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Found 18 with Last Name = 'kawabata' and Initial = 'a'
TargetProteinase-activated receptor 2(RAT)
The University of Calgary

Curated by PDSP Ki Database
LigandPNGBDBM85517(CAS_171436-38-7 | SL-NH2 | SLIGRL-NH2)
Affinity DataKi:  260nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetProteinase-activated receptor 2(RAT)
The University of Calgary

Curated by PDSP Ki Database
LigandPNGBDBM85518(tc-NH2 | trans-cinnamoyl-LIGRLO-NH2)
Affinity DataKi:  260nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetProteinase-activated receptor 2(RAT)
The University of Calgary

Curated by PDSP Ki Database
LigandPNGBDBM85516(CAS_141923-41-3 | P5-NH2 | SFLLR-NH2)
Affinity DataKi:  2.30E+3nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetProteinase-activated receptor 2(RAT)
The University of Calgary

Curated by PDSP Ki Database
LigandPNGBDBM85088(SFLLR-OH)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetVoltage-dependent T-type calcium channel subunit alpha-1H(Homo sapiens (Human))
University Of Toyama

Curated by ChEMBL
LigandPNGBDBM50463094(CHEMBL4248823)
Affinity DataIC50:  260nMAssay Description:Inhibition of human CaV3.2 expressed in HEK293 cells assessed as suppression of T-current amplitude after 10 mins by whole cell patch clamp methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetVoltage-dependent T-type calcium channel subunit alpha-1H(Homo sapiens (Human))
University Of Toyama

Curated by ChEMBL
LigandPNGBDBM50463095(CHEMBL4249364)
Affinity DataIC50:  390nMAssay Description:Inhibition of human CaV3.2 expressed in HEK293 cells assessed as suppression of T-current amplitude after 10 mins by whole cell patch clamp methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetVoltage-dependent T-type calcium channel subunit alpha-1H(Homo sapiens (Human))
University Of Toyama

Curated by ChEMBL
LigandPNGBDBM50463098(CHEMBL4238346)
Affinity DataIC50:  460nMAssay Description:Inhibition of human CaV3.2 expressed in HEK293 cells assessed as suppression of T-current amplitude after 10 mins by whole cell patch clamp methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetVoltage-dependent T-type calcium channel subunit alpha-1H(Homo sapiens (Human))
University Of Toyama

Curated by ChEMBL
LigandPNGBDBM50463097(CHEMBL4251381)
Affinity DataIC50:  480nMAssay Description:Inhibition of human CaV3.2 expressed in HEK293 cells assessed as suppression of T-current amplitude after 10 mins by whole cell patch clamp methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetVoltage-dependent T-type calcium channel subunit alpha-1H(Homo sapiens (Human))
University Of Toyama

Curated by ChEMBL
LigandPNGBDBM50463091(CHEMBL4240812)
Affinity DataIC50:  500nMAssay Description:Inhibition of human CaV3.2 expressed in HEK293 cells assessed as suppression of T-current amplitude after 10 mins by whole cell patch clamp methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetVoltage-dependent T-type calcium channel subunit alpha-1H(Homo sapiens (Human))
University Of Toyama

Curated by ChEMBL
LigandPNGBDBM50463096(CHEMBL4245811)
Affinity DataIC50:  640nMAssay Description:Inhibition of human CaV3.2 expressed in HEK293 cells assessed as suppression of T-current amplitude after 10 mins by whole cell patch clamp methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetVoltage-dependent T-type calcium channel subunit alpha-1H(Homo sapiens (Human))
University Of Toyama

Curated by ChEMBL
LigandPNGBDBM19460((2S)-5,7-dihydroxy-2-(4-hydroxyphenyl)-8-(3-methyl...)
Affinity DataIC50:  1.00E+3nMAssay Description:Inhibition of human CaV3.2 expressed in HEK293 cells assessed as suppression of T-current amplitude after 10 mins by whole cell patch clamp methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVoltage-dependent T-type calcium channel subunit alpha-1H(Homo sapiens (Human))
University Of Toyama

Curated by ChEMBL
LigandPNGBDBM50208611((2S)-2-(2,4-dihydroxyphenyl)-5,7-dihydroxy-8-[(2R)...)
Affinity DataIC50:  1.00E+3nMAssay Description:Inhibition of human CaV3.2 expressed in HEK293 cells assessed as suppression of T-current amplitude after 10 mins by whole cell patch clamp methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVoltage-dependent T-type calcium channel subunit alpha-1G(Homo sapiens (Human))
University Of Toyama

Curated by ChEMBL
LigandPNGBDBM58016(2-(4-hydroxyphenyl)-6-(3-methylbut-2-enyl)-5,7-bis...)
Affinity DataIC50:  1.00E+3nMAssay Description:Inhibition of human CaV3.1 expressed in HEK293 cells assessed as suppression of T-current after 10 mins by whole cell patch clamp methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVoltage-dependent T-type calcium channel subunit alpha-1G(Homo sapiens (Human))
University Of Toyama

Curated by ChEMBL
LigandPNGBDBM19460((2S)-5,7-dihydroxy-2-(4-hydroxyphenyl)-8-(3-methyl...)
Affinity DataIC50:  1.00E+3nMAssay Description:Inhibition of human CaV3.1 expressed in HEK293 cells assessed as suppression of T-current after 10 mins by whole cell patch clamp methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVoltage-dependent T-type calcium channel subunit alpha-1G(Homo sapiens (Human))
University Of Toyama

Curated by ChEMBL
LigandPNGBDBM50208611((2S)-2-(2,4-dihydroxyphenyl)-5,7-dihydroxy-8-[(2R)...)
Affinity DataIC50:  1.00E+3nMAssay Description:Inhibition of human CaV3.1 expressed in HEK293 cells assessed as suppression of T-current after 10 mins by whole cell patch clamp methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVoltage-dependent T-type calcium channel subunit alpha-1H(Homo sapiens (Human))
University Of Toyama

Curated by ChEMBL
LigandPNGBDBM58016(2-(4-hydroxyphenyl)-6-(3-methylbut-2-enyl)-5,7-bis...)
Affinity DataIC50:  1.00E+3nMAssay Description:Inhibition of human CaV3.2 expressed in HEK293 cells assessed as suppression of T-current amplitude after 10 mins by whole cell patch clamp methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVoltage-dependent T-type calcium channel subunit alpha-1H(Homo sapiens (Human))
University Of Toyama

Curated by ChEMBL
LigandPNGBDBM50463092(CHEMBL4242828)
Affinity DataIC50:  1.02E+3nMAssay Description:Inhibition of human CaV3.2 expressed in HEK293 cells assessed as suppression of T-current amplitude after 10 mins by whole cell patch clamp methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetVoltage-dependent T-type calcium channel subunit alpha-1H(Homo sapiens (Human))
University Of Toyama

Curated by ChEMBL
LigandPNGBDBM50463093(CHEMBL4237637)
Affinity DataIC50:  1.25E+3nMAssay Description:Inhibition of human CaV3.2 expressed in HEK293 cells assessed as suppression of T-current amplitude after 10 mins by whole cell patch clamp methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed