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Found 86 with Last Name = 'kawachi' and Initial = 'e'
TargetRetinoic acid receptor gamma(Homo sapiens (Human))
University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM31883(9-cis-retinoic acid (9cRA) | ALL-TRANS-RETINOIC AC...)
Affinity DataKi:  0.0400nMAssay Description:Agonistic activity of the compound towards retinoic acid receptor-gammaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMedMMDB

TargetRetinoic acid receptor gamma(Homo sapiens (Human))
University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM31892(9-cis retinoic acid | 9C-RA | CHEMBL705 | Panretin...)
Affinity DataKi:  1nMAssay Description:Agonistic activity of the compound towards retinoic acid receptor-gammaMore data for this Ligand-Target Pair
TargetRetinoic acid receptor alpha(Homo sapiens (Human))
University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM31883(9-cis-retinoic acid (9cRA) | ALL-TRANS-RETINOIC AC...)
Affinity DataKi:  3.30nMAssay Description:Agonistic activity of the compound towards retinoic acid receptor-alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRetinoic acid receptor RXR-beta(Homo sapiens (Human))
University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM31892(9-cis retinoic acid | 9C-RA | CHEMBL705 | Panretin...)
Affinity DataKi:  3.80nMAssay Description:Agonistic activity of the compound towards retinoid X receptor-betaMore data for this Ligand-Target Pair
TargetRetinoic acid receptor beta(Homo sapiens (Human))
University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM31883(9-cis-retinoic acid (9cRA) | ALL-TRANS-RETINOIC AC...)
Affinity DataKi:  4.10nMAssay Description:Agonistic activity of the compound towards retinoic acid receptor-betaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMedMMDB

TargetRetinoic acid receptor RXR-beta(Homo sapiens (Human))
University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50032675(4-[1-(3,5,5,8,8-pentamethyl-5,6,7,8-tetrahydronaph...)
Affinity DataKi:  5.90nMAssay Description:Selective activity of the compound towards retinoid X receptor-betaMore data for this Ligand-Target Pair
TargetRetinoic acid receptor alpha(Homo sapiens (Human))
University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50061625(4-[(5,5,8,8-tetramethyl-5,6,7,8-tetrahydronaphthal...)
Affinity DataKi:  6.5nMAssay Description:Agonistic activity of the compound towards retinoic acid receptor-alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMedDrugBank

TargetRetinoic acid receptor RXR-gamma(Homo sapiens (Human))
University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50032675(4-[1-(3,5,5,8,8-pentamethyl-5,6,7,8-tetrahydronaph...)
Affinity DataKi:  8.30nMAssay Description:Selective activity of the compound towards retinoid X receptor-gammaMore data for this Ligand-Target Pair
TargetRetinoic acid receptor RXR-gamma(Homo sapiens (Human))
University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM31892(9-cis retinoic acid | 9C-RA | CHEMBL705 | Panretin...)
Affinity DataKi:  11nMAssay Description:Agonistic activity of the compound towards retinoid X receptor-gammaMore data for this Ligand-Target Pair
TargetRetinoic acid receptor RXR-alpha(Homo sapiens (Human))
University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM31892(9-cis retinoic acid | 9C-RA | CHEMBL705 | Panretin...)
Affinity DataKi:  12nMAssay Description:Agonistic activity of the compound towards retinoid X receptor-alphaMore data for this Ligand-Target Pair
TargetRetinoic acid receptor RXR-alpha(Homo sapiens (Human))
University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50032675(4-[1-(3,5,5,8,8-pentamethyl-5,6,7,8-tetrahydronaph...)
Affinity DataKi:  16nMAssay Description:Selective activity of the compound towards retinoid X receptor-alphaMore data for this Ligand-Target Pair
TargetRetinoic acid receptor beta(Homo sapiens (Human))
University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50061625(4-[(5,5,8,8-tetramethyl-5,6,7,8-tetrahydronaphthal...)
Affinity DataKi:  30nMAssay Description:Agonistic activity of the compound towards retinoic acid receptor-betaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMedDrugBank

TargetRetinoic acid receptor beta(Homo sapiens (Human))
University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50032675(4-[1-(3,5,5,8,8-pentamethyl-5,6,7,8-tetrahydronaph...)
Affinity DataKi:  50nMAssay Description:Selective activity of the compound towards retinoic acid receptor-betaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRetinoic acid receptor RXR-beta(Homo sapiens (Human))
University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM31883(9-cis-retinoic acid (9cRA) | ALL-TRANS-RETINOIC AC...)
Affinity DataKi:  54nMAssay Description:Agonistic activity of the compound towards retinoid X receptor-betaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRetinoic acid receptor RXR-gamma(Homo sapiens (Human))
University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM31883(9-cis-retinoic acid (9cRA) | ALL-TRANS-RETINOIC AC...)
Affinity DataKi:  120nMAssay Description:Agonistic activity of the compound towards retinoid X receptor-gammaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRetinoic acid receptor gamma(Homo sapiens (Human))
University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50032675(4-[1-(3,5,5,8,8-pentamethyl-5,6,7,8-tetrahydronaph...)
Affinity DataKi:  130nMAssay Description:Selective activity of the compound towards retinoic acid receptor-gammaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRetinoic acid receptor alpha(Homo sapiens (Human))
University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50032675(4-[1-(3,5,5,8,8-pentamethyl-5,6,7,8-tetrahydronaph...)
Affinity DataKi:  180nMAssay Description:Selective activity of the compound towards retinoic acid receptor-alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRetinoic acid receptor beta(Homo sapiens (Human))
University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50061616(4-(5,7,7,10,10-Pentamethyl-7,8,9,10-tetrahydro-5H-...)
Affinity DataKi:  220nMAssay Description:Antagonistic activity of the compound towards retinoic acid receptor-betaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRetinoic acid receptor beta(Homo sapiens (Human))
University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50061618(4-(7,7,10,10-Tetramethyl-7,8,9,10-tetrahydro-5-thi...)
Affinity DataKi:  320nMAssay Description:Synergistic activity of the compound towards retinoic acid receptor-betaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRetinoic acid receptor beta(Homo sapiens (Human))
University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50061617(4-(7,7,10,10-Tetramethyl-7,8,9,10-tetrahydro-5-oxa...)
Affinity DataKi:  320nMAssay Description:Synergistic activity of the compound towards retinoic acid receptor-betaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRetinoic acid receptor RXR-alpha(Homo sapiens (Human))
University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM31883(9-cis-retinoic acid (9cRA) | ALL-TRANS-RETINOIC AC...)
Affinity DataKi:  330nMAssay Description:Agonisticactivity of the compound towards retinoid X receptor-alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRetinoic acid receptor RXR-beta(Homo sapiens (Human))
University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50061618(4-(7,7,10,10-Tetramethyl-7,8,9,10-tetrahydro-5-thi...)
Affinity DataKi:  400nMAssay Description:Synergistic activity of the compound towards retinoid X receptor-betaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRetinoic acid receptor gamma(Homo sapiens (Human))
University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50061615(4-(10,10,13,13,15-Pentamethyl-11,12,13,15-tetrahyd...)
Affinity DataKi:  490nMAssay Description:Antagonistic activity of the compound towards retinoic acid receptor-gammaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRetinoic acid receptor beta(Homo sapiens (Human))
University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50061615(4-(10,10,13,13,15-Pentamethyl-11,12,13,15-tetrahyd...)
Affinity DataKi:  500nMAssay Description:Antagonistic activity of the compound towards retinoic acid receptor-betaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRetinoic acid receptor RXR-gamma(Homo sapiens (Human))
University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50061618(4-(7,7,10,10-Tetramethyl-7,8,9,10-tetrahydro-5-thi...)
Affinity DataKi:  620nMAssay Description:Synergistic activity of the compound towards retinoid X receptor-gammaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRetinoic acid receptor RXR-beta(Homo sapiens (Human))
University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50061624(4-(5,7,7,10,10-Pentamethyl-7,8,9,10-tetrahydro-5H-...)
Affinity DataKi:  640nMAssay Description:Synergistic activity of the compound towards retinoid X receptor-betaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRetinoic acid receptor beta(Homo sapiens (Human))
University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50061624(4-(5,7,7,10,10-Pentamethyl-7,8,9,10-tetrahydro-5H-...)
Affinity DataKi:  680nMAssay Description:Synergistic activity of the compound towards retinoic acid receptor-betaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRetinoic acid receptor RXR-beta(Homo sapiens (Human))
University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50061619(4-(7,7,10,10-Tetramethyl-7,8,9,10-tetrahydro-5H-13...)
Affinity DataKi:  790nMAssay Description:Synergistic activity of the compound towards retinoid X receptor-betaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRetinoic acid receptor beta(Homo sapiens (Human))
University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50061619(4-(7,7,10,10-Tetramethyl-7,8,9,10-tetrahydro-5H-13...)
Affinity DataKi:  810nMAssay Description:Synergistic activity of the compound towards retinoic acid receptor-betaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRetinoic acid receptor alpha(Homo sapiens (Human))
University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50061618(4-(7,7,10,10-Tetramethyl-7,8,9,10-tetrahydro-5-thi...)
Affinity DataKi:  900nMAssay Description:Synergistic activity of the compound towards retinoic acid receptor-alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRetinoic acid receptor RXR-alpha(Homo sapiens (Human))
University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50061618(4-(7,7,10,10-Tetramethyl-7,8,9,10-tetrahydro-5-thi...)
Affinity DataKi:  900nMAssay Description:Synergistic activity of the compound towards retinoid X receptor-alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRetinoic acid receptor alpha(Homo sapiens (Human))
University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50061617(4-(7,7,10,10-Tetramethyl-7,8,9,10-tetrahydro-5-oxa...)
Affinity DataKi:  980nMAssay Description:Synergistic activity of the compound towards retinoic acid receptor-alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRetinoic acid receptor RXR-gamma(Homo sapiens (Human))
University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50061624(4-(5,7,7,10,10-Pentamethyl-7,8,9,10-tetrahydro-5H-...)
Affinity DataKi:  1.00E+3nMAssay Description:Synergistic activity of the compound towards retinoid X receptor-gammaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRetinoic acid receptor RXR-gamma(Homo sapiens (Human))
University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50061619(4-(7,7,10,10-Tetramethyl-7,8,9,10-tetrahydro-5H-13...)
Affinity DataKi:  1.00E+3nMAssay Description:Synergistic activity of the compound towards retinoid X receptor-gammaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRetinoic acid receptor RXR-beta(Homo sapiens (Human))
University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50061617(4-(7,7,10,10-Tetramethyl-7,8,9,10-tetrahydro-5-oxa...)
Affinity DataKi:  1.20E+3nMAssay Description:Synergistic activity of the compound towards retinoid X receptor-betaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRetinoic acid receptor alpha(Homo sapiens (Human))
University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50061615(4-(10,10,13,13,15-Pentamethyl-11,12,13,15-tetrahyd...)
Affinity DataKi:  1.30E+3nMAssay Description:Antagonistic activity of the compound towards retinoic acid receptor-alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRetinoic acid receptor alpha(Homo sapiens (Human))
University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50061616(4-(5,7,7,10,10-Pentamethyl-7,8,9,10-tetrahydro-5H-...)
Affinity DataKi:  1.40E+3nMAssay Description:Antagonistic activity of the compound towards retinoic acid receptor-alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRetinoic acid receptor RXR-gamma(Homo sapiens (Human))
University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50061615(4-(10,10,13,13,15-Pentamethyl-11,12,13,15-tetrahyd...)
Affinity DataKi:  1.50E+3nMAssay Description:Antagonistic activity of the compound towards retinoid X receptor-gammaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRetinoic acid receptor alpha(Homo sapiens (Human))
University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50061619(4-(7,7,10,10-Tetramethyl-7,8,9,10-tetrahydro-5H-13...)
Affinity DataKi:  1.60E+3nMAssay Description:Synergistic activity of the compound towards retinoic acid receptor-alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRetinoic acid receptor RXR-beta(Homo sapiens (Human))
University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50061615(4-(10,10,13,13,15-Pentamethyl-11,12,13,15-tetrahyd...)
Affinity DataKi:  1.70E+3nMAssay Description:Antagonistic activity of the compound towards retinoid X receptor-betaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRetinoic acid receptor RXR-alpha(Homo sapiens (Human))
University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50061619(4-(7,7,10,10-Tetramethyl-7,8,9,10-tetrahydro-5H-13...)
Affinity DataKi:  1.80E+3nMAssay Description:Synergistic activity of the compound towards retinoid X receptor-alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRetinoic acid receptor RXR-alpha(Homo sapiens (Human))
University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50061624(4-(5,7,7,10,10-Pentamethyl-7,8,9,10-tetrahydro-5H-...)
Affinity DataKi:  1.90E+3nMAssay Description:Synergistic activity of the compound towards retinoid X receptor-alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRetinoic acid receptor alpha(Homo sapiens (Human))
University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50061621(4-(5,7,7,10,10-Pentamethyl-7,8,9,10-tetrahydro-5H-...)
Affinity DataKi:  2.00E+3nMAssay Description:Synergistic activity of the compound towards retinoic acid receptor-alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRetinoic acid receptor RXR-gamma(Homo sapiens (Human))
University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50061617(4-(7,7,10,10-Tetramethyl-7,8,9,10-tetrahydro-5-oxa...)
Affinity DataKi:  2.10E+3nMAssay Description:Synergistic activity of the compound towards retinoid X receptor-gammaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRetinoic acid receptor RXR-alpha(Homo sapiens (Human))
University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50061617(4-(7,7,10,10-Tetramethyl-7,8,9,10-tetrahydro-5-oxa...)
Affinity DataKi:  3.80E+3nMAssay Description:Synergistic activity of the compound towards retinoid X receptor-alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRetinoic acid receptor RXR-alpha(Homo sapiens (Human))
University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50061615(4-(10,10,13,13,15-Pentamethyl-11,12,13,15-tetrahyd...)
Affinity DataKi:  3.80E+3nMAssay Description:Antagonistic activity of the compound towards retinoid X receptor-alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVitamin D3 receptor(Bos taurus)
Ochanomizu University

Curated by ChEMBL
LigandPNGBDBM50200182((1S,3R,5Z,7E)-9,10-secocholesta-5,7,10(19)-triene-...)
Affinity DataIC50:  0.0480nMAssay Description:Displacement of [3H]-1-alpha,25-(OH)2D3 from bovine thymus VDR incubated for 18 hrs by competitive binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVitamin D3 receptor(Bos taurus)
Ochanomizu University

Curated by ChEMBL
LigandPNGBDBM50565950(CHEMBL4776651)
Affinity DataIC50:  2.10nMAssay Description:Displacement of [3H]-1-alpha,25-(OH)2D3 from bovine thymus VDR incubated for 18 hrs by competitive binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
In DepthDetails ArticlePubMed
TargetVitamin D3 receptor(Bos taurus)
Ochanomizu University

Curated by ChEMBL
LigandPNGBDBM50565949(CHEMBL4794075)
Affinity DataIC50:  67nMAssay Description:Displacement of [3H]-1-alpha,25-(OH)2D3 from bovine thymus VDR incubated for 18 hrs by competitive binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
In DepthDetails ArticlePubMed
TargetAndrogen receptor(Homo sapiens (Human))
Ochanomizu University

Curated by ChEMBL
LigandPNGBDBM50123007(CHEMBL3622589)
Affinity DataIC50:  180nMAssay Description:Antagonist activity at wild type AR expressed in human SC cells assessed as inhibition of 1 nM DHT-induced cell proliferation after 3 days by WST-8 a...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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