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Found 384 with Last Name = 'edwards' and Initial = 'pj'
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Santhera Pharmaceuticals (Switzerland)

Curated by ChEMBL
LigandPNGBDBM50296131(CHEMBL564249 | N-(((S)-1-((R)-3-amino-4-(3-chlorop...)
Affinity DataIC50:  0.380nMAssay Description:Inhibition of DPP4 by continuous fluorimetric assayMore data for this Ligand-Target Pair
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Santhera Pharmaceuticals (Switzerland)

Curated by ChEMBL
LigandPNGBDBM50302961((R)-3-amino-1-((S)-2-(3-(1-(methylsulfonyl)azetidi...)
Affinity DataIC50:  1nMAssay Description:Inhibition of human recombinant DPP4 transfected in Pichia methanolica expression system after 10 mins by continuous fluorimetric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Santhera Pharmaceuticals (Switzerland)

Curated by ChEMBL
LigandPNGBDBM50296761(CHEMBL564105 | N-(((S)-1-((R)-3-amino-4-(2,4,5-tri...)
Affinity DataIC50:  1.10nMAssay Description:Inhibition of DPP4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Santhera Pharmaceuticals (Switzerland)

Curated by ChEMBL
LigandPNGBDBM50296768(CHEMBL554908 | N-(((S)-1-((R)-3-amino-4-(2,4,5-tri...)
Affinity DataIC50:  1.30nMAssay Description:Inhibition of DPP4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Santhera Pharmaceuticals (Switzerland)

Curated by ChEMBL
LigandPNGBDBM50296755(CHEMBL558452 | N-(((S)-1-((R)-3-amino-4-(2,4,5-tri...)
Affinity DataIC50:  1.5nMAssay Description:Inhibition of DPP4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Santhera Pharmaceuticals (Switzerland)

Curated by ChEMBL
LigandPNGBDBM50302972((R)-3-amino-1-((S)-2-(5-(3-methyloxetan-3-yl)-1,2,...)
Affinity DataIC50:  2nMAssay Description:Inhibition of human recombinant DPP4 transfected in Pichia methanolica expression system after 10 mins by continuous fluorimetric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Santhera Pharmaceuticals (Switzerland)

Curated by ChEMBL
LigandPNGBDBM50302958((R)-3-amino-1-((S)-2-(3-(1-(trifluoromethyl)cyclop...)
Affinity DataIC50:  2nMAssay Description:Inhibition of human recombinant DPP4 transfected in Pichia methanolica expression system after 10 mins by continuous fluorimetric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Santhera Pharmaceuticals (Switzerland)

Curated by ChEMBL
LigandPNGBDBM50302964((R)-3-amino-1-((S)-2-(3-(pyrazin-2-yl)-1,2,4-oxadi...)
Affinity DataIC50:  2nMAssay Description:Inhibition of human recombinant DPP4 transfected in Pichia methanolica expression system after 10 mins by continuous fluorimetric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Santhera Pharmaceuticals (Switzerland)

Curated by ChEMBL
LigandPNGBDBM50302956((R)-3-amino-1-((S)-2-(3-tert-butyl-1,2,4-oxadiazol...)
Affinity DataIC50:  2nMAssay Description:Inhibition of human recombinant DPP4 transfected in Pichia methanolica expression system after 10 mins by continuous fluorimetric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Santhera Pharmaceuticals (Switzerland)

Curated by ChEMBL
LigandPNGBDBM50296773(6-(((S)-1-((R)-3-amino-4-(2,4,5-trifluorophenyl)bu...)
Affinity DataIC50:  2nMAssay Description:Inhibition of DPP4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Santhera Pharmaceuticals (Switzerland)

Curated by ChEMBL
LigandPNGBDBM50296767(CHEMBL563901 | N-(((S)-1-((R)-3-amino-4-(2,4,5-tri...)
Affinity DataIC50:  2.20nMAssay Description:Inhibition of DPP4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Santhera Pharmaceuticals (Switzerland)

Curated by ChEMBL
LigandPNGBDBM50296772(2-(((S)-1-((R)-3-amino-4-(2,4,5-trifluorophenyl)bu...)
Affinity DataIC50:  2.30nMAssay Description:Inhibition of DPP4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
Boehringer Ingelheim (Canada)

Curated by ChEMBL
LigandPNGBDBM50492164(CHEMBL2381561)
Affinity DataIC50:  2.60nMAssay Description:Inhibition of HIV1 reverse transcriptase using poly(rA)/oligo(dT)15 as substrate after 60 mins by fluorescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
Boehringer Ingelheim (Canada)

Curated by ChEMBL
LigandPNGBDBM50492156(CHEMBL2397560)
Affinity DataIC50:  2.60nMAssay Description:Inhibition of HIV1 reverse transcriptase using poly(rA)/oligo(dT)15 as substrate after 60 mins by fluorescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Santhera Pharmaceuticals (Switzerland)

Curated by ChEMBL
LigandPNGBDBM50296754(CHEMBL558647 | N-(((S)-1-((R)-3-amino-4-(2,4,5-tri...)
Affinity DataIC50:  2.70nMAssay Description:Inhibition of DPP4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Santhera Pharmaceuticals (Switzerland)

Curated by ChEMBL
LigandPNGBDBM50296769(CHEMBL552069 | N-(((S)-1-((R)-3-amino-4-(2,4,5-tri...)
Affinity DataIC50:  2.70nMAssay Description:Inhibition of DPP4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
Boehringer Ingelheim (Canada)

Curated by ChEMBL
LigandPNGBDBM50492155(CHEMBL2397554)
Affinity DataIC50:  2.90nMAssay Description:Inhibition of HIV1 reverse transcriptase using poly(rA)/oligo(dT)15 as substrate after 60 mins by fluorescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Santhera Pharmaceuticals (Switzerland)

Curated by ChEMBL
LigandPNGBDBM50302966((R)-3-amino-1-((S)-2-(3-(3,5-difluoropyridin-2-yl)...)
Affinity DataIC50:  3nMAssay Description:Inhibition of human recombinant DPP4 transfected in Pichia methanolica expression system after 10 mins by continuous fluorimetric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
Boehringer Ingelheim (Canada)

Curated by ChEMBL
LigandPNGBDBM50492176(CHEMBL2397567)
Affinity DataIC50:  3nMAssay Description:Inhibition of HIV1 reverse transcriptase using poly(rA)/oligo(dT)15 as substrate after 60 mins by fluorescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Santhera Pharmaceuticals (Switzerland)

Curated by ChEMBL
LigandPNGBDBM50302957((R)-3-amino-1-((S)-2-(3-(cyclopropylmethyl)-1,2,4-...)
Affinity DataIC50:  3nMAssay Description:Inhibition of human recombinant DPP4 transfected in Pichia methanolica expression system after 10 mins by continuous fluorimetric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
Boehringer Ingelheim (Canada)

Curated by ChEMBL
LigandPNGBDBM50492175(CHEMBL2397583)
Affinity DataIC50:  3.10nMAssay Description:Inhibition of HIV1 reverse transcriptase using poly(rA)/oligo(dT)15 as substrate after 60 mins by fluorescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Santhera Pharmaceuticals (Switzerland)

Curated by ChEMBL
LigandPNGBDBM50296779(2-(((S)-1-((R)-3-amino-4-(2,4,5-trifluorophenyl)bu...)
Affinity DataIC50:  3.20nMAssay Description:Inhibition of DPP4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
Boehringer Ingelheim (Canada)

Curated by ChEMBL
LigandPNGBDBM50492163(CHEMBL2397557)
Affinity DataIC50:  3.20nMAssay Description:Inhibition of HIV1 reverse transcriptase using poly(rA)/oligo(dT)15 as substrate after 60 mins by fluorescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Santhera Pharmaceuticals (Switzerland)

Curated by ChEMBL
LigandPNGBDBM50296762(CHEMBL550114 | N-(((S)-1-((R)-3-amino-4-(2,4,5-tri...)
Affinity DataIC50:  3.5nMAssay Description:Inhibition of DPP4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
Boehringer Ingelheim (Canada)

Curated by ChEMBL
LigandPNGBDBM50492154(CHEMBL2397572)
Affinity DataIC50:  3.5nMAssay Description:Inhibition of HIV1 reverse transcriptase using poly(rA)/oligo(dT)15 as substrate after 60 mins by fluorescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Santhera Pharmaceuticals (Switzerland)

Curated by ChEMBL
LigandPNGBDBM50296781(6-(((S)-1-((R)-3-amino-4-(2,4,5-trifluorophenyl)bu...)
Affinity DataIC50:  3.5nMAssay Description:Inhibition of DPP4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Santhera Pharmaceuticals (Switzerland)

Curated by ChEMBL
LigandPNGBDBM50296765(CHEMBL558322 | N-(((S)-1-((R)-3-amino-4-(2,4,5-tri...)
Affinity DataIC50:  3.70nMAssay Description:Inhibition of DPP4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Santhera Pharmaceuticals (Switzerland)

Curated by ChEMBL
LigandPNGBDBM50296774((R)-3-amino-1-((S)-2-((4-(trifluoromethyl)pyrimidi...)
Affinity DataIC50:  3.90nMAssay Description:Inhibition of DPP4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
Boehringer Ingelheim (Canada)

Curated by ChEMBL
LigandPNGBDBM50492168(CHEMBL2397584)
Affinity DataIC50:  3.90nMAssay Description:Inhibition of HIV1 reverse transcriptase using poly(rA)/oligo(dT)15 as substrate after 60 mins by fluorescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Santhera Pharmaceuticals (Switzerland)

Curated by ChEMBL
LigandPNGBDBM50302959((R)-3-amino-1-((S)-2-(3-morpholino-1,2,4-oxadiazol...)
Affinity DataIC50:  4nMAssay Description:Inhibition of human recombinant DPP4 transfected in Pichia methanolica expression system after 10 mins by continuous fluorimetric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Santhera Pharmaceuticals (Switzerland)

Curated by ChEMBL
LigandPNGBDBM50302960((R)-3-amino-1-((S)-2-(3-(pyrrolidin-1-yl)-1,2,4-ox...)
Affinity DataIC50:  4nMAssay Description:Inhibition of human recombinant DPP4 transfected in Pichia methanolica expression system after 10 mins by continuous fluorimetric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Santhera Pharmaceuticals (Switzerland)

Curated by ChEMBL
LigandPNGBDBM50302965((R)-3-amino-1-((S)-2-(3-(pyrimidin-2-yl)-1,2,4-oxa...)
Affinity DataIC50:  4nMAssay Description:Inhibition of human recombinant DPP4 transfected in Pichia methanolica expression system after 10 mins by continuous fluorimetric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Santhera Pharmaceuticals (Switzerland)

Curated by ChEMBL
LigandPNGBDBM50296780(6-((((S)-1-((R)-3-amino-4-(2,4,5-trifluorophenyl)b...)
Affinity DataIC50:  4nMAssay Description:Inhibition of DPP4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
Boehringer Ingelheim (Canada)

Curated by ChEMBL
LigandPNGBDBM50492153(CHEMBL2397563)
Affinity DataIC50:  4.70nMAssay Description:Inhibition of HIV1 reverse transcriptase using poly(rA)/oligo(dT)15 as substrate after 60 mins by fluorescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Santhera Pharmaceuticals (Switzerland)

Curated by ChEMBL
LigandPNGBDBM50296766(CHEMBL557723 | N-(((S)-1-((R)-3-amino-4-(2,4,5-tri...)
Affinity DataIC50:  4.80nMAssay Description:Inhibition of DPP4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
Boehringer Ingelheim (Canada)

Curated by ChEMBL
LigandPNGBDBM50492174(CHEMBL2397586)
Affinity DataIC50:  4.80nMAssay Description:Inhibition of HIV1 reverse transcriptase using poly(rA)/oligo(dT)15 as substrate after 60 mins by fluorescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Santhera Pharmaceuticals (Switzerland)

Curated by ChEMBL
LigandPNGBDBM50302962((R)-1-((S)-2-(3-(1-acetylazetidin-3-yl)-1,2,4-oxad...)
Affinity DataIC50:  5nMAssay Description:Inhibition of human recombinant DPP4 transfected in Pichia methanolica expression system after 10 mins by continuous fluorimetric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
Boehringer Ingelheim (Canada)

Curated by ChEMBL
LigandPNGBDBM50492169(CHEMBL2397582)
Affinity DataIC50:  5nMAssay Description:Inhibition of HIV1 reverse transcriptase using poly(rA)/oligo(dT)15 as substrate after 60 mins by fluorescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
Boehringer Ingelheim (Canada)

Curated by ChEMBL
LigandPNGBDBM50492179(CHEMBL2397587)
Affinity DataIC50:  5nMAssay Description:Inhibition of HIV1 reverse transcriptase using poly(rA)/oligo(dT)15 as substrate after 60 mins by fluorescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
Boehringer Ingelheim (Canada)

Curated by ChEMBL
LigandPNGBDBM50492152(CHEMBL2397565)
Affinity DataIC50:  5.20nMAssay Description:Inhibition of HIV1 reverse transcriptase using poly(rA)/oligo(dT)15 as substrate after 60 mins by fluorescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Santhera Pharmaceuticals (Switzerland)

Curated by ChEMBL
LigandPNGBDBM50296776((R)-3-amino-1-((S)-2-((pyrimidin-2-ylamino)methyl)...)
Affinity DataIC50:  5.40nMAssay Description:Inhibition of DPP4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
Boehringer Ingelheim (Canada)

Curated by ChEMBL
LigandPNGBDBM50492151(CHEMBL2397588)
Affinity DataIC50:  5.5nMAssay Description:Inhibition of HIV1 reverse transcriptase using poly(rA)/oligo(dT)15 as substrate after 60 mins by fluorescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Santhera Pharmaceuticals (Switzerland)

Curated by ChEMBL
LigandPNGBDBM50296756(CHEMBL559602 | N-(((S)-1-((R)-3-amino-4-(2,4,5-tri...)
Affinity DataIC50:  5.60nMAssay Description:Inhibition of DPP4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
Boehringer Ingelheim (Canada)

Curated by ChEMBL
LigandPNGBDBM50492162(CHEMBL2397549)
Affinity DataIC50:  5.80nMAssay Description:Inhibition of HIV1 reverse transcriptase using poly(rA)/oligo(dT)15 as substrate after 60 mins by fluorescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
Boehringer Ingelheim (Canada)

Curated by ChEMBL
LigandPNGBDBM50492158(CHEMBL2397548)
Affinity DataIC50:  5.90nMAssay Description:Inhibition of HIV1 reverse transcriptase using poly(rA)/oligo(dT)15 as substrate after 60 mins by fluorescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
Boehringer Ingelheim (Canada)

Curated by ChEMBL
LigandPNGBDBM50492173(CHEMBL2397573)
Affinity DataIC50:  5.90nMAssay Description:Inhibition of HIV1 reverse transcriptase using poly(rA)/oligo(dT)15 as substrate after 60 mins by fluorescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Santhera Pharmaceuticals (Switzerland)

Curated by ChEMBL
LigandPNGBDBM50296763(CHEMBL557860 | N-(((S)-1-((R)-3-amino-4-(2,4,5-tri...)
Affinity DataIC50:  5.90nMAssay Description:Inhibition of DPP4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
Boehringer Ingelheim (Canada)

Curated by ChEMBL
LigandPNGBDBM50492150(CHEMBL2397559)
Affinity DataIC50:  6.10nMAssay Description:Inhibition of HIV1 reverse transcriptase using poly(rA)/oligo(dT)15 as substrate after 60 mins by fluorescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Santhera Pharmaceuticals (Switzerland)

Curated by ChEMBL
LigandPNGBDBM50296771((R)-3-amino-1-((S)-2-((2-(trifluoromethyl)pyrimidi...)
Affinity DataIC50:  6.10nMAssay Description:Inhibition of DPP4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Santhera Pharmaceuticals (Switzerland)

Curated by ChEMBL
LigandPNGBDBM50296778((R)-3-amino-1-((S)-2-((5-fluoropyridin-2-ylamino)m...)
Affinity DataIC50:  6.30nMAssay Description:Inhibition of DPP4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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