TargetAmine oxidase [flavin-containing] A(Homo sapiens (Human))
Universidade Federal Do Rio Grande Do Sul-Ufrgs
Curated by ChEMBL
Universidade Federal Do Rio Grande Do Sul-Ufrgs
Curated by ChEMBL
Affinity DataIC50: 4nMAssay Description:Inhibition of recombinant human MAO-A incubated for 30 mins by fluorescence-based methodMore data for this Ligand-Target Pair
TargetCholinesterase(Equus caballus (Horse))
Universidade Federal Do Rio Grande Do Sul-Ufrgs
Curated by ChEMBL
Universidade Federal Do Rio Grande Do Sul-Ufrgs
Curated by ChEMBL
Affinity DataIC50: 8nMAssay Description:Inhibition of equine serum BChE using (S)-butyrylthiocholine iodide as substrate measured for 6 mins by Ellman's methodMore data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] A(Rattus norvegicus (rat))
Universidad Aut£Noma Del Estado De Morelos
Curated by ChEMBL
Universidad Aut£Noma Del Estado De Morelos
Curated by ChEMBL
Affinity DataIC50: 8nMAssay Description:Inhibition of Wistar rat brain MAOA using kynuramine as substrate preincubated for 15 mins followed by substrate addition and measured after 15 mins ...More data for this Ligand-Target Pair
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
Universidade Federal Do Rio Grande Do Sul-Ufrgs
Curated by ChEMBL
Universidade Federal Do Rio Grande Do Sul-Ufrgs
Curated by ChEMBL
Affinity DataIC50: 70nMAssay Description:Inhibition of electric eel AchE using acetylthiocholine as substrate measured for 6 mins by Ellman's methodMore data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] B(Rattus norvegicus (rat))
Universidad Aut£Noma Del Estado De Morelos
Curated by ChEMBL
Universidad Aut£Noma Del Estado De Morelos
Curated by ChEMBL
Affinity DataIC50: 220nMAssay Description:Inhibition of Wistar rat brain MAOB using kynuramine as substrate preincubated for 15 mins followed by substrate addition and measured after 15 mins ...More data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] A(Homo sapiens (Human))
Universidade Federal Do Rio Grande Do Sul-Ufrgs
Curated by ChEMBL
Universidade Federal Do Rio Grande Do Sul-Ufrgs
Curated by ChEMBL
Affinity DataIC50: 900nMAssay Description:Inhibition of recombinant human MAO-A incubated for 30 mins by fluorescence-based methodMore data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] A(Rattus norvegicus (rat))
Universidad Aut£Noma Del Estado De Morelos
Curated by ChEMBL
Universidad Aut£Noma Del Estado De Morelos
Curated by ChEMBL
Affinity DataIC50: 1.30E+3nMAssay Description:Inhibition of Wistar rat brain MAOA using kynuramine as substrate preincubated for 15 mins followed by substrate addition and measured after 15 mins ...More data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] A(Homo sapiens (Human))
Universidade Federal Do Rio Grande Do Sul-Ufrgs
Curated by ChEMBL
Universidade Federal Do Rio Grande Do Sul-Ufrgs
Curated by ChEMBL
Affinity DataIC50: 1.40E+3nMAssay Description:Inhibition of recombinant human MAO-A incubated for 30 mins by fluorescence-based methodMore data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] A(Homo sapiens (Human))
Universidade Federal Do Rio Grande Do Sul-Ufrgs
Curated by ChEMBL
Universidade Federal Do Rio Grande Do Sul-Ufrgs
Curated by ChEMBL
Affinity DataIC50: 1.40E+3nMAssay Description:Inhibition of recombinant human MAO-A incubated for 30 mins by fluorescence-based methodMore data for this Ligand-Target Pair
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
Universidade Federal Do Rio Grande Do Sul-Ufrgs
Curated by ChEMBL
Universidade Federal Do Rio Grande Do Sul-Ufrgs
Curated by ChEMBL
Affinity DataIC50: 3.40E+3nMAssay Description:Inhibition of Electrophorus electricus AChE using acetylthiocholine iodide as substrate measured during 6 mins by Ellman's methodMore data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] B(Rattus norvegicus (rat))
Universidad Aut£Noma Del Estado De Morelos
Curated by ChEMBL
Universidad Aut£Noma Del Estado De Morelos
Curated by ChEMBL
Affinity DataIC50: 4.40E+3nMAssay Description:Inhibition of Wistar rat brain MAOB using kynuramine as substrate preincubated for 15 mins followed by substrate addition and measured after 15 mins ...More data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] B(Rattus norvegicus (rat))
Universidad Aut£Noma Del Estado De Morelos
Curated by ChEMBL
Universidad Aut£Noma Del Estado De Morelos
Curated by ChEMBL
Affinity DataIC50: 4.70E+3nMAssay Description:Inhibition of Wistar rat brain MAOB using kynuramine as substrate preincubated for 15 mins followed by substrate addition and measured after 15 mins ...More data for this Ligand-Target Pair
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
Universidade Federal Do Rio Grande Do Sul-Ufrgs
Curated by ChEMBL
Universidade Federal Do Rio Grande Do Sul-Ufrgs
Curated by ChEMBL
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of Electrophorus electricus AChE using acetylthiocholine iodide as substrate measured during 6 mins by Ellman's methodMore data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] A(Homo sapiens (Human))
Universidade Federal Do Rio Grande Do Sul-Ufrgs
Curated by ChEMBL
Universidade Federal Do Rio Grande Do Sul-Ufrgs
Curated by ChEMBL
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of recombinant human MAO-A incubated for 30 mins by fluorescence-based methodMore data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] A(Homo sapiens (Human))
Universidade Federal Do Rio Grande Do Sul-Ufrgs
Curated by ChEMBL
Universidade Federal Do Rio Grande Do Sul-Ufrgs
Curated by ChEMBL
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of recombinant human MAO-A incubated for 30 mins by fluorescence-based methodMore data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] A(Homo sapiens (Human))
Universidade Federal Do Rio Grande Do Sul-Ufrgs
Curated by ChEMBL
Universidade Federal Do Rio Grande Do Sul-Ufrgs
Curated by ChEMBL
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of recombinant human MAO-A incubated for 30 mins by fluorescence-based methodMore data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] A(Rattus norvegicus (rat))
Universidad Aut£Noma Del Estado De Morelos
Curated by ChEMBL
Universidad Aut£Noma Del Estado De Morelos
Curated by ChEMBL
Affinity DataIC50: 3.10E+4nMAssay Description:Inhibition of Wistar rat brain MAOA using kynuramine as substrate preincubated for 15 mins followed by substrate addition and measured after 15 mins ...More data for this Ligand-Target Pair