Affinity DataIC50: 1nMAssay Description:Inhibition of human NEP-mediated amyloid beta hydrolysisMore data for this Ligand-Target Pair
TargetM1 family aminopeptidase(Plasmodium falciparum (isolate FcB1 / Columbia))
University Of Lille
Curated by ChEMBL
University Of Lille
Curated by ChEMBL
Affinity DataIC50: 6nMAssay Description:Inhibition of Plasmodium falciparum FcB1 M1 aminopeptidaseMore data for this Ligand-Target Pair
Affinity DataIC50: 11nMAssay Description:Inhibition of human ACE-mediated amyloid beta hydrolysisMore data for this Ligand-Target Pair
TargetType II NADH:quinone oxidoreductase Ndh(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)
Cnrs
Curated by ChEMBL
Cnrs
Curated by ChEMBL
Affinity DataIC50: 12nMAssay Description:Inhibition of Mycobacterium tuberculosis recombinant type II NADH dehydrogenase ndh expressed in Escherichia coli assessed as rate of NADH oxidation ...More data for this Ligand-Target Pair
TargetType II NADH:quinone oxidoreductase Ndh(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)
Cnrs
Curated by ChEMBL
Cnrs
Curated by ChEMBL
Affinity DataIC50: 12nMAssay Description:Inhibition of Mycobacterium tuberculosis recombinant type II NADH dehydrogenase ndh expressed in Escherichia coli assessed as rate of NADH oxidation ...More data for this Ligand-Target Pair
TargetM1 family aminopeptidase(Plasmodium falciparum (isolate FcB1 / Columbia))
University Of Lille
Curated by ChEMBL
University Of Lille
Curated by ChEMBL
Affinity DataIC50: 13nMAssay Description:Inhibition of Plasmodium falciparum FcB1 M1 aminopeptidaseMore data for this Ligand-Target Pair
TargetType II NADH:quinone oxidoreductase Ndh(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)
Cnrs
Curated by ChEMBL
Cnrs
Curated by ChEMBL
Affinity DataIC50: 28nMAssay Description:Inhibition of Mycobacterium tuberculosis recombinant type II NADH dehydrogenase ndh expressed in Escherichia coli assessed as rate of NADH oxidation ...More data for this Ligand-Target Pair
Affinity DataIC50: 28nMAssay Description:Inhibitory activity against mammalian Aminopeptidase N (APN)More data for this Ligand-Target Pair
Affinity DataIC50: 29nMAssay Description:Inhibition of human erythrocyte carbonic anhydrase-2 assessed as hydrolysis of 4-nitrophenylacetateMore data for this Ligand-Target Pair
TargetType II NADH:quinone oxidoreductase Ndh(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)
Cnrs
Curated by ChEMBL
Cnrs
Curated by ChEMBL
Affinity DataIC50: 32nMAssay Description:Inhibition of Mycobacterium tuberculosis recombinant type II NADH dehydrogenase ndh expressed in Escherichia coli assessed as rate of NADH oxidation ...More data for this Ligand-Target Pair
TargetType II NADH:quinone oxidoreductase Ndh(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)
Cnrs
Curated by ChEMBL
Cnrs
Curated by ChEMBL
Affinity DataIC50: 37nMAssay Description:Inhibition of Mycobacterium smegmatis MC2 155 recombinant type II NADH dehydrogenase ndh expressed in Escherichia coli assessed as rate of NADH oxida...More data for this Ligand-Target Pair
TargetType II NADH:quinone oxidoreductase Ndh(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)
Cnrs
Curated by ChEMBL
Cnrs
Curated by ChEMBL
Affinity DataIC50: 41nMAssay Description:Inhibition of Mycobacterium smegmatis MC2 155 recombinant type II NADH dehydrogenase ndh expressed in Escherichia coli assessed as rate of NADH oxida...More data for this Ligand-Target Pair
TargetM1 family aminopeptidase(Plasmodium falciparum (isolate FcB1 / Columbia))
University Of Lille
Curated by ChEMBL
University Of Lille
Curated by ChEMBL
Affinity DataIC50: 41nMAssay Description:Inhibition of Plasmodium falciparum FcB1 M1 aminopeptidaseMore data for this Ligand-Target Pair
TargetType II NADH:quinone oxidoreductase Ndh(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)
Cnrs
Curated by ChEMBL
Cnrs
Curated by ChEMBL
Affinity DataIC50: 42nMAssay Description:Inhibition of Mycobacterium smegmatis MC2 155 recombinant type II NADH dehydrogenase ndh expressed in Escherichia coli assessed as rate of NADH oxida...More data for this Ligand-Target Pair
TargetM1 family aminopeptidase(Plasmodium falciparum (isolate FcB1 / Columbia))
University Of Lille
Curated by ChEMBL
University Of Lille
Curated by ChEMBL
Affinity DataIC50: 45nMAssay Description:Inhibition of Plasmodium falciparum FcB1 M1 aminopeptidaseMore data for this Ligand-Target Pair
TargetM1 family aminopeptidase(Plasmodium falciparum (isolate FcB1 / Columbia))
University Of Lille
Curated by ChEMBL
University Of Lille
Curated by ChEMBL
Affinity DataIC50: 46nMAssay Description:Inhibition of Plasmodium falciparum FcB1 M1 aminopeptidaseMore data for this Ligand-Target Pair
TargetM1 family aminopeptidase(Plasmodium falciparum (isolate FcB1 / Columbia))
University Of Lille
Curated by ChEMBL
University Of Lille
Curated by ChEMBL
Affinity DataIC50: 57nMAssay Description:Inhibition of Plasmodium falciparum FcB1 M1 aminopeptidaseMore data for this Ligand-Target Pair
TargetType II NADH:quinone oxidoreductase NdhA(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)
Cnrs
Curated by ChEMBL
Cnrs
Curated by ChEMBL
Affinity DataIC50: 57nMAssay Description:Inhibition of Mycobacterium smegmatis MC2 155 recombinant ndhA assessed as rate of NADH oxidation in the presence of an electron acceptor menadioneMore data for this Ligand-Target Pair
TargetType II NADH:quinone oxidoreductase NdhA(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)
Cnrs
Curated by ChEMBL
Cnrs
Curated by ChEMBL
Affinity DataIC50: 59nMAssay Description:Inhibition of Mycobacterium smegmatis MC2 155 recombinant ndhA assessed as rate of NADH oxidation in the presence of an electron acceptor menadioneMore data for this Ligand-Target Pair
Affinity DataIC50: 82nMAssay Description:Inhibition of microsomal neural aminopeptidase in pig kidneyMore data for this Ligand-Target Pair
TargetType II NADH:quinone oxidoreductase Ndh(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)
Cnrs
Curated by ChEMBL
Cnrs
Curated by ChEMBL
Affinity DataIC50: 88nMAssay Description:Inhibition of Mycobacterium smegmatis MC2 155 recombinant type II NADH dehydrogenase ndh expressed in Escherichia coli assessed as rate of NADH oxida...More data for this Ligand-Target Pair
TargetM1 family aminopeptidase(Plasmodium falciparum (isolate FcB1 / Columbia))
University Of Lille
Curated by ChEMBL
University Of Lille
Curated by ChEMBL
Affinity DataIC50: 91nMAssay Description:Inhibition of Plasmodium falciparum FcB1 M1 aminopeptidaseMore data for this Ligand-Target Pair
TargetType II NADH:quinone oxidoreductase NdhA(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)
Cnrs
Curated by ChEMBL
Cnrs
Curated by ChEMBL
Affinity DataIC50: 96nMAssay Description:Inhibition of Mycobacterium smegmatis MC2 155 recombinant ndhA assessed as rate of NADH oxidation in the presence of an electron acceptor menadioneMore data for this Ligand-Target Pair
Affinity DataIC50: 100nMAssay Description:Inhibition of human recombinant IDE-mediated amyloid beta (16 to 23) hydrolysis using ATTO 655-Cys-Lys-Leu-Val-Phe-Phe-Ala-Glu-Asp-Trp as substrate p...More data for this Ligand-Target Pair
TargetM1 family aminopeptidase(Plasmodium falciparum (isolate FcB1 / Columbia))
University Of Lille
Curated by ChEMBL
University Of Lille
Curated by ChEMBL
Affinity DataIC50: 107nMAssay Description:Inhibition of Plasmodium falciparum FcB1 M1 aminopeptidaseMore data for this Ligand-Target Pair
TargetM1 family aminopeptidase(Plasmodium falciparum (isolate FcB1 / Columbia))
University Of Lille
Curated by ChEMBL
University Of Lille
Curated by ChEMBL
Affinity DataIC50: 109nMAssay Description:Inhibition of Plasmodium falciparum FcB1 M1 aminopeptidaseMore data for this Ligand-Target Pair
TargetM1 family aminopeptidase(Plasmodium falciparum (isolate FcB1 / Columbia))
University Of Lille
Curated by ChEMBL
University Of Lille
Curated by ChEMBL
Affinity DataIC50: 125nMAssay Description:Inhibition of Plasmodium falciparum FcB1 M1 aminopeptidaseMore data for this Ligand-Target Pair
TargetM1 family aminopeptidase(Plasmodium falciparum (isolate FcB1 / Columbia))
University Of Lille
Curated by ChEMBL
University Of Lille
Curated by ChEMBL
Affinity DataIC50: 125nMAssay Description:Inhibition of Plasmodium falciparum FcB1 M1 aminopeptidaseMore data for this Ligand-Target Pair
TargetM1 family aminopeptidase(Plasmodium falciparum (isolate FcB1 / Columbia))
University Of Lille
Curated by ChEMBL
University Of Lille
Curated by ChEMBL
Affinity DataIC50: 130nMAssay Description:Inhibition of Plasmodium falciparum FcB1 M1 aminopeptidaseMore data for this Ligand-Target Pair
TargetM1 family aminopeptidase(Plasmodium falciparum (isolate FcB1 / Columbia))
University Of Lille
Curated by ChEMBL
University Of Lille
Curated by ChEMBL
Affinity DataIC50: 164nMAssay Description:Inhibition of Plasmodium falciparum FcB1 M1 aminopeptidaseMore data for this Ligand-Target Pair
TargetM1 family aminopeptidase(Plasmodium falciparum (isolate FcB1 / Columbia))
University Of Lille
Curated by ChEMBL
University Of Lille
Curated by ChEMBL
Affinity DataIC50: 170nMAssay Description:Inhibition of Plasmodium falciparum FcB1 M1 aminopeptidaseMore data for this Ligand-Target Pair
TargetType II NADH:quinone oxidoreductase Ndh(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)
Cnrs
Curated by ChEMBL
Cnrs
Curated by ChEMBL
Affinity DataIC50: 200nMAssay Description:Inhibition of Mycobacterium tuberculosis recombinant type II NADH dehydrogenase ndh expressed in Escherichia coli assessed as rate of NADH oxidation ...More data for this Ligand-Target Pair
TargetM1 family aminopeptidase(Plasmodium falciparum (isolate FcB1 / Columbia))
University Of Lille
Curated by ChEMBL
University Of Lille
Curated by ChEMBL
Affinity DataIC50: 206nMAssay Description:Inhibition of Plasmodium falciparum FcB1 M1 aminopeptidaseMore data for this Ligand-Target Pair
TargetM1 family aminopeptidase(Plasmodium falciparum (isolate FcB1 / Columbia))
University Of Lille
Curated by ChEMBL
University Of Lille
Curated by ChEMBL
Affinity DataIC50: 225nMAssay Description:Inhibition of Plasmodium falciparum FcB1 M1 aminopeptidaseMore data for this Ligand-Target Pair
TargetM1 family aminopeptidase(Plasmodium falciparum (isolate FcB1 / Columbia))
University Of Lille
Curated by ChEMBL
University Of Lille
Curated by ChEMBL
Affinity DataIC50: 231nMAssay Description:Inhibition of Plasmodium falciparum FcB1 M1 aminopeptidaseMore data for this Ligand-Target Pair
TargetM1 family aminopeptidase(Plasmodium falciparum (isolate FcB1 / Columbia))
University Of Lille
Curated by ChEMBL
University Of Lille
Curated by ChEMBL
Affinity DataIC50: 248nMAssay Description:Inhibition of Plasmodium falciparum FcB1 M1 aminopeptidaseMore data for this Ligand-Target Pair
TargetM1 family aminopeptidase(Plasmodium falciparum (isolate FcB1 / Columbia))
University Of Lille
Curated by ChEMBL
University Of Lille
Curated by ChEMBL
Affinity DataIC50: 253nMAssay Description:Inhibition of Plasmodium falciparum FcB1 M1 aminopeptidaseMore data for this Ligand-Target Pair
TargetM1 family aminopeptidase(Plasmodium falciparum (isolate FcB1 / Columbia))
University Of Lille
Curated by ChEMBL
University Of Lille
Curated by ChEMBL
Affinity DataIC50: 284nMAssay Description:Inhibitory activity for Plasmodium falciparum Zinc aminopeptidaseMore data for this Ligand-Target Pair
TargetType II NADH:quinone oxidoreductase NdhA(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)
Cnrs
Curated by ChEMBL
Cnrs
Curated by ChEMBL
Affinity DataIC50: 330nMAssay Description:Inhibition of Mycobacterium smegmatis MC2 155 recombinant ndhA assessed as rate of NADH oxidation in the presence of an electron acceptor menadioneMore data for this Ligand-Target Pair
TargetM1 family aminopeptidase(Plasmodium falciparum (isolate FcB1 / Columbia))
University Of Lille
Curated by ChEMBL
University Of Lille
Curated by ChEMBL
Affinity DataIC50: 330nMAssay Description:Inhibition of Plasmodium falciparum FcB1 M1 aminopeptidaseMore data for this Ligand-Target Pair
TargetType II NADH:quinone oxidoreductase Ndh(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)
Cnrs
Curated by ChEMBL
Cnrs
Curated by ChEMBL
Affinity DataIC50: 340nMAssay Description:Inhibition of Mycobacterium tuberculosis recombinant type II NADH dehydrogenase ndh expressed in Escherichia coli assessed as rate of NADH oxidation ...More data for this Ligand-Target Pair
TargetHTH-type transcriptional regulator EthR(Mycobacterium tuberculosis)
University Of Lille
Curated by ChEMBL
University Of Lille
Curated by ChEMBL
Affinity DataIC50: 400nMAssay Description:Inhibition of EthR binding to ethA promoter in 106-bp biotinylated DNA preincubated for 5 mins measured for 3 mins by surface plasmon resonance assayMore data for this Ligand-Target Pair
TargetM1 family aminopeptidase(Plasmodium falciparum (isolate FcB1 / Columbia))
University Of Lille
Curated by ChEMBL
University Of Lille
Curated by ChEMBL
Affinity DataIC50: 406nMAssay Description:Inhibition of Plasmodium falciparum FcB1 M1 aminopeptidaseMore data for this Ligand-Target Pair
Affinity DataIC50: 443nMAssay Description:Inhibition of pig kidney microsomal APNMore data for this Ligand-Target Pair
Affinity DataIC50: 443nMAssay Description:Inhibition of microsomal neural aminopeptidase in pig kidneyMore data for this Ligand-Target Pair
Affinity DataIC50: 452nMAssay Description:Inhibition of microsomal neural aminopeptidase in pig kidneyMore data for this Ligand-Target Pair
TargetType II NADH:quinone oxidoreductase Ndh(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)
Cnrs
Curated by ChEMBL
Cnrs
Curated by ChEMBL
Affinity DataIC50: 470nMAssay Description:Inhibition of Mycobacterium smegmatis MC2 155 recombinant type II NADH dehydrogenase ndh expressed in Escherichia coli assessed as rate of NADH oxida...More data for this Ligand-Target Pair
TargetM1 family aminopeptidase(Plasmodium falciparum (isolate FcB1 / Columbia))
University Of Lille
Curated by ChEMBL
University Of Lille
Curated by ChEMBL
Affinity DataIC50: 495nMAssay Description:Inhibition of Plasmodium falciparum FcB1 M1 aminopeptidaseMore data for this Ligand-Target Pair
TargetHTH-type transcriptional regulator EthR(Mycobacterium tuberculosis)
University Of Lille
Curated by ChEMBL
University Of Lille
Curated by ChEMBL
Affinity DataIC50: 500nMAssay Description:Inhibition of Mycobacterium tuberculosis EthR interaction to ethA promoter after 5 mins by surface plasmon resonance assayMore data for this Ligand-Target Pair
TargetM1 family aminopeptidase(Plasmodium falciparum (isolate FcB1 / Columbia))
University Of Lille
Curated by ChEMBL
University Of Lille
Curated by ChEMBL
Affinity DataIC50: 527nMAssay Description:Inhibition of Plasmodium falciparum FcB1 M1 aminopeptidaseMore data for this Ligand-Target Pair