TargetNeutrophil elastase(Homo sapiens (Human))
Sterling Winthrop Pharmaceutical Research Division
Curated by ChEMBL
Sterling Winthrop Pharmaceutical Research Division
Curated by ChEMBL
Affinity DataKi: 0.00700nMAssay Description:In vitro inhibition constant of human leukocyte elastase.More data for this Ligand-Target Pair
TargetNeutrophil elastase(Homo sapiens (Human))
Sterling Winthrop Pharmaceutical Research Division
Curated by ChEMBL
Sterling Winthrop Pharmaceutical Research Division
Curated by ChEMBL
Affinity DataKi: 0.00800nMAssay Description:In vitro inhibition constant of human leukocyte elastase.More data for this Ligand-Target Pair
TargetNeutrophil elastase(Homo sapiens (Human))
Sterling Winthrop Pharmaceutical Research Division
Curated by ChEMBL
Sterling Winthrop Pharmaceutical Research Division
Curated by ChEMBL
Affinity DataKi: 0.0100nMAssay Description:In vitro inhibition constant of human leukocyte elastase.More data for this Ligand-Target Pair
TargetNeutrophil elastase(Homo sapiens (Human))
Sterling Winthrop Pharmaceutical Research Division
Curated by ChEMBL
Sterling Winthrop Pharmaceutical Research Division
Curated by ChEMBL
Affinity DataKi: 0.0300nMAssay Description:In vitro inhibition constant of human leukocyte elastase.More data for this Ligand-Target Pair
TargetNeutrophil elastase(Homo sapiens (Human))
Sterling Winthrop Pharmaceutical Research Division
Curated by ChEMBL
Sterling Winthrop Pharmaceutical Research Division
Curated by ChEMBL
Affinity DataKi: 0.0600nMAssay Description:In vitro inhibition constant of human leukocyte elastase.More data for this Ligand-Target Pair
TargetNeutrophil elastase(Homo sapiens (Human))
Sterling Winthrop Pharmaceutical Research Division
Curated by ChEMBL
Sterling Winthrop Pharmaceutical Research Division
Curated by ChEMBL
Affinity DataKi: 0.170nMAssay Description:In vitro inhibition constant of human leukocyte elastase.More data for this Ligand-Target Pair
TargetNeutrophil elastase(Homo sapiens (Human))
Sterling Winthrop Pharmaceutical Research Division
Curated by ChEMBL
Sterling Winthrop Pharmaceutical Research Division
Curated by ChEMBL
Affinity DataKi: 1nMAssay Description:In vitro inhibition constant of human leukocyte elastase.More data for this Ligand-Target Pair
TargetNeutrophil elastase(Homo sapiens (Human))
Sterling Winthrop Pharmaceutical Research Division
Curated by ChEMBL
Sterling Winthrop Pharmaceutical Research Division
Curated by ChEMBL
Affinity DataKi: 2nMAssay Description:In vitro inhibition constant of human leukocyte elastase.More data for this Ligand-Target Pair
TargetNeutrophil elastase(Homo sapiens (Human))
Sterling Winthrop Pharmaceutical Research Division
Curated by ChEMBL
Sterling Winthrop Pharmaceutical Research Division
Curated by ChEMBL
Affinity DataKi: 2.70nMAssay Description:In vitro inhibition constant of human leukocyte elastase.More data for this Ligand-Target Pair
TargetNeutrophil elastase(Homo sapiens (Human))
Sterling Winthrop Pharmaceutical Research Division
Curated by ChEMBL
Sterling Winthrop Pharmaceutical Research Division
Curated by ChEMBL
Affinity DataKi: 4nMAssay Description:In vitro inhibition constant of human leukocyte elastase.More data for this Ligand-Target Pair
TargetNeutrophil elastase(Homo sapiens (Human))
Sterling Winthrop Pharmaceutical Research Division
Curated by ChEMBL
Sterling Winthrop Pharmaceutical Research Division
Curated by ChEMBL
Affinity DataKi: 8nMAssay Description:In vitro inhibition constant of human leukocyte elastase.More data for this Ligand-Target Pair
TargetNeutrophil elastase(Homo sapiens (Human))
Sterling Winthrop Pharmaceutical Research Division
Curated by ChEMBL
Sterling Winthrop Pharmaceutical Research Division
Curated by ChEMBL
Affinity DataKi: 8nMAssay Description:In vitro inhibition constant of human leukocyte elastase.More data for this Ligand-Target Pair
TargetNeutrophil elastase(Homo sapiens (Human))
Sterling Winthrop Pharmaceutical Research Division
Curated by ChEMBL
Sterling Winthrop Pharmaceutical Research Division
Curated by ChEMBL
Affinity DataKi: 8.5nMAssay Description:In vitro inhibition constant of human leukocyte elastase.More data for this Ligand-Target Pair
TargetNeutrophil elastase(Homo sapiens (Human))
Sterling Winthrop Pharmaceutical Research Division
Curated by ChEMBL
Sterling Winthrop Pharmaceutical Research Division
Curated by ChEMBL
Affinity DataKi: 18nMAssay Description:In vitro inhibition constant of human leukocyte elastase.More data for this Ligand-Target Pair
TargetNeutrophil elastase(Homo sapiens (Human))
Sterling Winthrop Pharmaceutical Research Division
Curated by ChEMBL
Sterling Winthrop Pharmaceutical Research Division
Curated by ChEMBL
Affinity DataKi: 26nMAssay Description:In vitro inhibition constant of human leukocyte elastase.More data for this Ligand-Target Pair
TargetNeutrophil elastase(Homo sapiens (Human))
Sterling Winthrop Pharmaceutical Research Division
Curated by ChEMBL
Sterling Winthrop Pharmaceutical Research Division
Curated by ChEMBL
Affinity DataKi: 31nMAssay Description:In vitro inhibition constant of human leukocyte elastase.More data for this Ligand-Target Pair
TargetNeutrophil elastase(Homo sapiens (Human))
Sterling Winthrop Pharmaceutical Research Division
Curated by ChEMBL
Sterling Winthrop Pharmaceutical Research Division
Curated by ChEMBL
Affinity DataKi: 37nMAssay Description:In vitro inhibition constant of human leukocyte elastase.More data for this Ligand-Target Pair
TargetNeutrophil elastase(Homo sapiens (Human))
Sterling Winthrop Pharmaceutical Research Division
Curated by ChEMBL
Sterling Winthrop Pharmaceutical Research Division
Curated by ChEMBL
Affinity DataKi: 102nMAssay Description:In vitro inhibition constant of human leukocyte elastase.More data for this Ligand-Target Pair
Affinity DataIC50: 0.120nMAssay Description:Inhibition of [125]I-Bolton Hunter Substance P([125]I-BHSP) binding to standard Tachykinin receptor 1 from rat forebrain membranes.More data for this Ligand-Target Pair
TargetcGMP-inhibited 3',5'-cyclic phosphodiesterase 3A/3B(Homo sapiens (Human))
Sterling Winthrop Pharmaceuticals Research Division
Curated by ChEMBL
Sterling Winthrop Pharmaceuticals Research Division
Curated by ChEMBL
Affinity DataIC50: 18nMAssay Description:In vitro inhibitory activity against cAMP phosphodiesterase III in dog aortaMore data for this Ligand-Target Pair
TargetcGMP-inhibited 3',5'-cyclic phosphodiesterase 3A/3B(Homo sapiens (Human))
Sterling Winthrop Pharmaceuticals Research Division
Curated by ChEMBL
Sterling Winthrop Pharmaceuticals Research Division
Curated by ChEMBL
Affinity DataIC50: 20nMAssay Description:In vitro inhibitory activity against cAMP phosphodiesterase III in dog aortaMore data for this Ligand-Target Pair
TargetcGMP-inhibited 3',5'-cyclic phosphodiesterase 3A/3B(Homo sapiens (Human))
Sterling Winthrop Pharmaceuticals Research Division
Curated by ChEMBL
Sterling Winthrop Pharmaceuticals Research Division
Curated by ChEMBL
Affinity DataIC50: 23nMAssay Description:In vitro inhibitory activity against cAMP phosphodiesterase III in dog aortaMore data for this Ligand-Target Pair
Affinity DataIC50: 24nMAssay Description:Inhibition of [125]I-Bolton Hunter Substance P([125]I-BHSP) binding to standard Tachykinin receptor 1 from rat forebrain membranes.More data for this Ligand-Target Pair
TargetcGMP-inhibited 3',5'-cyclic phosphodiesterase 3A/3B(Homo sapiens (Human))
Sterling Winthrop Pharmaceuticals Research Division
Curated by ChEMBL
Sterling Winthrop Pharmaceuticals Research Division
Curated by ChEMBL
Affinity DataIC50: 24nMAssay Description:In vitro inhibitory activity against cAMP phosphodiesterase III in dog aortaMore data for this Ligand-Target Pair
Affinity DataIC50: 48nMAssay Description:Inhibition of [125]I-Bolton Hunter Substance P([125]I-BHSP) binding to standard Tachykinin receptor 1 from rat forebrain membranes.More data for this Ligand-Target Pair
Affinity DataIC50: 50nMAssay Description:Inhibition of [125]I-Bolton Hunter Substance P([125]I-BHSP) binding to standard Tachykinin receptor 1 from rat forebrain membranes.More data for this Ligand-Target Pair
TargetcGMP-inhibited 3',5'-cyclic phosphodiesterase 3A/3B(Homo sapiens (Human))
Sterling Winthrop Pharmaceuticals Research Division
Curated by ChEMBL
Sterling Winthrop Pharmaceuticals Research Division
Curated by ChEMBL
Affinity DataIC50: 69nMAssay Description:In vitro inhibitory activity against cAMP phosphodiesterase III in dog aortaMore data for this Ligand-Target Pair
TargetcGMP-inhibited 3',5'-cyclic phosphodiesterase 3A/3B(Homo sapiens (Human))
Sterling Winthrop Pharmaceuticals Research Division
Curated by ChEMBL
Sterling Winthrop Pharmaceuticals Research Division
Curated by ChEMBL
Affinity DataIC50: 78nMAssay Description:In vitro inhibitory activity against cAMP phosphodiesterase III in dog aortaMore data for this Ligand-Target Pair
Affinity DataIC50: 86nMAssay Description:Inhibition of [125]I-Bolton Hunter Substance P([125]I-BHSP) binding to standard Tachykinin receptor 1 from rat forebrain membranes.More data for this Ligand-Target Pair
TargetcGMP-inhibited 3',5'-cyclic phosphodiesterase 3A/3B(Homo sapiens (Human))
Sterling Winthrop Pharmaceuticals Research Division
Curated by ChEMBL
Sterling Winthrop Pharmaceuticals Research Division
Curated by ChEMBL
Affinity DataIC50: 100nMAssay Description:In vitro inhibitory activity against cAMP phosphodiesterase III in dog aortaMore data for this Ligand-Target Pair
TargetcGMP-inhibited 3',5'-cyclic phosphodiesterase 3A/3B(Homo sapiens (Human))
Sterling Winthrop Pharmaceuticals Research Division
Curated by ChEMBL
Sterling Winthrop Pharmaceuticals Research Division
Curated by ChEMBL
Affinity DataIC50: 140nMAssay Description:In vitro inhibitory activity against cAMP phosphodiesterase III in dog aortaMore data for this Ligand-Target Pair
TargetcGMP-inhibited 3',5'-cyclic phosphodiesterase 3A/3B(Homo sapiens (Human))
Sterling Winthrop Pharmaceuticals Research Division
Curated by ChEMBL
Sterling Winthrop Pharmaceuticals Research Division
Curated by ChEMBL
Affinity DataIC50: 180nMAssay Description:In vitro inhibitory activity against cAMP phosphodiesterase III in dog aortaMore data for this Ligand-Target Pair
Affinity DataIC50: 180nMAssay Description:Inhibition of [125]I-Bolton Hunter Substance P([125]I-BHSP) binding to Tachykinin receptor 1 from rat forebrain membranes.More data for this Ligand-Target Pair
Affinity DataIC50: 200nMAssay Description:Inhibition of [125]I-Bolton Hunter Substance P([125]I-BHSP) binding to standard Tachykinin receptor 1 from rat forebrain membranes.More data for this Ligand-Target Pair
Affinity DataIC50: 220nMAssay Description:Inhibition of [125]I-Bolton Hunter Substance P([125]I-BHSP) binding to standard Tachykinin receptor 1 from rat forebrain membranes.More data for this Ligand-Target Pair
TargetcGMP-inhibited 3',5'-cyclic phosphodiesterase 3A/3B(Homo sapiens (Human))
Sterling Winthrop Pharmaceuticals Research Division
Curated by ChEMBL
Sterling Winthrop Pharmaceuticals Research Division
Curated by ChEMBL
Affinity DataIC50: 230nMAssay Description:In vitro inhibitory activity against cAMP phosphodiesterase III in dog aortaMore data for this Ligand-Target Pair
Affinity DataIC50: 320nMAssay Description:Inhibition of [125]I-Bolton Hunter Substance P([125]I-BHSP) binding to Tachykinin receptor 1 from rat forebrain membranes.More data for this Ligand-Target Pair
Affinity DataIC50: 320nMAssay Description:Inhibition of [125]I-Bolton Hunter Substance P([125]I-BHSP) binding to standard Tachykinin receptor 1 from rat forebrain membranes.More data for this Ligand-Target Pair
TargetcGMP-inhibited 3',5'-cyclic phosphodiesterase 3A/3B(Homo sapiens (Human))
Sterling Winthrop Pharmaceuticals Research Division
Curated by ChEMBL
Sterling Winthrop Pharmaceuticals Research Division
Curated by ChEMBL
Affinity DataIC50: 350nMAssay Description:In vitro inhibitory activity against cAMP phosphodiesterase III in dog aortaMore data for this Ligand-Target Pair
TargetcGMP-inhibited 3',5'-cyclic phosphodiesterase 3A/3B(Homo sapiens (Human))
Sterling Winthrop Pharmaceuticals Research Division
Curated by ChEMBL
Sterling Winthrop Pharmaceuticals Research Division
Curated by ChEMBL
Affinity DataIC50: 360nMAssay Description:In vitro inhibitory activity against cAMP phosphodiesterase III in dog aortaMore data for this Ligand-Target Pair
TargetcGMP-inhibited 3',5'-cyclic phosphodiesterase 3A/3B(Homo sapiens (Human))
Sterling Winthrop Pharmaceuticals Research Division
Curated by ChEMBL
Sterling Winthrop Pharmaceuticals Research Division
Curated by ChEMBL
Affinity DataIC50: 540nMAssay Description:In vitro inhibitory activity against cAMP phosphodiesterase III in dog aortaMore data for this Ligand-Target Pair
TargetcGMP-inhibited 3',5'-cyclic phosphodiesterase 3A/3B(Homo sapiens (Human))
Sterling Winthrop Pharmaceuticals Research Division
Curated by ChEMBL
Sterling Winthrop Pharmaceuticals Research Division
Curated by ChEMBL
Affinity DataIC50: 560nMAssay Description:In vitro inhibitory activity against cAMP phosphodiesterase III in dog aortaMore data for this Ligand-Target Pair
TargetcGMP-inhibited 3',5'-cyclic phosphodiesterase 3A/3B(Homo sapiens (Human))
Sterling Winthrop Pharmaceuticals Research Division
Curated by ChEMBL
Sterling Winthrop Pharmaceuticals Research Division
Curated by ChEMBL
Affinity DataIC50: 630nMAssay Description:In vitro inhibitory activity against cAMP phosphodiesterase III in dog aortaMore data for this Ligand-Target Pair
TargetcGMP-inhibited 3',5'-cyclic phosphodiesterase 3A/3B(Homo sapiens (Human))
Sterling Winthrop Pharmaceuticals Research Division
Curated by ChEMBL
Sterling Winthrop Pharmaceuticals Research Division
Curated by ChEMBL
Affinity DataIC50: 850nMAssay Description:In vitro inhibitory activity against cAMP phosphodiesterase III in dog aortaMore data for this Ligand-Target Pair
Affinity DataIC50: 1.20E+3nMAssay Description:Inhibition of [125]I-Bolton Hunter Substance P([125]I-BHSP) binding to standard Tachykinin receptor 1 from rat forebrain membranes.More data for this Ligand-Target Pair
TargetcGMP-inhibited 3',5'-cyclic phosphodiesterase 3A/3B(Homo sapiens (Human))
Sterling Winthrop Pharmaceuticals Research Division
Curated by ChEMBL
Sterling Winthrop Pharmaceuticals Research Division
Curated by ChEMBL
Affinity DataIC50: 1.30E+3nMAssay Description:In vitro inhibitory activity against cAMP phosphodiesterase III in dog aortaMore data for this Ligand-Target Pair
TargetcGMP-inhibited 3',5'-cyclic phosphodiesterase 3A/3B(Homo sapiens (Human))
Sterling Winthrop Pharmaceuticals Research Division
Curated by ChEMBL
Sterling Winthrop Pharmaceuticals Research Division
Curated by ChEMBL
Affinity DataIC50: 1.40E+3nMAssay Description:In vitro inhibitory activity against cAMP phosphodiesterase III in dog aortaMore data for this Ligand-Target Pair
Affinity DataIC50: 1.60E+3nMAssay Description:Inhibition of [125]I-Bolton Hunter Substance P([125]I-BHSP) binding to standard Tachykinin receptor 1 from rat forebrain membranes.More data for this Ligand-Target Pair
TargetcGMP-inhibited 3',5'-cyclic phosphodiesterase 3A/3B(Homo sapiens (Human))
Sterling Winthrop Pharmaceuticals Research Division
Curated by ChEMBL
Sterling Winthrop Pharmaceuticals Research Division
Curated by ChEMBL
Affinity DataIC50: 1.60E+3nMAssay Description:In vitro inhibitory activity against cAMP phosphodiesterase III in dog aortaMore data for this Ligand-Target Pair
TargetcGMP-inhibited 3',5'-cyclic phosphodiesterase 3A/3B(Homo sapiens (Human))
Sterling Winthrop Pharmaceuticals Research Division
Curated by ChEMBL
Sterling Winthrop Pharmaceuticals Research Division
Curated by ChEMBL
Affinity DataIC50: 2.00E+3nMAssay Description:In vitro inhibitory activity against cAMP phosphodiesterase III in dog aortaMore data for this Ligand-Target Pair