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Found 1268 with Last Name = 'gentile' and Initial = 'g'
TargetD(3) dopamine receptor(Homo sapiens (Human))
Imperial College

Curated by ChEMBL
LigandPNGBDBM50020217((4aR,10bR)-4-propyl-3,4,4a,5,6,10b-hexahydro-2H-na...)
Affinity DataKi:  0.200nMAssay Description:Agonistic activity at DRD3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Homo sapiens (Human))
Imperial College

Curated by ChEMBL
LigandPNGBDBM50312271((1S,5R)-3-(3-{[4-Methyl-5-(4-methyl-1,3-oxazol-5-y...)
Affinity DataKi:  0.501nMAssay Description:Antagonist activity at dopamine D3 receptor by GTPgammaS binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Homo sapiens (Human))
Imperial College

Curated by ChEMBL
LigandPNGBDBM50414563(CHEMBL559873)
Affinity DataKi:  0.631nMAssay Description:Binding affinity to human DRD3 receptor by GTPgammaS binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Homo sapiens (Human))
Imperial College

Curated by ChEMBL
LigandPNGBDBM50414563(CHEMBL559873)
Affinity DataKi:  0.631nMAssay Description:Antagonist activity at human D3 receptor expressed in CHO cells by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Homo sapiens (Human))
Imperial College

Curated by ChEMBL
LigandPNGBDBM50331549(CHEMBL567286 | [11C]-3-(2-oxo-3-(2-(4-(trifluorome...)
Affinity DataKi:  0.794nMAssay Description:Binding affinity to human dopamine D3 receptor by filtration binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Homo sapiens (Human))
Imperial College

Curated by ChEMBL
LigandPNGBDBM50331549(CHEMBL567286 | [11C]-3-(2-oxo-3-(2-(4-(trifluorome...)
Affinity DataKi:  0.794nMAssay Description:Antagonistic activity at human DRD3 receptor by filtration binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Rattus norvegicus (Rat))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50331549(CHEMBL567286 | [11C]-3-(2-oxo-3-(2-(4-(trifluorome...)
Affinity DataKi:  0.794nMAssay Description:Binding affinity to dopamine D3 receptor in rat native tissue by filtration binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Homo sapiens (Human))
Imperial College

Curated by ChEMBL
LigandPNGBDBM50411716(CHEMBL429132)
Affinity DataKi:  0.794nMAssay Description:Antagonist activity at human dopamine D3 receptor by cell based GTPgammaS binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Rattus norvegicus (Rat))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50331549(CHEMBL567286 | [11C]-3-(2-oxo-3-(2-(4-(trifluorome...)
Affinity DataKi:  0.794nMAssay Description:Antagonistic activity at rat DRD3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Homo sapiens (Human))
Imperial College

Curated by ChEMBL
LigandPNGBDBM50411713(CHEMBL255620)
Affinity DataKi:  1nMAssay Description:Antagonist activity at human dopamine D3 receptor by cell based GTPgammaS binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Homo sapiens (Human))
Imperial College

Curated by ChEMBL
LigandPNGBDBM50414436(CHEMBL560574)
Affinity DataKi:  1nMAssay Description:Antagonist activity at human dopamine D3 receptor expressed in CHO cells by [35S]GTP-gamma-S-based scintillation spectrometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Homo sapiens (Human))
Imperial College

Curated by ChEMBL
LigandPNGBDBM50331549(CHEMBL567286 | [11C]-3-(2-oxo-3-(2-(4-(trifluorome...)
Affinity DataKi:  1nMAssay Description:Antagonist activity at human dopamine D3 receptor expressed in CHO cells by [35S]GTP-gamma-S-based scintillation spectrometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Homo sapiens (Human))
Imperial College

Curated by ChEMBL
LigandPNGBDBM50414574(CHEMBL563580)
Affinity DataKi:  1.26nMAssay Description:Binding affinity to human DRD3 receptor by GTPgammaS binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Homo sapiens (Human))
Imperial College

Curated by ChEMBL
LigandPNGBDBM50414574(CHEMBL563580)
Affinity DataKi:  1.26nMAssay Description:Antagonist activity at human D3 receptor expressed in CHO cells by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Homo sapiens (Human))
Imperial College

Curated by ChEMBL
LigandPNGBDBM50416717(CHEMBL1224699)
Affinity DataKi:  1.26nMAssay Description:Antagonist activity at dopamine D3 receptor by GTPgammaS binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Homo sapiens (Human))
Imperial College

Curated by ChEMBL
LigandPNGBDBM50414406(CHEMBL561512)
Affinity DataKi:  1.26nMAssay Description:Antagonist activity at human dopamine D3 receptor expressed in CHO cells by [35S]GTP-gamma-S-based scintillation spectrometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Homo sapiens (Human))
Imperial College

Curated by ChEMBL
LigandPNGBDBM50414435(CHEMBL569846)
Affinity DataKi:  1.26nMAssay Description:Antagonist activity at human dopamine D3 receptor expressed in CHO cells by [35S]GTP-gamma-S-based scintillation spectrometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Homo sapiens (Human))
Imperial College

Curated by ChEMBL
LigandPNGBDBM50411402(CHEMBL244946)
Affinity DataKi:  1.58nMAssay Description:Antagonist activity at human D3 receptor expressed in CHO cells by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Homo sapiens (Human))
Imperial College

Curated by ChEMBL
LigandPNGBDBM50411402(CHEMBL244946)
Affinity DataKi:  1.58nMAssay Description:Binding affinity to human DRD3 receptor by GTPgammaS binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Homo sapiens (Human))
Imperial College

Curated by ChEMBL
LigandPNGBDBM50414578(CHEMBL558058)
Affinity DataKi:  1.58nMAssay Description:Binding affinity to human DRD3 receptor by GTPgammaS binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Homo sapiens (Human))
Imperial College

Curated by ChEMBL
LigandPNGBDBM50414578(CHEMBL558058)
Affinity DataKi:  1.58nMAssay Description:Antagonist activity at human D3 receptor expressed in CHO cells by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Homo sapiens (Human))
Imperial College

Curated by ChEMBL
LigandPNGBDBM50414409(CHEMBL565017)
Affinity DataKi:  1.58nMAssay Description:Antagonist activity at human dopamine D3 receptor expressed in CHO cells by [35S]GTP-gamma-S-based scintillation spectrometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Homo sapiens (Human))
Imperial College

Curated by ChEMBL
LigandPNGBDBM50414437(CHEMBL562624)
Affinity DataKi:  1.58nMAssay Description:Antagonist activity at human dopamine D3 receptor expressed in CHO cells by [35S]GTP-gamma-S-based scintillation spectrometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Homo sapiens (Human))
Imperial College

Curated by ChEMBL
LigandPNGBDBM50411678(CHEMBL273199)
Affinity DataKi:  1.58nMAssay Description:Antagonist activity at human dopamine D3 receptor by cell based GTPgammaS binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Homo sapiens (Human))
Imperial College

Curated by ChEMBL
LigandPNGBDBM50414413(CHEMBL556272)
Affinity DataKi:  1.58nMAssay Description:Antagonist activity at human dopamine D3 receptor expressed in CHO cells by [35S]GTP-gamma-S-based scintillation spectrometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Homo sapiens (Human))
Imperial College

Curated by ChEMBL
LigandPNGBDBM50411669(CHEMBL271631)
Affinity DataKi:  2.51nMAssay Description:Antagonist activity at human dopamine D3 receptor by cell based GTPgammaS binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Homo sapiens (Human))
Imperial College

Curated by ChEMBL
LigandPNGBDBM50414403(CHEMBL560177)
Affinity DataKi:  2.51nMAssay Description:Antagonist activity at human D3 receptor expressed in CHO cells by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Homo sapiens (Human))
Imperial College

Curated by ChEMBL
LigandPNGBDBM50414434(CHEMBL551914)
Affinity DataKi:  2.51nMAssay Description:Antagonist activity at human dopamine D3 receptor expressed in CHO cells by [35S]GTP-gamma-S-based scintillation spectrometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Homo sapiens (Human))
Imperial College

Curated by ChEMBL
LigandPNGBDBM50411672(CHEMBL256477)
Affinity DataKi:  2.51nMAssay Description:Antagonist activity at human dopamine D3 receptor by cell based GTPgammaS binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Homo sapiens (Human))
Imperial College

Curated by ChEMBL
LigandPNGBDBM50414572(CHEMBL563860)
Affinity DataKi:  2.51nMAssay Description:Binding affinity to human DRD3 receptor by GTPgammaS binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Homo sapiens (Human))
Imperial College

Curated by ChEMBL
LigandPNGBDBM50414557(CHEMBL562464)
Affinity DataKi:  2.51nMAssay Description:Binding affinity to human DRD3 receptor by GTPgammaS binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Homo sapiens (Human))
Imperial College

Curated by ChEMBL
LigandPNGBDBM50414570(CHEMBL563635)
Affinity DataKi:  2.51nMAssay Description:Antagonist activity at human D3 receptor expressed in CHO cells by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Homo sapiens (Human))
Imperial College

Curated by ChEMBL
LigandPNGBDBM50414572(CHEMBL563860)
Affinity DataKi:  2.51nMAssay Description:Antagonist activity at human D3 receptor expressed in CHO cells by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Homo sapiens (Human))
Imperial College

Curated by ChEMBL
LigandPNGBDBM50414570(CHEMBL563635)
Affinity DataKi:  2.51nMAssay Description:Binding affinity to human DRD3 receptor by GTPgammaS binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Homo sapiens (Human))
Imperial College

Curated by ChEMBL
LigandPNGBDBM50414403(CHEMBL560177)
Affinity DataKi:  2.51nMAssay Description:Binding affinity to human DRD3 receptor by GTPgammaS binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Homo sapiens (Human))
Imperial College

Curated by ChEMBL
LigandPNGBDBM50414403(CHEMBL560177)
Affinity DataKi:  2.51nMAssay Description:Antagonist activity at human dopamine D3 receptor expressed in CHO cells by [35S]GTP-gamma-S-based scintillation spectrometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Homo sapiens (Human))
Imperial College

Curated by ChEMBL
LigandPNGBDBM50414404(CHEMBL559029)
Affinity DataKi:  2.51nMAssay Description:Antagonist activity at human dopamine D3 receptor expressed in CHO cells by [35S]GTP-gamma-S-based scintillation spectrometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Homo sapiens (Human))
Imperial College

Curated by ChEMBL
LigandPNGBDBM50416713(CHEMBL1224638)
Affinity DataKi:  2.51nMAssay Description:Antagonist activity at dopamine D3 receptor by GTPgammaS binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Homo sapiens (Human))
Imperial College

Curated by ChEMBL
LigandPNGBDBM50416716(CHEMBL1224698)
Affinity DataKi:  2.51nMAssay Description:Antagonist activity at dopamine D3 receptor by GTPgammaS binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Homo sapiens (Human))
Imperial College

Curated by ChEMBL
LigandPNGBDBM50414557(CHEMBL562464)
Affinity DataKi:  2.51nMAssay Description:Antagonist activity at human D3 receptor expressed in CHO cells by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Homo sapiens (Human))
Imperial College

Curated by ChEMBL
LigandPNGBDBM50414412(CHEMBL559856)
Affinity DataKi:  2.51nMAssay Description:Antagonist activity at human dopamine D3 receptor expressed in CHO cells by [35S]GTP-gamma-S-based scintillation spectrometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Homo sapiens (Human))
Imperial College

Curated by ChEMBL
LigandPNGBDBM50411702(CHEMBL256015)
Affinity DataKi:  3.16nMAssay Description:Antagonist activity at human dopamine D3 receptor by cell based GTPgammaS binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Homo sapiens (Human))
Imperial College

Curated by ChEMBL
LigandPNGBDBM50411712(CHEMBL271083)
Affinity DataKi:  3.16nMAssay Description:Antagonist activity at human dopamine D3 receptor by cell based GTPgammaS binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Imperial College

Curated by ChEMBL
LigandPNGBDBM50414563(CHEMBL559873)
Affinity DataKi:  3.16nMAssay Description:Binding affinity to human DRD2 receptor by GTPgammaS binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Imperial College

Curated by ChEMBL
LigandPNGBDBM50414563(CHEMBL559873)
Affinity DataKi:  3.16nMAssay Description:Antagonist activity at human D2 receptor expressed in CHO cells by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Homo sapiens (Human))
Imperial College

Curated by ChEMBL
LigandPNGBDBM50414555(CHEMBL565075)
Affinity DataKi:  3.16nMAssay Description:Antagonist activity at human D3 receptor expressed in CHO cells by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Homo sapiens (Human))
Imperial College

Curated by ChEMBL
LigandPNGBDBM50414555(CHEMBL565075)
Affinity DataKi:  3.16nMAssay Description:Binding affinity to human DRD3 receptor by GTPgammaS binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Homo sapiens (Human))
Imperial College

Curated by ChEMBL
LigandPNGBDBM50414443(CHEMBL549894)
Affinity DataKi:  3.16nMAssay Description:Antagonist activity at human dopamine D3 receptor expressed in CHO cells by [35S]GTP-gamma-S-based scintillation spectrometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Homo sapiens (Human))
Imperial College

Curated by ChEMBL
LigandPNGBDBM50370572(CHEMBL85606 | SB-277011)
Affinity DataKi:  3.98nMAssay Description:Antagonist activity at human D3 receptor expressed in CHO cells by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Homo sapiens (Human))
Imperial College

Curated by ChEMBL
LigandPNGBDBM50416713(CHEMBL1224638)
Affinity DataKi:  3.98nMAssay Description:Antagonist activity at dopamine D3 receptor by GTPgammaS binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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