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Found 218 with Last Name = 'jensen' and Initial = 'hh'
TargetSodium-dependent serotonin transporter(Homo sapiens (Human))
Aarhus University

Curated by ChEMBL
LigandPNGBDBM50304053(CHEMBL595677 | methyl 8-methyl-3-(4-(thiophen-3-yl...)
Affinity DataKi:  0.580nMAssay Description:Displacement of [125I]methyl 3-(4-iodophenyl)-8-methyl-8-aza-bicyclo[3.2.1]octane-2-carboxylate from human recombinant SERT expressed in african gree...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Homo sapiens (Human))
Aarhus University

Curated by ChEMBL
LigandPNGBDBM50304049(1-[3beta-(4-Chloro-phenyl)tropane-2beta-carbonyl-o...)
Affinity DataKi:  0.860nMAssay Description:Displacement of [125I]methyl 3-(4-iodophenyl)-8-methyl-8-aza-bicyclo[3.2.1]octane-2-carboxylate from human recombinant SERT expressed in african gree...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Homo sapiens (Human))
Aarhus University

Curated by ChEMBL
LigandPNGBDBM50304049(1-[3beta-(4-Chloro-phenyl)tropane-2beta-carbonyl-o...)
Affinity DataKi:  1nMAssay Description:Displacement of [125I]methyl 3-(4-iodophenyl)-8-methyl-8-aza-bicyclo[3.2.1]octane-2-carboxylate from human recombinant DAT expressed in african green...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Homo sapiens (Human))
Aarhus University

Curated by ChEMBL
LigandPNGBDBM50304053(CHEMBL595677 | methyl 8-methyl-3-(4-(thiophen-3-yl...)
Affinity DataKi:  2.5nMAssay Description:Displacement of [125I]methyl 3-(4-iodophenyl)-8-methyl-8-aza-bicyclo[3.2.1]octane-2-carboxylate from human recombinant DAT expressed in african green...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Homo sapiens (Human))
Aarhus University

Curated by ChEMBL
LigandPNGBDBM50304045(CHEMBL608703 | methyl 3-(4-chlorophenyl)-8-methyl-...)
Affinity DataKi:  2.70nMAssay Description:Displacement of [125I]methyl 3-(4-iodophenyl)-8-methyl-8-aza-bicyclo[3.2.1]octane-2-carboxylate from human recombinant DAT expressed in african green...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Homo sapiens (Human))
Aarhus University

Curated by ChEMBL
LigandPNGBDBM50304046(1-[3beta-(4-Chloro-phenyl)tropane-2beta-carbonyl-o...)
Affinity DataKi:  3.5nMAssay Description:Displacement of [125I]methyl 3-(4-iodophenyl)-8-methyl-8-aza-bicyclo[3.2.1]octane-2-carboxylate from human recombinant SERT expressed in african gree...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Homo sapiens (Human))
Aarhus University

Curated by ChEMBL
LigandPNGBDBM22166(3-(4-iodophenyl)tropane-2-carboxylic acid methyl e...)
Affinity DataKi:  3.90nMAssay Description:Displacement of [125I]methyl 3-(4-iodophenyl)-8-methyl-8-aza-bicyclo[3.2.1]octane-2-carboxylate from human recombinant DAT expressed in african green...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Homo sapiens (Human))
Aarhus University

Curated by ChEMBL
LigandPNGBDBM50304046(1-[3beta-(4-Chloro-phenyl)tropane-2beta-carbonyl-o...)
Affinity DataKi:  3.90nMAssay Description:Displacement of [125I]methyl 3-(4-iodophenyl)-8-methyl-8-aza-bicyclo[3.2.1]octane-2-carboxylate from human recombinant DAT expressed in african green...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Homo sapiens (Human))
Aarhus University

Curated by ChEMBL
LigandPNGBDBM22166(3-(4-iodophenyl)tropane-2-carboxylic acid methyl e...)
Affinity DataKi:  4.20nMAssay Description:Displacement of [125I]methyl 3-(4-iodophenyl)-8-methyl-8-aza-bicyclo[3.2.1]octane-2-carboxylate from human recombinant SERT expressed in african gree...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Homo sapiens (Human))
Aarhus University

Curated by ChEMBL
LigandPNGBDBM50304047(1-[3beta-(4-Chlorophenyl)tropane-2beta-carbonyl-ox...)
Affinity DataKi:  5.5nMAssay Description:Displacement of [125I]methyl 3-(4-iodophenyl)-8-methyl-8-aza-bicyclo[3.2.1]octane-2-carboxylate from human recombinant DAT expressed in african green...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Homo sapiens (Human))
Aarhus University

Curated by ChEMBL
LigandPNGBDBM50010859(CHEMBL11 | IMIPRAMINE HYDROCHLORIDE | IMIPRAMINE P...)
Affinity DataKi:  5.70nMAssay Description:Inhibition of human SERT I179C mutant expressed in HEK293 MSR cells assessed as [3H]-5-HT uptake preincubated for 30 mins followed addition of [3H]-5...More data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Homo sapiens (Human))
Aarhus University

Curated by ChEMBL
LigandPNGBDBM50304048(1-[3beta-(4-Chlorophenyl)tropane-2beta-carbonyl-am...)
Affinity DataKi:  6.60nMAssay Description:Displacement of [125I]methyl 3-(4-iodophenyl)-8-methyl-8-aza-bicyclo[3.2.1]octane-2-carboxylate from human recombinant DAT expressed in african green...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent noradrenaline transporter(Homo sapiens (Human))
Aarhus University

Curated by ChEMBL
LigandPNGBDBM50304049(1-[3beta-(4-Chloro-phenyl)tropane-2beta-carbonyl-o...)
Affinity DataKi:  8.5nMAssay Description:Displacement of [125I]methyl 3-(4-iodophenyl)-8-methyl-8-aza-bicyclo[3.2.1]octane-2-carboxylate from human recombinant NET expressed in african green...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Homo sapiens (Human))
Aarhus University

Curated by ChEMBL
LigandPNGBDBM50304050(1-[3beta-(4-Chloro-phenyl)tropane-2beta-carbonyl-o...)
Affinity DataKi:  16nMAssay Description:Displacement of [125I]methyl 3-(4-iodophenyl)-8-methyl-8-aza-bicyclo[3.2.1]octane-2-carboxylate from human recombinant DAT expressed in african green...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent noradrenaline transporter(Homo sapiens (Human))
Aarhus University

Curated by ChEMBL
LigandPNGBDBM22166(3-(4-iodophenyl)tropane-2-carboxylic acid methyl e...)
Affinity DataKi:  19nMAssay Description:Displacement of [125I]methyl 3-(4-iodophenyl)-8-methyl-8-aza-bicyclo[3.2.1]octane-2-carboxylate from human recombinant NET expressed in african green...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent noradrenaline transporter(Homo sapiens (Human))
Aarhus University

Curated by ChEMBL
LigandPNGBDBM50304046(1-[3beta-(4-Chloro-phenyl)tropane-2beta-carbonyl-o...)
Affinity DataKi:  20nMAssay Description:Displacement of [125I]methyl 3-(4-iodophenyl)-8-methyl-8-aza-bicyclo[3.2.1]octane-2-carboxylate from human recombinant NET expressed in african green...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Homo sapiens (Human))
Aarhus University

Curated by ChEMBL
LigandPNGBDBM50304047(1-[3beta-(4-Chlorophenyl)tropane-2beta-carbonyl-ox...)
Affinity DataKi:  20nMAssay Description:Displacement of [125I]methyl 3-(4-iodophenyl)-8-methyl-8-aza-bicyclo[3.2.1]octane-2-carboxylate from human recombinant SERT expressed in african gree...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Homo sapiens (Human))
Aarhus University

Curated by ChEMBL
LigandPNGBDBM50304051(1-[3beta-(4-Chlorophenyl)tropane-2beta-carbonyl-am...)
Affinity DataKi:  20nMAssay Description:Displacement of [125I]methyl 3-(4-iodophenyl)-8-methyl-8-aza-bicyclo[3.2.1]octane-2-carboxylate from human recombinant DAT expressed in african green...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Homo sapiens (Human))
Aarhus University

Curated by ChEMBL
LigandPNGBDBM50304045(CHEMBL608703 | methyl 3-(4-chlorophenyl)-8-methyl-...)
Affinity DataKi:  21nMAssay Description:Displacement of [125I]methyl 3-(4-iodophenyl)-8-methyl-8-aza-bicyclo[3.2.1]octane-2-carboxylate from human recombinant SERT expressed in african gree...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Homo sapiens (Human))
Aarhus University

Curated by ChEMBL
LigandPNGBDBM50304052(1-[3beta-(4-Chlorophenyl)tropane-2beta-carbonyl-am...)
Affinity DataKi:  21nMAssay Description:Displacement of [125I]methyl 3-(4-iodophenyl)-8-methyl-8-aza-bicyclo[3.2.1]octane-2-carboxylate from human recombinant DAT expressed in african green...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent noradrenaline transporter(Homo sapiens (Human))
Aarhus University

Curated by ChEMBL
LigandPNGBDBM50304053(CHEMBL595677 | methyl 8-methyl-3-(4-(thiophen-3-yl...)
Affinity DataKi:  26nMAssay Description:Displacement of [125I]methyl 3-(4-iodophenyl)-8-methyl-8-aza-bicyclo[3.2.1]octane-2-carboxylate from human recombinant NET expressed in african green...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Homo sapiens (Human))
Aarhus University

Curated by ChEMBL
LigandPNGBDBM50168070(CHEMBL3798035)
Affinity DataKi:  27nMAssay Description:Inhibition of human SERT I179C mutant expressed in HEK293 MSR cells assessed as [3H]-5-HT uptake preincubated for 30 mins followed addition of [3H]-5...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Homo sapiens (Human))
Aarhus University

Curated by ChEMBL
LigandPNGBDBM50304050(1-[3beta-(4-Chloro-phenyl)tropane-2beta-carbonyl-o...)
Affinity DataKi:  27nMAssay Description:Displacement of [125I]methyl 3-(4-iodophenyl)-8-methyl-8-aza-bicyclo[3.2.1]octane-2-carboxylate from human recombinant SERT expressed in african gree...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Homo sapiens (Human))
Aarhus University

Curated by ChEMBL
LigandPNGBDBM50222175(2-(3,4-dichlorophenyl)-N-(furan-2-ylmethyl)cyclope...)
Affinity DataKi:  30nMAssay Description:Displacement of [125I]RTI55 from human DAT transfected in COS1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Homo sapiens (Human))
Aarhus University

Curated by ChEMBL
LigandPNGBDBM50010859(CHEMBL11 | IMIPRAMINE HYDROCHLORIDE | IMIPRAMINE P...)
Affinity DataKi:  31nMAssay Description:Inhibition of wild-type human SERT expressed in HEK293 MSR cells assessed as [3H]-5-HT uptake preincubated for 30 mins followed addition of [3H]-5HT ...More data for this Ligand-Target Pair
TargetSodium-dependent serotonin transporter(Homo sapiens (Human))
Aarhus University

Curated by ChEMBL
LigandPNGBDBM50168069(CHEMBL3797621)
Affinity DataKi:  35nMAssay Description:Inhibition of human SERT I179C mutant expressed in HEK293 MSR cells assessed as [3H]-5-HT uptake preincubated for 30 mins followed addition of [3H]-5...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent noradrenaline transporter(Homo sapiens (Human))
Aarhus University

Curated by ChEMBL
LigandPNGBDBM50304045(CHEMBL608703 | methyl 3-(4-chlorophenyl)-8-methyl-...)
Affinity DataKi:  39nMAssay Description:Displacement of [125I]methyl 3-(4-iodophenyl)-8-methyl-8-aza-bicyclo[3.2.1]octane-2-carboxylate from human recombinant NET expressed in african green...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Homo sapiens (Human))
Aarhus University

Curated by ChEMBL
LigandPNGBDBM50222179(CHEMBL248824 | m-tolyl 2-(3,4-dichlorophenyl)cyclo...)
Affinity DataKi:  60nMAssay Description:Displacement of [125I]RTI55 from human DAT transfected in COS1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Homo sapiens (Human))
Aarhus University

Curated by ChEMBL
LigandPNGBDBM50304054(1-[3beta-(4-Thiophene-3-yl-phenyl)tropane-2beta-ca...)
Affinity DataKi:  62nMAssay Description:Displacement of [125I]methyl 3-(4-iodophenyl)-8-methyl-8-aza-bicyclo[3.2.1]octane-2-carboxylate from human recombinant SERT expressed in african gree...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Homo sapiens (Human))
Aarhus University

Curated by ChEMBL
LigandPNGBDBM50304051(1-[3beta-(4-Chlorophenyl)tropane-2beta-carbonyl-am...)
Affinity DataKi:  65nMAssay Description:Displacement of [125I]methyl 3-(4-iodophenyl)-8-methyl-8-aza-bicyclo[3.2.1]octane-2-carboxylate from human recombinant SERT expressed in african gree...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Homo sapiens (Human))
Aarhus University

Curated by ChEMBL
LigandPNGBDBM50222191(2-(3,4-dichlorophenyl)-N-(2-fluoroethyl)cyclopent-...)
Affinity DataKi:  70nMAssay Description:Displacement of [125I]RTI55 from human DAT transfected in COS1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Homo sapiens (Human))
Aarhus University

Curated by ChEMBL
LigandPNGBDBM50304055(1,4-Di[3-(4-thiophene-3-yl-phenyl)tropane-2-carbon...)
Affinity DataKi:  93nMAssay Description:Displacement of [125I]methyl 3-(4-iodophenyl)-8-methyl-8-aza-bicyclo[3.2.1]octane-2-carboxylate from human recombinant DAT expressed in african green...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent noradrenaline transporter(Homo sapiens (Human))
Aarhus University

Curated by ChEMBL
LigandPNGBDBM50304051(1-[3beta-(4-Chlorophenyl)tropane-2beta-carbonyl-am...)
Affinity DataKi:  100nMAssay Description:Displacement of [125I]methyl 3-(4-iodophenyl)-8-methyl-8-aza-bicyclo[3.2.1]octane-2-carboxylate from human recombinant NET expressed in african green...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent noradrenaline transporter(Homo sapiens (Human))
Aarhus University

Curated by ChEMBL
LigandPNGBDBM50304050(1-[3beta-(4-Chloro-phenyl)tropane-2beta-carbonyl-o...)
Affinity DataKi:  120nMAssay Description:Displacement of [125I]methyl 3-(4-iodophenyl)-8-methyl-8-aza-bicyclo[3.2.1]octane-2-carboxylate from human recombinant NET expressed in african green...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Homo sapiens (Human))
Aarhus University

Curated by ChEMBL
LigandPNGBDBM50222184(2-(3,4-dichlorophenyl)-N-(thiophen-2-ylmethyl)cycl...)
Affinity DataKi:  140nMAssay Description:Displacement of [125I]RTI55 from human DAT transfected in COS1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Homo sapiens (Human))
Aarhus University

Curated by ChEMBL
LigandPNGBDBM50168069(CHEMBL3797621)
Affinity DataKi:  150nMAssay Description:Inhibition of wild-type human SERT expressed in HEK293 MSR cells assessed as [3H]-5-HT uptake preincubated for 30 mins followed addition of [3H]-5HT ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Homo sapiens (Human))
Aarhus University

Curated by ChEMBL
LigandPNGBDBM50304054(1-[3beta-(4-Thiophene-3-yl-phenyl)tropane-2beta-ca...)
Affinity DataKi:  160nMAssay Description:Displacement of [125I]methyl 3-(4-iodophenyl)-8-methyl-8-aza-bicyclo[3.2.1]octane-2-carboxylate from human recombinant DAT expressed in african green...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Homo sapiens (Human))
Aarhus University

Curated by ChEMBL
LigandPNGBDBM50304055(1,4-Di[3-(4-thiophene-3-yl-phenyl)tropane-2-carbon...)
Affinity DataKi:  160nMAssay Description:Displacement of [125I]methyl 3-(4-iodophenyl)-8-methyl-8-aza-bicyclo[3.2.1]octane-2-carboxylate from human recombinant SERT expressed in african gree...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Homo sapiens (Human))
Aarhus University

Curated by ChEMBL
LigandPNGBDBM50222188(CHEMBL401071 | phenyl 2-(3,4-dichlorophenyl)cyclop...)
Affinity DataKi:  170nMAssay Description:Displacement of [125I]RTI55 from human DAT transfected in COS1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent noradrenaline transporter(Homo sapiens (Human))
Aarhus University

Curated by ChEMBL
LigandPNGBDBM50304048(1-[3beta-(4-Chlorophenyl)tropane-2beta-carbonyl-am...)
Affinity DataKi:  180nMAssay Description:Displacement of [125I]methyl 3-(4-iodophenyl)-8-methyl-8-aza-bicyclo[3.2.1]octane-2-carboxylate from human recombinant NET expressed in african green...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Homo sapiens (Human))
Aarhus University

Curated by ChEMBL
LigandPNGBDBM50304056(1-[3beta-(4-Chlorophenyl)tropane-2beta-carbonyl-am...)
Affinity DataKi:  180nMAssay Description:Displacement of [125I]methyl 3-(4-iodophenyl)-8-methyl-8-aza-bicyclo[3.2.1]octane-2-carboxylate from human recombinant DAT expressed in african green...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Homo sapiens (Human))
Aarhus University

Curated by ChEMBL
LigandPNGBDBM50304057(1,4-Di[3beta-(4-thiophene-3-yl-phenyl)tropane-2bet...)
Affinity DataKi:  210nMAssay Description:Displacement of [125I]methyl 3-(4-iodophenyl)-8-methyl-8-aza-bicyclo[3.2.1]octane-2-carboxylate from human recombinant DAT expressed in african green...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Homo sapiens (Human))
Aarhus University

Curated by ChEMBL
LigandPNGBDBM50222183(CHEMBL403570 | o-tolyl 2-(3,4-dichlorophenyl)cyclo...)
Affinity DataKi:  220nMAssay Description:Displacement of [125I]RTI55 from human DAT transfected in COS1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Homo sapiens (Human))
Aarhus University

Curated by ChEMBL
LigandPNGBDBM50168070(CHEMBL3798035)
Affinity DataKi:  220nMAssay Description:Inhibition of wild-type human SERT expressed in HEK293 MSR cells assessed as [3H]-5-HT uptake preincubated for 30 mins followed addition of [3H]-5HT ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Homo sapiens (Human))
Aarhus University

Curated by ChEMBL
LigandPNGBDBM50304058(1,3-Di[3-(4-thiophene-3-yl-phenyl)tropane-2-carbon...)
Affinity DataKi:  230nMAssay Description:Displacement of [125I]methyl 3-(4-iodophenyl)-8-methyl-8-aza-bicyclo[3.2.1]octane-2-carboxylate from human recombinant DAT expressed in african green...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Homo sapiens (Human))
Aarhus University

Curated by ChEMBL
LigandPNGBDBM50304059(1,10-Di[3beta-(4-thiophene-3-yl-phenyl)tropane-2bc...)
Affinity DataKi:  250nMAssay Description:Displacement of [125I]methyl 3-(4-iodophenyl)-8-methyl-8-aza-bicyclo[3.2.1]octane-2-carboxylate from human recombinant SERT expressed in african gree...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Homo sapiens (Human))
Aarhus University

Curated by ChEMBL
LigandPNGBDBM50304057(1,4-Di[3beta-(4-thiophene-3-yl-phenyl)tropane-2bet...)
Affinity DataKi:  270nMAssay Description:Displacement of [125I]methyl 3-(4-iodophenyl)-8-methyl-8-aza-bicyclo[3.2.1]octane-2-carboxylate from human recombinant SERT expressed in african gree...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Homo sapiens (Human))
Aarhus University

Curated by ChEMBL
LigandPNGBDBM50168064(CHEMBL3799668)
Affinity DataKi:  270nMAssay Description:Inhibition of human SERT I179C mutant expressed in HEK293 MSR cells assessed as [3H]-5-HT uptake preincubated for 30 mins followed addition of [3H]-5...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Homo sapiens (Human))
Aarhus University

Curated by ChEMBL
LigandPNGBDBM50168071(CHEMBL3797849)
Affinity DataKi:  280nMAssay Description:Inhibition of human SERT I179C mutant expressed in HEK293 MSR cells assessed as [3H]-5-HT uptake preincubated for 30 mins followed addition of [3H]-5...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Homo sapiens (Human))
Aarhus University

Curated by ChEMBL
LigandPNGBDBM50168063(CHEMBL3799416)
Affinity DataKi:  290nMAssay Description:Inhibition of human SERT I179C mutant expressed in HEK293 MSR cells assessed as [3H]-5-HT uptake preincubated for 30 mins followed addition of [3H]-5...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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