Affinity DataIC50: 1.10nMAssay Description:Inhibition of Influenza A virus (A/California/07/09 (H1N1)) neuraminidase activity using 4-MUNANA as substrate preincubated for 60 mins followed by s...More data for this Ligand-Target Pair
Affinity DataIC50: 1.30nMAssay Description:Inhibition of Influenza A virus (A/chicken/Bangli/BBVD-563/2007(H5N1)) clade 2 neuraminidase activity using 4-MUNANA as substrate preincubated for 60...More data for this Ligand-Target Pair
Affinity DataIC50: 1.40nMAssay Description:Inhibition of Influenza A virus (A/swine/Shepparton/6/2009 (H1N1)) neuraminidase activity using 4-MUNANA as substrate preincubated for 60 mins follow...More data for this Ligand-Target Pair
Affinity DataIC50: 1.90nMAssay Description:Inhibition of Influenza A virus (A/Mississippi/03/01 (H1N1)) neuraminidase activity using 4-MUNANA as substrate preincubated for 60 mins followed by ...More data for this Ligand-Target Pair
Affinity DataIC50: 2.20nMAssay Description:Inhibition of Influenza A virus (A/Mississippi/03/01 (H1N1)) neuraminidase H274Y mutant using 4-MUNANA as substrate preincubated for 60 mins followed...More data for this Ligand-Target Pair
Affinity DataIC50: 2.5nMAssay Description:Inhibition of Influenza A virus (A/chicken/Vietnam/08/2004 (H5N1)) clade 1 neuraminidase activity using 4-MUNANA as substrate preincubated for 60 min...More data for this Ligand-Target Pair
TargetNeuraminidase(Influenza A virus (A/Brisbane/59/2007(H1N1)))
Csiro Manufacturing
Curated by ChEMBL
Csiro Manufacturing
Curated by ChEMBL
Affinity DataIC50: 3.40nMAssay Description:Inhibition of Influenza A virus (A/Fukui/45/04(H3N2)) neuraminidase E119V mutant activity using 4-MUNANA as substrate preincubated for 60 mins follow...More data for this Ligand-Target Pair
TargetNeuraminidase(Influenza A virus (strain A/Memphis/1/1971 H3N2))
Csiro Manufacturing
Curated by ChEMBL
Csiro Manufacturing
Curated by ChEMBL
Affinity DataIC50: 3.80nMAssay Description:Inhibition of Influenza A virus (A/Fukui/45/04(H3N2)) neuraminidase activity using 4-MUNANA as substrate preincubated for 60 mins followed by substra...More data for this Ligand-Target Pair
Affinity DataIC50: 5.80nMAssay Description:Inhibition of Influenza A virus (A/swine/Shepparton/6/2009 (H1N1)) neuraminidase activity using 4-MUNANA as substrate measured every min for 60 mins ...More data for this Ligand-Target Pair
Affinity DataIC50: 6nMAssay Description:Inhibition of Influenza A virus (A/Mississippi/03/01 (H1N1)) neuraminidase H274Y mutant using 4-MUNANA as substrate measured every min for 60 mins by...More data for this Ligand-Target Pair
Affinity DataIC50: 7.80nMAssay Description:Inhibition of Influenza A virus (A/Mississippi/03/01 (H1N1)) neuraminidase activity using 4-MUNANA as substrate measured every min for 60 mins by flu...More data for this Ligand-Target Pair
Affinity DataIC50: 8.90nMAssay Description:Inhibition of Influenza B virus (B/Perth/211/2001) neuraminidase activity using 4-MUNANA as substrate preincubated for 60 mins followed by substrate ...More data for this Ligand-Target Pair
Affinity DataIC50: 11nMAssay Description:Inhibition of Influenza A virus (A/chicken/Bangli/BBVD-563/2007(H5N1)) clade 2 neuraminidase activity using 4-MUNANA as substrate measured every min ...More data for this Ligand-Target Pair
Affinity DataIC50: 12nMAssay Description:Inhibition of Influenza A virus (A/chicken/Vietnam/08/2004 (H5N1)) clade 1 neuraminidase activity using 4-MUNANA as substrate measured every min for ...More data for this Ligand-Target Pair
Affinity DataIC50: 12nMAssay Description:Inhibition of Influenza A virus (A/California/07/09 (H1N1)) neuraminidase activity using 4-MUNANA as substrate measured every min for 60 mins by fluo...More data for this Ligand-Target Pair
TargetReverse transcriptase(Human immunodeficiency virus 1)
Mcgill University Aids Centre
Curated by ChEMBL
Mcgill University Aids Centre
Curated by ChEMBL
Affinity DataIC50: 18nMAssay Description:Inhibition of Human immunodeficiency virus 1 subtype B reverse transcriptase DNA-dependent DNA polymerase activity by gel-based primer extension assa...More data for this Ligand-Target Pair
TargetReverse transcriptase(Human immunodeficiency virus 1)
Mcgill University Aids Centre
Curated by ChEMBL
Mcgill University Aids Centre
Curated by ChEMBL
Affinity DataIC50: 19nMAssay Description:Inhibition of RNA-dependent DNA polymerase activity of wild type HIV1 subtype B reverse transcriptase by filter-based filtration assayMore data for this Ligand-Target Pair
Affinity DataIC50: 24nMAssay Description:Inhibition of Influenza A virus (A/Mississippi/03/01 (H1N1)) neuraminidase H274Y mutant using 4-MUNANA as substrate measured every min for 60 mins by...More data for this Ligand-Target Pair
Affinity DataIC50: 27nMAssay Description:Inhibition of Influenza B virus (B/Perth/211/2001) neuraminidase activity using 4-MUNANA as substrate preincubated for 60 mins followed by substrate ...More data for this Ligand-Target Pair
TargetReverse transcriptase(Human immunodeficiency virus 1)
Mcgill University Aids Centre
Curated by ChEMBL
Mcgill University Aids Centre
Curated by ChEMBL
Affinity DataIC50: 30nMAssay Description:Inhibition of RNA-dependent DNA polymerase activity of wild type HIV1 subtype B reverse transcriptase by filter-based filtration assayMore data for this Ligand-Target Pair
Affinity DataIC50: 32nMAssay Description:Inhibition of Influenza B virus (B/Perth/211/2001) neuraminidase D197E mutant activity using 4-MUNANA as substrate preincubated for 60 mins followed ...More data for this Ligand-Target Pair
TargetNeuraminidase(Influenza A virus (strain A/Memphis/1/1971 H3N2))
Csiro Manufacturing
Curated by ChEMBL
Csiro Manufacturing
Curated by ChEMBL
Affinity DataIC50: 32nMAssay Description:Inhibition of Influenza A virus (A/Fukui/45/04(H3N2)) neuraminidase activity using 4-MUNANA as substrate measured every min for 60 mins by fluorescen...More data for this Ligand-Target Pair
TargetReverse transcriptase(Human immunodeficiency virus 1)
Mcgill University Aids Centre
Curated by ChEMBL
Mcgill University Aids Centre
Curated by ChEMBL
Affinity DataIC50: 36nMAssay Description:Inhibition of DNA-dependent DNA polymerase activity of wild-type Human immunodeficiency virus 1 subtype B reverse transcriptase Y181C mutant by filte...More data for this Ligand-Target Pair
Affinity DataIC50: 37nMAssay Description:Inhibition of Influenza A virus (A/Mississippi/03/01 (H1N1)) neuraminidase activity using 4-MUNANA as substrate preincubated for 60 mins followed by ...More data for this Ligand-Target Pair
Affinity DataIC50: 40nMAssay Description:Inhibition of Influenza B virus (B/Perth/211/2001) neuraminidase activity using 4-MUNANA as substrate preincubated for 60 mins followed by substrate ...More data for this Ligand-Target Pair
Affinity DataIC50: 48nMAssay Description:Inhibition of Influenza A virus (A/Mississippi/03/01 (H1N1)) neuraminidase activity using 4-MUNANA as substrate measured every min for 60 mins by flu...More data for this Ligand-Target Pair
TargetNeuraminidase(Influenza A virus (A/Brisbane/59/2007(H1N1)))
Csiro Manufacturing
Curated by ChEMBL
Csiro Manufacturing
Curated by ChEMBL
Affinity DataIC50: 52nMAssay Description:Inhibition of Influenza A virus (A/Fukui/45/04(H3N2)) neuraminidase E119V mutant activity using 4-MUNANA as substrate measured every min for 60 mins ...More data for this Ligand-Target Pair
TargetReverse transcriptase(Human immunodeficiency virus 1)
Mcgill University Aids Centre
Curated by ChEMBL
Mcgill University Aids Centre
Curated by ChEMBL
Affinity DataIC50: 57nMAssay Description:Inhibition of DNA-dependent DNA polymerase activity of wild type HIV1 subtype B reverse transcriptase by gel-based primer extension assayMore data for this Ligand-Target Pair
Affinity DataIC50: 61nMAssay Description:Inhibition of Influenza A virus (A/Mississippi/03/01 (H1N1)) neuraminidase activity using 4-MUNANA as substrate measured every min for 60 mins by flu...More data for this Ligand-Target Pair
Affinity DataIC50: 65nMAssay Description:Inhibition of Influenza B virus (B/Perth/211/2001) neuraminidase activity using 4-MUNANA as substrate preincubated for 60 mins followed by substrate ...More data for this Ligand-Target Pair
TargetReverse transcriptase(Human immunodeficiency virus 1)
Mcgill University Aids Centre
Curated by ChEMBL
Mcgill University Aids Centre
Curated by ChEMBL
Affinity DataIC50: 68nMAssay Description:Inhibition of RNA-dependent DNA polymerase activity of wild type HIV1 subtype B reverse transcriptase by filter-based filtration assayMore data for this Ligand-Target Pair
Affinity DataIC50: 69nMAssay Description:Inhibition of Influenza A virus (A/Mississippi/03/01 (H1N1)) neuraminidase activity using 4-MUNANA as substrate preincubated for 60 mins followed by ...More data for this Ligand-Target Pair
Affinity DataIC50: 76nMAssay Description:Inhibition of Influenza B virus (B/Perth/211/2001) neuraminidase activity using 4-MUNANA as substrate measured every min for 60 mins by fluorescence ...More data for this Ligand-Target Pair
Affinity DataIC50: 80nMAssay Description:Inhibition of Influenza A virus (A/Mississippi/03/01 (H1N1)) neuraminidase activity using 4-MUNANA as substrate preincubated for 60 mins followed by ...More data for this Ligand-Target Pair
TargetReverse transcriptase(Human immunodeficiency virus 1)
Mcgill University Aids Centre
Curated by ChEMBL
Mcgill University Aids Centre
Curated by ChEMBL
Affinity DataIC50: 93nMAssay Description:Inhibition of RNA-dependent DNA polymerase activity of wild-type Human immunodeficiency virus 1 subtype B reverse transcriptase by filter-based filtr...More data for this Ligand-Target Pair
TargetReverse transcriptase(Human immunodeficiency virus 1)
Mcgill University Aids Centre
Curated by ChEMBL
Mcgill University Aids Centre
Curated by ChEMBL
Affinity DataIC50: 97nMAssay Description:Inhibition of Human immunodeficiency virus 1 subtype B reverse transcriptase DNA-dependent DNA polymerase activity by gel-based primer extension assa...More data for this Ligand-Target Pair
Affinity DataIC50: 98nMAssay Description:Inhibition of Influenza A virus (A/Mississippi/03/01 (H1N1)) neuraminidase H274Y mutant using 4-MUNANA as substrate measured every min for 60 mins by...More data for this Ligand-Target Pair
TargetNeuraminidase(Influenza A virus (A/Brisbane/59/2007(H1N1)))
Csiro Manufacturing
Curated by ChEMBL
Csiro Manufacturing
Curated by ChEMBL
Affinity DataIC50: 102nMAssay Description:Inhibition of Influenza A virus (A/Fukui/45/04(H3N2)) neuraminidase E119V mutant activity using 4-MUNANA as substrate preincubated for 60 mins follow...More data for this Ligand-Target Pair
Affinity DataIC50: 104nMAssay Description:Inhibition of Influenza A virus (A/Mississippi/03/01 (H1N1)) neuraminidase H274Y mutant using 4-MUNANA as substrate preincubated for 60 mins followed...More data for this Ligand-Target Pair
TargetReverse transcriptase(Human immunodeficiency virus 1)
Mcgill University Aids Centre
Curated by ChEMBL
Mcgill University Aids Centre
Curated by ChEMBL
Affinity DataIC50: 107nMAssay Description:Inhibition of DNA-dependent DNA polymerase activity of wild-type Human immunodeficiency virus 1 subtype B reverse transcriptase Y181C mutant by filte...More data for this Ligand-Target Pair
TargetReverse transcriptase protein(Human immunodeficiency virus 1)
Mcgill University Aids Centre
Curated by ChEMBL
Mcgill University Aids Centre
Curated by ChEMBL
Affinity DataIC50: 112nMAssay Description:Inhibition of Human immunodeficiency virus 1 subtype B reverse transcriptase G190A mutant by filter-based filtration assayMore data for this Ligand-Target Pair
Affinity DataIC50: 116nMAssay Description:Inhibition of Influenza A virus (A/Mississippi/03/01 (H1N1)) neuraminidase activity using 4-MUNANA as substrate measured every min for 60 mins by flu...More data for this Ligand-Target Pair
Affinity DataIC50: 116nMAssay Description:Inhibition of Influenza A virus (A/Mississippi/03/01 (H1N1)) neuraminidase H274Y mutant using 4-MUNANA as substrate preincubated for 60 mins followed...More data for this Ligand-Target Pair
TargetReverse transcriptase(Human immunodeficiency virus 1)
Mcgill University Aids Centre
Curated by ChEMBL
Mcgill University Aids Centre
Curated by ChEMBL
Affinity DataIC50: 126nMAssay Description:Inhibition of DNA-dependent DNA polymerase activity of wild type HIV1 subtype B reverse transcriptase by gel-based primer extension assayMore data for this Ligand-Target Pair
TargetReverse transcriptase(Human immunodeficiency virus 1)
Mcgill University Aids Centre
Curated by ChEMBL
Mcgill University Aids Centre
Curated by ChEMBL
Affinity DataIC50: 126nMAssay Description:Inhibition of Human immunodeficiency virus 1 subtype B reverse transcriptase Y181C mutant by filter-based filtration assayMore data for this Ligand-Target Pair
TargetReverse transcriptase protein(Human immunodeficiency virus 1)
Mcgill University Aids Centre
Curated by ChEMBL
Mcgill University Aids Centre
Curated by ChEMBL
Affinity DataIC50: 129nMAssay Description:Inhibition of DNA-dependent DNA polymerase activity of wild-type Human immunodeficiency virus 1 subtype B reverse transcriptase G190A mutant by filte...More data for this Ligand-Target Pair
TargetReverse transcriptase(Human immunodeficiency virus 1)
Mcgill University Aids Centre
Curated by ChEMBL
Mcgill University Aids Centre
Curated by ChEMBL
Affinity DataIC50: 131nMAssay Description:Inhibition of DNA-dependent DNA polymerase activity of wild type HIV1 subtype B reverse transcriptase by gel-based primer extension assayMore data for this Ligand-Target Pair
Affinity DataIC50: 133nMAssay Description:Inhibition of Influenza A virus (A/Mississippi/03/01 (H1N1)) neuraminidase H274Y mutant using 4-MUNANA as substrate preincubated for 60 mins followed...More data for this Ligand-Target Pair
Affinity DataIC50: 139nMAssay Description:Inhibition of Influenza A virus (A/Mississippi/03/01 (H1N1)) neuraminidase H274Y mutant using 4-MUNANA as substrate measured every min for 60 mins by...More data for this Ligand-Target Pair
Affinity DataIC50: 167nMAssay Description:Inhibition of Influenza B virus (B/Perth/211/2001) neuraminidase activity using 4-MUNANA as substrate measured every min for 60 mins by fluorescence ...More data for this Ligand-Target Pair