TargetCoagulation factor XI(Homo sapiens (Human))
Ecole Polytechnique F�D�Rale De Lausanne (Epfl)
Curated by ChEMBL
Ecole Polytechnique F�D�Rale De Lausanne (Epfl)
Curated by ChEMBL
Affinity DataKi: 0.900nMAssay Description:Inhibition of biotinylated human FXIa assessed as inhibition of p-nitroaniline release using Pyr-Pro-Arg-pNA as substrate measured for 20 minsMore data for this Ligand-Target Pair
TargetCoagulation factor XI(Homo sapiens (Human))
Ecole Polytechnique F�D�Rale De Lausanne (Epfl)
Curated by ChEMBL
Ecole Polytechnique F�D�Rale De Lausanne (Epfl)
Curated by ChEMBL
Affinity DataKi: 2.40nMAssay Description:Inhibition of biotinylated human FXIa assessed as inhibition of p-nitroaniline release using Pyr-Pro-Arg-pNA as substrate measured for 20 minsMore data for this Ligand-Target Pair
TargetCoagulation factor XI(Homo sapiens (Human))
Ecole Polytechnique F�D�Rale De Lausanne (Epfl)
Curated by ChEMBL
Ecole Polytechnique F�D�Rale De Lausanne (Epfl)
Curated by ChEMBL
Affinity DataKi: 2.60nMAssay Description:Inhibition of biotinylated human FXIa assessed as inhibition of p-nitroaniline release using Pyr-Pro-Arg-pNA as substrate measured for 20 minsMore data for this Ligand-Target Pair
TargetCoagulation factor XI(Homo sapiens (Human))
Ecole Polytechnique F�D�Rale De Lausanne (Epfl)
Curated by ChEMBL
Ecole Polytechnique F�D�Rale De Lausanne (Epfl)
Curated by ChEMBL
Affinity DataKi: 2.80nMAssay Description:Inhibition of biotinylated human FXIa assessed as inhibition of p-nitroaniline release using Pyr-Pro-Arg-pNA as substrate measured for 20 minsMore data for this Ligand-Target Pair
TargetCoagulation factor XI(Homo sapiens (Human))
Ecole Polytechnique F�D�Rale De Lausanne (Epfl)
Curated by ChEMBL
Ecole Polytechnique F�D�Rale De Lausanne (Epfl)
Curated by ChEMBL
Affinity DataKi: 7.70nMAssay Description:Inhibition of biotinylated human FXIa assessed as inhibition of p-nitroaniline release using Pyr-Pro-Arg-pNA as substrate measured for 20 minsMore data for this Ligand-Target Pair
TargetCoagulation factor XI(Homo sapiens (Human))
Ecole Polytechnique F�D�Rale De Lausanne (Epfl)
Curated by ChEMBL
Ecole Polytechnique F�D�Rale De Lausanne (Epfl)
Curated by ChEMBL
Affinity DataKi: 31nMAssay Description:Inhibition of biotinylated human FXIa assessed as inhibition of p-nitroaniline release using Pyr-Pro-Arg-pNA as substrate measured for 20 minsMore data for this Ligand-Target Pair
TargetCoagulation factor XI(Homo sapiens (Human))
Ecole Polytechnique F�D�Rale De Lausanne (Epfl)
Curated by ChEMBL
Ecole Polytechnique F�D�Rale De Lausanne (Epfl)
Curated by ChEMBL
Affinity DataKi: 62nMAssay Description:Inhibition of biotinylated human FXIa assessed as inhibition of p-nitroaniline release using Pyr-Pro-Arg-pNA as substrate measured for 20 minsMore data for this Ligand-Target Pair
TargetCoagulation factor XI(Homo sapiens (Human))
Ecole Polytechnique F�D�Rale De Lausanne (Epfl)
Curated by ChEMBL
Ecole Polytechnique F�D�Rale De Lausanne (Epfl)
Curated by ChEMBL
Affinity DataKi: 72nMAssay Description:Inhibition of biotinylated human FXIa assessed as inhibition of p-nitroaniline release using Pyr-Pro-Arg-pNA as substrate measured for 20 minsMore data for this Ligand-Target Pair
TargetCoagulation factor XI(Homo sapiens (Human))
Ecole Polytechnique F�D�Rale De Lausanne (Epfl)
Curated by ChEMBL
Ecole Polytechnique F�D�Rale De Lausanne (Epfl)
Curated by ChEMBL
Affinity DataKi: 100nMAssay Description:Inhibition of biotinylated human FXIa assessed as inhibition of p-nitroaniline release using Pyr-Pro-Arg-pNA as substrate measured for 20 minsMore data for this Ligand-Target Pair
TargetCoagulation factor XI(Homo sapiens (Human))
Ecole Polytechnique F�D�Rale De Lausanne (Epfl)
Curated by ChEMBL
Ecole Polytechnique F�D�Rale De Lausanne (Epfl)
Curated by ChEMBL
Affinity DataKi: 260nMAssay Description:Inhibition of biotinylated human FXIa assessed as inhibition of p-nitroaniline release using Pyr-Pro-Arg-pNA as substrate measured for 20 minsMore data for this Ligand-Target Pair
TargetCoagulation factor XI(Homo sapiens (Human))
Ecole Polytechnique F�D�Rale De Lausanne (Epfl)
Curated by ChEMBL
Ecole Polytechnique F�D�Rale De Lausanne (Epfl)
Curated by ChEMBL
Affinity DataKi: 270nMAssay Description:Inhibition of biotinylated human FXIa assessed as inhibition of p-nitroaniline release using Pyr-Pro-Arg-pNA as substrate measured for 20 minsMore data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily M member 2(Homo sapiens (Human))
Queen'S Center For Biomedical Research
Curated by ChEMBL
Queen'S Center For Biomedical Research
Curated by ChEMBL
Affinity DataIC50: 25nMAssay Description:Concentration required to achieve 50% inhibition against 4-hydroxyphenylpyruvate dioxygenase from pig liver; (observed value)More data for this Ligand-Target Pair
Affinity DataIC50: 70nMAssay Description:Concentration required to achieve 50% inhibition against 4-Hydroxyphenylpyruvate dioxygenase (HPPD) from pig liver; (observed value)More data for this Ligand-Target Pair
TargetProtein-glutamine gamma-glutamyltransferase, liver(Cavia porcellus)
Institute Of Physical And Chemical Research (Riken)
Curated by ChEMBL
Institute Of Physical And Chemical Research (Riken)
Curated by ChEMBL
Affinity DataIC50: 81nMAssay Description:Inhibition of guinea pig liver transglutaminaseMore data for this Ligand-Target Pair
TargetProtein-glutamine gamma-glutamyltransferase, liver(Cavia porcellus)
Institute Of Physical And Chemical Research (Riken)
Curated by ChEMBL
Institute Of Physical And Chemical Research (Riken)
Curated by ChEMBL
Affinity DataIC50: 100nMAssay Description:Inhibition of guinea pig liver transglutaminaseMore data for this Ligand-Target Pair
TargetSolute carrier organic anion transporter family member 4C1(Homo sapiens)
Tohoku University
Curated by ChEMBL
Tohoku University
Curated by ChEMBL
Affinity DataIC50: 120nMAssay Description:TP_TRANSPORTER: inhibition of Digoxin uptake in OATP4C1-expressing MDCK cellsMore data for this Ligand-Target Pair
TargetProtein-glutamine gamma-glutamyltransferase, liver(Cavia porcellus)
Institute Of Physical And Chemical Research (Riken)
Curated by ChEMBL
Institute Of Physical And Chemical Research (Riken)
Curated by ChEMBL
Affinity DataIC50: 120nMAssay Description:Inhibition of guinea pig liver transglutaminaseMore data for this Ligand-Target Pair
TargetProtein-glutamine gamma-glutamyltransferase, liver(Cavia porcellus)
Institute Of Physical And Chemical Research (Riken)
Curated by ChEMBL
Institute Of Physical And Chemical Research (Riken)
Curated by ChEMBL
Affinity DataIC50: 190nMAssay Description:Inhibition of guinea pig liver transglutaminaseMore data for this Ligand-Target Pair
TargetProtein-glutamine gamma-glutamyltransferase, liver(Cavia porcellus)
Institute Of Physical And Chemical Research (Riken)
Curated by ChEMBL
Institute Of Physical And Chemical Research (Riken)
Curated by ChEMBL
Affinity DataIC50: 210nMAssay Description:Inhibition of guinea pig liver transglutaminaseMore data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily M member 2(Homo sapiens (Human))
Queen'S Center For Biomedical Research
Curated by ChEMBL
Queen'S Center For Biomedical Research
Curated by ChEMBL
Affinity DataIC50: 210nMAssay Description:Inhibition of human FLAG-tagged TRPM2 expressed in HEK293 cells assessed as reduction in ADPR-induced intracellular calcium flux after 30 to 60 mins ...More data for this Ligand-Target Pair
TargetProtein-glutamine gamma-glutamyltransferase, liver(Cavia porcellus)
Institute Of Physical And Chemical Research (Riken)
Curated by ChEMBL
Institute Of Physical And Chemical Research (Riken)
Curated by ChEMBL
Affinity DataIC50: 230nMAssay Description:Inhibition of guinea pig liver transglutaminaseMore data for this Ligand-Target Pair
TargetProtein-glutamine gamma-glutamyltransferase, liver(Cavia porcellus)
Institute Of Physical And Chemical Research (Riken)
Curated by ChEMBL
Institute Of Physical And Chemical Research (Riken)
Curated by ChEMBL
Affinity DataIC50: 320nMAssay Description:Inhibition of guinea pig liver transglutaminaseMore data for this Ligand-Target Pair
TargetProtein-glutamine gamma-glutamyltransferase, liver(Cavia porcellus)
Institute Of Physical And Chemical Research (Riken)
Curated by ChEMBL
Institute Of Physical And Chemical Research (Riken)
Curated by ChEMBL
Affinity DataIC50: 320nMAssay Description:Inhibition of guinea pig liver transglutaminaseMore data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily M member 2(Rattus norvegicus)
Queen'S Center For Biomedical Research
Curated by ChEMBL
Queen'S Center For Biomedical Research
Curated by ChEMBL
Affinity DataIC50: 330nMAssay Description:Inhibition of TRPM2 in rat INS-1 cells assessed as reduction in ADPR-induced intracellular calcium flux measured after 60 mins by whole cell patch cl...More data for this Ligand-Target Pair
TargetProtein-glutamine gamma-glutamyltransferase, liver(Cavia porcellus)
Institute Of Physical And Chemical Research (Riken)
Curated by ChEMBL
Institute Of Physical And Chemical Research (Riken)
Curated by ChEMBL
Affinity DataIC50: 360nMAssay Description:Inhibition of guinea pig liver transglutaminaseMore data for this Ligand-Target Pair
TargetProtein-glutamine gamma-glutamyltransferase, liver(Cavia porcellus)
Institute Of Physical And Chemical Research (Riken)
Curated by ChEMBL
Institute Of Physical And Chemical Research (Riken)
Curated by ChEMBL
Affinity DataIC50: 420nMAssay Description:Inhibition of guinea pig liver transglutaminaseMore data for this Ligand-Target Pair
TargetProtein-glutamine gamma-glutamyltransferase, liver(Cavia porcellus)
Institute Of Physical And Chemical Research (Riken)
Curated by ChEMBL
Institute Of Physical And Chemical Research (Riken)
Curated by ChEMBL
Affinity DataIC50: 420nMAssay Description:Inhibition of guinea pig liver transglutaminaseMore data for this Ligand-Target Pair
TargetProtein-glutamine gamma-glutamyltransferase, liver(Cavia porcellus)
Institute Of Physical And Chemical Research (Riken)
Curated by ChEMBL
Institute Of Physical And Chemical Research (Riken)
Curated by ChEMBL
Affinity DataIC50: 440nMAssay Description:Inhibition of guinea pig liver transglutaminaseMore data for this Ligand-Target Pair
TargetProtein-glutamine gamma-glutamyltransferase, liver(Cavia porcellus)
Institute Of Physical And Chemical Research (Riken)
Curated by ChEMBL
Institute Of Physical And Chemical Research (Riken)
Curated by ChEMBL
Affinity DataIC50: 470nMAssay Description:Inhibition of guinea pig liver transglutaminaseMore data for this Ligand-Target Pair
TargetSolute carrier organic anion transporter family member 4C1(Homo sapiens)
Tohoku University
Curated by ChEMBL
Tohoku University
Curated by ChEMBL
Affinity DataIC50: 490nMAssay Description:TP_TRANSPORTER: inhibition of Digoxin uptake in OATP4C1-expressing MDCK cellsMore data for this Ligand-Target Pair
TargetProtein-glutamine gamma-glutamyltransferase, liver(Cavia porcellus)
Institute Of Physical And Chemical Research (Riken)
Curated by ChEMBL
Institute Of Physical And Chemical Research (Riken)
Curated by ChEMBL
Affinity DataIC50: 530nMAssay Description:Inhibition of guinea pig liver transglutaminaseMore data for this Ligand-Target Pair
TargetProtein-glutamine gamma-glutamyltransferase, liver(Cavia porcellus)
Institute Of Physical And Chemical Research (Riken)
Curated by ChEMBL
Institute Of Physical And Chemical Research (Riken)
Curated by ChEMBL
Affinity DataIC50: 550nMAssay Description:Inhibition of guinea pig liver transglutaminaseMore data for this Ligand-Target Pair
TargetProtein-glutamine gamma-glutamyltransferase, liver(Cavia porcellus)
Institute Of Physical And Chemical Research (Riken)
Curated by ChEMBL
Institute Of Physical And Chemical Research (Riken)
Curated by ChEMBL
Affinity DataIC50: 570nMAssay Description:Inhibition of guinea pig liver transglutaminaseMore data for this Ligand-Target Pair
TargetProtein-glutamine gamma-glutamyltransferase, liver(Cavia porcellus)
Institute Of Physical And Chemical Research (Riken)
Curated by ChEMBL
Institute Of Physical And Chemical Research (Riken)
Curated by ChEMBL
Affinity DataIC50: 590nMAssay Description:Inhibition of guinea pig liver transglutaminaseMore data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily M member 2(Homo sapiens (Human))
Queen'S Center For Biomedical Research
Curated by ChEMBL
Queen'S Center For Biomedical Research
Curated by ChEMBL
Affinity DataIC50: 600nMAssay Description:Concentration required to achieve 50% inhibition against 4-hydroxyphenylpyruvate dioxygenase from pig liver; (observed value)More data for this Ligand-Target Pair
TargetProtein-glutamine gamma-glutamyltransferase, liver(Cavia porcellus)
Institute Of Physical And Chemical Research (Riken)
Curated by ChEMBL
Institute Of Physical And Chemical Research (Riken)
Curated by ChEMBL
Affinity DataIC50: 610nMAssay Description:Inhibition of guinea pig liver transglutaminaseMore data for this Ligand-Target Pair
TargetProtein-glutamine gamma-glutamyltransferase, liver(Cavia porcellus)
Institute Of Physical And Chemical Research (Riken)
Curated by ChEMBL
Institute Of Physical And Chemical Research (Riken)
Curated by ChEMBL
Affinity DataIC50: 650nMAssay Description:Inhibition of guinea pig liver transglutaminaseMore data for this Ligand-Target Pair
TargetProtein-glutamine gamma-glutamyltransferase, liver(Cavia porcellus)
Institute Of Physical And Chemical Research (Riken)
Curated by ChEMBL
Institute Of Physical And Chemical Research (Riken)
Curated by ChEMBL
Affinity DataIC50: 670nMAssay Description:Inhibition of guinea pig liver transglutaminaseMore data for this Ligand-Target Pair
TargetProtein-glutamine gamma-glutamyltransferase, liver(Cavia porcellus)
Institute Of Physical And Chemical Research (Riken)
Curated by ChEMBL
Institute Of Physical And Chemical Research (Riken)
Curated by ChEMBL
Affinity DataIC50: 680nMAssay Description:Inhibition of guinea pig liver transglutaminaseMore data for this Ligand-Target Pair
TargetProtein-glutamine gamma-glutamyltransferase, liver(Cavia porcellus)
Institute Of Physical And Chemical Research (Riken)
Curated by ChEMBL
Institute Of Physical And Chemical Research (Riken)
Curated by ChEMBL
Affinity DataIC50: 700nMAssay Description:Inhibition of guinea pig liver transglutaminaseMore data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily M member 7(Mus musculus)
Queen'S Center For Biomedical Research
Curated by ChEMBL
Queen'S Center For Biomedical Research
Curated by ChEMBL
Affinity DataIC50: 760nMAssay Description:Concentration required to achieve 50% inhibition against 4-Hydroxyphenylpyruvate dioxygenase (HPPD) from pig liver; (observed value)More data for this Ligand-Target Pair
TargetProtein-glutamine gamma-glutamyltransferase, liver(Cavia porcellus)
Institute Of Physical And Chemical Research (Riken)
Curated by ChEMBL
Institute Of Physical And Chemical Research (Riken)
Curated by ChEMBL
Affinity DataIC50: 770nMAssay Description:Inhibition of guinea pig liver transglutaminaseMore data for this Ligand-Target Pair
TargetProtein-glutamine gamma-glutamyltransferase, liver(Cavia porcellus)
Institute Of Physical And Chemical Research (Riken)
Curated by ChEMBL
Institute Of Physical And Chemical Research (Riken)
Curated by ChEMBL
Affinity DataIC50: 800nMAssay Description:Inhibition of guinea pig liver transglutaminaseMore data for this Ligand-Target Pair
TargetProtein-glutamine gamma-glutamyltransferase, liver(Cavia porcellus)
Institute Of Physical And Chemical Research (Riken)
Curated by ChEMBL
Institute Of Physical And Chemical Research (Riken)
Curated by ChEMBL
Affinity DataIC50: 830nMAssay Description:Inhibition of guinea pig liver transglutaminaseMore data for this Ligand-Target Pair
TargetProtein-glutamine gamma-glutamyltransferase, liver(Cavia porcellus)
Institute Of Physical And Chemical Research (Riken)
Curated by ChEMBL
Institute Of Physical And Chemical Research (Riken)
Curated by ChEMBL
Affinity DataIC50: 830nMAssay Description:Inhibition of guinea pig liver transglutaminaseMore data for this Ligand-Target Pair
TargetProtein-glutamine gamma-glutamyltransferase, liver(Cavia porcellus)
Institute Of Physical And Chemical Research (Riken)
Curated by ChEMBL
Institute Of Physical And Chemical Research (Riken)
Curated by ChEMBL
Affinity DataIC50: 840nMAssay Description:Inhibition of guinea pig liver transglutaminaseMore data for this Ligand-Target Pair
TargetProtein-glutamine gamma-glutamyltransferase, liver(Cavia porcellus)
Institute Of Physical And Chemical Research (Riken)
Curated by ChEMBL
Institute Of Physical And Chemical Research (Riken)
Curated by ChEMBL
Affinity DataIC50: 850nMAssay Description:Inhibition of guinea pig liver transglutaminaseMore data for this Ligand-Target Pair
TargetProtein-glutamine gamma-glutamyltransferase, liver(Cavia porcellus)
Institute Of Physical And Chemical Research (Riken)
Curated by ChEMBL
Institute Of Physical And Chemical Research (Riken)
Curated by ChEMBL
Affinity DataIC50: 920nMAssay Description:Inhibition of guinea pig liver transglutaminaseMore data for this Ligand-Target Pair
TargetProtein-glutamine gamma-glutamyltransferase, liver(Cavia porcellus)
Institute Of Physical And Chemical Research (Riken)
Curated by ChEMBL
Institute Of Physical And Chemical Research (Riken)
Curated by ChEMBL
Affinity DataIC50: 980nMAssay Description:Inhibition of guinea pig liver transglutaminaseMore data for this Ligand-Target Pair
TargetProtein-glutamine gamma-glutamyltransferase, liver(Cavia porcellus)
Institute Of Physical And Chemical Research (Riken)
Curated by ChEMBL
Institute Of Physical And Chemical Research (Riken)
Curated by ChEMBL
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of guinea pig liver transglutaminaseMore data for this Ligand-Target Pair