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Found 17 with Last Name = 'henriques' and Initial = 'at'
TargetAmine oxidase [flavin-containing] A(Homo sapiens (Human))
Universidade Federal Do Rio Grande Do Sul-Ufrgs

Curated by ChEMBL
LigandPNGBDBM15581(CHEMBL8706 | CLG | CLORGILINE | Clorgyline | N-[3-...)
Affinity DataIC50:  4nMAssay Description:Inhibition of recombinant human MAO-A incubated for 30 mins by fluorescence-based methodMore data for this Ligand-Target Pair
TargetCholinesterase(Equus caballus (Horse))
Universidade Federal Do Rio Grande Do Sul-Ufrgs

Curated by ChEMBL
LigandPNGBDBM8961(1,2,3,4-tetrahydro-9-acridinamine | 1,2,3,4-tetrah...)
Affinity DataIC50:  8nMAssay Description:Inhibition of equine serum BChE using (S)-butyrylthiocholine iodide as substrate measured for 6 mins by Ellman's methodMore data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] A(Rattus norvegicus (rat))
Universidad Aut£Noma Del Estado De Morelos

Curated by ChEMBL
LigandPNGBDBM15581(CHEMBL8706 | CLG | CLORGILINE | Clorgyline | N-[3-...)
Affinity DataIC50:  8nMAssay Description:Inhibition of Wistar rat brain MAOA using kynuramine as substrate preincubated for 15 mins followed by substrate addition and measured after 15 mins ...More data for this Ligand-Target Pair
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
Universidade Federal Do Rio Grande Do Sul-Ufrgs

Curated by ChEMBL
LigandPNGBDBM8961(1,2,3,4-tetrahydro-9-acridinamine | 1,2,3,4-tetrah...)
Affinity DataIC50:  70nMAssay Description:Inhibition of electric eel AchE using acetylthiocholine as substrate measured for 6 mins by Ellman's methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] B(Rattus norvegicus (rat))
Universidad Aut£Noma Del Estado De Morelos

Curated by ChEMBL
LigandPNGBDBM50172756(Benzyl-methyl-prop-2-ynyl-amine | CHEMBL673 | Euto...)
Affinity DataIC50:  220nMAssay Description:Inhibition of Wistar rat brain MAOB using kynuramine as substrate preincubated for 15 mins followed by substrate addition and measured after 15 mins ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] A(Homo sapiens (Human))
Universidade Federal Do Rio Grande Do Sul-Ufrgs

Curated by ChEMBL
LigandPNGBDBM50539725(CHEMBL4636378)
Affinity DataIC50:  900nMAssay Description:Inhibition of recombinant human MAO-A incubated for 30 mins by fluorescence-based methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] A(Rattus norvegicus (rat))
Universidad Aut£Noma Del Estado De Morelos

Curated by ChEMBL
LigandPNGBDBM50537505(CHEMBL4518615)
Affinity DataIC50:  1.30E+3nMAssay Description:Inhibition of Wistar rat brain MAOA using kynuramine as substrate preincubated for 15 mins followed by substrate addition and measured after 15 mins ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] A(Homo sapiens (Human))
Universidade Federal Do Rio Grande Do Sul-Ufrgs

Curated by ChEMBL
LigandPNGBDBM50539724(CHEMBL4639218)
Affinity DataIC50:  1.40E+3nMAssay Description:Inhibition of recombinant human MAO-A incubated for 30 mins by fluorescence-based methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] A(Homo sapiens (Human))
Universidade Federal Do Rio Grande Do Sul-Ufrgs

Curated by ChEMBL
LigandPNGBDBM50539723(CHEMBL4636394)
Affinity DataIC50:  1.40E+3nMAssay Description:Inhibition of recombinant human MAO-A incubated for 30 mins by fluorescence-based methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
Universidade Federal Do Rio Grande Do Sul-Ufrgs

Curated by ChEMBL
LigandPNGBDBM50279525(CHEMBL4163934)
Affinity DataIC50:  3.40E+3nMAssay Description:Inhibition of Electrophorus electricus AChE using acetylthiocholine iodide as substrate measured during 6 mins by Ellman's methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] B(Rattus norvegicus (rat))
Universidad Aut£Noma Del Estado De Morelos

Curated by ChEMBL
LigandPNGBDBM50537505(CHEMBL4518615)
Affinity DataIC50:  4.40E+3nMAssay Description:Inhibition of Wistar rat brain MAOB using kynuramine as substrate preincubated for 15 mins followed by substrate addition and measured after 15 mins ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] B(Rattus norvegicus (rat))
Universidad Aut£Noma Del Estado De Morelos

Curated by ChEMBL
LigandPNGBDBM50537506(CHEMBL4574182)
Affinity DataIC50:  4.70E+3nMAssay Description:Inhibition of Wistar rat brain MAOB using kynuramine as substrate preincubated for 15 mins followed by substrate addition and measured after 15 mins ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
Universidade Federal Do Rio Grande Do Sul-Ufrgs

Curated by ChEMBL
LigandPNGBDBM50279524(CHEMBL4174584)
Affinity DataIC50:  1.00E+4nMAssay Description:Inhibition of Electrophorus electricus AChE using acetylthiocholine iodide as substrate measured during 6 mins by Ellman's methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] A(Homo sapiens (Human))
Universidade Federal Do Rio Grande Do Sul-Ufrgs

Curated by ChEMBL
LigandPNGBDBM50539726(CHEMBL4645049)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of recombinant human MAO-A incubated for 30 mins by fluorescence-based methodMore data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] A(Homo sapiens (Human))
Universidade Federal Do Rio Grande Do Sul-Ufrgs

Curated by ChEMBL
LigandPNGBDBM50539727(CHEMBL4640837)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of recombinant human MAO-A incubated for 30 mins by fluorescence-based methodMore data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] A(Homo sapiens (Human))
Universidade Federal Do Rio Grande Do Sul-Ufrgs

Curated by ChEMBL
LigandPNGBDBM50539728(CHEMBL4637405)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of recombinant human MAO-A incubated for 30 mins by fluorescence-based methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] A(Rattus norvegicus (rat))
Universidad Aut£Noma Del Estado De Morelos

Curated by ChEMBL
LigandPNGBDBM50537506(CHEMBL4574182)
Affinity DataIC50:  3.10E+4nMAssay Description:Inhibition of Wistar rat brain MAOA using kynuramine as substrate preincubated for 15 mins followed by substrate addition and measured after 15 mins ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed