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Found 22 Enz. Inhib. hit(s) with Target = 'Neuraminidase' and Ligand = 'BDBM50271298'
TargetNeuraminidase(Influenza B virus)
Csiro Manufacturing

Curated by ChEMBL
LigandPNGBDBM50271298(CHEMBL4128362)
Affinity DataIC50:  65nMAssay Description:Inhibition of Influenza B virus (B/Perth/211/2001) neuraminidase activity using 4-MUNANA as substrate preincubated for 60 mins followed by substrate ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuraminidase(Influenza A virus)
Csiro Manufacturing

Curated by ChEMBL
LigandPNGBDBM50271298(CHEMBL4128362)
Affinity DataIC50:  80nMAssay Description:Inhibition of Influenza A virus (A/Mississippi/03/01 (H1N1)) neuraminidase activity using 4-MUNANA as substrate preincubated for 60 mins followed by ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuraminidase(Influenza A virus)
Csiro Manufacturing

Curated by ChEMBL
LigandPNGBDBM50271298(CHEMBL4128362)
Affinity DataIC50:  116nMAssay Description:Inhibition of Influenza A virus (A/Mississippi/03/01 (H1N1)) neuraminidase H274Y mutant using 4-MUNANA as substrate preincubated for 60 mins followed...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuraminidase(Influenza A virus)
Csiro Manufacturing

Curated by ChEMBL
LigandPNGBDBM50271298(CHEMBL4128362)
Affinity DataIC50:  116nMAssay Description:Inhibition of Influenza A virus (A/Mississippi/03/01 (H1N1)) neuraminidase activity using 4-MUNANA as substrate measured every min for 60 mins by flu...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuraminidase(Influenza A virus)
Csiro Manufacturing

Curated by ChEMBL
LigandPNGBDBM50271298(CHEMBL4128362)
Affinity DataIC50:  139nMAssay Description:Inhibition of Influenza A virus (A/Mississippi/03/01 (H1N1)) neuraminidase H274Y mutant using 4-MUNANA as substrate measured every min for 60 mins by...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuraminidase(Influenza B virus (B/Lee/40))
Csiro Manufacturing

Curated by ChEMBL
LigandPNGBDBM50271298(CHEMBL4128362)
Affinity DataIC50:  174nMAssay Description:Inhibition of Influenza B virus (B/Perth/211/2001) neuraminidase D197E mutant activity using 4-MUNANA as substrate preincubated for 60 mins followed ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuraminidase(Influenza A virus (A/Brisbane/59/2007(H1N1)))
Csiro Manufacturing

Curated by ChEMBL
LigandPNGBDBM50271298(CHEMBL4128362)
Affinity DataIC50:  238nMAssay Description:Inhibition of Influenza A virus (A/Fukui/45/04(H3N2)) neuraminidase E119V mutant activity using 4-MUNANA as substrate preincubated for 60 mins follow...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuraminidase(Influenza B virus)
Csiro Manufacturing

Curated by ChEMBL
LigandPNGBDBM50271298(CHEMBL4128362)
Affinity DataIC50:  414nMAssay Description:Inhibition of Influenza B virus (B/Perth/211/2001) neuraminidase activity using 4-MUNANA as substrate measured every min for 60 mins by fluorescence ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuraminidase(Influenza A virus (A/Brisbane/59/2007(H1N1)))
Csiro Manufacturing

Curated by ChEMBL
LigandPNGBDBM50271298(CHEMBL4128362)
Affinity DataIC50:  465nMAssay Description:Inhibition of Influenza A virus (A/Fukui/45/04(H3N2)) neuraminidase E119V mutant activity using 4-MUNANA as substrate measured every min for 60 mins ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuraminidase(Influenza A virus)
Csiro Manufacturing

Curated by ChEMBL
LigandPNGBDBM50271298(CHEMBL4128362)
Affinity DataIC50:  470nMAssay Description:Inhibition of Influenza A virus (A/swine/Shepparton/6/2009 (H1N1)) neuraminidase activity using 4-MUNANA as substrate preincubated for 60 mins follow...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuraminidase(Influenza A virus)
Csiro Manufacturing

Curated by ChEMBL
LigandPNGBDBM50271298(CHEMBL4128362)
Affinity DataIC50:  601nMAssay Description:Inhibition of Influenza A virus (A/California/07/09 (H1N1)) neuraminidase activity using 4-MUNANA as substrate preincubated for 60 mins followed by s...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuraminidase(Influenza A virus)
Csiro Manufacturing

Curated by ChEMBL
LigandPNGBDBM50271298(CHEMBL4128362)
Affinity DataIC50:  791nMAssay Description:Inhibition of Influenza A virus (A/California/07/09 (H1N1)) neuraminidase activity using 4-MUNANA as substrate measured every min for 60 mins by fluo...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuraminidase(Influenza A virus)
Csiro Manufacturing

Curated by ChEMBL
LigandPNGBDBM50271298(CHEMBL4128362)
Affinity DataIC50:  791nMAssay Description:Inhibition of Influenza A virus (A/swine/Shepparton/6/2009 (H1N1)) neuraminidase activity using 4-MUNANA as substrate measured every min for 60 mins ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuraminidase(Influenza A virus)
Csiro Manufacturing

Curated by ChEMBL
LigandPNGBDBM50271298(CHEMBL4128362)
Affinity DataIC50:  863nMAssay Description:Inhibition of Influenza A virus (A/chicken/Bangli/BBVD-563/2007(H5N1)) clade 2 neuraminidase activity using 4-MUNANA as substrate preincubated for 60...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuraminidase(Influenza A virus)
Csiro Manufacturing

Curated by ChEMBL
LigandPNGBDBM50271298(CHEMBL4128362)
Affinity DataIC50:  889nMAssay Description:Inhibition of Influenza A virus (A/chicken/Bangli/BBVD-563/2007(H5N1)) clade 2 neuraminidase activity using 4-MUNANA as substrate measured every min ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuraminidase(Influenza A virus)
Csiro Manufacturing

Curated by ChEMBL
LigandPNGBDBM50271298(CHEMBL4128362)
Affinity DataIC50:  1.15E+3nMAssay Description:Inhibition of Influenza A virus (A/NWS/G70C(H1N9)) neuraminidase E119G mutant activity using 4-MUNANA as substrate preincubated for 60 mins followed ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuraminidase(Influenza A virus)
Csiro Manufacturing

Curated by ChEMBL
LigandPNGBDBM50271298(CHEMBL4128362)
Affinity DataIC50:  1.20E+3nMAssay Description:Inhibition of Influenza A virus (A/NWS/G70C(H1N9)) neuraminidase E119G mutant activity using 4-MUNANA as substrate measured every min for 60 mins by ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuraminidase(Influenza B virus (B/Lee/40))
Csiro Manufacturing

Curated by ChEMBL
LigandPNGBDBM50271298(CHEMBL4128362)
Affinity DataIC50:  1.26E+3nMAssay Description:Inhibition of Influenza B virus (B/Perth/211/2001) neuraminidase D197E mutant activity using 4-MUNANA as substrate measured every min for 60 mins by ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuraminidase(Influenza A virus (strain A/Memphis/1/1971 H3N2))
Csiro Manufacturing

Curated by ChEMBL
LigandPNGBDBM50271298(CHEMBL4128362)
Affinity DataIC50:  1.38E+3nMAssay Description:Inhibition of Influenza A virus (A/Fukui/45/04(H3N2)) neuraminidase activity using 4-MUNANA as substrate preincubated for 60 mins followed by substra...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuraminidase(Influenza A virus)
Csiro Manufacturing

Curated by ChEMBL
LigandPNGBDBM50271298(CHEMBL4128362)
Affinity DataIC50:  1.66E+3nMAssay Description:Inhibition of Influenza A virus (A/chicken/Vietnam/08/2004 (H5N1)) clade 1 neuraminidase activity using 4-MUNANA as substrate preincubated for 60 min...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuraminidase(Influenza A virus (strain A/Memphis/1/1971 H3N2))
Csiro Manufacturing

Curated by ChEMBL
LigandPNGBDBM50271298(CHEMBL4128362)
Affinity DataIC50:  1.67E+3nMAssay Description:Inhibition of Influenza A virus (A/Fukui/45/04(H3N2)) neuraminidase activity using 4-MUNANA as substrate measured every min for 60 mins by fluorescen...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuraminidase(Influenza A virus)
Csiro Manufacturing

Curated by ChEMBL
LigandPNGBDBM50271298(CHEMBL4128362)
Affinity DataIC50:  2.17E+3nMAssay Description:Inhibition of Influenza A virus (A/chicken/Vietnam/08/2004 (H5N1)) clade 1 neuraminidase activity using 4-MUNANA as substrate measured every min for ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed