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Found 246 with Last Name = 'freeman' and Initial = 'ra'
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
University of North Texas

Curated by PDSP Ki Database
LigandPNGBDBM21397(8-[4-(4-fluorophenyl)-4-keto-butyl]-1-phenyl-1,3,8...)
Affinity DataKi:  0.0100nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Rattus norvegicus (Rat))
Wake Forest University School Of Medicine

Curated by ChEMBL
LigandPNGBDBM50099807(CHEMBL54866 | N-(9-Benzyl-9-aza-bicyclo[3.3.1]non-...)
Affinity DataKi:  0.0400nMAssay Description:Binding affinity for dopamine receptor D3 expressed in Sf9 cells using [125I]-IABN the radioligand.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Rattus norvegicus (Rat))
Wake Forest University School Of Medicine

Curated by ChEMBL
LigandPNGBDBM50099821(4-Bromo-1-methoxy-naphthalene-2-carboxylic acid (9...)
Affinity DataKi:  0.0400nMAssay Description:Binding affinity for dopamine receptor D3 expressed in Sf9 cells using [125I]-IABN the radioligand.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
University of North Texas

Curated by PDSP Ki Database
LigandPNGBDBM50008735((+)-3-(tert-butyl)-(3S,4aS,13bS)-2,3,4,4a,8,9,13b,...)
Affinity DataKi:  0.0500nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
University of North Texas

Curated by PDSP Ki Database
LigandPNGBDBM50099807(CHEMBL54866 | N-(9-Benzyl-9-aza-bicyclo[3.3.1]non-...)
Affinity DataKi:  0.0500nMAssay Description:Binding affinity for dopamine receptor D2 long expressed in Sf9 cells using [125I]-IABN radioligand.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Rattus norvegicus (Rat))
Wake Forest University School Of Medicine

Curated by ChEMBL
LigandPNGBDBM50099794(4-Bromo-1-methoxy-naphthalene-2-carboxylic acid (1...)
Affinity DataKi:  0.200nMAssay Description:Binding affinity for dopamine receptor D3 expressed in Sf9 cells using [125I]-IABN the radioligand.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
University of North Texas

Curated by PDSP Ki Database
LigandPNGBDBM50099821(4-Bromo-1-methoxy-naphthalene-2-carboxylic acid (9...)
Affinity DataKi:  0.200nMAssay Description:Binding affinity for dopamine receptor D2 long expressed in Sf9 cells using [125I]-IABN radioligand.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
University of North Texas

Curated by PDSP Ki Database
LigandPNGBDBM50241107(1-(3-(4-(5-chloro-2-oxo-2,3-dihydrobenzo[d]imidazo...)
Affinity DataKi:  0.200nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
University of North Texas

Curated by PDSP Ki Database
LigandPNGBDBM78433(2-[4-[3-[2-(trifluoromethyl)-10-phenothiazinyl]pro...)
Affinity DataKi:  0.25nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
University of North Texas

Curated by PDSP Ki Database
LigandPNGBDBM79172(2-[4-[(3Z)-3-[2-(trifluoromethyl)-9-thioxanthenyli...)
Affinity DataKi:  0.25nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Rattus norvegicus (Rat))
Wake Forest University School Of Medicine

Curated by ChEMBL
LigandPNGBDBM50137621(4-Bromo-1-methoxy-naphthalene-2-carboxylic acid (1...)
Affinity DataKi:  0.400nMAssay Description:Binding affinity at dopamine receptor D3 on Sf9 cells by [125I]-IABN displacement.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Rattus norvegicus (Rat))
Wake Forest University School Of Medicine

Curated by ChEMBL
LigandPNGBDBM50099800(4-Bromo-1-methoxy-naphthalene-2-carboxylic acid (1...)
Affinity DataKi:  0.400nMAssay Description:Binding affinity for dopamine receptor D3 expressed in Sf9 cells using [125I]-IABN the radioligand.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
University of North Texas

Curated by PDSP Ki Database
LigandPNGBDBM79181(10-[3-(4-methyl-1-piperazinyl)propyl]-2-(trifluoro...)
Affinity DataKi:  0.410nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
University of North Texas

Curated by PDSP Ki Database
LigandPNGBDBM21398(4-[4-(4-Chloro-phenyl)-4-hydroxy-piperidin-1-yl]-1...)
Affinity DataKi:  0.440nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Rattus norvegicus (Rat))
Wake Forest University School Of Medicine

Curated by ChEMBL
LigandPNGBDBM50119390(Benzo[b]thiophene-2-carboxylic acid {4-[4-(2,3-dic...)
Affinity DataKi:  0.5nMAssay Description:Binding affinity at dopamine receptor D3 on Sf9 cells by [125I]-IABN displacement.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Rattus norvegicus (Rat))
Wake Forest University School Of Medicine

Curated by ChEMBL
LigandPNGBDBM50129426(CHEMBL69451 | N-(4-(4-(2,3-dichlorophenyl)piperazi...)
Affinity DataKi:  0.600nMAssay Description:Binding affinity towards rat Dopamine receptor D3 in Sf9 cells expressing in recombinant baculovirus (Bv) using [125I]-IABN as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
Wake Forest University School Of Medicine

Curated by ChEMBL
LigandPNGBDBM50099802(4-Bromo-1-methoxy-naphthalene-2-carboxylic acid (1...)
Affinity DataKi:  0.700nMAssay Description:Binding affinity for sigma-1 receptor measured on guinea pig brain membranes using [3H]-(+)-pentazocine as radioligand.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Rattus norvegicus (Rat))
Wake Forest University School Of Medicine

Curated by ChEMBL
LigandPNGBDBM50099806(4-Bromo-1-methoxy-naphthalene-2-carboxylic acid (1...)
Affinity DataKi:  0.800nMAssay Description:Binding affinity for dopamine receptor D3 expressed in Sf9 cells using [125I]-IABN the radioligand.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Rattus norvegicus (Rat))
Wake Forest University School Of Medicine

Curated by ChEMBL
LigandPNGBDBM50122056(Biphenyl-4-carboxylic acid {4-[4-(2,3-dichloro-phe...)
Affinity DataKi:  0.900nMAssay Description:Binding affinity at dopamine receptor D3 on Sf9 cells by [125I]-IABN displacement.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Rattus norvegicus (Rat))
Wake Forest University School Of Medicine

Curated by ChEMBL
LigandPNGBDBM50099817(4-Bromo-1-methoxy-naphthalene-2-carboxylic acid (1...)
Affinity DataKi:  1nMAssay Description:Binding affinity for dopamine receptor D3 expressed in Sf9 cells using [125I]-IABN the radioligand.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
Wake Forest University School Of Medicine

Curated by ChEMBL
LigandPNGBDBM50099808(4-Bromo-1-methoxy-naphthalene-2-carboxylic acid (1...)
Affinity DataKi:  1.10nMAssay Description:Binding affinity for sigma-1 receptor measured on guinea pig brain membranes using [3H]-(+)-pentazocine as radioligand.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
Wake Forest University School Of Medicine

Curated by ChEMBL
LigandPNGBDBM50099797(4-Bromo-1-methoxy-naphthalene-2-carboxylic acid (1...)
Affinity DataKi:  1.10nMAssay Description:Binding affinity for sigma-1 receptor measured on guinea pig brain membranes using [3H]-(+)-pentazocine as radioligand.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Rattus norvegicus (Rat))
Wake Forest University School Of Medicine

Curated by ChEMBL
LigandPNGBDBM50099799(4-Bromo-1-methoxy-naphthalene-2-carboxylic acid (1...)
Affinity DataKi:  1.10nMAssay Description:Binding affinity for dopamine receptor D3 expressed in Sf9 cells using [125I]-IABN the radioligand.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Rattus norvegicus (Rat))
Wake Forest University School Of Medicine

Curated by ChEMBL
LigandPNGBDBM50071959(9H-Fluorene-2-carboxylic acid {4-[4-(2,3-dichloro-...)
Affinity DataKi:  1.10nMAssay Description:Binding affinity towards rat Dopamine receptor D3 in Sf9 cells expressing in recombinant baculovirus (Bv) using [125I]-IABN as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
Wake Forest University School Of Medicine

Curated by ChEMBL
LigandPNGBDBM50099826(4-Bromo-1-methoxy-naphthalene-2-carboxylic acid (1...)
Affinity DataKi:  1.20nMAssay Description:Binding affinity for sigma-1 receptor measured on guinea pig brain membranes using [3H]-(+)-pentazocine as radioligand.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
Wake Forest University School Of Medicine

Curated by ChEMBL
LigandPNGBDBM50099820(4-Bromo-1-methoxy-naphthalene-2-carboxylic acid (1...)
Affinity DataKi:  1.20nMAssay Description:Binding affinity for sigma-1 receptor measured on guinea pig brain membranes using [3H]-(+)-pentazocine as radioligand.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
University of North Texas

Curated by PDSP Ki Database
LigandPNGBDBM50132693(4-Amino-N-(1-benzyl-piperidin-4-yl)-5-chloro-2-met...)
Affinity DataKi:  1.20nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Rattus norvegicus (Rat))
Wake Forest University School Of Medicine

Curated by ChEMBL
LigandPNGBDBM50129433(CHEMBL71327 | N-{(E)-4-[4-(2,3-Dichloro-phenyl)-pi...)
Affinity DataKi:  1.30nMAssay Description:Binding affinity towards rat Dopamine receptor D3 in Sf9 cells expressing in recombinant baculovirus (Bv) using [125I]-IABN as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Rattus norvegicus (Rat))
Wake Forest University School Of Medicine

Curated by ChEMBL
LigandPNGBDBM50129428(CHEMBL302374 | N-{4-[4-(2,3-Dichloro-phenyl)-piper...)
Affinity DataKi:  1.40nMAssay Description:Binding affinity towards rat Dopamine receptor D3 in Sf9 cells expressing in recombinant baculovirus (Bv) using [125I]-IABN as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Rattus norvegicus (Rat))
Wake Forest University School Of Medicine

Curated by ChEMBL
LigandPNGBDBM50071959(9H-Fluorene-2-carboxylic acid {4-[4-(2,3-dichloro-...)
Affinity DataKi:  1.40nMAssay Description:Binding affinity at dopamine receptor D3 on Sf9 cells by [125I]-IABN displacement.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Rattus norvegicus (Rat))
Wake Forest University School Of Medicine

Curated by ChEMBL
LigandPNGBDBM50104122(9-Oxo-9H-fluorene-4-carboxylic acid {4-[4-(2,3-dic...)
Affinity DataKi:  1.40nMAssay Description:Binding affinity at dopamine receptor D3 on Sf9 cells by [125I]-IABN displacement.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Rattus norvegicus (Rat))
Wake Forest University School Of Medicine

Curated by ChEMBL
LigandPNGBDBM50099809(4-Bromo-1-methoxy-naphthalene-2-carboxylic acid (1...)
Affinity DataKi:  1.40nMAssay Description:Binding affinity for dopamine receptor D3 expressed in Sf9 cells using [125I]-IABN the radioligand.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
Wake Forest University School Of Medicine

Curated by ChEMBL
LigandPNGBDBM21398(4-[4-(4-Chloro-phenyl)-4-hydroxy-piperidin-1-yl]-1...)
Affinity DataKi:  1.5nMAssay Description:Binding affinity for sigma-1 receptor measured on guinea pig brain membranes using [3H]-(+)-pentazocine as radioligandMore data for this Ligand-Target Pair
TargetD(3) dopamine receptor(Rattus norvegicus (Rat))
Wake Forest University School Of Medicine

Curated by ChEMBL
LigandPNGBDBM50104122(9-Oxo-9H-fluorene-4-carboxylic acid {4-[4-(2,3-dic...)
Affinity DataKi:  1.60nMAssay Description:Binding affinity towards rat Dopamine receptor D3 in Sf9 cells expressing in recombinant baculovirus (Bv) using [125I]-IABN as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Rattus norvegicus (Rat))
Wake Forest University School Of Medicine

Curated by ChEMBL
LigandPNGBDBM50099814(4-Bromo-1-methoxy-naphthalene-2-carboxylic acid ((...)
Affinity DataKi:  1.60nMAssay Description:Binding affinity for dopamine receptor D3 expressed in Sf9 cells using [125I]-IABN the radioligand.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
Wake Forest University School Of Medicine

Curated by ChEMBL
LigandPNGBDBM50099803(4-Bromo-1-methoxy-naphthalene-2-carboxylic acid (1...)
Affinity DataKi:  1.70nMAssay Description:Binding affinity for sigma-1 receptor measured on guinea pig brain membranes using [3H]-(+)-pentazocine as radioligand.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
University of North Texas

Curated by PDSP Ki Database
LigandPNGBDBM50099794(4-Bromo-1-methoxy-naphthalene-2-carboxylic acid (1...)
Affinity DataKi:  1.80nMAssay Description:Binding affinity for dopamine receptor D2 long expressed in Sf9 cells using [125I]-IABN radioligand.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Rattus norvegicus (Rat))
Wake Forest University School Of Medicine

Curated by ChEMBL
LigandPNGBDBM50129432(CHEMBL262724 | Quinoxaline-2-carboxylic acid {4-[4...)
Affinity DataKi:  1.90nMAssay Description:Binding affinity towards rat Dopamine receptor D3 in Sf9 cells expressing in recombinant baculovirus (Bv) using [125I]-IABN as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Rattus norvegicus (Rat))
Wake Forest University School Of Medicine

Curated by ChEMBL
LigandPNGBDBM50099798(4-Bromo-1-methoxy-naphthalene-2-carboxylic acid (1...)
Affinity DataKi:  1.90nMAssay Description:Binding affinity for dopamine receptor D3 expressed in Sf9 cells using [125I]-IABN the radioligand.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
Wake Forest University School Of Medicine

Curated by ChEMBL
LigandPNGBDBM50099816(4-Bromo-1-methoxy-naphthalene-2-carboxylic acid (1...)
Affinity DataKi:  1.90nMAssay Description:Binding affinity for sigma-1 receptor measured on guinea pig brain membranes using [3H]-(+)-pentazocine as radioligand.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Rattus norvegicus (Rat))
Wake Forest University School Of Medicine

Curated by ChEMBL
LigandPNGBDBM50104130(9-Oxo-9H-fluorene-4-carboxylic acid {5-[4-(2,3-dic...)
Affinity DataKi:  2nMAssay Description:Binding affinity towards rat Dopamine receptor D3 in Sf9 cells expressing in recombinant baculovirus (Bv) using [125I]-IABN as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Rattus norvegicus (Rat))
Wake Forest University School Of Medicine

Curated by ChEMBL
LigandPNGBDBM50137626(5-Bromo-N-{4-[4-(2,3-dichloro-phenyl)-piperazin-1-...)
Affinity DataKi:  2.10nMAssay Description:Binding affinity at dopamine receptor D3 on Sf9 cells by [125I]-IABN displacement.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Rattus norvegicus (Rat))
Wake Forest University School Of Medicine

Curated by ChEMBL
LigandPNGBDBM50099796(4-Bromo-1-methoxy-naphthalene-2-carboxylic acid (1...)
Affinity DataKi:  2.40nMAssay Description:Binding affinity for dopamine receptor D3 expressed in Sf9 cells using [125I]-IABN the radioligand.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
Wake Forest University School Of Medicine

Curated by ChEMBL
LigandPNGBDBM50099795(4-Bromo-1-methoxy-naphthalene-2-carboxylic acid (1...)
Affinity DataKi:  2.5nMAssay Description:Binding affinity for sigma-1 receptor measured on guinea pig brain membranes using [3H]-(+)-pentazocine as radioligand.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Rattus norvegicus (Rat))
Wake Forest University School Of Medicine

Curated by ChEMBL
LigandPNGBDBM50099812(4-Bromo-1-methoxy-naphthalene-2-carboxylic acid (1...)
Affinity DataKi:  2.5nMAssay Description:Binding affinity for dopamine receptor D3 expressed in Sf9 cells using [125I]-IABN the radioligand.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Rattus norvegicus (Rat))
Wake Forest University School Of Medicine

Curated by ChEMBL
LigandPNGBDBM50129425(5-Fluoro-1H-indole-2-carboxylic acid {4-[4-(2,3-di...)
Affinity DataKi:  2.60nMAssay Description:Binding affinity towards rat Dopamine receptor D3 in Sf9 cells expressing in recombinant baculovirus (Bv) using [125I]-IABN as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Rattus norvegicus (Rat))
Wake Forest University School Of Medicine

Curated by ChEMBL
LigandPNGBDBM50099805(4-Bromo-1-methoxy-naphthalene-2-carboxylic acid (1...)
Affinity DataKi:  2.60nMAssay Description:Binding affinity for dopamine receptor D3 expressed in Sf9 cells using [125I]-IABN the radioligand.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Rattus norvegicus (Rat))
Wake Forest University School Of Medicine

Curated by ChEMBL
LigandPNGBDBM50099803(4-Bromo-1-methoxy-naphthalene-2-carboxylic acid (1...)
Affinity DataKi:  2.90nMAssay Description:Binding affinity for dopamine receptor D3 expressed in Sf9 cells using [125I]-IABN the radioligand.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
Wake Forest University School Of Medicine

Curated by ChEMBL
LigandPNGBDBM50099817(4-Bromo-1-methoxy-naphthalene-2-carboxylic acid (1...)
Affinity DataKi:  3.20nMAssay Description:Binding affinity for sigma-1 receptor measured on guinea pig brain membranes using [3H]-(+)-pentazocine as radioligand.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Rattus norvegicus (Rat))
Wake Forest University School Of Medicine

Curated by ChEMBL
LigandPNGBDBM50099815(4-Bromo-1-methoxy-naphthalene-2-carboxylic acid ((...)
Affinity DataKi:  3.20nMAssay Description:Binding affinity for dopamine receptor D3 expressed in Sf9 cells using [125I]-IABN the radioligand.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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