TargetBeta-1 adrenergic receptor(Rattus norvegicus (Rat))
National Institute of Diabetes
Curated by ChEMBL
National Institute of Diabetes
Curated by ChEMBL
Affinity DataKi: 60nMAssay Description:Compound was evaluated for the inhibition of binding of [3H]-dihydroalprenolol from beta-1 adrenergic receptor of rat cerebral cortical membranesMore data for this Ligand-Target Pair
TargetBeta-1 adrenergic receptor(Rattus norvegicus (Rat))
National Institute of Diabetes
Curated by ChEMBL
National Institute of Diabetes
Curated by ChEMBL
Affinity DataKi: 120nMAssay Description:Compound was evaluated for the inhibition of binding of [3H]-dihydroalprenolol from beta-1 adrenergic receptor of rat cerebral cortical membranesMore data for this Ligand-Target Pair
TargetBeta-1 adrenergic receptor(Rattus norvegicus (Rat))
National Institute of Diabetes
Curated by ChEMBL
National Institute of Diabetes
Curated by ChEMBL
Affinity DataKi: 670nMAssay Description:Compound was evaluated for the inhibition of binding of [3H]-dihydroalprenolol from beta-1 adrenergic receptor of rat cerebral cortical membranesMore data for this Ligand-Target Pair
Affinity DataKi: 2.23E+3nMAssay Description:Inhibitory constant was determined in an HIV-1 reverse transcriptase assay in which the [3H]dTTP concentration was varied (i.e. 40, 20, 10, 6, and 4 ...More data for this Ligand-Target Pair
TargetBeta-1 adrenergic receptor(Rattus norvegicus (Rat))
National Institute of Diabetes
Curated by ChEMBL
National Institute of Diabetes
Curated by ChEMBL
Affinity DataKi: 8.70E+4nMAssay Description:Compound was evaluated for the inhibition of binding of [3H]-dihydroalprenolol from beta-1 adrenergic receptor of rat cerebral cortical membranesMore data for this Ligand-Target Pair
Affinity DataIC50: 22nMAssay Description:Compound concentration that causes 50 % inhibition of HIV-1 peptide-derived reverse transcriptase (RT) obtained from HIV-1-infected H9 cell culturesMore data for this Ligand-Target Pair
Affinity DataIC50: 620nMAssay Description:Compound concentration that causes 50 % inhibition of HIV-1 peptide-derived reverse transcriptase (RT)More data for this Ligand-Target Pair
Affinity DataIC50: 6.95E+3nMAssay Description:Compound concentration that causes 50 % inhibition of HIV-1 peptide-derived reverse transcriptase (RT)More data for this Ligand-Target Pair
TargetBeta-1/Beta-2/Beta-3 adrenergic receptor(Rattus norvegicus (Rat))
National Institute of Diabetes
Curated by ChEMBL
National Institute of Diabetes
Curated by ChEMBL
Affinity DataEC50: 7nMAssay Description:Beta adrenergic receptor agonistic activity for the stimulation of accumulation of cyclic AMP in cultured C6 glioma cellsMore data for this Ligand-Target Pair
TargetBeta-1/Beta-2/Beta-3 adrenergic receptor(Rattus norvegicus (Rat))
National Institute of Diabetes
Curated by ChEMBL
National Institute of Diabetes
Curated by ChEMBL
Affinity DataEC50: 8.20nMAssay Description:Beta adrenergic receptor agonistic activity for the stimulation of accumulation of cyclic AMP in cultured C6 glioma cellsMore data for this Ligand-Target Pair
TargetBeta-1/Beta-2/Beta-3 adrenergic receptor(Rattus norvegicus (Rat))
National Institute of Diabetes
Curated by ChEMBL
National Institute of Diabetes
Curated by ChEMBL
Affinity DataEC50: 9.20nMAssay Description:Activity was evaluated by measuring the inhibition of isolated hog H+/K+ ATPaseMore data for this Ligand-Target Pair
Affinity DataEC50: 38nMAssay Description:Agonistic activity (beta2- adrenergic) for the percent maximal relaxation of isolated guinea pig tracheaMore data for this Ligand-Target Pair
Affinity DataEC50: 8.60nMAssay Description:Agonistic activity (beta-1 adrenergic receptor) for the percent maximal increase in contraction rate of isolated guinea pig atriaMore data for this Ligand-Target Pair
Affinity DataEC50: 130nMAssay Description:Agonistic activity (beta2- adrenergic) for the percent maximal relaxation of isolated guinea pig tracheaMore data for this Ligand-Target Pair
Affinity DataEC50: 58nMAssay Description:Agonistic activity (beta2- adrenergic) for the percent maximal relaxation of isolated guinea pig tracheaMore data for this Ligand-Target Pair
Affinity DataEC50: 6nMAssay Description:Agonistic activity (beta-1 adrenergic receptor) for the percent maximal increase in contraction rate of isolated guinea pig atriaMore data for this Ligand-Target Pair
Affinity DataEC50: 4.70nMAssay Description:Agonistic activity (beta-1 adrenergic receptor) for the percent maximal increase in contraction rate of isolated guinea pig atriaMore data for this Ligand-Target Pair
Affinity DataEC50: 175nMAssay Description:Agonistic activity (beta-1 adrenergic receptor) for the percent maximal increase in contraction rate of isolated guinea pig atriaMore data for this Ligand-Target Pair