiazol-3-yl]pyridine | ...)
Affinity DataIC50:  100nMAssay Description:Inhibition of Photinus pyralis luciferaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLuciferin 4-monooxygenase(Photinus pyralis)
National Human Genome Research Institute

Curated by ChEMBL
LigandPNGBDBM50238226(2-(5-biphenyl-4-yl-[1,2,4]oxadiazol-3-yl)-pyridine...)
Affinity DataIC50:  100nMAssay Description:Inhibition of Photinus pyralis luciferaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase JAK3(Homo sapiens (Human))
Ligand Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50311641(9-(2,3-difluorobenzyl)-2-(6-fluoro-1H-benzo[d]imid...)
Affinity DataIC50:  108nMAssay Description:Inhibition of human JAK3 (508-1124) by time resolved fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase JAK3(Homo sapiens (Human))
Ligand Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50311635(2-(1H-benzo[d]imidazol-1-yl)-9-(tetrahydro-2H-pyra...)
Affinity DataIC50:  115nMAssay Description:Inhibition of human JAK3 (508-1124) by time resolved fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLuciferin 4-monooxygenase(Photinus pyralis)
National Human Genome Research Institute

Curated by ChEMBL
LigandPNGBDBM37601(3-(1H-benzimidazol-2-yl)-7-(diethylamino)-1-benzop...)
Affinity DataIC50:  120nMAssay Description:Inhibition of Photinus pyralis luciferase by Steady-Glo reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLuciferin 4-monooxygenase(Photinus pyralis)
National Human Genome Research Institute

Curated by ChEMBL
LigandPNGBDBM50238226(2-(5-biphenyl-4-yl-[1,2,4]oxadiazol-3-yl)-pyridine...)
Affinity DataIC50:  140nMAssay Description:Inhibition of Photinus pyralis luciferase by Steady-Glo reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLuciferin 4-monooxygenase(Photinus pyralis)
National Human Genome Research Institute

Curated by ChEMBL
LigandPNGBDBM39048(5-(2-chloranyl-4-methyl-phenyl)-3-phenyl-1,2,4-oxa...)
Affinity DataIC50:  150nMAssay Description:Inhibition of Photinus pyralis luciferaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLuciferin 4-monooxygenase(Photinus pyralis)
National Human Genome Research Institute

Curated by ChEMBL
LigandPNGBDBM38943(2-(1,3-benzothiazol-2-yl)-1-phthalazinone | 2-(1,3...)
Affinity DataIC50:  150nMAssay Description:Inhibition of Photinus pyralis luciferase by Easy lite assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLuciferin 4-monooxygenase(Photinus pyralis)
National Human Genome Research Institute

Curated by ChEMBL
LigandPNGBDBM50293101(5-(2,4-dimethoxyphenyl)-3-phenyl-1,2,4-oxadiazole ...)
Affinity DataIC50:  150nMAssay Description:Inhibition of Photinus pyralis luciferaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLuciferin 4-monooxygenase(Photinus pyralis)
National Human Genome Research Institute

Curated by ChEMBL
LigandPNGBDBM39048(5-(2-chloranyl-4-methyl-phenyl)-3-phenyl-1,2,4-oxa...)
Affinity DataIC50:  160nMAssay Description:Inhibition of Photinus pyralis luciferase by Steady-Glo reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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