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Found 41 with Last Name = 'kende' and Initial = 'as'
TargetThromboxane A2 receptor(Homo sapiens (Human))
Procter & Gamble Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50035622((5Z,13E,15S)-9alpha,11alpha,15-trihydroxyprosta-5,...)
Affinity DataIC50: >0.00100nMAssay Description:In vitro binding of the compound at TP human prostaglandin receptor using [3H]-SQ-29,548 as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin F2-alpha receptor(Homo sapiens (Human))
Procter & Gamble Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50106547(7-[3,5-Dihydroxy-2-(3-hydroxy-4-phenoxy-but-1-enyl...)
Affinity DataIC50:  2nMAssay Description:In vitro binding of the compound at FP human prostaglandin receptor using [3H]-PGF-2 alpha as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin F2-alpha receptor(Homo sapiens (Human))
Procter & Gamble Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50035622((5Z,13E,15S)-9alpha,11alpha,15-trihydroxyprosta-5,...)
Affinity DataIC50:  3nMAssay Description:In vitro binding of the compound at FP human prostaglandin receptor using [3H]-PGF-2 alpha as radioligandMore data for this Ligand-Target Pair
TargetProstaglandin E2 receptor EP1 subtype(Homo sapiens (Human))
Procter & Gamble Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50106547(7-[3,5-Dihydroxy-2-(3-hydroxy-4-phenoxy-but-1-enyl...)
Affinity DataIC50:  38nMAssay Description:Functional activity in RAT-1 cells, transiently transfected with human prostaglandin EP1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin F2-alpha receptor(Homo sapiens (Human))
Procter & Gamble Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50106548(CHEMBL440164 | {6-[3,5-Dihydroxy-2-(3-hydroxy-4-ph...)
Affinity DataIC50:  42nMAssay Description:In vitro binding of the compound at FP human prostaglandin receptor using [3H]-PGF-2 alpha as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin E2 receptor EP3 subtype(Homo sapiens (Human))
Procter & Gamble Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50035622((5Z,13E,15S)-9alpha,11alpha,15-trihydroxyprosta-5,...)
Affinity DataIC50:  110nMAssay Description:In vitro binding of the compound at EP3 human prostaglandin receptor using [3H]-PGE-2 as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin F2-alpha receptor(Homo sapiens (Human))
Procter & Gamble Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50106546(CHEMBL134546 | {6-[3,5-Dihydroxy-2-(3-hydroxy-oct-...)
Affinity DataIC50:  114nMAssay Description:In vitro binding of the compound at FP human prostaglandin receptor using [3H]-PGF-2 alpha as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin E2 receptor EP3 subtype(Homo sapiens (Human))
Procter & Gamble Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50106547(7-[3,5-Dihydroxy-2-(3-hydroxy-4-phenoxy-but-1-enyl...)
Affinity DataIC50:  186nMAssay Description:Functional activity in RAT-1 cells, transiently transfected with human prostaglandin EP3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin E2 receptor EP1 subtype(Homo sapiens (Human))
Procter & Gamble Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50035622((5Z,13E,15S)-9alpha,11alpha,15-trihydroxyprosta-5,...)
Affinity DataIC50:  220nMAssay Description:In vitro binding of the compound at EP1 human prostaglandin receptor using [3H]-PGE-2 as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin F2-alpha receptor(Homo sapiens (Human))
Procter & Gamble Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50106549(CHEMBL336781 | {6-[3,5-Dihydroxy-2-(3-hydroxy-oct-...)
Affinity DataIC50:  311nMAssay Description:In vitro binding of the compound at FP human prostaglandin receptor using [3H]-PGF-2 alpha as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThromboxane A2 receptor(Homo sapiens (Human))
Procter & Gamble Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50106547(7-[3,5-Dihydroxy-2-(3-hydroxy-4-phenoxy-but-1-enyl...)
Affinity DataIC50:  510nMAssay Description:Functional activity in RAT-1 cells, transiently transfected with human prostaglandin TP receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin F2-alpha receptor(Homo sapiens (Human))
Procter & Gamble Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50106553(CHEMBL336543 | {6-[3,5-Dihydroxy-2-(3-hydroxy-oct-...)
Affinity DataIC50:  1.00E+3nMAssay Description:In vitro binding of the compound at FP human prostaglandin receptor using [3H]- PGF-2 alpha as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin F2-alpha receptor(Homo sapiens (Human))
Procter & Gamble Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50106552(CHEMBL133945 | {6-[3,5-Dihydroxy-2-(3-hydroxy-oct-...)
Affinity DataIC50:  4.10E+3nMAssay Description:In vitro binding of the compound at FP human prostaglandin receptor using [3H]-PGF-2 alpha as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin E2 receptor EP4 subtype(Homo sapiens (Human))
Procter & Gamble Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50035622((5Z,13E,15S)-9alpha,11alpha,15-trihydroxyprosta-5,...)
Affinity DataIC50:  4.20E+3nMAssay Description:In vitro binding of the compound at EP4 human prostaglandin receptor using [3H]-PGE-2 as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin D2 receptor(Homo sapiens (Human))
Procter & Gamble Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50035622((5Z,13E,15S)-9alpha,11alpha,15-trihydroxyprosta-5,...)
Affinity DataIC50:  4.50E+3nMAssay Description:In vitro binding of the compound at DP human prostaglandin receptor using [3H]- PGD-2 as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin F2-alpha receptor(Homo sapiens (Human))
Procter & Gamble Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50106551(Butyl-{6-[3,5-dihydroxy-2-(3-hydroxy-oct-1-enyl)-c...)
Affinity DataIC50:  6.70E+3nMAssay Description:In vitro binding of the compound at FP human prostaglandin receptor using [3H]-PGF-2 alpha as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin E2 receptor EP2 subtype(Homo sapiens (Human))
Procter & Gamble Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50106546(CHEMBL134546 | {6-[3,5-Dihydroxy-2-(3-hydroxy-oct-...)
Affinity DataIC50: >1.00E+4nMAssay Description:In vitro binding of the compound at EP2 human prostaglandin receptor using [3H]-PGE-2 as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThromboxane A2 receptor(Homo sapiens (Human))
Procter & Gamble Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50106548(CHEMBL440164 | {6-[3,5-Dihydroxy-2-(3-hydroxy-4-ph...)
Affinity DataIC50: >1.00E+4nMAssay Description:In vitro binding of the compound at TP human prostaglandin receptor using [3H]-SQ-29,548 as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin E2 receptor EP1 subtype(Homo sapiens (Human))
Procter & Gamble Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50106548(CHEMBL440164 | {6-[3,5-Dihydroxy-2-(3-hydroxy-4-ph...)
Affinity DataIC50: >1.00E+4nMAssay Description:In vitro binding of the compound at EP1 human prostaglandin receptor using [3H]-PGE-2 as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin F2-alpha receptor(Homo sapiens (Human))
Procter & Gamble Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50106550(CHEMBL334810 | {6-[3,5-Dihydroxy-2-(3-hydroxy-oct-...)
Affinity DataIC50: >1.00E+4nMAssay Description:In vitro binding of the compound at FP human prostaglandin receptor using [3H]- PGF-2 alpha as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin E2 receptor EP3 subtype(Homo sapiens (Human))
Procter & Gamble Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50106548(CHEMBL440164 | {6-[3,5-Dihydroxy-2-(3-hydroxy-4-ph...)
Affinity DataIC50: >1.00E+4nMAssay Description:In vitro binding of the compound at EP3 human prostaglandin receptor using [3H]-PGE-2 as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin D2 receptor(Homo sapiens (Human))
Procter & Gamble Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50106548(CHEMBL440164 | {6-[3,5-Dihydroxy-2-(3-hydroxy-4-ph...)
Affinity DataIC50: >1.00E+4nMAssay Description:In vitro binding of the compound at DP human prostaglandin receptor using [3H]- PGD-2 as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin E2 receptor EP3 subtype(Homo sapiens (Human))
Procter & Gamble Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50106546(CHEMBL134546 | {6-[3,5-Dihydroxy-2-(3-hydroxy-oct-...)
Affinity DataIC50: >1.00E+4nMAssay Description:In vitro binding of the compound at EP3 human prostaglandin receptor using [3H]-PGE-2 as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin E2 receptor EP1 subtype(Homo sapiens (Human))
Procter & Gamble Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50106546(CHEMBL134546 | {6-[3,5-Dihydroxy-2-(3-hydroxy-oct-...)
Affinity DataIC50: >1.00E+4nMAssay Description:In vitro binding of the compound at EP1 human prostaglandin receptor using [3H]-PGE-2 as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin E2 receptor EP2 subtype(Homo sapiens (Human))
Procter & Gamble Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50106548(CHEMBL440164 | {6-[3,5-Dihydroxy-2-(3-hydroxy-4-ph...)
Affinity DataIC50: >1.00E+4nMAssay Description:In vitro binding of the compound at EP2 human prostaglandin receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstacyclin receptor(Homo sapiens (Human))
Procter & Gamble Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50106548(CHEMBL440164 | {6-[3,5-Dihydroxy-2-(3-hydroxy-4-ph...)
Affinity DataIC50: >1.00E+4nMAssay Description:In vitro binding of the compound at prostanoid IP receptor using [3H]-Iloprost as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstacyclin receptor(Homo sapiens (Human))
Procter & Gamble Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50106546(CHEMBL134546 | {6-[3,5-Dihydroxy-2-(3-hydroxy-oct-...)
Affinity DataIC50: >1.00E+4nMAssay Description:In vitro binding of the compound at prostanoid IP receptor using [3H]-Iloprost as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThromboxane A2 receptor(Homo sapiens (Human))
Procter & Gamble Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50106546(CHEMBL134546 | {6-[3,5-Dihydroxy-2-(3-hydroxy-oct-...)
Affinity DataIC50: >1.00E+4nMAssay Description:In vitro binding of the compound at TP human prostaglandin receptor using [3H]-SQ-29,548 as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin D2 receptor(Homo sapiens (Human))
Procter & Gamble Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50106546(CHEMBL134546 | {6-[3,5-Dihydroxy-2-(3-hydroxy-oct-...)
Affinity DataIC50: >1.00E+4nMAssay Description:In vitro binding of the compound at DP human prostaglandin receptor using [3H]- PGD-2 as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin E2 receptor EP4 subtype(Homo sapiens (Human))
Procter & Gamble Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50106546(CHEMBL134546 | {6-[3,5-Dihydroxy-2-(3-hydroxy-oct-...)
Affinity DataIC50: >1.00E+4nMAssay Description:In vitro binding of the compound at EP4 human prostaglandin receptor using [3H]-PGE-2 as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin E2 receptor EP4 subtype(Homo sapiens (Human))
Procter & Gamble Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50106548(CHEMBL440164 | {6-[3,5-Dihydroxy-2-(3-hydroxy-4-ph...)
Affinity DataIC50: >1.00E+4nMAssay Description:In vitro binding of the compound at EP4 human prostaglandin receptor using [3H]-PGE-2 as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin E2 receptor EP2 subtype(Homo sapiens (Human))
Procter & Gamble Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50035622((5Z,13E,15S)-9alpha,11alpha,15-trihydroxyprosta-5,...)
Affinity DataIC50: >1.00E+5nMAssay Description:In vitro binding of the compound at EP2 human prostaglandin receptor using [3H]-PGE-2 as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstacyclin receptor(Homo sapiens (Human))
Procter & Gamble Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50035622((5Z,13E,15S)-9alpha,11alpha,15-trihydroxyprosta-5,...)
Affinity DataIC50: >1.00E+5nMAssay Description:In vitro binding of the compound at prostanoid IP receptor using [3H]-Iloprost as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMedDrugBank

TargetAryl hydrocarbon receptor(Mus musculus (Mouse))
University of Wisconsin

LigandPNGBDBM92708(Photoaffinity ligand, 5)
Affinity DataKd:  13nMpH: 7.5 T: 2°CAssay Description:The equilibrium dissocation constants, KD values for the photoaffinity ligands were determined by a competitive binding assay. More data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails PubMed
TargetAryl hydrocarbon receptor(Mus musculus (Mouse))
University of Wisconsin

LigandPNGBDBM92711(Photoaffinity ligand, 8)
Affinity DataKd:  11nMpH: 7.5 T: 2°CAssay Description:The equilibrium dissocation constants, KD values for the photoaffinity ligands were determined by a competitive binding assay. More data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails PubMed
TargetAryl hydrocarbon receptor(Mus musculus (Mouse))
University of Wisconsin

LigandPNGBDBM92704(Photoaffinity ligand, 1)
Affinity DataKd:  0.440nMpH: 7.5 T: 2°CAssay Description:The equilibrium dissocation constants, KD values for the photoaffinity ligands were determined by a competitive binding assay. More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetAryl hydrocarbon receptor(Mus musculus (Mouse))
University of Wisconsin

LigandPNGBDBM92706(Photoaffinity ligand, 3)
Affinity DataKd:  0.490nMpH: 7.5 T: 2°CAssay Description:The equilibrium dissocation constants, KD values for the photoaffinity ligands were determined by a competitive binding assay. More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetAryl hydrocarbon receptor(Mus musculus (Mouse))
University of Wisconsin

LigandPNGBDBM92710(Photoaffinity ligand, 7)
Affinity DataKd:  113nMpH: 7.5 T: 2°CAssay Description:The equilibrium dissocation constants, KD values for the photoaffinity ligands were determined by a competitive binding assay. More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetAryl hydrocarbon receptor(Mus musculus (Mouse))
University of Wisconsin

LigandPNGBDBM92705(Photoaffinity ligand, 2)
Affinity DataKd:  2.10nMpH: 7.5 T: 2°CAssay Description:The equilibrium dissocation constants, KD values for the photoaffinity ligands were determined by a competitive binding assay. More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetAryl hydrocarbon receptor(Mus musculus (Mouse))
University of Wisconsin

LigandPNGBDBM92709(Photoaffinity ligand, 6)
Affinity DataKd:  8.10nMpH: 7.5 T: 2°CAssay Description:The equilibrium dissocation constants, KD values for the photoaffinity ligands were determined by a competitive binding assay. More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetAryl hydrocarbon receptor(Mus musculus (Mouse))
University of Wisconsin

LigandPNGBDBM92707(Photoaffinity ligand, 4)
Affinity DataKd:  0.760nMpH: 7.5 T: 2°CAssay Description:The equilibrium dissocation constants, KD values for the photoaffinity ligands were determined by a competitive binding assay. More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed