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Found 344 with Last Name = 'goossens' and Initial = 'jf'
TargetType-1 angiotensin II receptor(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50042235(2-butyl-3-{[2'-(1H-tetrazol-5-yl)[1,1'-biphenyl]-4...)
Affinity DataKi:  2nMAssay Description:In vitro binding affinity towards Angiotensin II receptor, type 1 of human hepatoma cell line PLC-PRF-5More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50042235(2-butyl-3-{[2'-(1H-tetrazol-5-yl)[1,1'-biphenyl]-4...)
Affinity DataKi:  2nMAssay Description:Binding affinity against AT1 in human hepatoma cell line, PLC-PRF-5More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50224081(CHEMBL235733 | N3-(1-(3,5-dimethyl)adamantyl)-7-ch...)
Affinity DataKi:  5.30nMAssay Description:Inhibition of human CB2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM21278(5-(4-chlorophenyl)-1-(2,4-dichlorophenyl)-4-methyl...)
Affinity DataKi:  5.37nMAssay Description:Displacement of [3H]SR-141716A from human CB1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMedDrugBank

TargetCannabinoid receptor 2(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50067499((6aR,10aR)-3(1,1-dimethylheptyl)-9-hydroxymethyl)-...)
Affinity DataKi:  7.30nMAssay Description:Displacement of [3H]CP-55940 from human CB2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 2(Homo sapiens (Human))
University Of Lille

Curated by ChEMBL
LigandPNGBDBM50428509(CHEMBL2331608)
Affinity DataKi:  8.90nMAssay Description:Inhibition of human carbonic anhydrase 2 preincubated for 10 mins by CO2 hydration stopped-flow assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 2(Homo sapiens (Human))
University Of Lille

Curated by ChEMBL
LigandPNGBDBM50329603(CHEMBL1270532 | N-(Piperidino-1-ethyl)-1-[4-(amino...)
Affinity DataKi:  9nMAssay Description:Inhibition of human carbonic anhydrase 2 by stopped flow CO2 hydration assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM21281((11R)-2-methyl-11-(morpholin-4-ylmethyl)-3-(naphth...)
Affinity DataKi:  9.10nMAssay Description:Displacement of [3H]CP-55940 from human CB2 receptorMore data for this Ligand-Target Pair
TargetCarbonic anhydrase 2(Homo sapiens (Human))
University Of Lille

Curated by ChEMBL
LigandPNGBDBM50428503(CHEMBL2336615)
Affinity DataKi:  9.10nMAssay Description:Inhibition of human carbonic anhydrase 2 preincubated for 10 mins by CO2 hydration stopped-flow assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 2(Homo sapiens (Human))
University Of Lille

Curated by ChEMBL
LigandPNGBDBM50428512(CHEMBL2336626)
Affinity DataKi:  9.60nMAssay Description:Inhibition of human carbonic anhydrase 2 preincubated for 10 mins by CO2 hydration stopped-flow assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50089984(4'-(3-Butyl-1,4-dioxo-2,3-diaza-spiro[4.4]non-2-yl...)
Affinity DataKi:  10nMAssay Description:Binding affinity against AT1 in human hepatoma cell line, PLC-PRF-5More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 2(Homo sapiens (Human))
University Of Lille

Curated by ChEMBL
LigandPNGBDBM50329601(4-{2-Methyl-3-[(4-methylpiperazino)carbonyl]-5-(2-...)
Affinity DataKi:  10nMAssay Description:Inhibition of human carbonic anhydrase 2 by stopped flow CO2 hydration assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 2(Homo sapiens (Human))
University Of Lille

Curated by ChEMBL
LigandPNGBDBM50329602(CHEMBL1270531 | N-[2-(Pyrrolidinyl-1-ethyl)]-1-[4-...)
Affinity DataKi:  10nMAssay Description:Inhibition of human carbonic anhydrase 2 by stopped flow CO2 hydration assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 9(Homo sapiens (Human))
University Of Lille

Curated by ChEMBL
LigandPNGBDBM50329599(CHEMBL1270341 | N-[2-(Dimethylamino)ethyl]-1-[4-(a...)
Affinity DataKi:  10nMAssay Description:Inhibition of human carbonic anhydrase 9 by stopped flow CO2 hydration assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 9(Homo sapiens (Human))
University Of Lille

Curated by ChEMBL
LigandPNGBDBM50329600(CHEMBL1270437 | N-(Dimethylaminopropyl)-1-[4-(amin...)
Affinity DataKi:  11nMAssay Description:Inhibition of human carbonic anhydrase 9 by stopped flow CO2 hydration assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 2(Homo sapiens (Human))
University Of Lille

Curated by ChEMBL
LigandPNGBDBM10880(AZA | AZA2 | AZM acetazolamide | Acerazolamide, AA...)
Affinity DataKi:  12nMAssay Description:Inhibition of human carbonic anhydrase 2 preincubated for 10 mins by CO2 hydration stopped-flow assayMore data for this Ligand-Target Pair
TargetType-1 angiotensin II receptor(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50089996(4'-(3-Butyl-1,4-dioxo-2,3-diaza-spiro[4.4]non-2-yl...)
Affinity DataKi:  13nMAssay Description:Binding affinity against AT1 in human hepatoma cell line, PLC-PRF-5More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 9(Homo sapiens (Human))
University Of Lille

Curated by ChEMBL
LigandPNGBDBM50428520(CHEMBL2336632)
Affinity DataKi:  13nMAssay Description:Inhibition of human carbonic anhydrase 9 preincubated for 10 mins by CO2 hydration stopped-flow assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50180026(CHEMBL264521 | N3-(2-adamantyl)-4-oxo-1-pentyl-1,4...)
Affinity DataKi:  13.4nMAssay Description:Displacement of [3H]CP-55940 from human CB2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50224046(((+/-)-N3-(1-(1-adamantyl)ethyl)-4-oxo-1-pentyl-1,...)
Affinity DataKi:  14nMAssay Description:Inhibition of human CB2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50119657(8-Butyl-7-[2'-(1H-tetrazol-5-yl)-biphenyl-4-ylmeth...)
Affinity DataKi:  14nMAssay Description:In vitro binding affinity towards Angiotensin II receptor, type 1 of human hepatoma cell line PLC-PRF-5More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 9(Homo sapiens (Human))
University Of Lille

Curated by ChEMBL
LigandPNGBDBM50428518(CHEMBL2336620)
Affinity DataKi:  15nMAssay Description:Inhibition of human carbonic anhydrase 9 preincubated for 10 mins by CO2 hydration stopped-flow assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50072775(2-((1R,2R,5R)-5-hydroxy-2-(3-hydroxypropyl)cyclohe...)
Affinity DataKi:  15.4nMAssay Description:Displacement of [3H]CP-55940 from human CB2 receptorMore data for this Ligand-Target Pair
TargetCannabinoid receptor 2(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50180020(4-oxo-1-pentyl-1,4-dihydro-quinoline-3-carboxylic ...)
Affinity DataKi:  15.8nMAssay Description:Displacement of [3H]CP-55940 from human CB2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 2(Homo sapiens (Human))
University Of Lille

Curated by ChEMBL
LigandPNGBDBM50329600(CHEMBL1270437 | N-(Dimethylaminopropyl)-1-[4-(amin...)
Affinity DataKi:  16nMAssay Description:Inhibition of human carbonic anhydrase 2 by stopped flow CO2 hydration assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50180040(4-Oxo-1-pentyl-1,4-dihydro-quinoline-3-carboxylic ...)
Affinity DataKi:  16.4nMAssay Description:Displacement of [3H]CP-55940 from human CB2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 9(Homo sapiens (Human))
University Of Lille

Curated by ChEMBL
LigandPNGBDBM50428512(CHEMBL2336626)
Affinity DataKi:  17nMAssay Description:Inhibition of human carbonic anhydrase 9 preincubated for 10 mins by CO2 hydration stopped-flow assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50224077(CHEMBL236361 | N3-(1-(3,5-dimethyl)adamantyl)-1-pe...)
Affinity DataKi:  18.2nMAssay Description:Inhibition of human CB2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 9(Homo sapiens (Human))
University Of Lille

Curated by ChEMBL
LigandPNGBDBM50428501(CHEMBL2336617)
Affinity DataKi:  19nMAssay Description:Inhibition of human carbonic anhydrase 9 preincubated for 10 mins by CO2 hydration stopped-flow assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 9(Homo sapiens (Human))
University Of Lille

Curated by ChEMBL
LigandPNGBDBM50428511(CHEMBL2336627)
Affinity DataKi:  19nMAssay Description:Inhibition of human carbonic anhydrase 9 preincubated for 10 mins by CO2 hydration stopped-flow assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 9(Homo sapiens (Human))
University Of Lille

Curated by ChEMBL
LigandPNGBDBM50428516(CHEMBL2336622)
Affinity DataKi:  20nMAssay Description:Inhibition of human carbonic anhydrase 9 preincubated for 10 mins by CO2 hydration stopped-flow assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50180036((6aR,10aR)-3-(1,1-dimethylbutyl)-6a,7,10,10a-tetra...)
Affinity DataKi:  20.3nMAssay Description:Displacement of [3H]CP-55940 from human CB2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 9(Homo sapiens (Human))
University Of Lille

Curated by ChEMBL
LigandPNGBDBM50428503(CHEMBL2336615)
Affinity DataKi:  21nMAssay Description:Inhibition of human carbonic anhydrase 9 preincubated for 10 mins by CO2 hydration stopped-flow assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 9(Homo sapiens (Human))
University Of Lille

Curated by ChEMBL
LigandPNGBDBM50428519(CHEMBL2336619)
Affinity DataKi:  22nMAssay Description:Inhibition of human carbonic anhydrase 9 preincubated for 10 mins by CO2 hydration stopped-flow assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 9(Homo sapiens (Human))
University Of Lille

Curated by ChEMBL
LigandPNGBDBM50329606(CHEMBL1270836 | N-(2-Morpholinoethyl)-1-[4-(aminos...)
Affinity DataKi:  22nMAssay Description:Inhibition of human carbonic anhydrase 9 by stopped flow CO2 hydration assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 9(Homo sapiens (Human))
University Of Lille

Curated by ChEMBL
LigandPNGBDBM50428521(CHEMBL2336631)
Affinity DataKi:  23nMAssay Description:Inhibition of human carbonic anhydrase 9 preincubated for 10 mins by CO2 hydration stopped-flow assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50224059(CHEMBL235040 | N3-(1-(3,5-dimethyl)adamantyl)-4-ox...)
Affinity DataKi:  23.5nMAssay Description:Inhibition of human CB2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 9(Homo sapiens (Human))
University Of Lille

Curated by ChEMBL
LigandPNGBDBM10880(AZA | AZA2 | AZM acetazolamide | Acerazolamide, AA...)
Affinity DataKi:  25nMAssay Description:Inhibition of human carbonic anhydrase 9 preincubated for 10 mins by CO2 hydration stopped-flow assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50089990(2-Butyl-3-[2'-(1H-tetrazol-5-yl)-biphenyl-4-ylmeth...)
Affinity DataKi:  25nMAssay Description:Binding affinity against AT1 in human hepatoma cell line, PLC-PRF-5More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50089987(4'-(1,4-Dioxo-3-pentyl-2,3-diaza-spiro[4.4]non-2-y...)
Affinity DataKi:  25nMAssay Description:Binding affinity against AT1 in human hepatoma cell line, PLC-PRF-5More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50089990(2-Butyl-3-[2'-(1H-tetrazol-5-yl)-biphenyl-4-ylmeth...)
Affinity DataKi:  25nMAssay Description:In vitro binding affinity towards Angiotensin II receptor, type 1 of human hepatoma cell line PLC-PRF-5More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50224052(CHEMBL393792 | adamantane-1-carboxylic Acid (4-Oxo...)
Affinity DataKi:  25.5nMAssay Description:Inhibition of human CB2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 9(Homo sapiens (Human))
University Of Lille

Curated by ChEMBL
LigandPNGBDBM50428515(CHEMBL2336623)
Affinity DataKi:  26nMAssay Description:Inhibition of human carbonic anhydrase 9 preincubated for 10 mins by CO2 hydration stopped-flow assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50224051(((+/-)-N3-(1-(1-adamantyl)ethyl)-7-chloro-4-oxo-1-...)
Affinity DataKi:  26.1nMAssay Description:Inhibition of human CB2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 9(Homo sapiens (Human))
University Of Lille

Curated by ChEMBL
LigandPNGBDBM50428522(CHEMBL2336633)
Affinity DataKi:  27nMAssay Description:Inhibition of human carbonic anhydrase 9 preincubated for 10 mins by CO2 hydration stopped-flow assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 9(Homo sapiens (Human))
University Of Lille

Curated by ChEMBL
LigandPNGBDBM50428517(CHEMBL2336621)
Affinity DataKi:  27nMAssay Description:Inhibition of human carbonic anhydrase 9 preincubated for 10 mins by CO2 hydration stopped-flow assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 9(Homo sapiens (Human))
University Of Lille

Curated by ChEMBL
LigandPNGBDBM50428509(CHEMBL2331608)
Affinity DataKi:  27nMAssay Description:Inhibition of human carbonic anhydrase 9 preincubated for 10 mins by CO2 hydration stopped-flow assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50224063(CHEMBL235946 | N3-(1-(3,5-dimethyl)adamantyl)-8-ch...)
Affinity DataKi:  27.4nMAssay Description:Inhibition of human CB2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 9(Homo sapiens (Human))
University Of Lille

Curated by ChEMBL
LigandPNGBDBM50428500(CHEMBL2336618)
Affinity DataKi:  29nMAssay Description:Inhibition of human carbonic anhydrase 9 preincubated for 10 mins by CO2 hydration stopped-flow assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 9(Homo sapiens (Human))
University Of Lille

Curated by ChEMBL
LigandPNGBDBM50428510(CHEMBL2336628)
Affinity DataKi:  30nMAssay Description:Inhibition of human carbonic anhydrase 9 preincubated for 10 mins by CO2 hydration stopped-flow assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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