Affinity DataKi: 0.0100nMAssay Description:Inhibition of KDM5B (unknown origin) using biotin-H3K4me3 as substrate preincubated for 15 mins followed by substrate addition measured after 20 mins...More data for this Ligand-Target Pair
Affinity DataKi: 0.0200nMAssay Description:Inhibition of recombinant human N-terminal GST-tagged KDM4B (1 to 500 residues) expressed in baculovirus infected sf9 cells using biotin-H3K9me3 as s...More data for this Ligand-Target Pair
Affinity DataKi: 0.0500nMAssay Description:Inhibition of recombinant human N-terminal GST-tagged KDM4B (1 to 500 residues) expressed in baculovirus infected sf9 cells using biotin-H3K9me3 as s...More data for this Ligand-Target Pair
Affinity DataKi: 0.120nMAssay Description:Displacement of [125I]DOI from 5HT2A receptor expressed in HEK cellsMore data for this Ligand-Target Pair
Affinity DataKi: 0.150nMAssay Description:Displacement of [125I]DOI from 5HT2A receptor expressed in HEK cellsMore data for this Ligand-Target Pair
Affinity DataKi: 0.150nMAssay Description:Displacement of [125I]DOI from 5HT2A receptor expressed in HEK cellsMore data for this Ligand-Target Pair
Affinity DataKi: 0.180nMAssay Description:Displacement of [125I]DOI from 5HT2A receptor expressed in HEK cellsMore data for this Ligand-Target Pair
Affinity DataKi: 0.190nMAssay Description:Displacement of [125I]DOI from 5HT2A receptor expressed in HEK cellsMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 7(Rattus norvegicus (rat))
University Of Minnesota
Curated by ChEMBL
University Of Minnesota
Curated by ChEMBL
Affinity DataKi: 0.220nMAssay Description:Inhibition of recombinant human N-terminal GST-tagged KDM4B (1 to 500 residues) expressed in baculovirus infected sf9 cells using biotin-H3K9me3 as s...More data for this Ligand-Target Pair
Affinity DataKi: 0.220nMAssay Description:Displacement of [125I]DOI from 5HT2A receptor expressed in HEK cellsMore data for this Ligand-Target Pair
Affinity DataKi: 0.25nMAssay Description:Displacement of [125I]DOI from 5HT2A receptor expressed in HEK cellsMore data for this Ligand-Target Pair
Affinity DataKi: 0.260nMAssay Description:Displacement of [125I]DOI from 5HT2A receptor expressed in HEK cellsMore data for this Ligand-Target Pair
Affinity DataKi: 0.280nMAssay Description:Displacement of [125I]DOI from 5HT2A receptor expressed in HEK cellsMore data for this Ligand-Target Pair
Affinity DataKi: 0.280nMAssay Description:Displacement of [125I]DOI from 5HT2A receptor expressed in HEK cellsMore data for this Ligand-Target Pair
Affinity DataKi: 0.310nMAssay Description:Displacement of [125I]DOI from 5HT2A receptor expressed in HEK cellsMore data for this Ligand-Target Pair
Affinity DataKi: 0.330nMAssay Description:Displacement of [125I]DOI from 5HT2A receptor expressed in HEK cellsMore data for this Ligand-Target Pair
Affinity DataKi: 0.340nMAssay Description:Displacement of [125I]DOI from 5HT2A receptor expressed in HEK cellsMore data for this Ligand-Target Pair
Affinity DataKi: 0.360nMAssay Description:Displacement of [125I]DOI from 5HT2A receptor expressed in HEK cellsMore data for this Ligand-Target Pair
Affinity DataKi: 0.360nMAssay Description:Inhibition of KDM5B (unknown origin) using biotin-H3K4me3 as substrate preincubated for 15 mins followed by substrate addition measured after 20 mins...More data for this Ligand-Target Pair
Affinity DataKi: 0.410nMAssay Description:Displacement of [125I]DOI from 5HT2A receptor expressed in HEK cellsMore data for this Ligand-Target Pair
Affinity DataKi: 0.420nMAssay Description:Displacement of [125I]DOI from 5HT2A receptor expressed in HEK cellsMore data for this Ligand-Target Pair
Affinity DataKi: 0.430nMAssay Description:Displacement of [125I]DOI from 5HT2A receptor expressed in HEK cellsMore data for this Ligand-Target Pair
Affinity DataKi: 0.430nMAssay Description:Displacement of [125I]DOI from 5HT2A receptor expressed in HEK cellsMore data for this Ligand-Target Pair
Affinity DataKi: 0.479nMAssay Description:Inhibition of KDM5B (unknown origin) using biotin-H3K4me3 as substrate preincubated for 15 mins followed by substrate addition measured after 20 mins...More data for this Ligand-Target Pair
Affinity DataKi: 0.480nMAssay Description:Displacement of [125I]DOI from human recombinant 5HT2A receptor expressed in HEK293 cells after 1 hr by scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 0.510nMAssay Description:Displacement of [125I]DOI from human recombinant 5HT2A receptor expressed in HEK293 cells after 1 hr by scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 0.530nMAssay Description:Inhibition of KDM5B (unknown origin) using biotin-H3K4me3 as substrate preincubated for 15 mins followed by substrate addition measured after 20 mins...More data for this Ligand-Target Pair
Affinity DataKi: 0.540nMAssay Description:Displacement of [125I](+/-)DOI from human 5-HT2B receptor trasfected in CHO cell membrane after 60 mins by scintillation counting analysisMore data for this Ligand-Target Pair
Affinity DataKi: 0.540nMAssay Description:Displacement of [125I]DOI from 5HT2A receptor expressed in HEK cellsMore data for this Ligand-Target Pair
Affinity DataKi: 0.550nMAssay Description:Displacement of [125I]DOI from 5HT2A receptor expressed in HEK cellsMore data for this Ligand-Target Pair
Affinity DataKi: 0.580nMAssay Description:Displacement of [125I]DOI from 5HT2A receptor expressed in HEK cellsMore data for this Ligand-Target Pair
Affinity DataKi: 0.600nMAssay Description:Displacement of [125I]DOI from human recombinant 5HT2A receptor expressed in HEK293 cells by scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 0.600nMAssay Description:Displacement of [125I]DOI from human recombinant 5HT2A receptor expressed in HEK293 cells by scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 0.610nMAssay Description:Displacement of [125I]DOI from 5HT2A receptor expressed in HEK cellsMore data for this Ligand-Target Pair
Affinity DataKi: 0.630nMAssay Description:Displacement of [125I]DOI from 5HT2A receptor expressed in HEK cellsMore data for this Ligand-Target Pair
Affinity DataKi: 0.660nMAssay Description:Displacement of [125I]DOI from 5HT2A receptor expressed in HEK cellsMore data for this Ligand-Target Pair
Affinity DataKi: 0.690nMAssay Description:Displacement of [125I]DOI from 5HT2A receptor expressed in HEK cellsMore data for this Ligand-Target Pair
Affinity DataKi: 0.700nMAssay Description:Displacement of [125I]DOI from human recombinant 5HT2A receptor expressed in HEK293 cells by scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 0.700nMAssay Description:Inhibition of KDM5B (unknown origin) using biotin-H3K4me3 as substrate preincubated for 15 mins followed by substrate addition measured after 20 mins...More data for this Ligand-Target Pair
Affinity DataKi: 0.820nMAssay Description:Displacement of [125I]DOI from 5HT2A receptor expressed in HEK cellsMore data for this Ligand-Target Pair
Affinity DataKi: 0.840nMAssay Description:Displacement of [125I]DOI from 5HT2A receptor expressed in HEK cellsMore data for this Ligand-Target Pair
Affinity DataKi: 0.840nMAssay Description:Displacement of [125I]DOI from 5HT2A receptor expressed in HEK cellsMore data for this Ligand-Target Pair
Affinity DataKi: 0.860nMAssay Description:Displacement of [125I]DOI from 5HT2A receptor expressed in HEK cellsMore data for this Ligand-Target Pair
Affinity DataKi: 0.910nMAssay Description:Displacement of [125I]DOI from 5HT2A receptor expressed in HEK cellsMore data for this Ligand-Target Pair
Affinity DataKi: 0.960nMAssay Description:Displacement of [125I]DOI from 5HT2A receptor expressed in HEK cellsMore data for this Ligand-Target Pair
Affinity DataKi: 0.970nMAssay Description:Displacement of [125I](+/-)DOI from human 5-HT2B receptor trasfected in CHO cell membrane after 60 mins by scintillation counting analysisMore data for this Ligand-Target Pair
Affinity DataKi: 0.990nMAssay Description:Displacement of [125I]DOI from 5HT2A receptor expressed in HEK cellsMore data for this Ligand-Target Pair
Affinity DataKi: 0.990nMAssay Description:Displacement of [125I]DOI from 5HT2A receptor expressed in HEK cellsMore data for this Ligand-Target Pair
Affinity DataKi: 1nMAssay Description:Displacement of [125I](+/-)DOI from human 5-HT2B receptor trasfected in CHO cell membrane after 60 mins by scintillation counting analysisMore data for this Ligand-Target Pair
Affinity DataKi: 1.10nMAssay Description:Displacement of [125I]DOI from human recombinant 5HT2A receptor expressed in HEK293 cells after 1 hr by scintillation countingMore data for this Ligand-Target Pair