TargetMuscarinic acetylcholine receptor M2(Homo sapiens (Human))
Schering-Plough Research Institute
Curated by ChEMBL
Schering-Plough Research Institute
Curated by ChEMBL
Affinity DataKi: 0.0100nMAssay Description:Antagonistic activity of the compound against Muscarinic acetylcholine receptor M2More data for this Ligand-Target Pair
Affinity DataKi: 0.0650nMAssay Description:Binding affinity towards Muscarinic acetylcholine receptor M2More data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M2(Homo sapiens (Human))
Schering-Plough Research Institute
Curated by ChEMBL
Schering-Plough Research Institute
Curated by ChEMBL
Affinity DataKi: 0.140nMAssay Description:Antagonistic activity of the compound against muscarinic acetylcholine receptor M2More data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M2(Homo sapiens (Human))
Schering-Plough Research Institute
Curated by ChEMBL
Schering-Plough Research Institute
Curated by ChEMBL
Affinity DataKi: 0.200nMAssay Description:Antagonistic activity of the compound against muscarinic acetylcholine receptor M2More data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M2(Homo sapiens (Human))
Schering-Plough Research Institute
Curated by ChEMBL
Schering-Plough Research Institute
Curated by ChEMBL
Affinity DataKi: 0.230nMAssay Description:Antagonistic activity of the compound against Muscarinic acetylcholine receptor M2More data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M2(Homo sapiens (Human))
Schering-Plough Research Institute
Curated by ChEMBL
Schering-Plough Research Institute
Curated by ChEMBL
Affinity DataKi: 0.290nMAssay Description:Antagonistic activity of the compound against Muscarinic acetylcholine receptor M2More data for this Ligand-Target Pair
Affinity DataKi: 0.390nMAssay Description:Binding affinity towards Muscarinic acetylcholine receptor M2More data for this Ligand-Target Pair
Affinity DataKi: 0.400nMAssay Description:Binding affinity towards Muscarinic acetylcholine receptor M2More data for this Ligand-Target Pair
Affinity DataKi: 0.440nMAssay Description:Binding affinity towards Muscarinic acetylcholine receptor M2More data for this Ligand-Target Pair
Affinity DataKi: 0.510nMAssay Description:Binding affinity towards Muscarinic acetylcholine receptor M2More data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M2(Homo sapiens (Human))
Schering-Plough Research Institute
Curated by ChEMBL
Schering-Plough Research Institute
Curated by ChEMBL
Affinity DataKi: 0.510nMAssay Description:Antagonistic activity of the compound against muscarinic acetylcholine receptor M2More data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M2(Homo sapiens (Human))
Schering-Plough Research Institute
Curated by ChEMBL
Schering-Plough Research Institute
Curated by ChEMBL
Affinity DataKi: 0.510nMAssay Description:Binding affinity for human Muscarinic acetylcholine receptor M2More data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M2(Homo sapiens (Human))
Schering-Plough Research Institute
Curated by ChEMBL
Schering-Plough Research Institute
Curated by ChEMBL
Affinity DataKi: 0.510nMAssay Description:Antagonistic activity of the compound against muscarinic acetylcholine receptor M2More data for this Ligand-Target Pair
Affinity DataKi: 0.530nMAssay Description:Binding affinity towards Muscarinic acetylcholine receptor M2More data for this Ligand-Target Pair
Affinity DataKi: 0.530nMAssay Description:Binding affinity towards Muscarinic acetylcholine receptor M2More data for this Ligand-Target Pair
Affinity DataKi: 0.540nMAssay Description:Binding affinity towards Muscarinic acetylcholine receptor M2More data for this Ligand-Target Pair
Affinity DataKi: 0.680nMAssay Description:Binding affinity towards Muscarinic acetylcholine receptor M2More data for this Ligand-Target Pair
Affinity DataKi: 0.700nMAssay Description:Inhibition of recombinant human BACE1 expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 0.700nMAssay Description:Inhibition of recombinant human BACE1 expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 0.720nMAssay Description:Binding affinity towards Muscarinic acetylcholine receptor M2More data for this Ligand-Target Pair
Affinity DataKi: 0.780nMAssay Description:Binding affinity towards Muscarinic acetylcholine receptor M2More data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M2(Homo sapiens (Human))
Schering-Plough Research Institute
Curated by ChEMBL
Schering-Plough Research Institute
Curated by ChEMBL
Affinity DataKi: 0.810nMAssay Description:Antagonistic activity of the compound against muscarinic acetylcholine receptor M2More data for this Ligand-Target Pair
Affinity DataKi: 0.860nMAssay Description:Binding affinity towards Muscarinic acetylcholine receptor M2More data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M2(Homo sapiens (Human))
Schering-Plough Research Institute
Curated by ChEMBL
Schering-Plough Research Institute
Curated by ChEMBL
Affinity DataKi: 0.890nMAssay Description:Binding affinity for human Muscarinic acetylcholine receptor M2More data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M2(Homo sapiens (Human))
Schering-Plough Research Institute
Curated by ChEMBL
Schering-Plough Research Institute
Curated by ChEMBL
Affinity DataKi: 0.900nMAssay Description:Binding affinity for human Muscarinic acetylcholine receptor M2More data for this Ligand-Target Pair
Affinity DataKi: 0.900nMAssay Description:Binding affinity towards Muscarinic acetylcholine receptor M2More data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M2(Homo sapiens (Human))
Schering-Plough Research Institute
Curated by ChEMBL
Schering-Plough Research Institute
Curated by ChEMBL
Affinity DataKi: 0.990nMAssay Description:Antagonistic activity of the compound against Muscarinic acetylcholine receptor M2More data for this Ligand-Target Pair
Affinity DataKi: 1nMAssay Description:Inhibition of recombinant human BACE1 expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 1nMAssay Description:Inhibition of recombinant human BACE1 expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 1nMAssay Description:Inhibition of recombinant human BACE1 expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 1nMAssay Description:Inhibition of recombinant human BACE1 expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 1nMAssay Description:Inhibition of recombinant human BACE1 expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 1nMAssay Description:Binding affinity towards Muscarinic acetylcholine receptor M2More data for this Ligand-Target Pair
Affinity DataKi: 1nMAssay Description:Inhibition of recombinant human BACE1 expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 1nMAssay Description:Inhibition of recombinant human BACE1 expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 1nMAssay Description:Inhibition of recombinant human BACE1 expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 1.10nMAssay Description:Binding affinity towards Muscarinic acetylcholine receptor M2More data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M2(Homo sapiens (Human))
Schering-Plough Research Institute
Curated by ChEMBL
Schering-Plough Research Institute
Curated by ChEMBL
Affinity DataKi: 1.20nMAssay Description:Antagonistic activity of the compound against muscarinic acetylcholine receptor M2More data for this Ligand-Target Pair
Affinity DataKi: 1.20nMAssay Description:Binding affinity towards Muscarinic acetylcholine receptor M2More data for this Ligand-Target Pair
Affinity DataKi: 1.40nMAssay Description:Binding affinity towards Muscarinic acetylcholine receptor M2More data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M2(Homo sapiens (Human))
Schering-Plough Research Institute
Curated by ChEMBL
Schering-Plough Research Institute
Curated by ChEMBL
Affinity DataKi: 1.40nMAssay Description:Antagonistic activity of the compound against muscarinic acetylcholine receptor M2More data for this Ligand-Target Pair
Affinity DataKi: 1.40nMAssay Description:Inhibition of recombinant human BACE1 preincubated for 30 mins followed QSY7EISEVNLDAEFC-Eu-amide substrate addition measured after 90 mins by FRET a...More data for this Ligand-Target Pair
Affinity DataKi: 1.5nMAssay Description:Binding affinity towards Muscarinic acetylcholine receptor M2More data for this Ligand-Target Pair
Affinity DataKi: 1.60nMAssay Description:Binding affinity towards Muscarinic acetylcholine receptor M2More data for this Ligand-Target Pair
Affinity DataKi: 1.80nMAssay Description:Binding affinity towards Muscarinic acetylcholine receptor M2More data for this Ligand-Target Pair
Affinity DataKi: 2nMAssay Description:Inhibition of recombinant human BACE1 expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 2.30nMAssay Description:Binding affinity towards Muscarinic acetylcholine receptor M2More data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M2(Homo sapiens (Human))
Schering-Plough Research Institute
Curated by ChEMBL
Schering-Plough Research Institute
Curated by ChEMBL
Affinity DataKi: 2.40nMAssay Description:Binding affinity for human Muscarinic acetylcholine receptor M2More data for this Ligand-Target Pair
Affinity DataKi: 2.5nMAssay Description:Binding affinity towards Muscarinic acetylcholine receptor M2More data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M2(Homo sapiens (Human))
Schering-Plough Research Institute
Curated by ChEMBL
Schering-Plough Research Institute
Curated by ChEMBL
Affinity DataKi: 2.70nMAssay Description:Binding affinity for human Muscarinic acetylcholine receptor M2More data for this Ligand-Target Pair