TargetNeuronal acetylcholine receptor subunit alpha-2(Rattus norvegicus (Rat))
The Danish University of Pharmaceutical Sciences
Curated by PDSP Ki Database
The Danish University of Pharmaceutical Sciences
Curated by PDSP Ki Database
TargetNeuronal acetylcholine receptor subunit alpha-4(Rattus norvegicus (Rat))
The Danish University of Pharmaceutical Sciences
Curated by PDSP Ki Database
The Danish University of Pharmaceutical Sciences
Curated by PDSP Ki Database
TargetNeuronal acetylcholine receptor subunit alpha-4(Rattus norvegicus (Rat))
The Danish University of Pharmaceutical Sciences
Curated by PDSP Ki Database
The Danish University of Pharmaceutical Sciences
Curated by PDSP Ki Database
TargetNeuronal acetylcholine receptor subunit alpha-2(Rattus norvegicus (Rat))
The Danish University of Pharmaceutical Sciences
Curated by PDSP Ki Database
The Danish University of Pharmaceutical Sciences
Curated by PDSP Ki Database
TargetNeuronal acetylcholine receptor subunit alpha-3(Rattus norvegicus (Rat))
The Danish University of Pharmaceutical Sciences
Curated by PDSP Ki Database
The Danish University of Pharmaceutical Sciences
Curated by PDSP Ki Database
TargetNeuronal acetylcholine receptor subunit alpha-2(Rattus norvegicus (Rat))
The Danish University of Pharmaceutical Sciences
Curated by PDSP Ki Database
The Danish University of Pharmaceutical Sciences
Curated by PDSP Ki Database
TargetNeuronal acetylcholine receptor subunit alpha-4(Rattus norvegicus (Rat))
The Danish University of Pharmaceutical Sciences
Curated by PDSP Ki Database
The Danish University of Pharmaceutical Sciences
Curated by PDSP Ki Database
Affinity DataKi: 0.910nMAssay Description:Displacement of [3H]epibatidine from rat recombinant alpha4beta2 nAChR expressed in HEK293 cellsMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 2A(Homo sapiens (Human))
University Of Copenhagen
Curated by ChEMBL
University Of Copenhagen
Curated by ChEMBL
Affinity DataKi: 0.910nMAssay Description:Antagonist activity at human 5HT2A receptor expressed in HEK293 cells assessed as inhibition of 5HT-induced intracellular calcium release measured fo...More data for this Ligand-Target Pair
TargetGamma-aminobutyric acid receptor subunit alpha-1/beta-3/gamma-2(Homo sapiens (Human))
The Danish University Of Pharmaceutical Sciences
Curated by ChEMBL
The Danish University Of Pharmaceutical Sciences
Curated by ChEMBL
Affinity DataKi: 1.20nMAssay Description:Binding affinity at human GABAA alpha1beta3gamma2S expressed in Xenopus oocytes by voltage-clamp electrophysiologyMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-4(Rattus norvegicus (Rat))
The Danish University of Pharmaceutical Sciences
Curated by PDSP Ki Database
The Danish University of Pharmaceutical Sciences
Curated by PDSP Ki Database
TargetNeuronal acetylcholine receptor subunit alpha-2(Rattus norvegicus (Rat))
The Danish University of Pharmaceutical Sciences
Curated by PDSP Ki Database
The Danish University of Pharmaceutical Sciences
Curated by PDSP Ki Database
Target5-hydroxytryptamine receptor 2C(Homo sapiens (Human))
University Of Copenhagen
Curated by ChEMBL
University Of Copenhagen
Curated by ChEMBL
Affinity DataKi: 1.70nMAssay Description:Displacement of [3H]mesulergine from human 5HT2C receptor expressed in tsA201 cell membranes after 1 hr by scintillation counting analysisMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-7(Rattus norvegicus (Rat))
The Danish University of Pharmaceutical Sciences
Curated by PDSP Ki Database
The Danish University of Pharmaceutical Sciences
Curated by PDSP Ki Database
TargetNeuronal acetylcholine receptor subunit alpha-4(Rattus norvegicus (Rat))
The Danish University of Pharmaceutical Sciences
Curated by PDSP Ki Database
The Danish University of Pharmaceutical Sciences
Curated by PDSP Ki Database
Affinity DataKi: 2.10nMAssay Description:Displacement of [3H]epibatidine from rat recombinant alpha4beta2 nAChR expressed in HEK293 cellsMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-4(Rattus norvegicus (Rat))
The Danish University of Pharmaceutical Sciences
Curated by PDSP Ki Database
The Danish University of Pharmaceutical Sciences
Curated by PDSP Ki Database
Target5-hydroxytryptamine receptor 2C(Homo sapiens (Human))
University Of Copenhagen
Curated by ChEMBL
University Of Copenhagen
Curated by ChEMBL
Affinity DataKi: 2.5nMAssay Description:Antagonist activity at human 5HT2C receptor expressed in HEK293 cells assessed as inhibition of 5HT-induced intracellular calcium release measured fo...More data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 2A(Homo sapiens (Human))
University Of Copenhagen
Curated by ChEMBL
University Of Copenhagen
Curated by ChEMBL
Affinity DataKi: 2.5nMAssay Description:Antagonist activity at human 5HT2A receptor expressed in HEK293 cells assessed as inhibition of 5HT-induced intracellular calcium release measured fo...More data for this Ligand-Target Pair
TargetGamma-aminobutyric acid receptor subunit alpha-1/beta-3/gamma-2(Homo sapiens (Human))
The Danish University Of Pharmaceutical Sciences
Curated by ChEMBL
The Danish University Of Pharmaceutical Sciences
Curated by ChEMBL
Affinity DataKi: 3nMAssay Description:Binding affinity at human GABAA alpha1beta3gamma2S expressed in Xenopus oocytes by voltage-clamp electrophysiologyMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-2(Rattus norvegicus (Rat))
The Danish University of Pharmaceutical Sciences
Curated by PDSP Ki Database
The Danish University of Pharmaceutical Sciences
Curated by PDSP Ki Database
TargetNeuronal acetylcholine receptor subunit alpha-4(Rattus norvegicus (Rat))
The Danish University of Pharmaceutical Sciences
Curated by PDSP Ki Database
The Danish University of Pharmaceutical Sciences
Curated by PDSP Ki Database
Affinity DataKi: 3.80nMAssay Description:Displacement of [3H]epibatidine from rat recombinant alpha4beta2 nAChR expressed in HEK293 cellsMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-7(Rattus norvegicus (Rat))
The Danish University of Pharmaceutical Sciences
Curated by PDSP Ki Database
The Danish University of Pharmaceutical Sciences
Curated by PDSP Ki Database
TargetNeuronal acetylcholine receptor subunit alpha-2(Rattus norvegicus (Rat))
The Danish University of Pharmaceutical Sciences
Curated by PDSP Ki Database
The Danish University of Pharmaceutical Sciences
Curated by PDSP Ki Database
TargetNeuronal acetylcholine receptor subunit alpha-2(Rattus norvegicus (Rat))
The Danish University of Pharmaceutical Sciences
Curated by PDSP Ki Database
The Danish University of Pharmaceutical Sciences
Curated by PDSP Ki Database
TargetMuscarinic acetylcholine receptor M2(RAT)
The Danish University of Pharmaceutical Sciences
Curated by PDSP Ki Database
The Danish University of Pharmaceutical Sciences
Curated by PDSP Ki Database
TargetNeuronal acetylcholine receptor subunit alpha-4(Rattus norvegicus (Rat))
The Danish University of Pharmaceutical Sciences
Curated by PDSP Ki Database
The Danish University of Pharmaceutical Sciences
Curated by PDSP Ki Database
Affinity DataKi: 5.10nMAssay Description:Displacement of [3H]epibatidine from rat recombinant alpha4beta2 nAChR expressed in HEK293 cellsMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-3(Rattus norvegicus (Rat))
The Danish University of Pharmaceutical Sciences
Curated by PDSP Ki Database
The Danish University of Pharmaceutical Sciences
Curated by PDSP Ki Database
Affinity DataKi: 5.40nMAssay Description:Agonist activity at rat alpha-3-beta-4 nAChR expressed in HEK293 cells by FMP assayMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-4(Rattus norvegicus (Rat))
The Danish University of Pharmaceutical Sciences
Curated by PDSP Ki Database
The Danish University of Pharmaceutical Sciences
Curated by PDSP Ki Database
TargetNeuronal acetylcholine receptor subunit alpha-3(Rattus norvegicus (Rat))
The Danish University of Pharmaceutical Sciences
Curated by PDSP Ki Database
The Danish University of Pharmaceutical Sciences
Curated by PDSP Ki Database
Affinity DataKi: 7.70nMAssay Description:Agonist activity at rat alpha-3-beta-4 nAChR expressed in HEK293 cells by FMP assayMore data for this Ligand-Target Pair
TargetGamma-aminobutyric acid receptor subunit alpha-1/beta-3/gamma-2(Homo sapiens (Human))
The Danish University Of Pharmaceutical Sciences
Curated by ChEMBL
The Danish University Of Pharmaceutical Sciences
Curated by ChEMBL
Affinity DataKi: 8nMAssay Description:Antagonist activity at human GABAA alpha-1-beta-3-gamma-2S expressed in Xenopus oocytes by two-electrode voltage-clamp electrophysiologyMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 2C(Homo sapiens (Human))
University Of Copenhagen
Curated by ChEMBL
University Of Copenhagen
Curated by ChEMBL
Affinity DataKi: 8nMAssay Description:Antagonist activity at human 5HT2C receptor expressed in HEK293 cells assessed as inhibition of 5HT-induced intracellular calcium release measured fo...More data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 2A(Homo sapiens (Human))
University Of Copenhagen
Curated by ChEMBL
University Of Copenhagen
Curated by ChEMBL
Affinity DataKi: 8.10nMAssay Description:Antagonist activity at human 5HT2A receptor expressed in HEK293 cells assessed as inhibition of 5HT-induced intracellular calcium release measured fo...More data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-4(Rattus norvegicus (Rat))
The Danish University of Pharmaceutical Sciences
Curated by PDSP Ki Database
The Danish University of Pharmaceutical Sciences
Curated by PDSP Ki Database
TargetGamma-aminobutyric acid receptor subunit alpha-1/beta-3/gamma-2(Homo sapiens (Human))
The Danish University Of Pharmaceutical Sciences
Curated by ChEMBL
The Danish University Of Pharmaceutical Sciences
Curated by ChEMBL
Affinity DataKi: 9nMAssay Description:Antagonist activity at human GABAA alpha-1-beta-3-gamma-2S expressed in Xenopus oocytes by two-electrode voltage-clamp electrophysiologyMore data for this Ligand-Target Pair
TargetNicotinic acetylcholine receptor(RAT)
The Danish University of Pharmaceutical Sciences
Curated by PDSP Ki Database
The Danish University of Pharmaceutical Sciences
Curated by PDSP Ki Database
Target5-hydroxytryptamine receptor 2A(Homo sapiens (Human))
University Of Copenhagen
Curated by ChEMBL
University Of Copenhagen
Curated by ChEMBL
Affinity DataKi: 9.10nMAssay Description:Antagonist activity at human 5HT2A receptor expressed in HEK293 cells assessed as inhibition of 5HT-induced intracellular calcium release measured fo...More data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-2(Rattus norvegicus (Rat))
The Danish University of Pharmaceutical Sciences
Curated by PDSP Ki Database
The Danish University of Pharmaceutical Sciences
Curated by PDSP Ki Database
Target5-hydroxytryptamine receptor 2C(Homo sapiens (Human))
University Of Copenhagen
Curated by ChEMBL
University Of Copenhagen
Curated by ChEMBL
Affinity DataKi: 9.30nMAssay Description:Displacement of [3H]mesulergine from human 5HT2C receptor expressed in tsA201 cell membranes after 1 hr by scintillation counting analysisMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 2C(Homo sapiens (Human))
University Of Copenhagen
Curated by ChEMBL
University Of Copenhagen
Curated by ChEMBL
Affinity DataKi: 9.30nMAssay Description:Displacement of [3H]mesulergine from human 5HT2C receptor expressed in tsA201 cell membranes after 1 hr by scintillation counting analysisMore data for this Ligand-Target Pair
TargetGamma-aminobutyric acid receptor subunit alpha-1/beta-3/gamma-2(Homo sapiens (Human))
The Danish University Of Pharmaceutical Sciences
Curated by ChEMBL
The Danish University Of Pharmaceutical Sciences
Curated by ChEMBL
Affinity DataKi: 10nMAssay Description:Antagonist activity at human GABAA alpha-1-beta-3-gamma-2S expressed in Xenopus oocytes by two-electrode voltage-clamp electrophysiologyMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-4(Homo sapiens (Human))
Copenhagen University
Curated by ChEMBL
Copenhagen University
Curated by ChEMBL
Affinity DataKi: 13nMAssay Description:Displacement of [3H]epibatidine from alpha4beta2 nAChR (unknown origin) expressed in HEK293 cellsMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-4(Rattus norvegicus (Rat))
The Danish University of Pharmaceutical Sciences
Curated by PDSP Ki Database
The Danish University of Pharmaceutical Sciences
Curated by PDSP Ki Database
Affinity DataKi: 13nMAssay Description:Displacement of [3H]epibatidine from rat recombinant alpha4beta2 nAChR expressed in HEK293 cellsMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-4(Rattus norvegicus (Rat))
The Danish University of Pharmaceutical Sciences
Curated by PDSP Ki Database
The Danish University of Pharmaceutical Sciences
Curated by PDSP Ki Database
Affinity DataKi: 15nMAssay Description:Displacement of [3H]epibatidine from rat recombinant alpha4beta2 nAChR expressed in HEK293 cellsMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-4(Rattus norvegicus (Rat))
The Danish University of Pharmaceutical Sciences
Curated by PDSP Ki Database
The Danish University of Pharmaceutical Sciences
Curated by PDSP Ki Database
TargetGamma-aminobutyric acid receptor subunit alpha-1/beta-3/gamma-2(Homo sapiens (Human))
The Danish University Of Pharmaceutical Sciences
Curated by ChEMBL
The Danish University Of Pharmaceutical Sciences
Curated by ChEMBL
Affinity DataKi: 20nMAssay Description:Binding affinity at human GABAA alpha1beta3gamma2S expressed in Xenopus oocytes by voltage-clamp electrophysiologyMore data for this Ligand-Target Pair
TargetNicotinic acetylcholine receptor(RAT)
The Danish University of Pharmaceutical Sciences
Curated by PDSP Ki Database
The Danish University of Pharmaceutical Sciences
Curated by PDSP Ki Database
TargetNeuronal acetylcholine receptor subunit alpha-4(Rattus norvegicus (Rat))
The Danish University of Pharmaceutical Sciences
Curated by PDSP Ki Database
The Danish University of Pharmaceutical Sciences
Curated by PDSP Ki Database
Affinity DataKi: 20nMAssay Description:Displacement of [3H]epibatidine from rat recombinant alpha4beta2 nAChR expressed in HEK293 cellsMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-4(Rattus norvegicus (Rat))
The Danish University of Pharmaceutical Sciences
Curated by PDSP Ki Database
The Danish University of Pharmaceutical Sciences
Curated by PDSP Ki Database
Affinity DataKi: 22nMAssay Description:Displacement of [3H]epibatidine from rat recombinant alpha4beta2 nAChR expressed in HEK293 cellsMore data for this Ligand-Target Pair
TargetGamma-aminobutyric acid receptor subunit alpha-1/beta-3/gamma-2(Homo sapiens (Human))
The Danish University Of Pharmaceutical Sciences
Curated by ChEMBL
The Danish University Of Pharmaceutical Sciences
Curated by ChEMBL
Affinity DataKi: 22nMAssay Description:Binding affinity at human GABAA alpha1beta3gamma2S expressed in Xenopus oocytes by voltage-clamp electrophysiologyMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-3(Rattus norvegicus (Rat))
The Danish University of Pharmaceutical Sciences
Curated by PDSP Ki Database
The Danish University of Pharmaceutical Sciences
Curated by PDSP Ki Database
Affinity DataKi: 23nMAssay Description:Agonist activity at rat alpha-3-beta-4 nAChR expressed in HEK293 cells by FMP assayMore data for this Ligand-Target Pair
TargetNicotinic acetylcholine receptor(RAT)
The Danish University of Pharmaceutical Sciences
Curated by PDSP Ki Database
The Danish University of Pharmaceutical Sciences
Curated by PDSP Ki Database