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Found 2202 with Last Name = 'kazaks' and Initial = 'a'
TargetCarbonic anhydrase 12(Homo sapiens (Human))
Riga Technical University

Curated by ChEMBL
LigandPNGBDBM50207820(CHEMBL3985384)
Affinity DataKi:  0.820nMAssay Description:Inhibition of human recombinant transmembrane tumor associated carbonic anhydrase 12 preincubated for 10 mins prior to testing by stopped-flow CO2 hy...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 9(Homo sapiens (Human))
Riga Technical University

Curated by ChEMBL
LigandPNGBDBM50207818(CHEMBL3956725)
Affinity DataKi:  0.940nMAssay Description:Inhibition of human recombinant transmembrane tumor associated carbonic anhydrase 9 preincubated for 10 mins prior to testing by stopped-flow CO2 hyd...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 12(Homo sapiens (Human))
Riga Technical University

Curated by ChEMBL
LigandPNGBDBM50207818(CHEMBL3956725)
Affinity DataKi:  1.5nMAssay Description:Inhibition of human recombinant transmembrane tumor associated carbonic anhydrase 12 preincubated for 10 mins prior to testing by stopped-flow CO2 hy...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 9(Homo sapiens (Human))
Riga Technical University

Curated by ChEMBL
LigandPNGBDBM50207820(CHEMBL3985384)
Affinity DataKi:  1.70nMAssay Description:Inhibition of human recombinant transmembrane tumor associated carbonic anhydrase 9 preincubated for 10 mins prior to testing by stopped-flow CO2 hyd...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 2(Homo sapiens (Human))
Riga Technical University

Curated by ChEMBL
LigandPNGBDBM50207736(CHEMBL3947437)
Affinity DataKi:  2.90nMAssay Description:Inhibition of human recombinant cytosolic carbonic anhydrase 2 preincubated for 10 mins prior to testing by stopped-flow CO2 hydration assayMore data for this Ligand-Target Pair
TargetCarbonic anhydrase 2(Homo sapiens (Human))
Riga Technical University

Curated by ChEMBL
LigandPNGBDBM50207818(CHEMBL3956725)
Affinity DataKi:  3.70nMAssay Description:Inhibition of human recombinant cytosolic carbonic anhydrase 2 preincubated for 10 mins prior to testing by stopped-flow CO2 hydration assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 2(Homo sapiens (Human))
Riga Technical University

Curated by ChEMBL
LigandPNGBDBM50207737(CHEMBL3928543)
Affinity DataKi:  4.40nMAssay Description:Inhibition of human recombinant cytosolic carbonic anhydrase 2 preincubated for 10 mins prior to testing by stopped-flow CO2 hydration assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 12(Homo sapiens (Human))
Riga Technical University

Curated by ChEMBL
LigandPNGBDBM10880(AZA | AZA2 | AZM acetazolamide | Acerazolamide, AA...)
Affinity DataKi:  5nMAssay Description:Inhibition of human recombinant transmembrane CA12 catalytic domain after 6 hrs by stopped-flow CO2 hydration methodMore data for this Ligand-Target Pair
TargetCarbonic anhydrase 12(Homo sapiens (Human))
Riga Technical University

Curated by ChEMBL
LigandPNGBDBM50271176(CHEMBL4130085)
Affinity DataKi:  5nMAssay Description:Inhibition of recombinant human carbonic anhydrase 12 assessed as reduction in CO2 hydration pretreated for 15 mins followed by CO2 addition measured...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 2(Homo sapiens (Human))
Riga Technical University

Curated by ChEMBL
LigandPNGBDBM50207820(CHEMBL3985384)
Affinity DataKi:  5.10nMAssay Description:Inhibition of human recombinant cytosolic carbonic anhydrase 2 preincubated for 10 mins prior to testing by stopped-flow CO2 hydration assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 12(Homo sapiens (Human))
Riga Technical University

Curated by ChEMBL
LigandPNGBDBM50207736(CHEMBL3947437)
Affinity DataKi:  5.20nMAssay Description:Inhibition of human recombinant transmembrane tumor associated carbonic anhydrase 12 preincubated for 10 mins prior to testing by stopped-flow CO2 hy...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 12(Homo sapiens (Human))
Riga Technical University

Curated by ChEMBL
LigandPNGBDBM50271193(CHEMBL4129969)
Affinity DataKi:  5.20nMAssay Description:Inhibition of recombinant human carbonic anhydrase 12 assessed as reduction in CO2 hydration pretreated for 15 mins followed by CO2 addition measured...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 9(Homo sapiens (Human))
Riga Technical University

Curated by ChEMBL
LigandPNGBDBM50207844(CHEMBL3912159)
Affinity DataKi:  5.40nMAssay Description:Inhibition of human recombinant transmembrane tumor associated carbonic anhydrase 9 preincubated for 10 mins prior to testing by stopped-flow CO2 hyd...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 2(Homo sapiens (Human))
Riga Technical University

Curated by ChEMBL
LigandPNGBDBM50207843(CHEMBL3956141)
Affinity DataKi:  5.5nMAssay Description:Inhibition of human recombinant cytosolic carbonic anhydrase 2 preincubated for 10 mins prior to testing by stopped-flow CO2 hydration assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 12(Homo sapiens (Human))
Riga Technical University

Curated by ChEMBL
LigandPNGBDBM10880(AZA | AZA2 | AZM acetazolamide | Acerazolamide, AA...)
Affinity DataKi:  5.60nMAssay Description:Inhibition of human recombinant transmembrane tumor associated carbonic anhydrase 12 preincubated for 10 mins prior to testing by stopped-flow CO2 hy...More data for this Ligand-Target Pair
TargetCarbonic anhydrase 12(Homo sapiens (Human))
Riga Technical University

Curated by ChEMBL
LigandPNGBDBM10880(AZA | AZA2 | AZM acetazolamide | Acerazolamide, AA...)
Affinity DataKi:  5.60nMAssay Description:Inhibition of recombinant human carbonic anhydrase-12 assessed as reduction in CO2 hydration preincubated for 10 mins measured for 5 to 10 secs by st...More data for this Ligand-Target Pair
TargetCarbonic anhydrase 12(Homo sapiens (Human))
Riga Technical University

Curated by ChEMBL
LigandPNGBDBM10880(AZA | AZA2 | AZM acetazolamide | Acerazolamide, AA...)
Affinity DataKi:  5.70nMAssay Description:Inhibition of recombinant human carbonic anhydrase 12 assessed as reduction in CO2 hydration pretreated for 15 mins followed by CO2 addition measured...More data for this Ligand-Target Pair
TargetCarbonic anhydrase 12(Homo sapiens (Human))
Riga Technical University

Curated by ChEMBL
LigandPNGBDBM50207815(CHEMBL3977311)
Affinity DataKi:  5.90nMAssay Description:Inhibition of human recombinant transmembrane tumor associated carbonic anhydrase 12 preincubated for 10 mins prior to testing by stopped-flow CO2 hy...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 9(Homo sapiens (Human))
Riga Technical University

Curated by ChEMBL
LigandPNGBDBM50207843(CHEMBL3956141)
Affinity DataKi:  6.10nMAssay Description:Inhibition of human recombinant transmembrane tumor associated carbonic anhydrase 9 preincubated for 10 mins prior to testing by stopped-flow CO2 hyd...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 12(Homo sapiens (Human))
Riga Technical University

Curated by ChEMBL
LigandPNGBDBM50271194(CHEMBL4127617)
Affinity DataKi:  6.20nMAssay Description:Inhibition of recombinant human carbonic anhydrase 12 assessed as reduction in CO2 hydration pretreated for 15 mins followed by CO2 addition measured...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 12(Homo sapiens (Human))
Riga Technical University

Curated by ChEMBL
LigandPNGBDBM50271182(CHEMBL4129897)
Affinity DataKi:  6.30nMAssay Description:Inhibition of recombinant human carbonic anhydrase 12 assessed as reduction in CO2 hydration pretreated for 15 mins followed by CO2 addition measured...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 12(Homo sapiens (Human))
Riga Technical University

Curated by ChEMBL
LigandPNGBDBM50271198(CHEMBL4126627)
Affinity DataKi:  6.70nMAssay Description:Inhibition of recombinant human carbonic anhydrase 12 assessed as reduction in CO2 hydration pretreated for 15 mins followed by CO2 addition measured...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 12(Homo sapiens (Human))
Riga Technical University

Curated by ChEMBL
LigandPNGBDBM50271202(CHEMBL4126466)
Affinity DataKi:  6.80nMAssay Description:Inhibition of recombinant human carbonic anhydrase 12 assessed as reduction in CO2 hydration pretreated for 15 mins followed by CO2 addition measured...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 12(Homo sapiens (Human))
Riga Technical University

Curated by ChEMBL
LigandPNGBDBM50271196(CHEMBL4126396)
Affinity DataKi:  6.80nMAssay Description:Inhibition of recombinant human carbonic anhydrase 12 assessed as reduction in CO2 hydration pretreated for 15 mins followed by CO2 addition measured...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 9(Homo sapiens (Human))
Riga Technical University

Curated by ChEMBL
LigandPNGBDBM50207736(CHEMBL3947437)
Affinity DataKi:  7nMAssay Description:Inhibition of human recombinant transmembrane tumor associated carbonic anhydrase 9 preincubated for 10 mins prior to testing by stopped-flow CO2 hyd...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 12(Homo sapiens (Human))
Riga Technical University

Curated by ChEMBL
LigandPNGBDBM50426698(CHEMBL2326518)
Affinity DataKi:  7nMAssay Description:Inhibition of human recombinant transmembrane CA12 catalytic domain after 6 hrs by stopped-flow CO2 hydration methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 9(Homo sapiens (Human))
Riga Technical University

Curated by ChEMBL
LigandPNGBDBM50207842(CHEMBL3939285)
Affinity DataKi:  7.5nMAssay Description:Inhibition of human recombinant transmembrane tumor associated carbonic anhydrase 9 preincubated for 10 mins prior to testing by stopped-flow CO2 hyd...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 12(Homo sapiens (Human))
Riga Technical University

Curated by ChEMBL
LigandPNGBDBM50207844(CHEMBL3912159)
Affinity DataKi:  7.80nMAssay Description:Inhibition of human recombinant transmembrane tumor associated carbonic anhydrase 12 preincubated for 10 mins prior to testing by stopped-flow CO2 hy...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 12(Homo sapiens (Human))
Riga Technical University

Curated by ChEMBL
LigandPNGBDBM50207845(CHEMBL3968822)
Affinity DataKi:  8.20nMAssay Description:Inhibition of human recombinant transmembrane tumor associated carbonic anhydrase 12 preincubated for 10 mins prior to testing by stopped-flow CO2 hy...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 9(Homo sapiens (Human))
Riga Technical University

Curated by ChEMBL
LigandPNGBDBM50207815(CHEMBL3977311)
Affinity DataKi:  8.30nMAssay Description:Inhibition of human recombinant transmembrane tumor associated carbonic anhydrase 9 preincubated for 10 mins prior to testing by stopped-flow CO2 hyd...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 12(Homo sapiens (Human))
Riga Technical University

Curated by ChEMBL
LigandPNGBDBM50207738(CHEMBL3922422)
Affinity DataKi:  8.40nMAssay Description:Inhibition of human recombinant transmembrane tumor associated carbonic anhydrase 12 preincubated for 10 mins prior to testing by stopped-flow CO2 hy...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 12(Homo sapiens (Human))
Riga Technical University

Curated by ChEMBL
LigandPNGBDBM50426700(CHEMBL2326516)
Affinity DataKi:  9nMAssay Description:Inhibition of human recombinant transmembrane CA12 catalytic domain after 6 hrs by stopped-flow CO2 hydration methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 2(Homo sapiens (Human))
Riga Technical University

Curated by ChEMBL
LigandPNGBDBM50207738(CHEMBL3922422)
Affinity DataKi:  9.30nMAssay Description:Inhibition of human recombinant cytosolic carbonic anhydrase 2 preincubated for 10 mins prior to testing by stopped-flow CO2 hydration assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 12(Homo sapiens (Human))
Riga Technical University

Curated by ChEMBL
LigandPNGBDBM50242141(CHEMBL4090838)
Affinity DataKi:  10nMAssay Description:Inhibition of recombinant human carbonic anhydrase-12 assessed as reduction in CO2 hydration preincubated for 10 mins measured for 5 to 10 secs by st...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 9(Homo sapiens (Human))
Riga Technical University

Curated by ChEMBL
LigandPNGBDBM50207845(CHEMBL3968822)
Affinity DataKi:  11nMAssay Description:Inhibition of human recombinant transmembrane tumor associated carbonic anhydrase 9 preincubated for 10 mins prior to testing by stopped-flow CO2 hyd...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 9(Homo sapiens (Human))
Riga Technical University

Curated by ChEMBL
LigandPNGBDBM50207738(CHEMBL3922422)
Affinity DataKi:  11nMAssay Description:Inhibition of human recombinant transmembrane tumor associated carbonic anhydrase 9 preincubated for 10 mins prior to testing by stopped-flow CO2 hyd...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 9(Homo sapiens (Human))
Riga Technical University

Curated by ChEMBL
LigandPNGBDBM50207737(CHEMBL3928543)
Affinity DataKi:  11nMAssay Description:Inhibition of human recombinant transmembrane tumor associated carbonic anhydrase 9 preincubated for 10 mins prior to testing by stopped-flow CO2 hyd...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 12(Homo sapiens (Human))
Riga Technical University

Curated by ChEMBL
LigandPNGBDBM50426702(CHEMBL2326514)
Affinity DataKi:  12nMAssay Description:Inhibition of human recombinant transmembrane CA12 catalytic domain after 6 hrs by stopped-flow CO2 hydration methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 2(Homo sapiens (Human))
Riga Technical University

Curated by ChEMBL
LigandPNGBDBM10880(AZA | AZA2 | AZM acetazolamide | Acerazolamide, AA...)
Affinity DataKi:  12nMAssay Description:Inhibition of full length human recombinant CA2 cytosolic isoform after 6 hrs by stopped-flow CO2 hydration methodMore data for this Ligand-Target Pair
TargetCarbonic anhydrase 2(Homo sapiens (Human))
Riga Technical University

Curated by ChEMBL
LigandPNGBDBM10880(AZA | AZA2 | AZM acetazolamide | Acerazolamide, AA...)
Affinity DataKi:  12nMAssay Description:Inhibition of human recombinant cytosolic carbonic anhydrase 2 preincubated for 10 mins prior to testing by stopped-flow CO2 hydration assayMore data for this Ligand-Target Pair
TargetCarbonic anhydrase 12(Homo sapiens (Human))
Riga Technical University

Curated by ChEMBL
LigandPNGBDBM50271184(CHEMBL4128603)
Affinity DataKi:  12nMAssay Description:Inhibition of recombinant human carbonic anhydrase 12 assessed as reduction in CO2 hydration pretreated for 15 mins followed by CO2 addition measured...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 2(Homo sapiens (Human))
Riga Technical University

Curated by ChEMBL
LigandPNGBDBM10880(AZA | AZA2 | AZM acetazolamide | Acerazolamide, AA...)
Affinity DataKi:  12nMAssay Description:Inhibition of recombinant human carbonic anhydrase-2 assessed as reduction in CO2 hydration preincubated for 10 mins measured for 5 to 10 secs by sto...More data for this Ligand-Target Pair
TargetCarbonic anhydrase 2(Homo sapiens (Human))
Riga Technical University

Curated by ChEMBL
LigandPNGBDBM10880(AZA | AZA2 | AZM acetazolamide | Acerazolamide, AA...)
Affinity DataKi:  12nMAssay Description:Inhibition of recombinant human carbonic anhydrase 2 assessed as reduction in CO2 hydration pretreated for 15 mins followed by CO2 addition measured ...More data for this Ligand-Target Pair
TargetCarbonic anhydrase 12(Homo sapiens (Human))
Riga Technical University

Curated by ChEMBL
LigandPNGBDBM50426695(CHEMBL2326521)
Affinity DataKi:  13nMAssay Description:Inhibition of human recombinant transmembrane CA12 catalytic domain after 6 hrs by stopped-flow CO2 hydration methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 12(Homo sapiens (Human))
Riga Technical University

Curated by ChEMBL
LigandPNGBDBM50426701(CHEMBL2326515)
Affinity DataKi:  13nMAssay Description:Inhibition of human recombinant transmembrane CA12 catalytic domain after 6 hrs by stopped-flow CO2 hydration methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 12(Homo sapiens (Human))
Riga Technical University

Curated by ChEMBL
LigandPNGBDBM50207842(CHEMBL3939285)
Affinity DataKi:  13nMAssay Description:Inhibition of human recombinant transmembrane tumor associated carbonic anhydrase 12 preincubated for 10 mins prior to testing by stopped-flow CO2 hy...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 12(Homo sapiens (Human))
Riga Technical University

Curated by ChEMBL
LigandPNGBDBM50207819(CHEMBL3894409)
Affinity DataKi:  13nMAssay Description:Inhibition of human recombinant transmembrane tumor associated carbonic anhydrase 12 preincubated for 10 mins prior to testing by stopped-flow CO2 hy...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 12(Homo sapiens (Human))
Riga Technical University

Curated by ChEMBL
LigandPNGBDBM50207843(CHEMBL3956141)
Affinity DataKi:  13nMAssay Description:Inhibition of human recombinant transmembrane tumor associated carbonic anhydrase 12 preincubated for 10 mins prior to testing by stopped-flow CO2 hy...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 12(Homo sapiens (Human))
Riga Technical University

Curated by ChEMBL
LigandPNGBDBM50426697(CHEMBL2326519)
Affinity DataKi:  14nMAssay Description:Inhibition of human recombinant transmembrane CA12 catalytic domain after 6 hrs by stopped-flow CO2 hydration methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 12(Homo sapiens (Human))
Riga Technical University

Curated by ChEMBL
LigandPNGBDBM50426699(CHEMBL2326517)
Affinity DataKi:  16nMAssay Description:Inhibition of human recombinant transmembrane CA12 catalytic domain after 6 hrs by stopped-flow CO2 hydration methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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