TargetSomatostatin receptor type 2(Homo sapiens (Human))
University of Cambridge
Curated by PDSP Ki Database
University of Cambridge
Curated by PDSP Ki Database
TargetSomatostatin receptor type 5(Homo sapiens (Human))
University of Cambridge
Curated by PDSP Ki Database
University of Cambridge
Curated by PDSP Ki Database
TargetSomatostatin receptor type 1(Homo sapiens (Human))
University of Cambridge
Curated by PDSP Ki Database
University of Cambridge
Curated by PDSP Ki Database
TargetSomatostatin receptor type 3(Homo sapiens (Human))
University of Cambridge
Curated by PDSP Ki Database
University of Cambridge
Curated by PDSP Ki Database
TargetSomatostatin receptor type 4(Homo sapiens (Human))
University of Cambridge
Curated by PDSP Ki Database
University of Cambridge
Curated by PDSP Ki Database
TargetSomatostatin receptor type 2(Homo sapiens (Human))
University of Cambridge
Curated by PDSP Ki Database
University of Cambridge
Curated by PDSP Ki Database
TargetSomatostatin receptor type 5(Homo sapiens (Human))
University of Cambridge
Curated by PDSP Ki Database
University of Cambridge
Curated by PDSP Ki Database
TargetSomatostatin receptor type 3(Homo sapiens (Human))
University of Cambridge
Curated by PDSP Ki Database
University of Cambridge
Curated by PDSP Ki Database
TargetSomatostatin receptor type 4(Homo sapiens (Human))
University of Cambridge
Curated by PDSP Ki Database
University of Cambridge
Curated by PDSP Ki Database
TargetSomatostatin receptor type 4(Homo sapiens (Human))
University of Cambridge
Curated by PDSP Ki Database
University of Cambridge
Curated by PDSP Ki Database
Affinity DataIC50: 41nMAssay Description:Inhibitory concentration required for somatostatin 4 receptor in radioligand binding assay ([125I]-Tyr11-SRIF)More data for this Ligand-Target Pair
TargetSomatostatin receptor type 5(Homo sapiens (Human))
University of Cambridge
Curated by PDSP Ki Database
University of Cambridge
Curated by PDSP Ki Database
Affinity DataIC50: 41nMAssay Description:Inhibitory concentration required for somatostatin 5 receptor in radioligand binding assay ([125I]-Tyr11-SRIF)More data for this Ligand-Target Pair
TargetSomatostatin receptor type 5(Homo sapiens (Human))
University of Cambridge
Curated by PDSP Ki Database
University of Cambridge
Curated by PDSP Ki Database
Affinity DataIC50: 87nMAssay Description:Inhibitory concentration required for somatostatin 5 receptor in radioligand binding assay ([125I]-Tyr11-SRIF)More data for this Ligand-Target Pair
Affinity DataIC50: 100nMAssay Description:Inhibition of human recombinant CYP2D6More data for this Ligand-Target Pair
Affinity DataIC50: 190nMAssay Description:Inhibition of human CYP3A4 expressed in Escherichia coli using diethoxyfluorescein substrate measured in 25 to 30 mins by time dependent inhibition a...More data for this Ligand-Target Pair
Affinity DataIC50: 200nMAssay Description:Inhibition of CYP3A4 (unknown origin) using diethoxyfluorescein substrateMore data for this Ligand-Target Pair
Affinity DataIC50: 200nMAssay Description:Inhibition of human recombinant CYP2D6More data for this Ligand-Target Pair
Affinity DataIC50: 200nMAssay Description:Inhibition of human recombinant CYP2D6More data for this Ligand-Target Pair
Affinity DataIC50: 200nMAssay Description:Inhibition of human recombinant CYP2C9More data for this Ligand-Target Pair
TargetSomatostatin receptor type 2(Homo sapiens (Human))
University of Cambridge
Curated by PDSP Ki Database
University of Cambridge
Curated by PDSP Ki Database
Affinity DataIC50: 275nMAssay Description:Inhibitory concentration required for somatostatin 2 receptor in radioligand binding assay ([125I]-Tyr11-SRIF)More data for this Ligand-Target Pair
Affinity DataIC50: 300nMAssay Description:Inhibition of human recombinant CYP2D6More data for this Ligand-Target Pair
TargetSomatostatin receptor type 5(Homo sapiens (Human))
University of Cambridge
Curated by PDSP Ki Database
University of Cambridge
Curated by PDSP Ki Database
Affinity DataIC50: 316nMAssay Description:Compound was tested for inhibition of specific [125I]Tyr11-SRIF binding to human recombinant SST5 (somatostatin) receptor expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
TargetSomatostatin receptor type 5(Homo sapiens (Human))
University of Cambridge
Curated by PDSP Ki Database
University of Cambridge
Curated by PDSP Ki Database
Affinity DataIC50: 316nMAssay Description:Compound was tested for inhibition of specific [125I]Tyr11-SRIF binding to human recombinant SST5 (somatostatin) receptor expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
TargetSomatostatin receptor type 5(Homo sapiens (Human))
University of Cambridge
Curated by PDSP Ki Database
University of Cambridge
Curated by PDSP Ki Database
Affinity DataIC50: 398nMAssay Description:Compound was tested for inhibition of specific [125I]Tyr11-SRIF binding to human recombinant SST5 (somatostatin) receptor expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 400nMAssay Description:Inhibition of CYP3A4 (unknown origin) using phenylpiperazinylmethylbenzylresofurin substrateMore data for this Ligand-Target Pair
Affinity DataIC50: 400nMAssay Description:Inhibition of human recombinant CYP2C9More data for this Ligand-Target Pair
TargetSomatostatin receptor type 1(Homo sapiens (Human))
University of Cambridge
Curated by PDSP Ki Database
University of Cambridge
Curated by PDSP Ki Database
Affinity DataIC50: 407nMAssay Description:Inhibitory concentration required for somatostatin 1 receptor in radioligand binding assay ([125I]-Tyr11-SRIF)More data for this Ligand-Target Pair
Affinity DataIC50: 500nMAssay Description:Inhibition of human recombinant CYP2D6More data for this Ligand-Target Pair
Affinity DataIC50: 500nMAssay Description:Inhibition of CYP3A4 (unknown origin) using phenylpiperazinylmethylbenzylresofurin substrateMore data for this Ligand-Target Pair
TargetSomatostatin receptor type 5(Homo sapiens (Human))
University of Cambridge
Curated by PDSP Ki Database
University of Cambridge
Curated by PDSP Ki Database
Affinity DataIC50: 501nMAssay Description:Compound was tested for inhibition of specific [125I]Tyr11-SRIF binding to human recombinant SST5 (somatostatin) receptor expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
TargetSomatostatin receptor type 1(Homo sapiens (Human))
University of Cambridge
Curated by PDSP Ki Database
University of Cambridge
Curated by PDSP Ki Database
Affinity DataIC50: 501nMAssay Description:Inhibitory concentration required for somatostatin 1 receptor in radioligand binding assay ([125I]-Tyr11-SRIF)More data for this Ligand-Target Pair
Affinity DataIC50: 600nMAssay Description:Inhibition of CYP3A4 (unknown origin) using diethoxyfluorescein substrateMore data for this Ligand-Target Pair
Affinity DataIC50: 600nMAssay Description:Inhibition of human recombinant CYP2D6More data for this Ligand-Target Pair
Affinity DataIC50: 600nMAssay Description:Inhibition of human recombinant CYP2C9More data for this Ligand-Target Pair
Affinity DataIC50: 800nMAssay Description:Inhibition of human recombinant CYP3A4 using diethoxyfluorescein as substrateMore data for this Ligand-Target Pair
Affinity DataIC50: 900nMAssay Description:Inhibition of CYP3A4 (unknown origin) using diethoxyfluorescein substrateMore data for this Ligand-Target Pair
TargetSomatostatin receptor type 4(Homo sapiens (Human))
University of Cambridge
Curated by PDSP Ki Database
University of Cambridge
Curated by PDSP Ki Database
Affinity DataIC50: 1.05E+3nMAssay Description:Inhibitory concentration required for somatostatin 4 receptor in radioligand binding assay ([125I]-Tyr11-SRIF)More data for this Ligand-Target Pair
Affinity DataIC50: 1.10E+3nMAssay Description:Inhibition of human recombinant CYP2D6More data for this Ligand-Target Pair
TargetSomatostatin receptor type 3(Homo sapiens (Human))
University of Cambridge
Curated by PDSP Ki Database
University of Cambridge
Curated by PDSP Ki Database
Affinity DataIC50: 1.26E+3nMAssay Description:Inhibitory concentration required for somatostatin 3 receptor in radioligand binding assay ([125I]-Tyr11-SRIF)More data for this Ligand-Target Pair
Affinity DataIC50: 1.30E+3nMAssay Description:Inhibition of human recombinant CYP2D6More data for this Ligand-Target Pair
Affinity DataIC50: 1.40E+3nMAssay Description:Inhibition of CYP3A4 (unknown origin) using diethoxyfluorescein substrateMore data for this Ligand-Target Pair
Affinity DataIC50: 1.40E+3nMAssay Description:Inhibition of human CYP3A4 expressed in Escherichia coli using diethoxyfluorescein substrate measured in 25 to 30 mins by time dependent inhibition a...More data for this Ligand-Target Pair
TargetSomatostatin receptor type 5(Homo sapiens (Human))
University of Cambridge
Curated by PDSP Ki Database
University of Cambridge
Curated by PDSP Ki Database
Affinity DataIC50: 1.41E+3nMAssay Description:Compound was tested for inhibition of specific [125I]Tyr11-SRIF binding to human recombinant SST5 (somatostatin) receptor expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 1.50E+3nMAssay Description:Inhibition of CYP3A4 (unknown origin) using phenylpiperazinylmethylbenzylresofurin substrateMore data for this Ligand-Target Pair
Affinity DataIC50: 1.50E+3nMAssay Description:Inhibition of CYP3A4 (unknown origin) using phenylpiperazinylmethylbenzylresofurin substrateMore data for this Ligand-Target Pair
TargetSomatostatin receptor type 2(Homo sapiens (Human))
University of Cambridge
Curated by PDSP Ki Database
University of Cambridge
Curated by PDSP Ki Database
Affinity DataIC50: 1.59E+3nMAssay Description:Inhibitory concentration required for somatostatin 2 receptor in radioligand binding assay ([125I]-Tyr11-SRIF)More data for this Ligand-Target Pair
Affinity DataIC50: 1.60E+3nMAssay Description:Inhibition of human recombinant CYP2D6More data for this Ligand-Target Pair