Affinity DataKi: 0.800nMAssay Description:Competitive reversible inhibition of DPP4 (unknown origin)More data for this Ligand-Target Pair
Affinity DataKi: 87nMAssay Description:Displacement of 1,8-ANS from FABP4 (unknown origin) after 3 mins by fluorescence assayMore data for this Ligand-Target Pair
Target6-phosphogluconate dehydrogenase, decarboxylating(Rattus norvegicus)
Johns Hopkins University School Of Medicine
Curated by ChEMBL
Johns Hopkins University School Of Medicine
Curated by ChEMBL
Affinity DataKi: 100nMAssay Description:Inhibition of rat 6PGD assessed as inhibition constant by spectrophotometric methodMore data for this Ligand-Target Pair
Affinity DataKi: 200nMAssay Description:Displacement of 1,8-ANS from FABP4 (unknown origin) after 3 mins by fluorescence assayMore data for this Ligand-Target Pair
Affinity DataKi: 210nMAssay Description:Displacement of 1,8-ANS from FABP4 (unknown origin) after 3 mins by fluorescence assayMore data for this Ligand-Target Pair
Affinity DataKi: 230nMAssay Description:Displacement of 1,8-ANS from FABP4 (unknown origin) after 3 mins by fluorescence assayMore data for this Ligand-Target Pair
Affinity DataKi: 350nMAssay Description:Displacement of 1,8-ANS from FABP4 (unknown origin) after 3 mins by fluorescence assayMore data for this Ligand-Target Pair
Affinity DataKi: 400nMAssay Description:Displacement of 1,8-ANS from FABP4 (unknown origin) after 3 mins by fluorescence assayMore data for this Ligand-Target Pair
Affinity DataKi: 580nMAssay Description:Displacement of 1,8-ANS from FABP4 (unknown origin) after 3 mins by fluorescence assayMore data for this Ligand-Target Pair
Affinity DataKi: 590nMAssay Description:Displacement of 1,8-ANS from FABP4 (unknown origin) after 3 mins by fluorescence assayMore data for this Ligand-Target Pair
Affinity DataKi: 760nMAssay Description:Displacement of 1,8-ANS from FABP4 (unknown origin) after 3 mins by fluorescence assayMore data for this Ligand-Target Pair
Affinity DataKi: 820nMAssay Description:Displacement of 1,8-ANS from FABP4 (unknown origin) after 3 mins by fluorescence assayMore data for this Ligand-Target Pair
Affinity DataKi: 840nMAssay Description:Displacement of 1,8-ANS from FABP4 (unknown origin) after 3 mins by fluorescence assayMore data for this Ligand-Target Pair
Affinity DataKi: 910nMAssay Description:Displacement of 1,8-ANS from FABP4 (unknown origin) after 3 mins by fluorescence assayMore data for this Ligand-Target Pair
Affinity DataKi: 930nMAssay Description:Displacement of 1,8-ANS from FABP4 (unknown origin) after 3 mins by fluorescence assayMore data for this Ligand-Target Pair
Affinity DataKi: 1.15E+3nMAssay Description:Displacement of 1,8-ANS from FABP4 (unknown origin) after 3 mins by fluorescence assayMore data for this Ligand-Target Pair
Affinity DataKi: 1.16E+3nMAssay Description:Displacement of 1,8-ANS from FABP4 (unknown origin) after 3 mins by fluorescence assayMore data for this Ligand-Target Pair
Affinity DataKi: 1.19E+3nMAssay Description:Displacement of 1,8-ANS from FABP4 (unknown origin) after 3 mins by fluorescence assayMore data for this Ligand-Target Pair
Affinity DataKi: 1.28E+3nMAssay Description:Displacement of 1,8-ANS from FABP4 (unknown origin) after 3 mins by fluorescence assayMore data for this Ligand-Target Pair
Affinity DataKi: 1.66E+3nMAssay Description:Displacement of 1,8-ANS from FABP4 (unknown origin) after 3 mins by fluorescence assayMore data for this Ligand-Target Pair
Affinity DataKi: 1.67E+3nMAssay Description:Displacement of 1,8-ANS from FABP4 (unknown origin) after 3 mins by fluorescence assayMore data for this Ligand-Target Pair
Affinity DataKi: 1.85E+3nMAssay Description:Displacement of 1,8-ANS from FABP4 (unknown origin) after 3 mins by fluorescence assayMore data for this Ligand-Target Pair
Affinity DataKi: 1.95E+3nMAssay Description:Displacement of 1,8-ANS from FABP4 (unknown origin) after 3 mins by fluorescence assayMore data for this Ligand-Target Pair
Affinity DataKi: 2.12E+3nMAssay Description:Displacement of 1,8-ANS from FABP4 (unknown origin) after 3 mins by fluorescence assayMore data for this Ligand-Target Pair
Affinity DataKi: 2.16E+3nMAssay Description:Displacement of 1,8-ANS from FABP4 (unknown origin) after 3 mins by fluorescence assayMore data for this Ligand-Target Pair
Affinity DataKi: 2.55E+3nMAssay Description:Displacement of 1,8-ANS from FABP4 (unknown origin) after 3 mins by fluorescence assayMore data for this Ligand-Target Pair
Affinity DataKi: 2.69E+3nMAssay Description:Displacement of 1,8-ANS from FABP4 (unknown origin) after 3 mins by fluorescence assayMore data for this Ligand-Target Pair
Affinity DataKi: 2.76E+3nMAssay Description:Displacement of 1,8-ANS from FABP4 (unknown origin) after 3 mins by fluorescence assayMore data for this Ligand-Target Pair
Affinity DataKi: 4.32E+3nMAssay Description:Displacement of 1,8-ANS from FABP4 (unknown origin) after 3 mins by fluorescence assayMore data for this Ligand-Target Pair
Affinity DataKi: 4.84E+3nMAssay Description:Displacement of 1,8-ANS from FABP4 (unknown origin) after 3 mins by fluorescence assayMore data for this Ligand-Target Pair
TargetReplicase polyprotein 1ab(2019-nCoV)
Shanghai University Of Traditional Chinese Medicine
Curated by ChEMBL
Shanghai University Of Traditional Chinese Medicine
Curated by ChEMBL
Affinity DataKi: 6.09E+3nMAssay Description:Mixed type inhibition of SARS-CoV-2 3CL protease using Dabcyl-KNSTLQSGLRKE-Edan as substrate incubated for 30 mins and measured by Lineweaver-Burk pl...More data for this Ligand-Target Pair
Affinity DataKi: >6.14E+3nMAssay Description:Displacement of 1,8-ANS from FABP4 (unknown origin) after 3 mins by fluorescence assayMore data for this Ligand-Target Pair
Affinity DataKi: >6.14E+3nMAssay Description:Displacement of 1,8-ANS from FABP4 (unknown origin) after 3 mins by fluorescence assayMore data for this Ligand-Target Pair
Affinity DataKi: >6.14E+3nMAssay Description:Displacement of 1,8-ANS from FABP4 (unknown origin) after 3 mins by fluorescence assayMore data for this Ligand-Target Pair
Affinity DataKi: >6.14E+3nMAssay Description:Displacement of 1,8-ANS from FABP4 (unknown origin) after 3 mins by fluorescence assayMore data for this Ligand-Target Pair
Affinity DataKi: >6.14E+3nMAssay Description:Displacement of 1,8-ANS from FABP4 (unknown origin) after 3 mins by fluorescence assayMore data for this Ligand-Target Pair
Affinity DataKi: >6.14E+3nMAssay Description:Displacement of 1,8-ANS from FABP4 (unknown origin) after 3 mins by fluorescence assayMore data for this Ligand-Target Pair
Affinity DataKi: 6.51E+3nMAssay Description:Displacement of 1,8-ANS from FABP4 (unknown origin) after 3 mins by fluorescence assayMore data for this Ligand-Target Pair
Affinity DataKi: 7.38E+3nMAssay Description:Displacement of 1,8-ANS from FABP4 (unknown origin) after 3 mins by fluorescence assayMore data for this Ligand-Target Pair
TargetReplicase polyprotein 1ab(2019-nCoV)
Shanghai University Of Traditional Chinese Medicine
Curated by ChEMBL
Shanghai University Of Traditional Chinese Medicine
Curated by ChEMBL
Affinity DataKi: 7.64E+3nMAssay Description:Mixed type inhibition of SARS-CoV-2 3CL protease using Dabcyl-KNSTLQSGLRKE-Edan as substrate incubated for 30 mins and measured by Lineweaver-Burk pl...More data for this Ligand-Target Pair
Affinity DataKi: 7.75E+3nMAssay Description:Displacement of 1,8-ANS from FABP4 (unknown origin) after 3 mins by fluorescence assayMore data for this Ligand-Target Pair
Affinity DataIC50: 0.0830nMAssay Description:Inhibition of recombinant full length BTK (unknown origin) expressed in baculovirus infected Sf9 cells using Biotin-EQEDEPEGDYFEWLE-NH2 peptide as su...More data for this Ligand-Target Pair
Affinity DataIC50: 0.100nMAssay Description:Inhibition of 6-His-tagged recombinant full length BTK (unknown origin) expressed in baculovirus-transfected Sf9 cells using Biotin-EQEDEPEGDYFEWLE-N...More data for this Ligand-Target Pair
Affinity DataIC50: 0.100nMAssay Description:Inhibition of 6-His-tagged recombinant full length BTK (unknown origin) expressed in baculovirus-transfected Sf9 cells using Biotin-EQEDEPEGDYFEWLE-N...More data for this Ligand-Target Pair
Affinity DataIC50: 0.100nMAssay Description:Inhibition of 6-His-tagged recombinant full length BTK (unknown origin) expressed in baculovirus-transfected Sf9 cells using Biotin-EQEDEPEGDYFEWLE-N...More data for this Ligand-Target Pair
Affinity DataIC50: 0.100nMAssay Description:Inhibition of cathepsin S using FR-aminoluciferin as substrate preincubated for 15 mins before substrate addition measured after 1 hr by luminescence...More data for this Ligand-Target Pair
Affinity DataIC50: 0.100nMAssay Description:Inhibition of recombinant full-length His6-tagged BTK (unknown origin) expressed in baculovirus infected Sf9 cells using biotinylated A5 peptide as s...More data for this Ligand-Target Pair
Affinity DataIC50: 0.100nMAssay Description:Inhibition of human DPP4 preincubated for 30 mins followed by Gly-Pro-AMC addition measured for 50 mins by continuous fluorescence assayMore data for this Ligand-Target Pair
Affinity DataIC50: 0.100nMAssay Description:Inhibition of recombinant full length BTK (unknown origin) expressed in baculovirus infected Sf9 cells using Biotin-EQEDEPEGDYFEWLE-NH2 peptide as su...More data for this Ligand-Target Pair
Affinity DataIC50: 0.100nMAssay Description:Inhibition of recombinant full length BTK (unknown origin) expressed in baculovirus infected Sf9 cells using Biotin-EQEDEPEGDYFEWLE-NH2 peptide as su...More data for this Ligand-Target Pair