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Found 33 with Last Name = 'hu' and Initial = 'xq'
TargetAcetylcholinesterase(Rattus norvegicus (rat))
Hunan University

Curated by ChEMBL
LigandPNGBDBM50026058(CHEMBL3335259)
Affinity DataKi:  2.75E+3nMAssay Description:Inhibition of Sprague-Dawley rat brain AChE by Michaelis-Menten equationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Rattus norvegicus (rat))
Hunan University

Curated by ChEMBL
LigandPNGBDBM50026058(CHEMBL3335259)
Affinity DataKi:  4.58E+3nMAssay Description:Inhibition of Sprague-Dawley rat brain AChE using acetylthiocholin iodide as substrate by Michaelis-Menten equationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Rattus norvegicus (rat))
Hunan University

Curated by ChEMBL
LigandPNGBDBM50026058(CHEMBL3335259)
Affinity DataIC50:  4.15E+3nMAssay Description:Inhibition of Sprague-Dawley rat brain AChE using acetylthiocholin iodide as substrate preincubated for 25 mins by Ellman's/UV-vis spectroscopy analy...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetE3 ubiquitin-protein ligase CBL-B(Homo sapiens)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50570684(CHEMBL4872230)
Affinity DataIC50:  7.84E+3nMAssay Description:Binding affinity to recombinant His-tagged Cbl-b (unknown origin) (39 to 368 residues) expressed in Escherichia coli BL21 (DE3) using FITC-DGpYPEPA-N...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Rattus norvegicus (rat))
Hunan University

Curated by ChEMBL
LigandPNGBDBM10620((S)-3-(1-(dimethylamino)ethyl)phenyl ethyl(methyl)...)
Affinity DataIC50:  1.05E+4nMAssay Description:Inhibition of Sprague-Dawley rat brain AChE using acetylthiocholin iodide as substrate preincubated for 25 mins by Ellman's/UV-vis spectroscopy analy...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetE3 ubiquitin-protein ligase CBL-B(Homo sapiens)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50570682(CHEMBL4846771)
Affinity DataIC50:  1.06E+4nMAssay Description:Binding affinity to recombinant His-tagged Cbl-b (unknown origin) (39 to 368 residues) expressed in Escherichia coli BL21 (DE3) using FITC-DGpYPEPA-N...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetE3 ubiquitin-protein ligase CBL-B(Homo sapiens)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50570683(CHEMBL4853735)
Affinity DataIC50:  1.13E+4nMAssay Description:Binding affinity to recombinant His-tagged Cbl-b (unknown origin) (39 to 368 residues) expressed in Escherichia coli BL21 (DE3) using FITC-DGpYPEPA-N...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Rattus norvegicus (rat))
Hunan University

Curated by ChEMBL
LigandPNGBDBM50026061(CHEMBL3335261)
Affinity DataIC50:  1.24E+4nMAssay Description:Inhibition of Sprague-Dawley rat brain AChE using acetylthiocholin iodide as substrate preincubated for 25 mins by Ellman's/UV-vis spectroscopy analy...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Rattus norvegicus (rat))
Hunan University

Curated by ChEMBL
LigandPNGBDBM50026062(CHEMBL3335256)
Affinity DataIC50:  1.51E+4nMAssay Description:Inhibition of Sprague-Dawley rat brain AChE using acetylthiocholin iodide as substrate preincubated for 25 mins by Ellman's/UV-vis spectroscopy analy...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Rattus norvegicus (rat))
Hunan University

Curated by ChEMBL
LigandPNGBDBM50026064(CHEMBL3335258)
Affinity DataIC50:  1.61E+4nMAssay Description:Inhibition of Sprague-Dawley rat brain AChE using acetylthiocholin iodide as substrate preincubated for 25 mins by Ellman's/UV-vis spectroscopy analy...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Rattus norvegicus (rat))
Hunan University

Curated by ChEMBL
LigandPNGBDBM50026065(CHEMBL3335255)
Affinity DataIC50:  1.88E+4nMAssay Description:Inhibition of Sprague-Dawley rat brain AChE using acetylthiocholin iodide as substrate preincubated for 25 mins by Ellman's/UV-vis spectroscopy analy...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetE3 ubiquitin-protein ligase CBL-B(Homo sapiens)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50570689(CHEMBL4867045)
Affinity DataIC50:  2.73E+4nMAssay Description:Binding affinity to recombinant His-tagged Cbl-b (unknown origin) (39 to 368 residues) expressed in Escherichia coli BL21 (DE3) using FITC-DGpYPEPA-N...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetE3 ubiquitin-protein ligase CBL-B(Homo sapiens)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50570690(CHEMBL4874562)
Affinity DataIC50:  4.63E+4nMAssay Description:Binding affinity to recombinant His-tagged Cbl-b (unknown origin) (39 to 368 residues) expressed in Escherichia coli BL21 (DE3) using FITC-DGpYPEPA-N...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Rattus norvegicus (rat))
Hunan University

Curated by ChEMBL
LigandPNGBDBM50026063(CHEMBL3335257)
Affinity DataIC50:  5.48E+4nMAssay Description:Inhibition of Sprague-Dawley rat brain AChE using acetylthiocholin iodide as substrate preincubated for 25 mins by Ellman's/UV-vis spectroscopy analy...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetE3 ubiquitin-protein ligase CBL-B(Homo sapiens)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50570688(CHEMBL4858812)
Affinity DataIC50:  1.04E+5nMAssay Description:Binding affinity to recombinant His-tagged Cbl-b (unknown origin) (39 to 368 residues) expressed in Escherichia coli BL21 (DE3) using FITC-DGpYPEPA-N...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Rattus norvegicus (rat))
Hunan University

Curated by ChEMBL
LigandPNGBDBM50026060(CHEMBL3335260)
Affinity DataIC50:  2.65E+5nMAssay Description:Inhibition of Sprague-Dawley rat brain AChE using acetylthiocholin iodide as substrate preincubated for 25 mins by Ellman's/UV-vis spectroscopy analy...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetE3 ubiquitin-protein ligase CBL-B(Homo sapiens)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50570686(CHEMBL4865503)
Affinity DataIC50:  3.99E+5nMAssay Description:Binding affinity to recombinant His-tagged Cbl-b (unknown origin) (39 to 368 residues) expressed in Escherichia coli BL21 (DE3) using FITC-DGpYPEPA-N...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetE3 ubiquitin-protein ligase CBL-B(Homo sapiens)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50570687(CHEMBL4849701)
Affinity DataIC50: >1.00E+6nMAssay Description:Binding affinity to recombinant His-tagged Cbl-b (unknown origin) (39 to 368 residues) expressed in Escherichia coli BL21 (DE3) using FITC-DGpYPEPA-N...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetE3 ubiquitin-protein ligase CBL-B(Homo sapiens)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50570685(CHEMBL4858228)
Affinity DataIC50: >1.00E+6nMAssay Description:Binding affinity to recombinant His-tagged Cbl-b (unknown origin) (39 to 368 residues) expressed in Escherichia coli BL21 (DE3) using FITC-DGpYPEPA-N...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetE3 ubiquitin-protein ligase CBL-B(Homo sapiens)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50570688(CHEMBL4858812)
Affinity DataKd:  5.71E+4nMAssay Description:Binding affinity to recombinant His-tagged Cbl-b (unknown origin) (39 to 368 residues) expressed in Escherichia coli BL21 (DE3) assessed as dissociat...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetE3 ubiquitin-protein ligase CBL-B(Homo sapiens)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50570689(CHEMBL4867045)
Affinity DataKd:  2.44E+4nMAssay Description:Binding affinity to recombinant His-tagged Cbl-b (unknown origin) (39 to 368 residues) expressed in Escherichia coli BL21 (DE3) assessed as dissociat...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetE3 ubiquitin-protein ligase CBL-B(Homo sapiens)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50570690(CHEMBL4874562)
Affinity DataKd:  1.85E+4nMAssay Description:Binding affinity to recombinant His-tagged Cbl-b (unknown origin) (39 to 368 residues) expressed in Escherichia coli BL21 (DE3) assessed as dissociat...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetE3 ubiquitin-protein ligase CBL-B(Homo sapiens)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50570691(CHEMBL4869894)
Affinity DataKd:  8.28E+3nMAssay Description:Binding affinity to recombinant His-tagged Cbl-b (unknown origin) (39 to 368 residues) expressed in Escherichia coli BL21 (DE3) assessed as dissociat...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetE3 ubiquitin-protein ligase CBL-B(Homo sapiens)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50570692(CHEMBL4870377)
Affinity DataKd:  763nMAssay Description:Binding affinity to recombinant His-tagged Cbl-b (unknown origin) (39 to 368 residues) expressed in Escherichia coli BL21 (DE3) assessed as dissociat...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetE3 ubiquitin-protein ligase CBL-B(Homo sapiens)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50570693(CHEMBL4875389)
Affinity DataKd:  2.98E+4nMAssay Description:Binding affinity to recombinant His-tagged Cbl-b (unknown origin) (39 to 368 residues) expressed in Escherichia coli BL21 (DE3) assessed as dissociat...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetE3 ubiquitin-protein ligase CBL-B(Homo sapiens)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50570694(CHEMBL4870845)
Affinity DataKd:  3.55E+4nMAssay Description:Binding affinity to recombinant His-tagged Cbl-b (unknown origin) (39 to 368 residues) expressed in Escherichia coli BL21 (DE3) assessed as dissociat...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetE3 ubiquitin-protein ligase CBL-B(Homo sapiens)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50570695(CHEMBL4850928)
Affinity DataKd:  4.34E+4nMAssay Description:Binding affinity to recombinant His-tagged Cbl-b (unknown origin) (39 to 368 residues) expressed in Escherichia coli BL21 (DE3) assessed as dissociat...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetE3 ubiquitin-protein ligase CBL-B(Homo sapiens)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50570696(CHEMBL4866454)
Affinity DataKd:  2.29E+4nMAssay Description:Binding affinity to recombinant His-tagged Cbl-b (unknown origin) (39 to 368 residues) expressed in Escherichia coli BL21 (DE3) assessed as dissociat...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetE3 ubiquitin-protein ligase CBL-B(Homo sapiens)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50570686(CHEMBL4865503)
Affinity DataKd:  9.83E+4nMAssay Description:Binding affinity to recombinant His-tagged Cbl-b (unknown origin) (39 to 368 residues) expressed in Escherichia coli BL21 (DE3) assessed as dissociat...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetE3 ubiquitin-protein ligase CBL-B(Homo sapiens)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50570684(CHEMBL4872230)
Affinity DataKd:  5.55E+3nMAssay Description:Binding affinity to recombinant His-tagged Cbl-b (unknown origin) (39 to 368 residues) expressed in Escherichia coli BL21 (DE3) assessed as dissociat...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetE3 ubiquitin-protein ligase CBL-B(Homo sapiens)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50570683(CHEMBL4853735)
Affinity DataKd:  2.24E+4nMAssay Description:Binding affinity to recombinant His-tagged Cbl-b (unknown origin) (39 to 368 residues) expressed in Escherichia coli BL21 (DE3) assessed as dissociat...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetE3 ubiquitin-protein ligase CBL-B(Homo sapiens)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50570682(CHEMBL4846771)
Affinity DataKd:  2.44E+4nMAssay Description:Binding affinity to recombinant His-tagged Cbl-b (unknown origin) (39 to 368 residues) expressed in Escherichia coli BL21 (DE3) assessed as dissociat...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetE3 ubiquitin-protein ligase CBL-B(Homo sapiens)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50570697(CHEMBL4850791)
Affinity DataKd:  3.35E+4nMAssay Description:Binding affinity to recombinant His-tagged Cbl-b (unknown origin) (39 to 368 residues) expressed in Escherichia coli BL21 (DE3) assessed as dissociat...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed