Affinity DataKi: 0.340nMAssay Description:Binding affinity to human D3 receptor expressed in CHO cells assessed as inhibition constant by scintillation counting methodMore data for this Ligand-Target Pair
Ligand Info
TargetNeuropeptide Y receptor type 2(Homo sapiens (Human))
Bristol-Myers Squibb
Curated by PDSP Ki Database
Bristol-Myers Squibb
Curated by PDSP Ki Database
Affinity DataKi: 0.700nMAssay Description:Binding affinity to human D3 receptor expressed in CHO cells assessed as inhibition constant by scintillation counting methodMore data for this Ligand-Target Pair
Ligand Info
TargetNeuropeptide Y receptor type 2(Homo sapiens (Human))
Bristol-Myers Squibb
Curated by PDSP Ki Database
Bristol-Myers Squibb
Curated by PDSP Ki Database
Affinity DataKi: 0.860nMAssay Description:Binding affinity to human D3 receptor expressed in CHO cells assessed as inhibition constant by scintillation counting methodMore data for this Ligand-Target Pair
Ligand Info
Affinity DataKi: 0.920nMAssay Description:Binding affinity to human D3 receptor expressed in CHO cells assessed as inhibition constant by scintillation counting methodMore data for this Ligand-Target Pair
Ligand Info
Affinity DataKi: 0.920nMAssay Description:Inhibition of human D3 receptor expressed in CHO cells assessed as inhibition constant by scintillation counting methodMore data for this Ligand-Target Pair
Ligand Info
TargetNeuropeptide Y receptor type 2(Homo sapiens (Human))
Bristol-Myers Squibb
Curated by PDSP Ki Database
Bristol-Myers Squibb
Curated by PDSP Ki Database
Affinity DataKi: 1nMAssay Description:Displacement of [3H]-Histamine from human histamine 4 receptor transfected in HEK293T cells incubated for 16 hrs by liquid scintillation counter anal...More data for this Ligand-Target Pair
Affinity DataKi: 1.40nMAssay Description:Binding affinity to human D3 receptor expressed in CHO cells assessed as inhibition constant by scintillation counting methodMore data for this Ligand-Target Pair
Ligand Info
TargetNeuropeptide Y receptor type 2(Homo sapiens (Human))
Bristol-Myers Squibb
Curated by PDSP Ki Database
Bristol-Myers Squibb
Curated by PDSP Ki Database
Affinity DataKi: 2.5nMAssay Description:Displacement of [3H]-Histamine from human histamine 3 receptor transfected in HEK293T cells incubated for 16 hrs by liquid scintillation counter anal...More data for this Ligand-Target Pair
Affinity DataKi: 3.10nMAssay Description:Binding affinity to human D3 receptor expressed in CHO cells assessed as inhibition constant by scintillation counting methodMore data for this Ligand-Target Pair
Ligand Info
TargetNeuropeptide Y receptor type 2(Homo sapiens (Human))
Bristol-Myers Squibb
Curated by PDSP Ki Database
Bristol-Myers Squibb
Curated by PDSP Ki Database
TargetNeuropeptide Y receptor type 2(Homo sapiens (Human))
Bristol-Myers Squibb
Curated by PDSP Ki Database
Bristol-Myers Squibb
Curated by PDSP Ki Database
Affinity DataKi: 4nMAssay Description:Displacement of [3H]-Histamine from human histamine 3 receptor transfected in HEK293T cells incubated for 16 hrs by liquid scintillation counter anal...More data for this Ligand-Target Pair
TargetNeuropeptide Y receptor type 2(Homo sapiens (Human))
Bristol-Myers Squibb
Curated by PDSP Ki Database
Bristol-Myers Squibb
Curated by PDSP Ki Database
Affinity DataKi: 6.30nMAssay Description:Displacement of [3H]-Histamine from human histamine 3 receptor transfected in HEK293T cells incubated for 16 hrs by liquid scintillation counter anal...More data for this Ligand-Target Pair
Affinity DataKi: >10nMAssay Description:Binding affinity to human D3 receptor expressed in CHO cells assessed as inhibition constant by scintillation counting methodMore data for this Ligand-Target Pair
Ligand Info
Affinity DataKi: >10nMAssay Description:Binding affinity to human D3 receptor expressed in CHO cells assessed as inhibition constant by scintillation counting methodMore data for this Ligand-Target Pair
Ligand Info
Affinity DataKi: >10nMAssay Description:Binding affinity to human D3 receptor expressed in CHO cells assessed as inhibition constant by scintillation counting methodMore data for this Ligand-Target Pair
Ligand Info
Affinity DataKi: >10nMAssay Description:Binding affinity to human D3 receptor expressed in CHO cells assessed as inhibition constant by scintillation counting methodMore data for this Ligand-Target Pair
Ligand Info
Affinity DataKi: >10nMAssay Description:Binding affinity to human D3 receptor expressed in CHO cells assessed as inhibition constant by scintillation counting methodMore data for this Ligand-Target Pair
Ligand Info
TargetNeuropeptide Y receptor type 2(Homo sapiens (Human))
Bristol-Myers Squibb
Curated by PDSP Ki Database
Bristol-Myers Squibb
Curated by PDSP Ki Database
Affinity DataKi: 16nMAssay Description:Displacement of [3H]-Histamine from human histamine 3 receptor transfected in HEK293T cells incubated for 16 hrs by liquid scintillation counter anal...More data for this Ligand-Target Pair
Affinity DataKi: 16nMAssay Description:Inhibition of human H3 receptor assessed as inhibition constant incubated for 90 mins by scintillation counting methodMore data for this Ligand-Target Pair
Affinity DataKi: 36nMAssay Description:Competitive inhibition of N-terminal His-tagged human OGA using 4-Mu-GlcNAc as substrate assessed as inhibition constant by measuring liberation of n...More data for this Ligand-Target Pair
Affinity DataKi: 40nMAssay Description:Displacement of [3H]-Histamine from human histamine 3 receptor transfected in HEK293T cells incubated for 16 hrs by liquid scintillation counter anal...More data for this Ligand-Target Pair
Affinity DataKi: 47nMAssay Description:Competitive inhibition of cow HexA/HexB (unknown origin) using pNP-GlcNAc as substrate assessed as inhibition constant by measuring liberation of nit...More data for this Ligand-Target Pair
Affinity DataKi: 50nMAssay Description:Inhibition of OGA (unknown origin) using pNP-O-GlcNAc as substrate assessed as inhibition constant incubated for 30 minsMore data for this Ligand-Target Pair
Affinity DataKi: 54nMAssay Description:Binding affinity to human D3 receptor expressed in CHO cells assessed as inhibition constant by scintillation counting methodMore data for this Ligand-Target Pair
Affinity DataKi: 79nMAssay Description:Displacement of [3H]-Histamine from human histamine 4 receptor transfected in HEK293T cells incubated for 16 hrs by liquid scintillation counter anal...More data for this Ligand-Target Pair
Affinity DataKi: 83nMAssay Description:Competitive inhibition of N-terminal His-tagged human OGA using 4-Mu-GlcNAc as substrate assessed as inhibition constant by measuring liberation of n...More data for this Ligand-Target Pair
Affinity DataKi: 125nMAssay Description:Competitive inhibition of cow HexA/HexB (unknown origin) using pNP-GlcNAc as substrate assessed as inhibition constant by measuring liberation of nit...More data for this Ligand-Target Pair
Affinity DataKi: 130nMAssay Description:Inhibition of HexA/HexB (unknown origin)More data for this Ligand-Target Pair
Affinity DataKi: 154nMAssay Description:Competitive inhibition of cow HexA/HexB (unknown origin) using pNP-GlcNAc as substrate assessed as inhibition constant by measuring liberation of nit...More data for this Ligand-Target Pair
Affinity DataKi: 155nMAssay Description:Competitive inhibition of N-terminal His-tagged human OGA using pNP-GlcNAc as chromogenic substrate assessed as inhibition constant by measuring libe...More data for this Ligand-Target Pair
TargetEndoplasmic reticulum mannosyl-oligosaccharide 1,2-alpha-mannosidase(Homo sapiens (Human))
Universidade Do Porto 687
Curated by ChEMBL
Universidade Do Porto 687
Curated by ChEMBL
Affinity DataKi: 160nMAssay Description:Inhibition of human ER alpha mannosidase 1More data for this Ligand-Target Pair
Affinity DataKi: 167nMAssay Description:Competitive inhibition of N-terminal His-tagged human OGA using pNP-GlcNAc as chromogenic substrate assessed as inhibition constant by measuring libe...More data for this Ligand-Target Pair
Affinity DataKi: 170nMAssay Description:Competitive inhibition of cow HexA/HexB (unknown origin) using pNP-GlcNAc as substrate assessed as inhibition constant by measuring liberation of nit...More data for this Ligand-Target Pair
Affinity DataKi: 190nMAssay Description:Competitive inhibition of N-terminal His-tagged human OGA using pNP-GlcNAc as chromogenic substrate assessed as inhibition constant by measuring libe...More data for this Ligand-Target Pair
Affinity DataKi: 205nMAssay Description:Competitive inhibition of cow HexA/HexB (unknown origin) using pNP-GlcNAc as substrate assessed as inhibition constant by measuring liberation of nit...More data for this Ligand-Target Pair
TargetEndoplasmic reticulum mannosyl-oligosaccharide 1,2-alpha-mannosidase(Homo sapiens (Human))
Universidade Do Porto 687
Curated by ChEMBL
Universidade Do Porto 687
Curated by ChEMBL
Affinity DataKi: 230nMAssay Description:Inhibition of human ER alpha mannosidase 1More data for this Ligand-Target Pair
Affinity DataKi: 270nMAssay Description:Competitive inhibition of N-terminal His-tagged human OGA using pNP-GlcNAc as chromogenic substrate assessed as inhibition constant by measuring libe...More data for this Ligand-Target Pair
Affinity DataKi: 270nMAssay Description:Binding affinity to human H3 receptor assessed as inhibition constant incubated for 90 mins by scintillation counting methodMore data for this Ligand-Target Pair
Ligand Info
TargetEndoplasmic reticulum mannosyl-oligosaccharide 1,2-alpha-mannosidase(Homo sapiens (Human))
Universidade Do Porto 687
Curated by ChEMBL
Universidade Do Porto 687
Curated by ChEMBL
Affinity DataKi: 310nMAssay Description:Inhibition of human ER alpha mannosidase 1More data for this Ligand-Target Pair
TargetEndoplasmic reticulum mannosyl-oligosaccharide 1,2-alpha-mannosidase(Homo sapiens (Human))
Universidade Do Porto 687
Curated by ChEMBL
Universidade Do Porto 687
Curated by ChEMBL
Affinity DataKi: 310nMAssay Description:Inhibition of human ER alpha mannosidase 1More data for this Ligand-Target Pair
Affinity DataKi: 332nMAssay Description:Competitive inhibition of cow HexA/HexB (unknown origin) using pNP-GlcNAc as substrate assessed as inhibition constant by measuring liberation of nit...More data for this Ligand-Target Pair
Affinity DataKi: 398nMAssay Description:Displacement of [3H]-Histamine from human histamine 3 receptor transfected in HEK293T cells incubated for 16 hrs by liquid scintillation counter anal...More data for this Ligand-Target Pair
Affinity DataKi: 413nMAssay Description:Competitive inhibition of cow HexA/HexB (unknown origin) using pNP-GlcNAc as substrate assessed as inhibition constant by measuring liberation of nit...More data for this Ligand-Target Pair