Affinity DataKi: 0.0100nMAssay Description:Inhibition of GCP2 by top scintillation counter in presence of 30 nM NAA[3]GMore data for this Ligand-Target Pair
TargetPoly [ADP-ribose] polymerase 1(Homo sapiens (Human))
Johns Hopkins University Brain Science Institute
Curated by ChEMBL
Johns Hopkins University Brain Science Institute
Curated by ChEMBL
TargetPoly [ADP-ribose] polymerase 1(Homo sapiens (Human))
Johns Hopkins University Brain Science Institute
Curated by ChEMBL
Johns Hopkins University Brain Science Institute
Curated by ChEMBL
Affinity DataKi: 60nMAssay Description:Competitive inhibition of recombinant human DAAO expressed in HEK cells by double reciprocal plot analysis in presence of D-serineMore data for this Ligand-Target Pair
TargetAldehyde dehydrogenase family 1 member A3(Homo sapiens (Human))
University Of Pisa
Curated by ChEMBL
University Of Pisa
Curated by ChEMBL
Affinity DataKi: 120nMAssay Description:Competitive inhibition of human recombinant ALDH1A3 pre-incubated for 5 mins before acetaldehyde addition by continuous spectrometric assay relative ...More data for this Ligand-Target Pair
TargetAldehyde dehydrogenase family 1 member A3(Homo sapiens (Human))
University Of Pisa
Curated by ChEMBL
University Of Pisa
Curated by ChEMBL
Affinity DataKi: 540nMAssay Description:Competitive inhibition of recombinant human 6His-tagged ALDH1A3 expressed in Escherichia coli BL21(DE3) using varying level of acetaldehyde as substr...More data for this Ligand-Target Pair
Affinity DataKi: 920nMAssay Description:Competitive inhibition of human recombinant ALDH1A2 pre-incubated for 5 mins before acetaldehyde addition by continuous spectrometric assay relative ...More data for this Ligand-Target Pair
TargetInosine-5'-monophosphate dehydrogenase(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)
National Institute Of Allergy And Infectious Diseases
Curated by ChEMBL
National Institute Of Allergy And Infectious Diseases
Curated by ChEMBL
Affinity DataKi: 1.10E+3nMAssay Description:Inhibition of Mycobacterium tuberculosis IMPDH2 Y487C mutant using IMP as substrate by spectrophotometric methodMore data for this Ligand-Target Pair
TargetInosine-5'-monophosphate dehydrogenase 2(Homo sapiens (Human))
National Institute Of Allergy And Infectious Diseases
Curated by ChEMBL
National Institute Of Allergy And Infectious Diseases
Curated by ChEMBL
Affinity DataKi: 2.00E+3nMAssay Description:Inhibition of human IMPDH2 using IMP as substrate by spectrophotometric methodMore data for this Ligand-Target Pair
TargetGlutaminase kidney isoform, mitochondrial(Homo sapiens (Human))
Johns Hopkins University
Curated by ChEMBL
Johns Hopkins University
Curated by ChEMBL
Affinity DataKi: 2.00E+3nMAssay Description:Uncompetitive inhibition of human kidney glutaminase (124 to 669) assessed as reduction of glutamine hydrolysis by double-reciprocal plot analysisMore data for this Ligand-Target Pair
TargetInosine-5'-monophosphate dehydrogenase 2(Homo sapiens (Human))
National Institute Of Allergy And Infectious Diseases
Curated by ChEMBL
National Institute Of Allergy And Infectious Diseases
Curated by ChEMBL
Affinity DataKi: 2.30E+3nMAssay Description:Inhibition of human IMPDH2 using IMP as substrate by spectrophotometric methodMore data for this Ligand-Target Pair
TargetInosine-5'-monophosphate dehydrogenase 2(Homo sapiens (Human))
National Institute Of Allergy And Infectious Diseases
Curated by ChEMBL
National Institute Of Allergy And Infectious Diseases
Curated by ChEMBL
Affinity DataKi: 2.90E+3nMAssay Description:Inhibition of human IMPDH2 using IMP as substrate by spectrophotometric methodMore data for this Ligand-Target Pair
TargetInosine-5'-monophosphate dehydrogenase 2(Homo sapiens (Human))
National Institute Of Allergy And Infectious Diseases
Curated by ChEMBL
National Institute Of Allergy And Infectious Diseases
Curated by ChEMBL
Affinity DataKi: 3.30E+3nMAssay Description:Inhibition of human IMPDH2 using IMP as substrate by spectrophotometric methodMore data for this Ligand-Target Pair
TargetGMP reductase 2(Homo sapiens)
National Institute Of Allergy And Infectious Diseases
Curated by ChEMBL
National Institute Of Allergy And Infectious Diseases
Curated by ChEMBL
Affinity DataKi: >5.00E+3nMAssay Description:Inhibition of human GMPR2 using GMP as substrate by spectrophotometric methodMore data for this Ligand-Target Pair
TargetGMP reductase 2(Homo sapiens)
National Institute Of Allergy And Infectious Diseases
Curated by ChEMBL
National Institute Of Allergy And Infectious Diseases
Curated by ChEMBL
Affinity DataKi: >5.00E+3nMAssay Description:Inhibition of human GMPR2 using GMP as substrate by spectrophotometric methodMore data for this Ligand-Target Pair
TargetGMP reductase 2(Homo sapiens)
National Institute Of Allergy And Infectious Diseases
Curated by ChEMBL
National Institute Of Allergy And Infectious Diseases
Curated by ChEMBL
Affinity DataKi: >5.00E+3nMAssay Description:Inhibition of human GMPR2 using GMP as substrate by spectrophotometric methodMore data for this Ligand-Target Pair
TargetGMP reductase 2(Homo sapiens)
National Institute Of Allergy And Infectious Diseases
Curated by ChEMBL
National Institute Of Allergy And Infectious Diseases
Curated by ChEMBL
Affinity DataKi: >5.00E+3nMAssay Description:Inhibition of human GMPR2 using GMP as substrate by spectrophotometric methodMore data for this Ligand-Target Pair
TargetGMP reductase 2(Homo sapiens)
National Institute Of Allergy And Infectious Diseases
Curated by ChEMBL
National Institute Of Allergy And Infectious Diseases
Curated by ChEMBL
Affinity DataKi: >5.00E+3nMAssay Description:Inhibition of human GMPR2 using GMP as substrate by spectrophotometric methodMore data for this Ligand-Target Pair
TargetGMP reductase 2(Homo sapiens)
National Institute Of Allergy And Infectious Diseases
Curated by ChEMBL
National Institute Of Allergy And Infectious Diseases
Curated by ChEMBL
Affinity DataKi: >5.00E+3nMAssay Description:Inhibition of human GMPR2 using GMP as substrate by spectrophotometric methodMore data for this Ligand-Target Pair
TargetInosine-5'-monophosphate dehydrogenase 2(Homo sapiens (Human))
National Institute Of Allergy And Infectious Diseases
Curated by ChEMBL
National Institute Of Allergy And Infectious Diseases
Curated by ChEMBL
Affinity DataKi: >5.00E+3nMAssay Description:Inhibition of human IMPDH2 using IMP as substrate by spectrophotometric methodMore data for this Ligand-Target Pair
TargetInosine-5'-monophosphate dehydrogenase 2(Homo sapiens (Human))
National Institute Of Allergy And Infectious Diseases
Curated by ChEMBL
National Institute Of Allergy And Infectious Diseases
Curated by ChEMBL
Affinity DataKi: >5.00E+3nMAssay Description:Inhibition of human IMPDH2 using IMP as substrate by spectrophotometric methodMore data for this Ligand-Target Pair
TargetGMP reductase 2(Homo sapiens)
National Institute Of Allergy And Infectious Diseases
Curated by ChEMBL
National Institute Of Allergy And Infectious Diseases
Curated by ChEMBL
Affinity DataKi: >5.00E+3nMAssay Description:Inhibition of human GMPR2 using GMP as substrate by spectrophotometric methodMore data for this Ligand-Target Pair
TargetGMP reductase 2(Homo sapiens)
National Institute Of Allergy And Infectious Diseases
Curated by ChEMBL
National Institute Of Allergy And Infectious Diseases
Curated by ChEMBL
Affinity DataKi: >5.00E+3nMAssay Description:Inhibition of human GMPR2 using GMP as substrate by spectrophotometric methodMore data for this Ligand-Target Pair
TargetGMP reductase 2(Homo sapiens)
National Institute Of Allergy And Infectious Diseases
Curated by ChEMBL
National Institute Of Allergy And Infectious Diseases
Curated by ChEMBL
Affinity DataKi: >5.00E+3nMAssay Description:Inhibition of human GMPR2 using GMP as substrate by spectrophotometric methodMore data for this Ligand-Target Pair
TargetGMP reductase 2(Homo sapiens)
National Institute Of Allergy And Infectious Diseases
Curated by ChEMBL
National Institute Of Allergy And Infectious Diseases
Curated by ChEMBL
Affinity DataKi: >5.00E+3nMAssay Description:Inhibition of human GMPR2 using GMP as substrate by spectrophotometric methodMore data for this Ligand-Target Pair
TargetGMP reductase 2(Homo sapiens)
National Institute Of Allergy And Infectious Diseases
Curated by ChEMBL
National Institute Of Allergy And Infectious Diseases
Curated by ChEMBL
Affinity DataKi: >5.00E+3nMAssay Description:Inhibition of human GMPR2 using GMP as substrate by spectrophotometric methodMore data for this Ligand-Target Pair
TargetInosine-5'-monophosphate dehydrogenase 2(Homo sapiens (Human))
National Institute Of Allergy And Infectious Diseases
Curated by ChEMBL
National Institute Of Allergy And Infectious Diseases
Curated by ChEMBL
Affinity DataKi: >5.00E+3nMAssay Description:Inhibition of human IMPDH2 using IMP as substrate by spectrophotometric methodMore data for this Ligand-Target Pair
TargetInosine-5'-monophosphate dehydrogenase 2(Homo sapiens (Human))
National Institute Of Allergy And Infectious Diseases
Curated by ChEMBL
National Institute Of Allergy And Infectious Diseases
Curated by ChEMBL
Affinity DataKi: >5.00E+3nMAssay Description:Inhibition of human IMPDH2 using IMP as substrate by spectrophotometric methodMore data for this Ligand-Target Pair
TargetInosine-5'-monophosphate dehydrogenase 2(Homo sapiens (Human))
National Institute Of Allergy And Infectious Diseases
Curated by ChEMBL
National Institute Of Allergy And Infectious Diseases
Curated by ChEMBL
Affinity DataKi: >5.00E+3nMAssay Description:Inhibition of human IMPDH2 using IMP as substrate by spectrophotometric methodMore data for this Ligand-Target Pair
TargetInosine-5'-monophosphate dehydrogenase 2(Homo sapiens (Human))
National Institute Of Allergy And Infectious Diseases
Curated by ChEMBL
National Institute Of Allergy And Infectious Diseases
Curated by ChEMBL
Affinity DataKi: >5.00E+3nMAssay Description:Inhibition of human IMPDH2 using IMP as substrate by spectrophotometric methodMore data for this Ligand-Target Pair
TargetInosine-5'-monophosphate dehydrogenase 2(Homo sapiens (Human))
National Institute Of Allergy And Infectious Diseases
Curated by ChEMBL
National Institute Of Allergy And Infectious Diseases
Curated by ChEMBL
Affinity DataKi: >5.00E+3nMAssay Description:Inhibition of human IMPDH2 using IMP as substrate by spectrophotometric methodMore data for this Ligand-Target Pair
TargetGMP reductase 2(Homo sapiens)
National Institute Of Allergy And Infectious Diseases
Curated by ChEMBL
National Institute Of Allergy And Infectious Diseases
Curated by ChEMBL
Affinity DataKi: >5.00E+3nMAssay Description:Inhibition of human GMPR2 using GMP as substrate by spectrophotometric methodMore data for this Ligand-Target Pair
TargetGMP reductase 2(Homo sapiens)
National Institute Of Allergy And Infectious Diseases
Curated by ChEMBL
National Institute Of Allergy And Infectious Diseases
Curated by ChEMBL
Affinity DataKi: >5.00E+3nMAssay Description:Inhibition of human GMPR2 using GMP as substrate by spectrophotometric methodMore data for this Ligand-Target Pair
TargetGMP reductase 2(Homo sapiens)
National Institute Of Allergy And Infectious Diseases
Curated by ChEMBL
National Institute Of Allergy And Infectious Diseases
Curated by ChEMBL
Affinity DataKi: >5.00E+3nMAssay Description:Inhibition of human GMPR2 using GMP as substrate by spectrophotometric methodMore data for this Ligand-Target Pair
TargetGMP reductase 2(Homo sapiens)
National Institute Of Allergy And Infectious Diseases
Curated by ChEMBL
National Institute Of Allergy And Infectious Diseases
Curated by ChEMBL
Affinity DataKi: >5.00E+3nMAssay Description:Inhibition of human GMPR2 using GMP as substrate by spectrophotometric methodMore data for this Ligand-Target Pair
TargetGMP reductase 2(Homo sapiens)
National Institute Of Allergy And Infectious Diseases
Curated by ChEMBL
National Institute Of Allergy And Infectious Diseases
Curated by ChEMBL
Affinity DataKi: >5.00E+3nMAssay Description:Inhibition of human GMPR2 using GMP as substrate by spectrophotometric methodMore data for this Ligand-Target Pair
TargetInosine-5'-monophosphate dehydrogenase 2(Homo sapiens (Human))
National Institute Of Allergy And Infectious Diseases
Curated by ChEMBL
National Institute Of Allergy And Infectious Diseases
Curated by ChEMBL
Affinity DataKi: >5.00E+3nMAssay Description:Inhibition of human IMPDH2 using IMP as substrate by spectrophotometric methodMore data for this Ligand-Target Pair
TargetGMP reductase 2(Homo sapiens)
National Institute Of Allergy And Infectious Diseases
Curated by ChEMBL
National Institute Of Allergy And Infectious Diseases
Curated by ChEMBL
Affinity DataKi: >5.00E+3nMAssay Description:Inhibition of human GMPR2 using GMP as substrate by spectrophotometric methodMore data for this Ligand-Target Pair
TargetInosine-5'-monophosphate dehydrogenase 2(Homo sapiens (Human))
National Institute Of Allergy And Infectious Diseases
Curated by ChEMBL
National Institute Of Allergy And Infectious Diseases
Curated by ChEMBL
Affinity DataKi: >5.00E+3nMAssay Description:Inhibition of human IMPDH2 using IMP as substrate by spectrophotometric methodMore data for this Ligand-Target Pair
TargetInosine-5'-monophosphate dehydrogenase 2(Homo sapiens (Human))
National Institute Of Allergy And Infectious Diseases
Curated by ChEMBL
National Institute Of Allergy And Infectious Diseases
Curated by ChEMBL
Affinity DataKi: >5.00E+3nMAssay Description:Inhibition of human IMPDH2 using IMP as substrate by spectrophotometric methodMore data for this Ligand-Target Pair
TargetInosine-5'-monophosphate dehydrogenase 2(Homo sapiens (Human))
National Institute Of Allergy And Infectious Diseases
Curated by ChEMBL
National Institute Of Allergy And Infectious Diseases
Curated by ChEMBL
Affinity DataKi: >5.00E+3nMAssay Description:Inhibition of human IMPDH2 using IMP as substrate by spectrophotometric methodMore data for this Ligand-Target Pair
TargetInosine-5'-monophosphate dehydrogenase 2(Homo sapiens (Human))
National Institute Of Allergy And Infectious Diseases
Curated by ChEMBL
National Institute Of Allergy And Infectious Diseases
Curated by ChEMBL
Affinity DataKi: >5.00E+3nMAssay Description:Inhibition of human IMPDH2 using IMP as substrate by spectrophotometric methodMore data for this Ligand-Target Pair
TargetInosine-5'-monophosphate dehydrogenase 2(Homo sapiens (Human))
National Institute Of Allergy And Infectious Diseases
Curated by ChEMBL
National Institute Of Allergy And Infectious Diseases
Curated by ChEMBL
Affinity DataKi: >5.00E+3nMAssay Description:Inhibition of human IMPDH2 using IMP as substrate by spectrophotometric methodMore data for this Ligand-Target Pair
TargetInosine-5'-monophosphate dehydrogenase 2(Homo sapiens (Human))
National Institute Of Allergy And Infectious Diseases
Curated by ChEMBL
National Institute Of Allergy And Infectious Diseases
Curated by ChEMBL
Affinity DataKi: >5.00E+3nMAssay Description:Inhibition of human IMPDH2 using IMP as substrate by spectrophotometric methodMore data for this Ligand-Target Pair
TargetInosine-5'-monophosphate dehydrogenase 2(Homo sapiens (Human))
National Institute Of Allergy And Infectious Diseases
Curated by ChEMBL
National Institute Of Allergy And Infectious Diseases
Curated by ChEMBL
Affinity DataKi: >5.00E+3nMAssay Description:Inhibition of human IMPDH2 using IMP as substrate by spectrophotometric methodMore data for this Ligand-Target Pair
TargetInosine-5'-monophosphate dehydrogenase 2(Homo sapiens (Human))
National Institute Of Allergy And Infectious Diseases
Curated by ChEMBL
National Institute Of Allergy And Infectious Diseases
Curated by ChEMBL
Affinity DataKi: >5.00E+3nMAssay Description:Inhibition of human IMPDH2 using IMP as substrate by spectrophotometric methodMore data for this Ligand-Target Pair
TargetInosine-5'-monophosphate dehydrogenase 2(Homo sapiens (Human))
National Institute Of Allergy And Infectious Diseases
Curated by ChEMBL
National Institute Of Allergy And Infectious Diseases
Curated by ChEMBL
Affinity DataKi: >5.00E+3nMAssay Description:Inhibition of human IMPDH2 using IMP as substrate by spectrophotometric methodMore data for this Ligand-Target Pair
TargetInosine-5'-monophosphate dehydrogenase 2(Homo sapiens (Human))
National Institute Of Allergy And Infectious Diseases
Curated by ChEMBL
National Institute Of Allergy And Infectious Diseases
Curated by ChEMBL
Affinity DataKi: >5.00E+3nMAssay Description:Inhibition of human IMPDH2 using IMP as substrate by spectrophotometric methodMore data for this Ligand-Target Pair
TargetGMP reductase 2(Homo sapiens)
National Institute Of Allergy And Infectious Diseases
Curated by ChEMBL
National Institute Of Allergy And Infectious Diseases
Curated by ChEMBL
Affinity DataKi: >5.00E+3nMAssay Description:Inhibition of human GMPR2 using GMP as substrate by spectrophotometric methodMore data for this Ligand-Target Pair
TargetGMP reductase 2(Homo sapiens)
National Institute Of Allergy And Infectious Diseases
Curated by ChEMBL
National Institute Of Allergy And Infectious Diseases
Curated by ChEMBL
Affinity DataKi: >5.00E+3nMAssay Description:Inhibition of human GMPR2 using GMP as substrate by spectrophotometric methodMore data for this Ligand-Target Pair