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Found 815 with Last Name = 'distinto' and Initial = 's'
TargetCannabinoid receptor 2(Homo sapiens (Human))
University Of Innsbruck

Curated by ChEMBL
LigandPNGBDBM50180036((6aR,10aR)-3-(1,1-dimethylbutyl)-6a,7,10,10a-tetra...)
Affinity DataKi:  0.0230nMAssay Description:Displacement of [3H]CP-55940 from human recombinant CB2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 2(Homo sapiens (Human))
University Of Cagliari

Curated by ChEMBL
LigandPNGBDBM50106422(CHEMBL3601892)
Affinity DataKi:  0.0700nMAssay Description:Inhibition of human carbonic anhydrase-2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(MOUSE)
Uos Of Cagliari

Curated by ChEMBL
LigandPNGBDBM50180022(5-(4-chloro-3-methyl-phenyl)-1-(4-methyl-benzyl)-1...)
Affinity DataKi:  0.280nMAssay Description:Displacement of [3H]-CP-55940 from cannabinoid CB2 receptor in CD1 mouse spleen membranes after 1 hr by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 12(Homo sapiens (Human))
University Of Cagliari

Curated by ChEMBL
LigandPNGBDBM50106422(CHEMBL3601892)
Affinity DataKi:  0.460nMAssay Description:Inhibition of human carbonic anhydrase-12More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
University Of Innsbruck

Curated by ChEMBL
LigandPNGBDBM50180036((6aR,10aR)-3-(1,1-dimethylbutyl)-6a,7,10,10a-tetra...)
Affinity DataKi:  0.797nMAssay Description:Displacement of [3H]CP-55940 from human recombinant CB1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] B(Bos taurus)
Universit?????? Degli Studi Di Roma "La Sapienza

Curated by ChEMBL
LigandPNGBDBM50476106(CHEMBL385117)
Affinity DataKi:  0.813nMAssay Description:Inhibition of bovine brain mitochondria MAOBMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
University Of Innsbruck

Curated by ChEMBL
LigandPNGBDBM50228072(1,9-dihydroxy-3-(1',1'-dimethylheptyl)-6H-benzo[c]...)
Affinity DataKi:  0.820nMAssay Description:Displacement of [3H]CP-55940 from human recombinant CB2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] B(Bos taurus)
Universit?????? Degli Studi Di Roma "La Sapienza

Curated by ChEMBL
LigandPNGBDBM11014((-)-(S)1 | (5S)-5-(4-chlorophenyl)-3-(4-methylphen...)
Affinity DataKi:  1nM ΔG°:  -53.6kJ/molepH: 7.4 T: 2°CAssay Description:MAO A and MAO B activities were determined spectrophotometrically using kynuramine as substrates. Fluorimetric measurements were recorded with a Perk...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(MOUSE)
Uos Of Cagliari

Curated by ChEMBL
LigandPNGBDBM50000092((-)-(etorphine) | (-)-morphine | (1S,5R,13R,14S)-1...)
Affinity DataKi:  1.20nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in CD1 mouse brain membranes after 1 hr by liquid scintillation countingMore data for this Ligand-Target Pair
TargetMu-type opioid receptor(MOUSE)
Uos Of Cagliari

Curated by ChEMBL
LigandPNGBDBM50000092((-)-(etorphine) | (-)-morphine | (1S,5R,13R,14S)-1...)
Affinity DataKi:  1.20nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in CD1 mouse whole brain minus cerebellum membranes by liquid scintillation countingMore data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] B(Bos taurus)
Universit?????? Degli Studi Di Roma "La Sapienza

Curated by ChEMBL
LigandPNGBDBM50476100(CHEMBL220548)
Affinity DataKi:  1.30nMAssay Description:Inhibition of bovine brain mitochondria MAOBMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
University Of Innsbruck

Curated by ChEMBL
LigandPNGBDBM50265650(2-(N-(2,5-dimethoxyphenyl)-4-methylphenylsulfonami...)
Affinity DataKi:  1.35nMAssay Description:Displacement of [3H]CP-55940 from human recombinant CB2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] B(Bos taurus)
Universit?????? Degli Studi Di Roma "La Sapienza

Curated by ChEMBL
LigandPNGBDBM11004(1-thiocarbamoyl-3,5-diaryl-4,5-dihydro-(1H)-pyrazo...)
Affinity DataKi:  1.5nM ΔG°:  -52.6kJ/molepH: 7.4 T: 2°CAssay Description:MAO A and MAO B activities were determined spectrophotometrically using kynuramine as substrates. Fluorimetric measurements were recorded with a Perk...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
University Of Innsbruck

Curated by ChEMBL
LigandPNGBDBM50265648(8-hexyl-3,5,5-trimethyl-2,3,4,5-tetrahydro-1H-chro...)
Affinity DataKi:  1.78nMAssay Description:Displacement of [3H]CP-55940 from human recombinant CB2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 1(Homo sapiens (Human))
University Of Cagliari

Curated by ChEMBL
LigandPNGBDBM50106422(CHEMBL3601892)
Affinity DataKi:  1.80nMAssay Description:Inhibition of human carbonic anhydrase-1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
University Of Innsbruck

Curated by ChEMBL
LigandPNGBDBM50265687(CHEMBL496781 | N-(2-ethylphenyl)-2-(5-(2-methoxyph...)
Affinity DataKi:  2.10nMAssay Description:Displacement of [3H]CP-55940 from human recombinant CB2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 12(Homo sapiens (Human))
University Of Cagliari

Curated by ChEMBL
LigandPNGBDBM50367288(CHEMBL4175989)
Affinity DataKi:  2.40nMAssay Description:Binding affinity to human carbonic anhydrase 12 by stopped flow CO2 hydration methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] B(Bos taurus)
Universit?????? Degli Studi Di Roma "La Sapienza

Curated by ChEMBL
LigandPNGBDBM11015((+)-(R)1 | (5R)-5-(4-chlorophenyl)-3-(4-methylphen...)
Affinity DataKi:  2.70nM ΔG°:  -51.0kJ/molepH: 7.4 T: 2°CAssay Description:MAO A and MAO B activities were determined spectrophotometrically using kynuramine as substrates. Fluorimetric measurements were recorded with a Perk...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 12(Homo sapiens (Human))
University Of Cagliari

Curated by ChEMBL
LigandPNGBDBM50367330(CHEMBL4168142)
Affinity DataKi:  3.40nMAssay Description:Binding affinity to human carbonic anhydrase 12 by stopped flow CO2 hydration methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
University Of Innsbruck

Curated by ChEMBL
LigandPNGBDBM50180036((6aR,10aR)-3-(1,1-dimethylbutyl)-6a,7,10,10a-tetra...)
Affinity DataKi:  3.40nMAssay Description:Binding affinity to CB2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 12(Homo sapiens (Human))
University Of Cagliari

Curated by ChEMBL
LigandPNGBDBM50367290(CHEMBL4160871)
Affinity DataKi:  3.60nMAssay Description:Binding affinity to human carbonic anhydrase 12 by stopped flow CO2 hydration methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] A(Bos taurus)
Sapienza University of Rome

LigandPNGBDBM11006(1-thiocarbamoyl-3,5-diaryl-4,5-dihydro-(1H)-pyrazo...)
Affinity DataKi:  4nM ΔG°:  -50.0kJ/molepH: 7.4 T: 2°CAssay Description:MAO A and MAO B activities were determined spectrophotometrically using kynuramine as substrates. Fluorimetric measurements were recorded with a Perk...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] B(Bos taurus)
Universit?????? Degli Studi Di Roma "La Sapienza

Curated by ChEMBL
LigandPNGBDBM50476107(CHEMBL375007)
Affinity DataKi:  4.10nMAssay Description:Inhibition of bovine brain mitochondria MAOBMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 12(Homo sapiens (Human))
University Of Cagliari

Curated by ChEMBL
LigandPNGBDBM50271176(CHEMBL4130085)
Affinity DataKi:  5nMAssay Description:Inhibition of recombinant human carbonic anhydrase 12 assessed as reduction in CO2 hydration pretreated for 15 mins followed by CO2 addition measured...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] A(Bos taurus)
Sapienza University of Rome

LigandPNGBDBM11016((-)-(S)4 | (5S)-5-(4-chlorophenyl)-3-(4-fluorophen...)
Affinity DataKi:  5nM ΔG°:  -49.4kJ/molepH: 7.4 T: 2°CAssay Description:MAO A and MAO B activities were determined spectrophotometrically using kynuramine as substrates. Fluorimetric measurements were recorded with a Perk...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 12(Homo sapiens (Human))
University Of Cagliari

Curated by ChEMBL
LigandPNGBDBM50271193(CHEMBL4129969)
Affinity DataKi:  5.20nMAssay Description:Inhibition of recombinant human carbonic anhydrase 12 assessed as reduction in CO2 hydration pretreated for 15 mins followed by CO2 addition measured...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 12(Homo sapiens (Human))
University Of Cagliari

Curated by ChEMBL
LigandPNGBDBM50106418(CHEMBL3601889)
Affinity DataKi:  5.30nMAssay Description:Inhibition of human carbonic anhydrase-12More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 12(Homo sapiens (Human))
University Of Cagliari

Curated by ChEMBL
LigandPNGBDBM50106416(CHEMBL3601887)
Affinity DataKi:  5.5nMAssay Description:Inhibition of human carbonic anhydrase-12More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 12(Homo sapiens (Human))
University Of Cagliari

Curated by ChEMBL
LigandPNGBDBM10880(AZA | AZA2 | AZM acetazolamide | Acerazolamide, AA...)
Affinity DataKi:  5.70nMAssay Description:Inhibition of recombinant human carbonic anhydrase 12 assessed as reduction in CO2 hydration pretreated for 15 mins followed by CO2 addition measured...More data for this Ligand-Target Pair
TargetCarbonic anhydrase 12(Homo sapiens (Human))
University Of Cagliari

Curated by ChEMBL
LigandPNGBDBM10880(AZA | AZA2 | AZM acetazolamide | Acerazolamide, AA...)
Affinity DataKi:  5.70nMAssay Description:Inhibition of human carbonic anhydrase-12More data for this Ligand-Target Pair
TargetCarbonic anhydrase 12(Homo sapiens (Human))
University Of Cagliari

Curated by ChEMBL
LigandPNGBDBM10880(AZA | AZA2 | AZM acetazolamide | Acerazolamide, AA...)
Affinity DataKi:  5.70nMAssay Description:Inhibition of recombinant human carbonic anhydrase 12 incubated for 6 hrs prior to testing measured for 10 to 100 secs by phenol red-based stopped-fl...More data for this Ligand-Target Pair
TargetCarbonic anhydrase 12(Homo sapiens (Human))
University Of Cagliari

Curated by ChEMBL
LigandPNGBDBM10880(AZA | AZA2 | AZM acetazolamide | Acerazolamide, AA...)
Affinity DataKi:  5.70nMAssay Description:Binding affinity to human carbonic anhydrase 12 by stopped flow CO2 hydration methodMore data for this Ligand-Target Pair
TargetCarbonic anhydrase 12(Homo sapiens (Human))
University Of Cagliari

Curated by ChEMBL
LigandPNGBDBM50106419(CHEMBL3601886)
Affinity DataKi:  5.80nMAssay Description:Inhibition of human carbonic anhydrase-12More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] B(Bos taurus)
Universit?????? Degli Studi Di Roma "La Sapienza

Curated by ChEMBL
LigandPNGBDBM11010(1-thiocarbamoyl-3,5-diaryl-4,5-dihydro-(1H)-pyrazo...)
Affinity DataKi:  6nM ΔG°:  -49.0kJ/molepH: 7.4 T: 2°CAssay Description:MAO A and MAO B activities were determined spectrophotometrically using kynuramine as substrates. Fluorimetric measurements were recorded with a Perk...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 12(Homo sapiens (Human))
University Of Cagliari

Curated by ChEMBL
LigandPNGBDBM10880(AZA | AZA2 | AZM acetazolamide | Acerazolamide, AA...)
Affinity DataKi:  6nMAssay Description:Inhibition of human CA12 by Lineweaver-Burk plot analysisMore data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] A(Bos taurus)
Sapienza University of Rome

LigandPNGBDBM11005(1-thiocarbamoyl-3,5-diaryl-4,5-dihydro-(1H)-pyrazo...)
Affinity DataKi:  6nM ΔG°:  -49.0kJ/molepH: 7.4 T: 2°CAssay Description:MAO A and MAO B activities were determined spectrophotometrically using kynuramine as substrates. Fluorimetric measurements were recorded with a Perk...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] A(Bos taurus)
Sapienza University of Rome

LigandPNGBDBM11007(1-thiocarbamoyl-3,5-diaryl-4,5-dihydro-(1H)-pyrazo...)
Affinity DataKi:  6nM ΔG°:  -49.0kJ/molepH: 7.4 T: 2°CAssay Description:MAO A and MAO B activities were determined spectrophotometrically using kynuramine as substrates. Fluorimetric measurements were recorded with a Perk...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
University Of Innsbruck

Curated by ChEMBL
LigandPNGBDBM50265747((4-methylnaphthalen-1-yl)(1-propyl-1H-indol-3-yl)m...)
Affinity DataKi:  6.10nMAssay Description:Displacement of [3H]CP-55940 from human recombinant CB2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 12(Homo sapiens (Human))
University Of Cagliari

Curated by ChEMBL
LigandPNGBDBM50106423(CHEMBL3601891)
Affinity DataKi:  6.10nMAssay Description:Inhibition of human carbonic anhydrase-12More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 12(Homo sapiens (Human))
University Of Cagliari

Curated by ChEMBL
LigandPNGBDBM50271194(CHEMBL4127617)
Affinity DataKi:  6.20nMAssay Description:Inhibition of recombinant human carbonic anhydrase 12 assessed as reduction in CO2 hydration pretreated for 15 mins followed by CO2 addition measured...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 12(Homo sapiens (Human))
University Of Cagliari

Curated by ChEMBL
LigandPNGBDBM50106424(CHEMBL3601890)
Affinity DataKi:  6.20nMAssay Description:Inhibition of human carbonic anhydrase-12More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 12(Homo sapiens (Human))
University Of Cagliari

Curated by ChEMBL
LigandPNGBDBM50271182(CHEMBL4129897)
Affinity DataKi:  6.30nMAssay Description:Inhibition of recombinant human carbonic anhydrase 12 assessed as reduction in CO2 hydration pretreated for 15 mins followed by CO2 addition measured...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 12(Homo sapiens (Human))
University Of Cagliari

Curated by ChEMBL
LigandPNGBDBM50106421(CHEMBL3601893)
Affinity DataKi:  6.30nMAssay Description:Inhibition of human carbonic anhydrase-12More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 12(Homo sapiens (Human))
University Of Cagliari

Curated by ChEMBL
LigandPNGBDBM50106413(CHEMBL3601883)
Affinity DataKi:  6.40nMAssay Description:Inhibition of human carbonic anhydrase-12More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 12(Homo sapiens (Human))
University Of Cagliari

Curated by ChEMBL
LigandPNGBDBM50106420(CHEMBL3601885)
Affinity DataKi:  6.70nMAssay Description:Inhibition of human carbonic anhydrase-12More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 12(Homo sapiens (Human))
University Of Cagliari

Curated by ChEMBL
LigandPNGBDBM50271198(CHEMBL4126627)
Affinity DataKi:  6.70nMAssay Description:Inhibition of recombinant human carbonic anhydrase 12 assessed as reduction in CO2 hydration pretreated for 15 mins followed by CO2 addition measured...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 12(Homo sapiens (Human))
University Of Cagliari

Curated by ChEMBL
LigandPNGBDBM50271196(CHEMBL4126396)
Affinity DataKi:  6.80nMAssay Description:Inhibition of recombinant human carbonic anhydrase 12 assessed as reduction in CO2 hydration pretreated for 15 mins followed by CO2 addition measured...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 12(Homo sapiens (Human))
University Of Cagliari

Curated by ChEMBL
LigandPNGBDBM50271202(CHEMBL4126466)
Affinity DataKi:  6.80nMAssay Description:Inhibition of recombinant human carbonic anhydrase 12 assessed as reduction in CO2 hydration pretreated for 15 mins followed by CO2 addition measured...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 12(Homo sapiens (Human))
University Of Cagliari

Curated by ChEMBL
LigandPNGBDBM50106412(CHEMBL3601884)
Affinity DataKi:  7nMAssay Description:Inhibition of human carbonic anhydrase-12More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] A(Bos taurus)
Sapienza University of Rome

LigandPNGBDBM11008(1-thiocarbamoyl-3,5-diaryl-4,5-dihydro-(1H)-pyrazo...)
Affinity DataKi:  7nM ΔG°:  -48.6kJ/molepH: 7.4 T: 2°CAssay Description:MAO A and MAO B activities were determined spectrophotometrically using kynuramine as substrates. Fluorimetric measurements were recorded with a Perk...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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