TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
Ushinsky Yaroslavl State Pedagogical University
Curated by ChEMBL
Ushinsky Yaroslavl State Pedagogical University
Curated by ChEMBL
Affinity DataIC50: 2.70nMAssay Description:Inhibition of human recombinant MAO-B expressed in insect cells microsomes assessed as inhibition of 4-hydroxyquinoline formation using kynuramine as...More data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
Ushinsky Yaroslavl State Pedagogical University
Curated by ChEMBL
Ushinsky Yaroslavl State Pedagogical University
Curated by ChEMBL
Affinity DataIC50: 48nMAssay Description:Inhibition of human recombinant MAO-B expressed in insect cells microsomes assessed as inhibition of 4-hydroxyquinoline formation using kynuramine as...More data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
Ushinsky Yaroslavl State Pedagogical University
Curated by ChEMBL
Ushinsky Yaroslavl State Pedagogical University
Curated by ChEMBL
Affinity DataIC50: 79nMAssay Description:Inhibition of human recombinant MAO-B expressed in insect cells microsomes assessed as inhibition of 4-hydroxyquinoline formation using kynuramine as...More data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
Ushinsky Yaroslavl State Pedagogical University
Curated by ChEMBL
Ushinsky Yaroslavl State Pedagogical University
Curated by ChEMBL
Affinity DataIC50: 79nMAssay Description:Inhibition of human recombinant MAO-B expressed in insect cells microsomes assessed as inhibition of 4-hydroxyquinoline formation using kynuramine as...More data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
Ushinsky Yaroslavl State Pedagogical University
Curated by ChEMBL
Ushinsky Yaroslavl State Pedagogical University
Curated by ChEMBL
Affinity DataIC50: 91nMAssay Description:Inhibition of human recombinant MAO-B expressed in insect cells microsomes assessed as inhibition of 4-hydroxyquinoline formation using kynuramine as...More data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
Ushinsky Yaroslavl State Pedagogical University
Curated by ChEMBL
Ushinsky Yaroslavl State Pedagogical University
Curated by ChEMBL
Affinity DataIC50: 168nMAssay Description:Inhibition of human recombinant MAO-B expressed in insect cells microsomes assessed as inhibition of 4-hydroxyquinoline formation using kynuramine as...More data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
Ushinsky Yaroslavl State Pedagogical University
Curated by ChEMBL
Ushinsky Yaroslavl State Pedagogical University
Curated by ChEMBL
Affinity DataIC50: 210nMAssay Description:Inhibition of human recombinant MAO-B expressed in insect cells microsomes assessed as inhibition of 4-hydroxyquinoline formation using kynuramine as...More data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
Ushinsky Yaroslavl State Pedagogical University
Curated by ChEMBL
Ushinsky Yaroslavl State Pedagogical University
Curated by ChEMBL
Affinity DataIC50: 318nMAssay Description:Inhibition of human recombinant MAO-B expressed in insect cells microsomes assessed as inhibition of 4-hydroxyquinoline formation using kynuramine as...More data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
Ushinsky Yaroslavl State Pedagogical University
Curated by ChEMBL
Ushinsky Yaroslavl State Pedagogical University
Curated by ChEMBL
Affinity DataIC50: 439nMAssay Description:Inhibition of human recombinant MAO-B expressed in insect cells microsomes assessed as inhibition of 4-hydroxyquinoline formation using kynuramine as...More data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
Ushinsky Yaroslavl State Pedagogical University
Curated by ChEMBL
Ushinsky Yaroslavl State Pedagogical University
Curated by ChEMBL
Affinity DataIC50: 571nMAssay Description:Inhibition of human recombinant MAO-B expressed in insect cells microsomes assessed as inhibition of 4-hydroxyquinoline formation using kynuramine as...More data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
Ushinsky Yaroslavl State Pedagogical University
Curated by ChEMBL
Ushinsky Yaroslavl State Pedagogical University
Curated by ChEMBL
Affinity DataIC50: 767nMAssay Description:Inhibition of human recombinant MAO-B expressed in insect cells microsomes assessed as inhibition of 4-hydroxyquinoline formation using kynuramine as...More data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
Ushinsky Yaroslavl State Pedagogical University
Curated by ChEMBL
Ushinsky Yaroslavl State Pedagogical University
Curated by ChEMBL
Affinity DataIC50: 975nMAssay Description:Inhibition of human recombinant MAO-B expressed in insect cells microsomes assessed as inhibition of 4-hydroxyquinoline formation using kynuramine as...More data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
Ushinsky Yaroslavl State Pedagogical University
Curated by ChEMBL
Ushinsky Yaroslavl State Pedagogical University
Curated by ChEMBL
Affinity DataIC50: 1.17E+3nMAssay Description:Inhibition of human recombinant MAO-B expressed in insect cells microsomes assessed as inhibition of 4-hydroxyquinoline formation using kynuramine as...More data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] A(Homo sapiens (Human))
Ushinsky Yaroslavl State Pedagogical University
Curated by ChEMBL
Ushinsky Yaroslavl State Pedagogical University
Curated by ChEMBL
Affinity DataIC50: 3.92E+3nMAssay Description:Inhibition of human recombinant MAO-A expressed in insect cells microsomes assessed as inhibition of 4-hydroxyquinoline formation using kynuramine as...More data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
Ushinsky Yaroslavl State Pedagogical University
Curated by ChEMBL
Ushinsky Yaroslavl State Pedagogical University
Curated by ChEMBL
Affinity DataIC50: 1.01E+4nMAssay Description:Inhibition of human recombinant MAO-B expressed in insect cells microsomes assessed as inhibition of 4-hydroxyquinoline formation using kynuramine as...More data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
Ushinsky Yaroslavl State Pedagogical University
Curated by ChEMBL
Ushinsky Yaroslavl State Pedagogical University
Curated by ChEMBL
Affinity DataIC50: 1.17E+4nMAssay Description:Inhibition of human recombinant MAO-B expressed in insect cells microsomes assessed as inhibition of 4-hydroxyquinoline formation using kynuramine as...More data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] A(Homo sapiens (Human))
Ushinsky Yaroslavl State Pedagogical University
Curated by ChEMBL
Ushinsky Yaroslavl State Pedagogical University
Curated by ChEMBL
Affinity DataIC50: 1.36E+4nMAssay Description:Inhibition of human recombinant MAO-A expressed in insect cells microsomes assessed as inhibition of 4-hydroxyquinoline formation using kynuramine as...More data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] A(Homo sapiens (Human))
Ushinsky Yaroslavl State Pedagogical University
Curated by ChEMBL
Ushinsky Yaroslavl State Pedagogical University
Curated by ChEMBL
Affinity DataIC50: 1.61E+4nMAssay Description:Inhibition of human recombinant MAO-A expressed in insect cells microsomes assessed as inhibition of 4-hydroxyquinoline formation using kynuramine as...More data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] A(Homo sapiens (Human))
Ushinsky Yaroslavl State Pedagogical University
Curated by ChEMBL
Ushinsky Yaroslavl State Pedagogical University
Curated by ChEMBL
Affinity DataIC50: 2.43E+4nMAssay Description:Inhibition of human recombinant MAO-A expressed in insect cells microsomes assessed as inhibition of 4-hydroxyquinoline formation using kynuramine as...More data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] B(Mus musculus)
Ushinsky Yaroslavl State Pedagogical University
Curated by ChEMBL
Ushinsky Yaroslavl State Pedagogical University
Curated by ChEMBL
Affinity DataIC50: 2.48E+4nMAssay Description:Inhibition of MAO-B in mouse brain assessed as reduction in H2O2 production incubated for 30 mins using benzylamine as substrate by Amplex red reagen...More data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] A(Homo sapiens (Human))
Ushinsky Yaroslavl State Pedagogical University
Curated by ChEMBL
Ushinsky Yaroslavl State Pedagogical University
Curated by ChEMBL
Affinity DataIC50: 3.44E+4nMAssay Description:Inhibition of human recombinant MAO-A expressed in insect cells microsomes assessed as inhibition of 4-hydroxyquinoline formation using kynuramine as...More data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] A(Homo sapiens (Human))
Ushinsky Yaroslavl State Pedagogical University
Curated by ChEMBL
Ushinsky Yaroslavl State Pedagogical University
Curated by ChEMBL
Affinity DataIC50: 3.96E+4nMAssay Description:Inhibition of human recombinant MAO-A expressed in insect cells microsomes assessed as inhibition of 4-hydroxyquinoline formation using kynuramine as...More data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] A(Homo sapiens (Human))
Ushinsky Yaroslavl State Pedagogical University
Curated by ChEMBL
Ushinsky Yaroslavl State Pedagogical University
Curated by ChEMBL
Affinity DataIC50: 4.62E+4nMAssay Description:Inhibition of human recombinant MAO-A expressed in insect cells microsomes assessed as inhibition of 4-hydroxyquinoline formation using kynuramine as...More data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] A(Homo sapiens (Human))
Ushinsky Yaroslavl State Pedagogical University
Curated by ChEMBL
Ushinsky Yaroslavl State Pedagogical University
Curated by ChEMBL
Affinity DataIC50: 5.59E+4nMAssay Description:Inhibition of human recombinant MAO-A expressed in insect cells microsomes assessed as inhibition of 4-hydroxyquinoline formation using kynuramine as...More data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] A(Homo sapiens (Human))
Ushinsky Yaroslavl State Pedagogical University
Curated by ChEMBL
Ushinsky Yaroslavl State Pedagogical University
Curated by ChEMBL
Affinity DataIC50: 6.14E+4nMAssay Description:Inhibition of human recombinant MAO-A expressed in insect cells microsomes assessed as inhibition of 4-hydroxyquinoline formation using kynuramine as...More data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] A(Homo sapiens (Human))
Ushinsky Yaroslavl State Pedagogical University
Curated by ChEMBL
Ushinsky Yaroslavl State Pedagogical University
Curated by ChEMBL
Affinity DataIC50: 6.28E+4nMAssay Description:Inhibition of human recombinant MAO-A expressed in insect cells microsomes assessed as inhibition of 4-hydroxyquinoline formation using kynuramine as...More data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] A(Homo sapiens (Human))
Ushinsky Yaroslavl State Pedagogical University
Curated by ChEMBL
Ushinsky Yaroslavl State Pedagogical University
Curated by ChEMBL
Affinity DataIC50: 6.39E+4nMAssay Description:Inhibition of human recombinant MAO-A expressed in insect cells microsomes assessed as inhibition of 4-hydroxyquinoline formation using kynuramine as...More data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] A(Homo sapiens (Human))
Ushinsky Yaroslavl State Pedagogical University
Curated by ChEMBL
Ushinsky Yaroslavl State Pedagogical University
Curated by ChEMBL
Affinity DataIC50: 6.80E+4nMAssay Description:Inhibition of human recombinant MAO-A expressed in insect cells microsomes assessed as inhibition of 4-hydroxyquinoline formation using kynuramine as...More data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] A(Homo sapiens (Human))
Ushinsky Yaroslavl State Pedagogical University
Curated by ChEMBL
Ushinsky Yaroslavl State Pedagogical University
Curated by ChEMBL
Affinity DataIC50: 8.38E+4nMAssay Description:Inhibition of human recombinant MAO-A expressed in insect cells microsomes assessed as inhibition of 4-hydroxyquinoline formation using kynuramine as...More data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
Ushinsky Yaroslavl State Pedagogical University
Curated by ChEMBL
Ushinsky Yaroslavl State Pedagogical University
Curated by ChEMBL
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of human recombinant MAO-B expressed in insect cells microsomes assessed as inhibition of 4-hydroxyquinoline formation using kynuramine as...More data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] A(Homo sapiens (Human))
Ushinsky Yaroslavl State Pedagogical University
Curated by ChEMBL
Ushinsky Yaroslavl State Pedagogical University
Curated by ChEMBL
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of human recombinant MAO-A expressed in insect cells microsomes assessed as inhibition of 4-hydroxyquinoline formation using kynuramine as...More data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] A(Homo sapiens (Human))
Ushinsky Yaroslavl State Pedagogical University
Curated by ChEMBL
Ushinsky Yaroslavl State Pedagogical University
Curated by ChEMBL
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of human recombinant MAO-A expressed in insect cells microsomes assessed as inhibition of 4-hydroxyquinoline formation using kynuramine as...More data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] A(Homo sapiens (Human))
Ushinsky Yaroslavl State Pedagogical University
Curated by ChEMBL
Ushinsky Yaroslavl State Pedagogical University
Curated by ChEMBL
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of human recombinant MAO-A expressed in insect cells microsomes assessed as inhibition of 4-hydroxyquinoline formation using kynuramine as...More data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
Ushinsky Yaroslavl State Pedagogical University
Curated by ChEMBL
Ushinsky Yaroslavl State Pedagogical University
Curated by ChEMBL
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of human recombinant MAO-B expressed in insect cells microsomes assessed as inhibition of 4-hydroxyquinoline formation using kynuramine as...More data for this Ligand-Target Pair