Compile Data Set for Download or QSAR
maximum 50k data
Found 3 Enz. Inhib. hit(s) with Target = 'Substance-P receptor' and Ligand = 'BDBM50002373'
TargetSubstance-P receptor(Rattus norvegicus (rat))
Rochester

Curated by ChEMBL
LigandPNGBDBM50002373(1-(1-ethynyl)-15a,17a-dimethyl-(1R,15aS,17aS)-2,3,...)
Affinity DataIC50:  24nMAssay Description:Inhibition of [125]I-Bolton Hunter Substance P([125]I-BHSP) binding to standard Tachykinin receptor 1 from rat forebrain membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(Rattus norvegicus (rat))
Rochester

Curated by ChEMBL
LigandPNGBDBM50002373(1-(1-ethynyl)-15a,17a-dimethyl-(1R,15aS,17aS)-2,3,...)
Affinity DataIC50:  48nMAssay Description:Inhibition of [125]I-Bolton Hunter Substance P([125]I-BHSP) binding to standard Tachykinin receptor 1 from rat forebrain membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(Rattus norvegicus (rat))
Rochester

Curated by ChEMBL
LigandPNGBDBM50002373(1-(1-ethynyl)-15a,17a-dimethyl-(1R,15aS,17aS)-2,3,...)
Affinity DataIC50:  50nMAssay Description:Inhibition of [125]I-Bolton Hunter Substance P([125]I-BHSP) binding to standard Tachykinin receptor 1 from rat forebrain membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed