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Found 265 with Last Name = 'hénichart' and Initial = 'jp'
TargetType-1 angiotensin II receptor(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50042235(2-butyl-3-{[2'-(1H-tetrazol-5-yl)[1,1'-biphenyl]-4...)
Affinity DataKi:  2nMAssay Description:Binding affinity against AT1 in human hepatoma cell line, PLC-PRF-5More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50042235(2-butyl-3-{[2'-(1H-tetrazol-5-yl)[1,1'-biphenyl]-4...)
Affinity DataKi:  2nMAssay Description:In vitro binding affinity towards Angiotensin II receptor, type 1 of human hepatoma cell line PLC-PRF-5More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50224081(CHEMBL235733 | N3-(1-(3,5-dimethyl)adamantyl)-7-ch...)
Affinity DataKi:  5.30nMAssay Description:Inhibition of human CB2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM21278(5-(4-chlorophenyl)-1-(2,4-dichlorophenyl)-4-methyl...)
Affinity DataKi:  5.37nMAssay Description:Displacement of [3H]SR-141716A from human CB1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMedDrugBank

TargetCannabinoid receptor 2(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50067499((6aR,10aR)-3(1,1-dimethylheptyl)-9-hydroxymethyl)-...)
Affinity DataKi:  7.30nMAssay Description:Displacement of [3H]CP-55940 from human CB2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM21281((11R)-2-methyl-11-(morpholin-4-ylmethyl)-3-(naphth...)
Affinity DataKi:  9.10nMAssay Description:Displacement of [3H]CP-55940 from human CB2 receptorMore data for this Ligand-Target Pair
TargetType-1 angiotensin II receptor(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50089984(4'-(3-Butyl-1,4-dioxo-2,3-diaza-spiro[4.4]non-2-yl...)
Affinity DataKi:  10nMAssay Description:Binding affinity against AT1 in human hepatoma cell line, PLC-PRF-5More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50089996(4'-(3-Butyl-1,4-dioxo-2,3-diaza-spiro[4.4]non-2-yl...)
Affinity DataKi:  13nMAssay Description:Binding affinity against AT1 in human hepatoma cell line, PLC-PRF-5More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50180026(CHEMBL264521 | N3-(2-adamantyl)-4-oxo-1-pentyl-1,4...)
Affinity DataKi:  13.4nMAssay Description:Displacement of [3H]CP-55940 from human CB2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50119657(8-Butyl-7-[2'-(1H-tetrazol-5-yl)-biphenyl-4-ylmeth...)
Affinity DataKi:  14nMAssay Description:In vitro binding affinity towards Angiotensin II receptor, type 1 of human hepatoma cell line PLC-PRF-5More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50224046(((+/-)-N3-(1-(1-adamantyl)ethyl)-4-oxo-1-pentyl-1,...)
Affinity DataKi:  14nMAssay Description:Inhibition of human CB2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50072775(2-((1R,2R,5R)-5-hydroxy-2-(3-hydroxypropyl)cyclohe...)
Affinity DataKi:  15.4nMAssay Description:Displacement of [3H]CP-55940 from human CB2 receptorMore data for this Ligand-Target Pair
TargetCannabinoid receptor 2(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50180020(4-oxo-1-pentyl-1,4-dihydro-quinoline-3-carboxylic ...)
Affinity DataKi:  15.8nMAssay Description:Displacement of [3H]CP-55940 from human CB2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50180040(4-Oxo-1-pentyl-1,4-dihydro-quinoline-3-carboxylic ...)
Affinity DataKi:  16.4nMAssay Description:Displacement of [3H]CP-55940 from human CB2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50224077(CHEMBL236361 | N3-(1-(3,5-dimethyl)adamantyl)-1-pe...)
Affinity DataKi:  18.2nMAssay Description:Inhibition of human CB2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50180036((6aR,10aR)-3-(1,1-dimethylbutyl)-6a,7,10,10a-tetra...)
Affinity DataKi:  20.3nMAssay Description:Displacement of [3H]CP-55940 from human CB2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50224059(CHEMBL235040 | N3-(1-(3,5-dimethyl)adamantyl)-4-ox...)
Affinity DataKi:  23.5nMAssay Description:Inhibition of human CB2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50089987(4'-(1,4-Dioxo-3-pentyl-2,3-diaza-spiro[4.4]non-2-y...)
Affinity DataKi:  25nMAssay Description:Binding affinity against AT1 in human hepatoma cell line, PLC-PRF-5More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50089990(2-Butyl-3-[2'-(1H-tetrazol-5-yl)-biphenyl-4-ylmeth...)
Affinity DataKi:  25nMAssay Description:Binding affinity against AT1 in human hepatoma cell line, PLC-PRF-5More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50089990(2-Butyl-3-[2'-(1H-tetrazol-5-yl)-biphenyl-4-ylmeth...)
Affinity DataKi:  25nMAssay Description:In vitro binding affinity towards Angiotensin II receptor, type 1 of human hepatoma cell line PLC-PRF-5More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50224052(CHEMBL393792 | adamantane-1-carboxylic Acid (4-Oxo...)
Affinity DataKi:  25.5nMAssay Description:Inhibition of human CB2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50224051(((+/-)-N3-(1-(1-adamantyl)ethyl)-7-chloro-4-oxo-1-...)
Affinity DataKi:  26.1nMAssay Description:Inhibition of human CB2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50224063(CHEMBL235946 | N3-(1-(3,5-dimethyl)adamantyl)-8-ch...)
Affinity DataKi:  27.4nMAssay Description:Inhibition of human CB2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50224061(CHEMBL392288 | N3-(1-(3,5-dimethyl)adamantyl)-4-ox...)
Affinity DataKi:  30.9nMAssay Description:Inhibition of human CB2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50089986(4'-(2,4-Dibutyl-4-methyl-3,5-dioxo-pyrazolidin-1-y...)
Affinity DataKi:  32nMAssay Description:Binding affinity against AT1 in human hepatoma cell line, PLC-PRF-5More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50089988(4'-(3-Butyl-1,4-dioxo-2,3-diaza-spiro[4.4]non-2-yl...)
Affinity DataKi:  32nMAssay Description:Binding affinity against AT1 in human hepatoma cell line, PLC-PRF-5More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50180021((R)-N3-(1-phenylethyl)-4-oxo-1-pentyl-1,4-dihydroq...)
Affinity DataKi:  37.1nMAssay Description:Displacement of [3H]CP-55940 from human CB2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50089993(4'-(1,4-Dioxo-3-propyl-2,3-diaza-spiro[4.4]non-2-y...)
Affinity DataKi:  40nMAssay Description:Binding affinity against AT1 in human hepatoma cell line, PLC-PRF-5More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50089992(4'-(2-Butyl-4,4-dimethyl-3,5-dioxo-pyrazolidin-1-y...)
Affinity DataKi:  42nMAssay Description:Binding affinity against AT1 in human hepatoma cell line, PLC-PRF-5More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50224062(CHEMBL235487 | N3-((1-adamantyl)methyl)-4-oxo-1-pe...)
Affinity DataKi:  50.6nMAssay Description:Inhibition of human CB2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50180022(5-(4-chloro-3-methyl-phenyl)-1-(4-methyl-benzyl)-1...)
Affinity DataKi:  51.7nMAssay Description:Displacement of [3H]CP-55940 from human CB2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50224064(CHEMBL235732 | N3-(1-(3,5-dimethyl)adamantyl)-6-ch...)
Affinity DataKi:  54.6nMAssay Description:Inhibition of human CB2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50180028((+)-N3-(1-(1,2,3,4-tetrahydronaphthyl))-4-oxo-1-pe...)
Affinity DataKi:  60.2nMAssay Description:Displacement of [3H]CP-55940 from human CB2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50180044((RS)-N3-(1-phenylethyl)-4-oxo-1-pentyl-1,4-dihydro...)
Affinity DataKi:  70.8nMAssay Description:Displacement of [3H]CP-55940 from human CB2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50119658(7-Butyl-8-[2'-(1H-tetrazol-5-yl)-biphenyl-4-ylmeth...)
Affinity DataKi:  80nMAssay Description:In vitro binding affinity towards Angiotensin II receptor, type 1 of human hepatoma cell line PLC-PRF-5More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50224083(CHEMBL238047 | N3-(1-(3,5-dimethyl)adamantyl)-4-ox...)
Affinity DataKi:  83.4nMAssay Description:Inhibition of human CB2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50224068(CHEMBL235042 | N3-(1-(3,5-dimethyl)adamantyl)-4-ox...)
Affinity DataKi:  93nMAssay Description:Inhibition of human CB2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50224050(CHEMBL393931 | N3-(1-(3,5-dimethyl)adamantyl)-4-ox...)
Affinity DataKi:  119nMAssay Description:Inhibition of human CB2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50224074(((+/-)-N3-(1-(1,2,3,4-tetrahydronaphthyl))-6-chlor...)
Affinity DataKi:  121nMAssay Description:Inhibition of human CB2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50224074(((+/-)-N3-(1-(1,2,3,4-tetrahydronaphthyl))-6-chlor...)
Affinity DataKi:  121nMAssay Description:Inhibition of human CB2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50180038((R)-N3-(1-(1-naphthyl)ethyl)-4-oxo-1-pentyl-1,4-di...)
Affinity DataKi:  125nMAssay Description:Displacement of [3H]CP-55940 from human CB2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50224045(((+/-))-N3-(1-(1-adamantyl)ethyl)-6-chloro-4-oxo-1...)
Affinity DataKi:  144nMAssay Description:Inhibition of human CB2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50224045(((+/-))-N3-(1-(1-adamantyl)ethyl)-6-chloro-4-oxo-1...)
Affinity DataKi:  144nMAssay Description:Inhibition of human CB2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50224045(((+/-))-N3-(1-(1-adamantyl)ethyl)-6-chloro-4-oxo-1...)
Affinity DataKi:  144nMAssay Description:Inhibition of human CB2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50224054(CHEMBL392952 | N3-(1-adamantyl)-4-oxo-1-(2-(morpho...)
Affinity DataKi:  152nMAssay Description:Inhibition of human CB2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50224072(3-(naphthalene-1-carbonyl)-1-pentyl-1,4-dihydroqui...)
Affinity DataKi:  154nMAssay Description:Inhibition of human CB2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50089989(2-Phenyl-3-[2'-(1H-tetrazol-5-yl)-biphenyl-4-ylmet...)
Affinity DataKi:  158nMAssay Description:Binding affinity against AT1 in human hepatoma cell line, PLC-PRF-5More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50224069(CHEMBL394230 | N3-(1-(3,5-dimethyl)adamantyl)-4-ox...)
Affinity DataKi:  160nMAssay Description:Inhibition of human CB2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50180030((RS)-N3-(1-(1-naphthyl)ethyl)-4-oxo-1-pentyl-1,4-d...)
Affinity DataKi:  174nMAssay Description:Displacement of [3H]CP-55940 from human CB2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50224082(CHEMBL236539 | N3-(1-(3,5-dimethyl)adamantyl)-2-me...)
Affinity DataKi:  200nMAssay Description:Inhibition of human CB2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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