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Found 1013 with Last Name = 'gordon' and Initial = 'da'
TargetApelin receptor(Homo sapiens (Human))
Bristol Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50567169(CHEMBL4873876)
Affinity DataKi:  0.0740nMAssay Description:Displacement of [3H]Apelin-13 from human APJ receptor stably expressed in human HEK293 cell membrane incubated for 120 mins by TopCount scintillation...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetApelin receptor(Homo sapiens (Human))
Bristol Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50014619(CHEMBL3184840)
Affinity DataKi:  0.170nMAssay Description:Displacement of [3H]Apelin-13 from human APJ receptor stably expressed in human HEK293 cell membrane incubated for 120 mins by TopCount scintillation...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMotilin receptor(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50143028(8'N-[1-[1-carbamoyl-3-phenyl-(1S)-propylcarbamoyl]...)
Affinity DataKi:  0.700nMAssay Description:In vitro binding affinity towards human motilin receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target11-beta-hydroxysteroid dehydrogenase 1(Homo sapiens (Human))
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50507371(BMS-823778)
Affinity DataKi:  0.900nMAssay Description:Inhibition of recombinant human 11beta-HSD1 expressed in HEK293 cell microsomes using [3H]cortisone as substrate after 4 hrs by homogeneous immuno-ra...More data for this Ligand-Target Pair
TargetMotilin receptor(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50143032(8'N-[1-(1-carbamoyl-3-phenylpropylcarbamoyl)-3-phe...)
Affinity DataKi:  1nMAssay Description:In vitro binding affinity towards human motilin receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMotilin receptor(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50143038(8'N-[1-[1-carbamoyl-3-phenyl-(1S)-propylcarbamoyl]...)
Affinity DataKi:  2nMAssay Description:In vitro binding affinity towards human motilin receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMotilin receptor(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50143039(8'N-[1-[1-carbamoyl-3-phenyl-(1R)-propylcarbamoyl]...)
Affinity DataKi:  2.70nMAssay Description:In vitro binding affinity towards human motilin receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMotilin receptor(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50143037(CHEMBL411576 | MOTILIN)
Affinity DataKi:  3.10nMAssay Description:In vitro binding affinity towards human motilin receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMotilin receptor(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50344952((2R,3S,4R,5R,8R,9S,10S,11R,12S)-5-ethyl-11-((2S,3R...)
Affinity DataKi:  3.40nMAssay Description:In vitro binding affinity towards human motilin receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target11-beta-hydroxysteroid dehydrogenase 1(Homo sapiens (Human))
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50239606(CHEMBL4080667)
Affinity DataKi:  3.80nMAssay Description:Inhibition of 11beta-HSD1 in human microsomes using [3H]cortisone as substrate preincubated for 10 mins followed by substrate addition measured after...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGrowth hormone secretagogue receptor type 1(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50371684(CHEMBL270666)
Affinity DataKi:  5.70nMAssay Description:Agonist activity at human GHS receptor expressed in H4 glioma cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGrowth hormone secretagogue receptor type 1(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50371688(CHEMBL404545)
Affinity DataKi:  7.5nMAssay Description:Agonist activity at human GHS receptor expressed in H4 glioma cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target11-beta-hydroxysteroid dehydrogenase 1(Homo sapiens (Human))
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50202086(CHEMBL219142 | N-[(E)-5-hydroxy-2-adamantyl]-2-{4-...)
Affinity DataKi:  8nMAssay Description:Inhibition of human 11beta-HSD-1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGrowth hormone secretagogue receptor type 1(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50264523((S)-N-benzyl-2-(3-chlorophenoxy)-N-((R)-pyrrolidin...)
Affinity DataKi:  30nMAssay Description:Binding affinity to GHSR (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGrowth hormone secretagogue receptor type 1(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50264552((S)-2-(3-Chloro-phenoxy)-N-(2-methyl-benzyl)-N-(R)...)
Affinity DataKi:  30nMAssay Description:Binding affinity to GHSR (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGrowth hormone secretagogue receptor type 1(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50371686(CHEMBL271876)
Affinity DataKi:  40nMAssay Description:Agonist activity at human GHS receptor expressed in H4 glioma cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGrowth hormone secretagogue receptor type 1(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50264357(2-(3-Chloro-phenoxy)-N-(2-methyl-benzyl)-N-(R)-1-p...)
Affinity DataKi:  90nMAssay Description:Binding affinity to GHSR (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGrowth hormone secretagogue receptor type 1(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50222142((S,E)-2-amino-N-(2-(benzyloxy)-1-(1-cinnamyl-1H-te...)
Affinity DataKi:  190nMAssay Description:Displacement of [125I]Ghrelin from human GHSR1a after 1 hrMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGrowth hormone secretagogue receptor type 1(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50371687(CHEMBL272085)
Affinity DataKi:  197nMAssay Description:Agonist activity at human GHS receptor expressed in H4 glioma cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGrowth hormone secretagogue receptor type 1(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50222164((S)-2-amino-N-(2-(benzyloxy)-1-(1-(3-phenylpropyl)...)
Affinity DataKi:  200nMAssay Description:Agonist activity at human GHS receptor expressed in H4 glioma cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGrowth hormone secretagogue receptor type 1(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50222164((S)-2-amino-N-(2-(benzyloxy)-1-(1-(3-phenylpropyl)...)
Affinity DataKi:  200nMAssay Description:Displacement of [125I]Ghrelin from human GHSR1a after 1 hrMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGrowth hormone secretagogue receptor type 1(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50371683(CHEMBL410060)
Affinity DataKi:  240nMAssay Description:Agonist activity at human GHS receptor expressed in H4 glioma cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGrowth hormone secretagogue receptor type 1(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50264521((S)-N-(4-acetamidophenyl)-2-(3-chlorophenoxy)-N-((...)
Affinity DataKi:  250nMAssay Description:Binding affinity to GHSR (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGrowth hormone secretagogue receptor type 1(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50264486(CHEMBL489401 | N-(4-acetamidophenyl)-2-(3-chloroph...)
Affinity DataKi:  260nMAssay Description:Binding affinity to GHSR (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGrowth hormone secretagogue receptor type 1(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50371693(CHEMBL402086)
Affinity DataKi:  298nMAssay Description:Agonist activity at human GHS receptor expressed in H4 glioma cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGrowth hormone secretagogue receptor type 1(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50264256(CHEMBL489370 | N-benzyl-2-(3-chlorophenoxy)-N-((R)...)
Affinity DataKi:  300nMAssay Description:Binding affinity to GHSR (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGrowth hormone secretagogue receptor type 1(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50222147((S)-benzyl 5-(5-(1-(2-amino-2-methylpropanamido)-2...)
Affinity DataKi:  320nMAssay Description:Displacement of [125I]Ghrelin from human GHSR1a after 1 hrMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target11-beta-hydroxysteroid dehydrogenase 1(Mus musculus (mouse))
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50507371(BMS-823778)
Affinity DataKi:  380nMAssay Description:Inhibition of recombinant mouse 11beta-HSD1 expressed in HEK293 cell microsomes using [3H]cortisone as substrate after 4 hrs by homogeneous immuno-ra...More data for this Ligand-Target Pair
TargetGrowth hormone secretagogue receptor type 1(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50222136(CHEMBL235793 | methyl 2-(5-((S)-1-(2-amino-2-methy...)
Affinity DataKi:  470nMAssay Description:Displacement of [125I]Ghrelin from human GHSR1a after 1 hrMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGrowth hormone secretagogue receptor type 1(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50371685(CHEMBL270876)
Affinity DataKi:  503nMAssay Description:Agonist activity at human GHS receptor expressed in H4 glioma cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGrowth hormone secretagogue receptor type 1(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50371691(CHEMBL270851)
Affinity DataKi:  611nMAssay Description:Agonist activity at human GHS receptor expressed in H4 glioma cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGrowth hormone secretagogue receptor type 1(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50371689(CHEMBL256235)
Affinity DataKi:  696nMAssay Description:Agonist activity at human GHS receptor expressed in H4 glioma cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGrowth hormone secretagogue receptor type 1(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50371689(CHEMBL256235)
Affinity DataKi:  696nMAssay Description:Agonist activity at human GHS receptor expressed in H4 glioma cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGrowth hormone secretagogue receptor type 1(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50371697(CHEMBL404336)
Affinity DataKi:  737nMAssay Description:Agonist activity at human GHS receptor expressed in H4 glioma cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGrowth hormone secretagogue receptor type 1(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50371697(CHEMBL404336)
Affinity DataKi:  737nMAssay Description:Agonist activity at human GHS receptor expressed in H4 glioma cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGrowth hormone secretagogue receptor type 1(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50222157(2-amino-N-{(S)-2-benzyloxy-1-[1-(2-phenethylcarbam...)
Affinity DataKi:  780nMAssay Description:Displacement of [125I]Ghrelin from human GHSR1a after 1 hrMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGrowth hormone secretagogue receptor type 1(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50222166(2-amino-N-((S)-2-benzyloxy-1-{1-[2-(3-phenyl-propy...)
Affinity DataKi:  820nMAssay Description:Displacement of [125I]Ghrelin from human GHSR1a after 1 hrMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGrowth hormone secretagogue receptor type 1(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50222162((S)-2-amino-N-(2-(benzyloxy)-1-(1-(2-(1-(methylsul...)
Affinity DataKi:  970nMAssay Description:Displacement of [125I]Ghrelin from human GHSR1a after 1 hrMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGrowth hormone secretagogue receptor type 1(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50222167(2-amino-N-{(S)-1-[1-(2-benzylcarbamoyl-ethyl)-1H-t...)
Affinity DataKi:  1.07E+3nMAssay Description:Displacement of [125I]Ghrelin from human GHSR1a after 1 hrMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGrowth hormone secretagogue receptor type 1(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50222173((S)-2-amino-N-(2-(benzyloxy)-1-(2-(2-(1-(methylsul...)
Affinity DataKi:  1.27E+3nMAssay Description:Displacement of [125I]Ghrelin from human GHSR1a after 1 hrMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGrowth hormone secretagogue receptor type 1(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50222150(2-amino-N-{(R)-1-[1-(2-butylcarbamoyl-ethyl)-1H-te...)
Affinity DataKi:  1.37E+3nMAssay Description:Displacement of [125I]Ghrelin from human GHSR1a after 1 hrMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGrowth hormone secretagogue receptor type 1(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50371695(CHEMBL403180)
Affinity DataKi:  1.38E+3nMAssay Description:Agonist activity at human GHS receptor expressed in H4 glioma cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGrowth hormone secretagogue receptor type 1(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50371695(CHEMBL403180)
Affinity DataKi:  1.38E+3nMAssay Description:Agonist activity at human GHS receptor expressed in H4 glioma cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGrowth hormone secretagogue receptor type 1(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50222151(2-amino-N-((S)-2-(benzyloxy)-1-(1-((1-(methylsulfo...)
Affinity DataKi:  1.59E+3nMAssay Description:Displacement of [125I]Ghrelin from human GHSR1a after 1 hrMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGrowth hormone secretagogue receptor type 1(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50222161((S)-2-amino-N-(2-(benzyloxy)-1-(1-(3-(2-(N-methylm...)
Affinity DataKi:  1.72E+3nMAssay Description:Displacement of [125I]Ghrelin from human GHSR1a after 1 hrMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGrowth hormone secretagogue receptor type 1(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50222146((S)-4-(5-(1-(2-amino-2-methylpropanamido)-2-(benzy...)
Affinity DataKi:  1.78E+3nMAssay Description:Displacement of [125I]Ghrelin from human GHSR1a after 1 hrMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGrowth hormone secretagogue receptor type 1(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50222153((S)-2-amino-N-(1-(1-benzyl-1H-tetrazol-5-yl)-2-(be...)
Affinity DataKi:  1.90E+3nMAssay Description:Displacement of [125I]Ghrelin from human GHSR1a after 1 hrMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGrowth hormone secretagogue receptor type 1(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50222165(2-amino-N-{(S)-2-benzyloxy-1-[1-(2-butylcarbamoyl-...)
Affinity DataKi:  2.19E+3nMAssay Description:Displacement of [125I]Ghrelin from human GHSR1a after 1 hrMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGrowth hormone secretagogue receptor type 1(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50222143((S)-N-(1-(1-(2-(methylsulfonamido)phenethyl)-1H-te...)
Affinity DataKi:  2.20E+3nMAssay Description:Displacement of [125I]Ghrelin from human GHSR1a after 1 hrMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGrowth hormone secretagogue receptor type 1(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50264524((R)-2-(3-Chloro-phenoxy)-N-(2-methyl-benzyl)-N-(R)...)
Affinity DataKi:  2.20E+3nMAssay Description:Binding affinity to GHSR (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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