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Found 1378 with Last Name = 'findlay' and Initial = 'ad'
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
Pharmaxis

Curated by ChEMBL
LigandPNGBDBM50589703(CHEMBL5196906)
Affinity DataKi:  8nMAssay Description:Time dependent inhibition of human recombinant MAO-B assessed as inhibition constantMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetLysyl oxidase homolog 2(Homo sapiens (Human))
Pharmaxis

Curated by ChEMBL
LigandPNGBDBM50505638(CHEMBL4457578)
Affinity DataKi:  83nMAssay Description:Time-dependent inhibition of recombinant human C-terminal His-tagged LOLX2 (1-774 residues) expressed in mouse myeloma cells assessed as apparent inh...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetRetina-specific copper amine oxidase(Homo sapiens (Human))
Pharmaxis

Curated by ChEMBL
LigandPNGBDBM50589703(CHEMBL5196906)
Affinity DataKi:  710nMAssay Description:Time dependent inhibition of human recombinant SSAO assessed as inhibition constantMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetAmine oxidase [flavin-containing] B(Mus musculus)
Pharmaxis

Curated by ChEMBL
LigandPNGBDBM50589703(CHEMBL5196906)
Affinity DataIC50:  0.400nMAssay Description:Inhibition of mouse muscle MAO-BMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
Pharmaxis

Curated by ChEMBL
LigandPNGBDBM50589702(CHEMBL5186190)
Affinity DataIC50:  2nMAssay Description:Inhibition of human recombinant MAO-BMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
Pharmaxis

Curated by ChEMBL
LigandPNGBDBM50589700(CHEMBL5204901)
Affinity DataIC50:  2nMAssay Description:Inhibition of human recombinant MAO-BMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
Pharmaxis

Curated by ChEMBL
LigandPNGBDBM50246766(CHEMBL489079 | Mofegiline | US9302986, Mofegiline)
Affinity DataIC50:  2nMAssay Description:Inhibition of human recombinant MAO-BMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
Pharmaxis

Curated by ChEMBL
LigandPNGBDBM50589699(CHEMBL5197971)
Affinity DataIC50:  3nMAssay Description:Inhibition of human recombinant MAO-BMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
Pharmaxis

Curated by ChEMBL
LigandPNGBDBM50589698(CHEMBL5199917)
Affinity DataIC50:  3nMAssay Description:Inhibition of human recombinant MAO-BMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetRetina-specific copper amine oxidase(Homo sapiens (Human))
Pharmaxis

Curated by ChEMBL
LigandPNGBDBM50589695(CHEMBL5198317)
Affinity DataIC50:  4nMAssay Description:Inhibition of recombinant human SSAOMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
Pharmaxis

Curated by ChEMBL
LigandPNGBDBM50589695(CHEMBL5198317)
Affinity DataIC50:  4nMAssay Description:Inhibition of human recombinant MAO-BMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
Pharmaxis

Curated by ChEMBL
LigandPNGBDBM50246766(CHEMBL489079 | Mofegiline | US9302986, Mofegiline)
Affinity DataIC50:  5nMpH: 7.4 T: 2°CAssay Description:Recombinant human MAO-B (0.06 mg/mL; Sigma Aldrich) was used as source of MAO-B enzyme activities. The assay was performed in a similar way as for hu...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetLysyl oxidase homolog 2(Homo sapiens (Human))
Pharmaxis

Curated by ChEMBL
LigandPNGBDBM50505638(CHEMBL4457578)
Affinity DataIC50:  5nMAssay Description:Inhibition of recombinant human C-terminal His-tagged LOLX2 (1-774 residues) expressed in mouse myeloma cells using putrescine as substrate preincuba...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetLysyl oxidase homolog 2(Homo sapiens (Human))
Pharmaxis

Curated by ChEMBL
LigandPNGBDBM50505633(CHEMBL4448713)
Affinity DataIC50:  5nMAssay Description:Inhibition of recombinant human C-terminal His-tagged LOLX2 (1-774 residues) expressed in mouse myeloma cells using putrescine as substrate preincuba...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetLysyl oxidase homolog 2(Homo sapiens (Human))
Pharmaxis

Curated by ChEMBL
LigandPNGBDBM50505638(CHEMBL4457578)
Affinity DataIC50:  5nMAssay Description:Inhibition of recombinant human C-terminal His-tagged LOLX2 (1-774 residues) expressed in mouse myeloma cells using putrescine as substrate preincuba...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
Pharmaxis

Curated by ChEMBL
LigandPNGBDBM50589703(CHEMBL5196906)
Affinity DataIC50:  5nMAssay Description:Inhibition of human recombinant MAO-BMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetRetina-specific copper amine oxidase(Homo sapiens (Human))
Pharmaxis

Curated by ChEMBL
LigandPNGBDBM50589700(CHEMBL5204901)
Affinity DataIC50:  5nMAssay Description:Inhibition of recombinant human SSAOMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetMembrane primary amine oxidase(Rattus norvegicus (Rat))
Pharmaxis

Curated by ChEMBL
LigandPNGBDBM50589703(CHEMBL5196906)
Affinity DataIC50:  5nMAssay Description:Inhibition of rat SSAOMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetRetina-specific copper amine oxidase(Homo sapiens (Human))
Pharmaxis

Curated by ChEMBL
LigandPNGBDBM50589696(CHEMBL5201033)
Affinity DataIC50:  6nMAssay Description:Inhibition of recombinant human SSAOMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetLysyl oxidase homolog 2(Mus musculus)
Pharmaxis

Curated by ChEMBL
LigandPNGBDBM50505638(CHEMBL4457578)
Affinity DataIC50:  6nMAssay Description:Inhibition of recombinant mouse C-terminal His-tagged LOLX2 (26-776 residues) expressed in mouse myeloma cells using putrescine as substrate preincub...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetLysyl oxidase homolog 2(Rattus norvegicus)
Pharmaxis

Curated by ChEMBL
LigandPNGBDBM50505638(CHEMBL4457578)
Affinity DataIC50:  6nMAssay Description:Inhibition of recombinant rat LOLX2 using putrescine as substrate preincubated with enzyme for 30 mins followed by substrate addition and measured ev...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
Pharmaxis

Curated by ChEMBL
LigandPNGBDBM50589696(CHEMBL5201033)
Affinity DataIC50:  9nMAssay Description:Inhibition of human recombinant MAO-BMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetLysyl oxidase homolog 2(Homo sapiens (Human))
Pharmaxis

Curated by ChEMBL
LigandPNGBDBM50505638(CHEMBL4457578)
Affinity DataIC50:  9nMAssay Description:Inhibition of LOXL2 in human IMR90 cells using putrescine as substrate preincubated with enzyme for 30 mins followed by substrate addition and measur...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetRetina-specific copper amine oxidase(Homo sapiens (Human))
Pharmaxis

Curated by ChEMBL
LigandPNGBDBM50246766(CHEMBL489079 | Mofegiline | US9302986, Mofegiline)
Affinity DataIC50:  10nMAssay Description:Inhibition of recombinant human SSAOMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetRetina-specific copper amine oxidase(Homo sapiens (Human))
Pharmaxis

Curated by ChEMBL
LigandPNGBDBM50589702(CHEMBL5186190)
Affinity DataIC50:  11nMAssay Description:Inhibition of recombinant human SSAOMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetRetina-specific copper amine oxidase(Homo sapiens (Human))
Pharmaxis

Curated by ChEMBL
LigandPNGBDBM50589699(CHEMBL5197971)
Affinity DataIC50:  12nMAssay Description:Inhibition of recombinant human SSAOMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
Pharmaxis

Curated by ChEMBL
LigandPNGBDBM50589697(CHEMBL5194056)
Affinity DataIC50:  13nMAssay Description:Inhibition of human recombinant MAO-BMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetLysyl oxidase homolog 2(Homo sapiens (Human))
Pharmaxis

Curated by ChEMBL
LigandPNGBDBM50505640(CHEMBL4556859)
Affinity DataIC50:  13nMAssay Description:Inhibition of recombinant human C-terminal His-tagged LOLX2 (1-774 residues) expressed in mouse myeloma cells using putrescine as substrate preincuba...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetLysyl oxidase homolog 2(Homo sapiens (Human))
Pharmaxis

Curated by ChEMBL
LigandPNGBDBM50505638(CHEMBL4457578)
Affinity DataIC50:  13nMAssay Description:Inhibition of recombinant human C-terminal His-tagged LOLX2 (1-774 residues) expressed in mouse myeloma cells assessed as inhibition of collagen oxid...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetLysyl oxidase homolog 2(Homo sapiens (Human))
Pharmaxis

Curated by ChEMBL
LigandPNGBDBM50505638(CHEMBL4457578)
Affinity DataIC50:  13nMAssay Description:Inhibition of recombinant human LOXL2 assessed as inhibition of collagen cross linking compound replenishment for 5 days and measured on day 7 by UPL...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetLysyl oxidase homolog 3(Homo sapiens (Human))
Pharmaxis

Curated by ChEMBL
LigandPNGBDBM50505638(CHEMBL4457578)
Affinity DataIC50:  16nMAssay Description:Inhibition of recombinant C-terminal His-tagged human LOXL3 (1 to 753 residues) expressed in CHO cells using putrescine as substrate preincubated wit...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetRetina-specific copper amine oxidase(Homo sapiens (Human))
Pharmaxis

Curated by ChEMBL
LigandPNGBDBM50589697(CHEMBL5194056)
Affinity DataIC50:  19nMAssay Description:Inhibition of recombinant human SSAOMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetRetina-specific copper amine oxidase(Homo sapiens (Human))
Pharmaxis

Curated by ChEMBL
LigandPNGBDBM50589703(CHEMBL5196906)
Affinity DataIC50:  19nMAssay Description:Inhibition of recombinant human SSAOMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetLysyl oxidase homolog 2(Homo sapiens (Human))
Pharmaxis

Curated by ChEMBL
LigandPNGBDBM50505653(CHEMBL4458907)
Affinity DataIC50:  20nMAssay Description:Inhibition of recombinant human C-terminal His-tagged LOLX2 (1-774 residues) expressed in mouse myeloma cells using putrescine as substrate preincuba...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetLysyl oxidase homolog 2(Homo sapiens (Human))
Pharmaxis

Curated by ChEMBL
LigandPNGBDBM50505658(CHEMBL4581458)
Affinity DataIC50:  20nMAssay Description:Inhibition of recombinant human C-terminal His-tagged LOLX2 (1-774 residues) expressed in mouse myeloma cells using putrescine as substrate preincuba...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLysyl oxidase homolog 2(Homo sapiens (Human))
Pharmaxis

Curated by ChEMBL
LigandPNGBDBM50505647(CHEMBL4531065)
Affinity DataIC50:  20nMAssay Description:Inhibition of recombinant human C-terminal His-tagged LOLX2 (1-774 residues) expressed in mouse myeloma cells using putrescine as substrate preincuba...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetLysyl oxidase homolog 2(Homo sapiens (Human))
Pharmaxis

Curated by ChEMBL
LigandPNGBDBM50505657(CHEMBL4467234)
Affinity DataIC50:  20nMAssay Description:Inhibition of recombinant human C-terminal His-tagged LOLX2 (1-774 residues) expressed in mouse myeloma cells using putrescine as substrate preincuba...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetLysyl oxidase homolog 2(Homo sapiens (Human))
Pharmaxis

Curated by ChEMBL
LigandPNGBDBM50505643(CHEMBL4582216)
Affinity DataIC50:  25nMAssay Description:Inhibition of recombinant human C-terminal His-tagged LOLX2 (1-774 residues) expressed in mouse myeloma cells using putrescine as substrate preincuba...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
Pharmaxis

Curated by ChEMBL
LigandPNGBDBM50589701(CHEMBL5186898)
Affinity DataIC50:  26nMAssay Description:Inhibition of human recombinant MAO-BMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetRetina-specific copper amine oxidase(Homo sapiens (Human))
Pharmaxis

Curated by ChEMBL
LigandPNGBDBM50589703(CHEMBL5196906)
Affinity DataIC50:  29nMAssay Description:Inhibition of SSAO in HMEC cellsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetRetina-specific copper amine oxidase(Homo sapiens (Human))
Pharmaxis

Curated by ChEMBL
LigandPNGBDBM50589701(CHEMBL5186898)
Affinity DataIC50:  32nMAssay Description:Inhibition of recombinant human SSAOMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetLysyl oxidase homolog 2(Homo sapiens (Human))
Pharmaxis

Curated by ChEMBL
LigandPNGBDBM50505634(CHEMBL4569453)
Affinity DataIC50:  50nMAssay Description:Inhibition of recombinant human C-terminal His-tagged LOLX2 (1-774 residues) expressed in mouse myeloma cells using putrescine as substrate preincuba...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetLysyl oxidase homolog 2(Homo sapiens (Human))
Pharmaxis

Curated by ChEMBL
LigandPNGBDBM50505645(CHEMBL4550754)
Affinity DataIC50:  50nMAssay Description:Inhibition of recombinant human C-terminal His-tagged LOLX2 (1-774 residues) expressed in mouse myeloma cells using putrescine as substrate preincuba...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMembrane primary amine oxidase(Homo sapiens (Human))
Pharmaxis

Curated by ChEMBL
LigandPNGBDBM50505648(CHEMBL4562149)
Affinity DataIC50:  50nMAssay Description:Inhibition of recombinant human SSAO using benzylamine as substrate preincubated with enzyme for 30 mins followed by substrate addition and measured ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetLysyl oxidase homolog 2(Homo sapiens (Human))
Pharmaxis

Curated by ChEMBL
LigandPNGBDBM50505661(CHEMBL4574820)
Affinity DataIC50:  63nMAssay Description:Inhibition of recombinant human C-terminal His-tagged LOLX2 (1-774 residues) expressed in mouse myeloma cells using putrescine as substrate preincuba...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetLysyl oxidase homolog 2(Homo sapiens (Human))
Pharmaxis

Curated by ChEMBL
LigandPNGBDBM50505663(CHEMBL4451632)
Affinity DataIC50:  79nMAssay Description:Inhibition of recombinant human C-terminal His-tagged LOLX2 (1-774 residues) expressed in mouse myeloma cells using putrescine as substrate preincuba...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetLysyl oxidase homolog 2(Homo sapiens (Human))
Pharmaxis

Curated by ChEMBL
LigandPNGBDBM50505662(CHEMBL4446643)
Affinity DataIC50:  79nMAssay Description:Inhibition of recombinant human C-terminal His-tagged LOLX2 (1-774 residues) expressed in mouse myeloma cells using putrescine as substrate preincuba...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetLysyl oxidase homolog 2(Homo sapiens (Human))
Pharmaxis

Curated by ChEMBL
LigandPNGBDBM50505652(CHEMBL4463296)
Affinity DataIC50:  100nMAssay Description:Inhibition of recombinant human C-terminal His-tagged LOLX2 (1-774 residues) expressed in mouse myeloma cells using putrescine as substrate preincuba...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAmiloride-sensitive amine oxidase [copper-containing](Homo sapiens (Human))
Boehringer Ingelheim International

US Patent
LigandPNGBDBM220884(US9302986, 18)
Affinity DataIC50: <100nMpH: 7.4 T: 2°CAssay Description:Recombinant human DAO (2.4 μg/mL) was used as source of DAO enzyme activities. The assay was performed as described in the method for human SSAO/V...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetAmiloride-sensitive amine oxidase [copper-containing](Homo sapiens (Human))
Boehringer Ingelheim International

US Patent
LigandPNGBDBM220869(US9302986, 2)
Affinity DataIC50: <100nMpH: 7.4 T: 2°CAssay Description:Recombinant human DAO (2.4 μg/mL) was used as source of DAO enzyme activities. The assay was performed as described in the method for human SSAO/V...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
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