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Found 163 with Last Name = 'goto' and Initial = 'j'
TargetCoagulation factor XI(Homo sapiens (Human))
Ecole Polytechnique F�D�Rale De Lausanne (Epfl)

Curated by ChEMBL
LigandPNGBDBM50591671(CHEMBL5191603)
Affinity DataKi:  0.900nMAssay Description:Inhibition of biotinylated human FXIa assessed as inhibition of p-nitroaniline release using Pyr-Pro-Arg-pNA as substrate measured for 20 minsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetCoagulation factor XI(Homo sapiens (Human))
Ecole Polytechnique F�D�Rale De Lausanne (Epfl)

Curated by ChEMBL
LigandPNGBDBM50591673(CHEMBL5198400)
Affinity DataKi:  2.40nMAssay Description:Inhibition of biotinylated human FXIa assessed as inhibition of p-nitroaniline release using Pyr-Pro-Arg-pNA as substrate measured for 20 minsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetCoagulation factor XI(Homo sapiens (Human))
Ecole Polytechnique F�D�Rale De Lausanne (Epfl)

Curated by ChEMBL
LigandPNGBDBM50591672(CHEMBL5184798)
Affinity DataKi:  2.60nMAssay Description:Inhibition of biotinylated human FXIa assessed as inhibition of p-nitroaniline release using Pyr-Pro-Arg-pNA as substrate measured for 20 minsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetCoagulation factor XI(Homo sapiens (Human))
Ecole Polytechnique F�D�Rale De Lausanne (Epfl)

Curated by ChEMBL
LigandPNGBDBM50591674(CHEMBL5173140)
Affinity DataKi:  2.80nMAssay Description:Inhibition of biotinylated human FXIa assessed as inhibition of p-nitroaniline release using Pyr-Pro-Arg-pNA as substrate measured for 20 minsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetCoagulation factor XI(Homo sapiens (Human))
Ecole Polytechnique F�D�Rale De Lausanne (Epfl)

Curated by ChEMBL
LigandPNGBDBM50591676(CHEMBL5202369)
Affinity DataKi:  7.70nMAssay Description:Inhibition of biotinylated human FXIa assessed as inhibition of p-nitroaniline release using Pyr-Pro-Arg-pNA as substrate measured for 20 minsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetCoagulation factor XI(Homo sapiens (Human))
Ecole Polytechnique F�D�Rale De Lausanne (Epfl)

Curated by ChEMBL
LigandPNGBDBM50591678(CHEMBL5174448)
Affinity DataKi:  31nMAssay Description:Inhibition of biotinylated human FXIa assessed as inhibition of p-nitroaniline release using Pyr-Pro-Arg-pNA as substrate measured for 20 minsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetCoagulation factor XI(Homo sapiens (Human))
Ecole Polytechnique F�D�Rale De Lausanne (Epfl)

Curated by ChEMBL
LigandPNGBDBM50591681(CHEMBL5199320)
Affinity DataKi:  62nMAssay Description:Inhibition of biotinylated human FXIa assessed as inhibition of p-nitroaniline release using Pyr-Pro-Arg-pNA as substrate measured for 20 minsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetCoagulation factor XI(Homo sapiens (Human))
Ecole Polytechnique F�D�Rale De Lausanne (Epfl)

Curated by ChEMBL
LigandPNGBDBM50591677(CHEMBL5206023)
Affinity DataKi:  72nMAssay Description:Inhibition of biotinylated human FXIa assessed as inhibition of p-nitroaniline release using Pyr-Pro-Arg-pNA as substrate measured for 20 minsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetCoagulation factor XI(Homo sapiens (Human))
Ecole Polytechnique F�D�Rale De Lausanne (Epfl)

Curated by ChEMBL
LigandPNGBDBM50591679(CHEMBL5192767)
Affinity DataKi:  100nMAssay Description:Inhibition of biotinylated human FXIa assessed as inhibition of p-nitroaniline release using Pyr-Pro-Arg-pNA as substrate measured for 20 minsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetCoagulation factor XI(Homo sapiens (Human))
Ecole Polytechnique F�D�Rale De Lausanne (Epfl)

Curated by ChEMBL
LigandPNGBDBM50591680(CHEMBL5198001)
Affinity DataKi:  260nMAssay Description:Inhibition of biotinylated human FXIa assessed as inhibition of p-nitroaniline release using Pyr-Pro-Arg-pNA as substrate measured for 20 minsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetCoagulation factor XI(Homo sapiens (Human))
Ecole Polytechnique F�D�Rale De Lausanne (Epfl)

Curated by ChEMBL
LigandPNGBDBM50591675(CHEMBL5185899)
Affinity DataKi:  270nMAssay Description:Inhibition of biotinylated human FXIa assessed as inhibition of p-nitroaniline release using Pyr-Pro-Arg-pNA as substrate measured for 20 minsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetTransient receptor potential cation channel subfamily M member 2(Homo sapiens (Human))
Queen'S Center For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM27497(2-(dimethylamino)-N-(6-oxo-5,6-dihydrophenanthridi...)
Affinity DataIC50:  25nMAssay Description:Concentration required to achieve 50% inhibition against 4-hydroxyphenylpyruvate dioxygenase from pig liver; (observed value)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhospholipase A2(Apis mellifera)
Queen'S Center For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50242184(Scalaradial)
Affinity DataIC50:  70nMAssay Description:Concentration required to achieve 50% inhibition against 4-Hydroxyphenylpyruvate dioxygenase (HPPD) from pig liver; (observed value)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein-glutamine gamma-glutamyltransferase, liver(Cavia porcellus)
Institute Of Physical And Chemical Research (Riken)

Curated by ChEMBL
LigandPNGBDBM50481688(CHEMBL598522)
Affinity DataIC50:  81nMAssay Description:Inhibition of guinea pig liver transglutaminaseMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtein-glutamine gamma-glutamyltransferase, liver(Cavia porcellus)
Institute Of Physical And Chemical Research (Riken)

Curated by ChEMBL
LigandPNGBDBM50481690(CHEMBL597916)
Affinity DataIC50:  100nMAssay Description:Inhibition of guinea pig liver transglutaminaseMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSolute carrier organic anion transporter family member 4C1(Homo sapiens)
Tohoku University

Curated by ChEMBL
LigandPNGBDBM46356(DIGITOXIN | MLS000069787 | SMR000058529 | US106680...)
Affinity DataIC50:  120nMAssay Description:TP_TRANSPORTER: inhibition of Digoxin uptake in OATP4C1-expressing MDCK cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein-glutamine gamma-glutamyltransferase, liver(Cavia porcellus)
Institute Of Physical And Chemical Research (Riken)

Curated by ChEMBL
LigandPNGBDBM50481676(CHEMBL610215)
Affinity DataIC50:  120nMAssay Description:Inhibition of guinea pig liver transglutaminaseMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtein-glutamine gamma-glutamyltransferase, liver(Cavia porcellus)
Institute Of Physical And Chemical Research (Riken)

Curated by ChEMBL
LigandPNGBDBM50481720(CHEMBL598521)
Affinity DataIC50:  190nMAssay Description:Inhibition of guinea pig liver transglutaminaseMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtein-glutamine gamma-glutamyltransferase, liver(Cavia porcellus)
Institute Of Physical And Chemical Research (Riken)

Curated by ChEMBL
LigandPNGBDBM50481700(CHEMBL598529)
Affinity DataIC50:  210nMAssay Description:Inhibition of guinea pig liver transglutaminaseMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily M member 2(Homo sapiens (Human))
Queen'S Center For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50242184(Scalaradial)
Affinity DataIC50:  210nMAssay Description:Inhibition of human FLAG-tagged TRPM2 expressed in HEK293 cells assessed as reduction in ADPR-induced intracellular calcium flux after 30 to 60 mins ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein-glutamine gamma-glutamyltransferase, liver(Cavia porcellus)
Institute Of Physical And Chemical Research (Riken)

Curated by ChEMBL
LigandPNGBDBM50481721(CHEMBL611979)
Affinity DataIC50:  230nMAssay Description:Inhibition of guinea pig liver transglutaminaseMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtein-glutamine gamma-glutamyltransferase, liver(Cavia porcellus)
Institute Of Physical And Chemical Research (Riken)

Curated by ChEMBL
LigandPNGBDBM50481737(CHEMBL597079)
Affinity DataIC50:  320nMAssay Description:Inhibition of guinea pig liver transglutaminaseMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtein-glutamine gamma-glutamyltransferase, liver(Cavia porcellus)
Institute Of Physical And Chemical Research (Riken)

Curated by ChEMBL
LigandPNGBDBM50481678(CHEMBL597103)
Affinity DataIC50:  320nMAssay Description:Inhibition of guinea pig liver transglutaminaseMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily M member 2(Rattus norvegicus)
Queen'S Center For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50242184(Scalaradial)
Affinity DataIC50:  330nMAssay Description:Inhibition of TRPM2 in rat INS-1 cells assessed as reduction in ADPR-induced intracellular calcium flux measured after 60 mins by whole cell patch cl...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein-glutamine gamma-glutamyltransferase, liver(Cavia porcellus)
Institute Of Physical And Chemical Research (Riken)

Curated by ChEMBL
LigandPNGBDBM50481748(CHEMBL589994)
Affinity DataIC50:  360nMAssay Description:Inhibition of guinea pig liver transglutaminaseMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtein-glutamine gamma-glutamyltransferase, liver(Cavia porcellus)
Institute Of Physical And Chemical Research (Riken)

Curated by ChEMBL
LigandPNGBDBM50481682(CHEMBL598319)
Affinity DataIC50:  420nMAssay Description:Inhibition of guinea pig liver transglutaminaseMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtein-glutamine gamma-glutamyltransferase, liver(Cavia porcellus)
Institute Of Physical And Chemical Research (Riken)

Curated by ChEMBL
LigandPNGBDBM50481691(CHEMBL597917)
Affinity DataIC50:  420nMAssay Description:Inhibition of guinea pig liver transglutaminaseMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtein-glutamine gamma-glutamyltransferase, liver(Cavia porcellus)
Institute Of Physical And Chemical Research (Riken)

Curated by ChEMBL
LigandPNGBDBM50481767(CHEMBL599534)
Affinity DataIC50:  440nMAssay Description:Inhibition of guinea pig liver transglutaminaseMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtein-glutamine gamma-glutamyltransferase, liver(Cavia porcellus)
Institute Of Physical And Chemical Research (Riken)

Curated by ChEMBL
LigandPNGBDBM50481730(CHEMBL599729)
Affinity DataIC50:  470nMAssay Description:Inhibition of guinea pig liver transglutaminaseMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSolute carrier organic anion transporter family member 4C1(Homo sapiens)
Tohoku University

Curated by ChEMBL
LigandPNGBDBM225707(CS337 | Digoxigenin)
Affinity DataIC50:  490nMAssay Description:TP_TRANSPORTER: inhibition of Digoxin uptake in OATP4C1-expressing MDCK cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein-glutamine gamma-glutamyltransferase, liver(Cavia porcellus)
Institute Of Physical And Chemical Research (Riken)

Curated by ChEMBL
LigandPNGBDBM50481666(CHEMBL599107)
Affinity DataIC50:  530nMAssay Description:Inhibition of guinea pig liver transglutaminaseMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtein-glutamine gamma-glutamyltransferase, liver(Cavia porcellus)
Institute Of Physical And Chemical Research (Riken)

Curated by ChEMBL
LigandPNGBDBM50481675(CHEMBL582295)
Affinity DataIC50:  550nMAssay Description:Inhibition of guinea pig liver transglutaminaseMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtein-glutamine gamma-glutamyltransferase, liver(Cavia porcellus)
Institute Of Physical And Chemical Research (Riken)

Curated by ChEMBL
LigandPNGBDBM50481734(CHEMBL608737)
Affinity DataIC50:  570nMAssay Description:Inhibition of guinea pig liver transglutaminaseMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtein-glutamine gamma-glutamyltransferase, liver(Cavia porcellus)
Institute Of Physical And Chemical Research (Riken)

Curated by ChEMBL
LigandPNGBDBM50481771(4-(3-(Benzyl(Isopropyl)Amino)Propanoyl)Benzonitril...)
Affinity DataIC50:  590nMAssay Description:Inhibition of guinea pig liver transglutaminaseMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily M member 2(Homo sapiens (Human))
Queen'S Center For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM27502(3,4-dihydro-5-(4-(1-piperidinyl)butoxy)-1(2H)-isoq...)
Affinity DataIC50:  600nMAssay Description:Concentration required to achieve 50% inhibition against 4-hydroxyphenylpyruvate dioxygenase from pig liver; (observed value)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein-glutamine gamma-glutamyltransferase, liver(Cavia porcellus)
Institute Of Physical And Chemical Research (Riken)

Curated by ChEMBL
LigandPNGBDBM50481752(CHEMBL611978)
Affinity DataIC50:  610nMAssay Description:Inhibition of guinea pig liver transglutaminaseMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtein-glutamine gamma-glutamyltransferase, liver(Cavia porcellus)
Institute Of Physical And Chemical Research (Riken)

Curated by ChEMBL
LigandPNGBDBM50481674(CHEMBL590246)
Affinity DataIC50:  650nMAssay Description:Inhibition of guinea pig liver transglutaminaseMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtein-glutamine gamma-glutamyltransferase, liver(Cavia porcellus)
Institute Of Physical And Chemical Research (Riken)

Curated by ChEMBL
LigandPNGBDBM50481713(CHEMBL598910)
Affinity DataIC50:  670nMAssay Description:Inhibition of guinea pig liver transglutaminaseMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtein-glutamine gamma-glutamyltransferase, liver(Cavia porcellus)
Institute Of Physical And Chemical Research (Riken)

Curated by ChEMBL
LigandPNGBDBM50481770(CHEMBL599350)
Affinity DataIC50:  680nMAssay Description:Inhibition of guinea pig liver transglutaminaseMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtein-glutamine gamma-glutamyltransferase, liver(Cavia porcellus)
Institute Of Physical And Chemical Research (Riken)

Curated by ChEMBL
LigandPNGBDBM50481741(CHEMBL609903)
Affinity DataIC50:  700nMAssay Description:Inhibition of guinea pig liver transglutaminaseMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily M member 7(Mus musculus)
Queen'S Center For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50242184(Scalaradial)
Affinity DataIC50:  760nMAssay Description:Concentration required to achieve 50% inhibition against 4-Hydroxyphenylpyruvate dioxygenase (HPPD) from pig liver; (observed value)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein-glutamine gamma-glutamyltransferase, liver(Cavia porcellus)
Institute Of Physical And Chemical Research (Riken)

Curated by ChEMBL
LigandPNGBDBM50481699(CHEMBL602665)
Affinity DataIC50:  770nMAssay Description:Inhibition of guinea pig liver transglutaminaseMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtein-glutamine gamma-glutamyltransferase, liver(Cavia porcellus)
Institute Of Physical And Chemical Research (Riken)

Curated by ChEMBL
LigandPNGBDBM50481745(CHEMBL590249)
Affinity DataIC50:  800nMAssay Description:Inhibition of guinea pig liver transglutaminaseMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtein-glutamine gamma-glutamyltransferase, liver(Cavia porcellus)
Institute Of Physical And Chemical Research (Riken)

Curated by ChEMBL
LigandPNGBDBM50481655(CHEMBL599730)
Affinity DataIC50:  830nMAssay Description:Inhibition of guinea pig liver transglutaminaseMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtein-glutamine gamma-glutamyltransferase, liver(Cavia porcellus)
Institute Of Physical And Chemical Research (Riken)

Curated by ChEMBL
LigandPNGBDBM50481649(CHEMBL600082)
Affinity DataIC50:  830nMAssay Description:Inhibition of guinea pig liver transglutaminaseMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtein-glutamine gamma-glutamyltransferase, liver(Cavia porcellus)
Institute Of Physical And Chemical Research (Riken)

Curated by ChEMBL
LigandPNGBDBM50481677(CHEMBL598051)
Affinity DataIC50:  840nMAssay Description:Inhibition of guinea pig liver transglutaminaseMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtein-glutamine gamma-glutamyltransferase, liver(Cavia porcellus)
Institute Of Physical And Chemical Research (Riken)

Curated by ChEMBL
LigandPNGBDBM50481727(CHEMBL611080)
Affinity DataIC50:  850nMAssay Description:Inhibition of guinea pig liver transglutaminaseMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtein-glutamine gamma-glutamyltransferase, liver(Cavia porcellus)
Institute Of Physical And Chemical Research (Riken)

Curated by ChEMBL
LigandPNGBDBM50481671(CHEMBL590493)
Affinity DataIC50:  920nMAssay Description:Inhibition of guinea pig liver transglutaminaseMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtein-glutamine gamma-glutamyltransferase, liver(Cavia porcellus)
Institute Of Physical And Chemical Research (Riken)

Curated by ChEMBL
LigandPNGBDBM50481715(CHEMBL602862)
Affinity DataIC50:  980nMAssay Description:Inhibition of guinea pig liver transglutaminaseMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtein-glutamine gamma-glutamyltransferase, liver(Cavia porcellus)
Institute Of Physical And Chemical Research (Riken)

Curated by ChEMBL
LigandPNGBDBM50481661(CHEMBL598239)
Affinity DataIC50:  1.00E+3nMAssay Description:Inhibition of guinea pig liver transglutaminaseMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
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