Affinity DataKi: 0.300nMAssay Description:Antagonist activity against PGE2 activated EP1 receptor assessed as ability to inhibit intracellular calcium mobilisation by FLIPRMore data for this Ligand-Target Pair
Affinity DataKi: 32nMAssay Description:Displacement of [3H]PGE2 from human EP4 receptor expressed in HEK 293 (EBNA) cell membranes incubated for 60 mins by scintillation counting methodMore data for this Ligand-Target Pair
Affinity DataKi: 79nMAssay Description:Displacement of [3H]PGE2 from human EP4 receptor expressed in HEK 293 (EBNA) cell membranes incubated for 60 mins by scintillation counting methodMore data for this Ligand-Target Pair
Affinity DataKi: 158nMAssay Description:Displacement of [3H]PGE2 from human EP4 receptor expressed in HEK 293 (EBNA) cell membranes incubated for 60 mins by scintillation counting methodMore data for this Ligand-Target Pair
Affinity DataKi: 158nMAssay Description:Displacement of [3H]PGE2 from human EP4 receptor expressed in HEK 293 (EBNA) cell membranes incubated for 60 mins by scintillation counting methodMore data for this Ligand-Target Pair
Affinity DataKi: 200nMAssay Description:Displacement of [3H]PGE2 from human EP4 receptor expressed in HEK 293 (EBNA) cell membranes incubated for 60 mins by scintillation counting methodMore data for this Ligand-Target Pair
Affinity DataKi: 398nMAssay Description:Displacement of [3H]PGE2 from human EP4 receptor expressed in HEK 293 (EBNA) cell membranes incubated for 60 mins by scintillation counting methodMore data for this Ligand-Target Pair
Affinity DataKi: 631nMAssay Description:Displacement of [3H]PGE2 from human EP4 receptor expressed in HEK 293 (EBNA) cell membranes incubated for 60 mins by scintillation counting methodMore data for this Ligand-Target Pair
Affinity DataKi: 631nMAssay Description:Displacement of [3H]PGE2 from human EP4 receptor expressed in HEK 293 (EBNA) cell membranes incubated for 60 mins by scintillation counting methodMore data for this Ligand-Target Pair
Affinity DataKi: 2.00E+3nMAssay Description:Displacement of [3H]PGE2 from human EP4 receptor expressed in HEK 293 (EBNA) cell membranes incubated for 60 mins by scintillation counting methodMore data for this Ligand-Target Pair
Affinity DataKi: <6.31E+3nMAssay Description:Displacement of [3H]PGE2 from human EP4 receptor expressed in HEK 293 (EBNA) cell membranes incubated for 60 mins by scintillation counting methodMore data for this Ligand-Target Pair
Affinity DataIC50: 0.0390nMAssay Description:Inhibition of human recombinant rennin in buffer assessed as accumulation of angiotensin 1 using human tetradecapeptide by immunoassayMore data for this Ligand-Target Pair
Affinity DataIC50: 0.0400nMAssay Description:Inhibition of renin in bufferMore data for this Ligand-Target Pair
Affinity DataIC50: 0.0500nMAssay Description:Inhibition of renin in bufferMore data for this Ligand-Target Pair
Affinity DataIC50: 0.0500nMAssay Description:Inhibition of renin in bufferMore data for this Ligand-Target Pair
Affinity DataIC50: 0.0500nMAssay Description:Inhibition of renin in bufferMore data for this Ligand-Target Pair
Affinity DataIC50: 0.0700nMAssay Description:Inhibition of renin in bufferMore data for this Ligand-Target Pair
Affinity DataIC50: 0.0800nMAssay Description:Inhibition of renin in bufferMore data for this Ligand-Target Pair
Affinity DataIC50: 0.0800nMAssay Description:Inhibition of renin in bufferMore data for this Ligand-Target Pair
Affinity DataIC50: 0.0900nMAssay Description:Inhibition of renin in bufferMore data for this Ligand-Target Pair
Affinity DataIC50: 0.0900nMAssay Description:Inhibition of renin in bufferMore data for this Ligand-Target Pair
Affinity DataIC50: 0.0900nMAssay Description:Inhibition of renin in bufferMore data for this Ligand-Target Pair
Affinity DataIC50: 0.100nMAssay Description:Inhibition of renin in bufferMore data for this Ligand-Target Pair
Affinity DataIC50: 0.100nMAssay Description:Inhibition of renin in bufferMore data for this Ligand-Target Pair
Affinity DataIC50: 0.110nMAssay Description:Inhibition of renin in bufferMore data for this Ligand-Target Pair
Affinity DataIC50: 0.120nMAssay Description:Inhibition of renin in bufferMore data for this Ligand-Target Pair
Affinity DataIC50: 0.120nMAssay Description:Inhibition of renin in bufferMore data for this Ligand-Target Pair
Affinity DataIC50: 0.120nMAssay Description:Inhibition of renin in bufferMore data for this Ligand-Target Pair
Affinity DataIC50: 0.130nMAssay Description:Inhibition of renin in bufferMore data for this Ligand-Target Pair
Affinity DataIC50: 0.140nMAssay Description:Inhibition of renin in bufferMore data for this Ligand-Target Pair
Affinity DataIC50: 0.150nMAssay Description:Inhibition of renin in bufferMore data for this Ligand-Target Pair
Affinity DataIC50: 0.150nMAssay Description:Inhibition of renin in bufferMore data for this Ligand-Target Pair
Affinity DataIC50: 0.150nMAssay Description:Inhibition of renin in bufferMore data for this Ligand-Target Pair
Affinity DataIC50: 0.160nMAssay Description:Inhibition of renin in bufferMore data for this Ligand-Target Pair
Affinity DataIC50: 0.160nMAssay Description:Inhibition of human recombinant rennin in buffer assessed as accumulation of angiotensin 1 using human tetradecapeptide by immunoassayMore data for this Ligand-Target Pair
Affinity DataIC50: 0.170nMAssay Description:Inhibition of renin in bufferMore data for this Ligand-Target Pair
Affinity DataIC50: 0.170nMAssay Description:Inhibition of renin in bufferMore data for this Ligand-Target Pair
Affinity DataIC50: 0.170nMAssay Description:Inhibition of renin in bufferMore data for this Ligand-Target Pair
Affinity DataIC50: 0.180nMAssay Description:Inhibition of renin in bufferMore data for this Ligand-Target Pair
Affinity DataIC50: 0.180nMAssay Description:Inhibition of renin in bufferMore data for this Ligand-Target Pair
Affinity DataIC50: 0.180nMAssay Description:Inhibition of renin in bufferMore data for this Ligand-Target Pair
Affinity DataIC50: 0.180nMAssay Description:Inhibition of renin in bufferMore data for this Ligand-Target Pair
Affinity DataIC50: 0.180nMAssay Description:Inhibition of renin in bufferMore data for this Ligand-Target Pair
Affinity DataIC50: 0.180nMAssay Description:Inhibition of renin in bufferMore data for this Ligand-Target Pair
Affinity DataIC50: 0.200nMAssay Description:Inhibition of renin in plasmaMore data for this Ligand-Target Pair
Affinity DataIC50: 0.200nMAssay Description:Inhibition of human recombinant rennin in buffer assessed as accumulation of angiotensin 1 using human tetradecapeptide by immunoassayMore data for this Ligand-Target Pair
Affinity DataIC50: 0.200nMAssay Description:Inhibition of renin in bufferMore data for this Ligand-Target Pair