TargetMelatonin receptor type 1A(Homo sapiens (Human))
Glaxo Wellcome Research and Development
Curated by PDSP Ki Database
Glaxo Wellcome Research and Development
Curated by PDSP Ki Database
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Nida Addiction Research Center
Curated by PDSP Ki Database
Nida Addiction Research Center
Curated by PDSP Ki Database
TargetMelatonin receptor type 1A(GUINEA PIG)
Glaxo Wellcome Research and Development
Curated by PDSP Ki Database
Glaxo Wellcome Research and Development
Curated by PDSP Ki Database
TargetMelatonin receptor type 1B(Homo sapiens (Human))
Glaxo Wellcome Research and Development
Curated by PDSP Ki Database
Glaxo Wellcome Research and Development
Curated by PDSP Ki Database
TargetMelatonin receptor type 1B(Homo sapiens (Human))
Glaxo Wellcome Research and Development
Curated by PDSP Ki Database
Glaxo Wellcome Research and Development
Curated by PDSP Ki Database
TargetMelatonin receptor type 1A(Homo sapiens (Human))
Glaxo Wellcome Research and Development
Curated by PDSP Ki Database
Glaxo Wellcome Research and Development
Curated by PDSP Ki Database
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Nida Addiction Research Center
Curated by PDSP Ki Database
Nida Addiction Research Center
Curated by PDSP Ki Database
TargetMelatonin receptor type 1A(GUINEA PIG)
Glaxo Wellcome Research and Development
Curated by PDSP Ki Database
Glaxo Wellcome Research and Development
Curated by PDSP Ki Database
TargetMelatonin receptor type 1B(Homo sapiens (Human))
Glaxo Wellcome Research and Development
Curated by PDSP Ki Database
Glaxo Wellcome Research and Development
Curated by PDSP Ki Database
TargetMelatonin receptor type 1A(Homo sapiens (Human))
Glaxo Wellcome Research and Development
Curated by PDSP Ki Database
Glaxo Wellcome Research and Development
Curated by PDSP Ki Database
TargetMelatonin receptor type 1A(GUINEA PIG)
Glaxo Wellcome Research and Development
Curated by PDSP Ki Database
Glaxo Wellcome Research and Development
Curated by PDSP Ki Database
TargetMelatonin receptor type 1A(GUINEA PIG)
Glaxo Wellcome Research and Development
Curated by PDSP Ki Database
Glaxo Wellcome Research and Development
Curated by PDSP Ki Database
Target5-hydroxytryptamine receptor 1D(Homo sapiens (Human))
Glaxo Research and Development
Curated by PDSP Ki Database
Glaxo Research and Development
Curated by PDSP Ki Database
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Nida Addiction Research Center
Curated by PDSP Ki Database
Nida Addiction Research Center
Curated by PDSP Ki Database
TargetMelatonin receptor type 1B(Homo sapiens (Human))
Glaxo Wellcome Research and Development
Curated by PDSP Ki Database
Glaxo Wellcome Research and Development
Curated by PDSP Ki Database
TargetMelatonin receptor type 1A(Homo sapiens (Human))
Glaxo Wellcome Research and Development
Curated by PDSP Ki Database
Glaxo Wellcome Research and Development
Curated by PDSP Ki Database
TargetMelatonin receptor type 1B(Homo sapiens (Human))
Glaxo Wellcome Research and Development
Curated by PDSP Ki Database
Glaxo Wellcome Research and Development
Curated by PDSP Ki Database
TargetMelatonin receptor type 1B(Homo sapiens (Human))
Glaxo Wellcome Research and Development
Curated by PDSP Ki Database
Glaxo Wellcome Research and Development
Curated by PDSP Ki Database
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Nida Addiction Research Center
Curated by PDSP Ki Database
Nida Addiction Research Center
Curated by PDSP Ki Database
TargetMelatonin receptor type 1A(GUINEA PIG)
Glaxo Wellcome Research and Development
Curated by PDSP Ki Database
Glaxo Wellcome Research and Development
Curated by PDSP Ki Database
TargetMelatonin receptor type 1A(GUINEA PIG)
Glaxo Wellcome Research and Development
Curated by PDSP Ki Database
Glaxo Wellcome Research and Development
Curated by PDSP Ki Database
TargetMelatonin receptor type 1A(GUINEA PIG)
Glaxo Wellcome Research and Development
Curated by PDSP Ki Database
Glaxo Wellcome Research and Development
Curated by PDSP Ki Database
TargetMelatonin receptor type 1B(Homo sapiens (Human))
Glaxo Wellcome Research and Development
Curated by PDSP Ki Database
Glaxo Wellcome Research and Development
Curated by PDSP Ki Database
TargetMelatonin receptor type 1B(Homo sapiens (Human))
Glaxo Wellcome Research and Development
Curated by PDSP Ki Database
Glaxo Wellcome Research and Development
Curated by PDSP Ki Database
TargetMelatonin receptor type 1A(GUINEA PIG)
Glaxo Wellcome Research and Development
Curated by PDSP Ki Database
Glaxo Wellcome Research and Development
Curated by PDSP Ki Database
Affinity DataKi: <0.5nMAssay Description:Inhibition of FAM-labeled ZBA248 binding to recombinant human N-terminal His6-tagged BRD4 bromodomain 2 (333 to 460 residues) expressed in Rosetta2 D...More data for this Ligand-Target Pair
Affinity DataKi: <0.5nMAssay Description:Inhibition of FAM-labeled ZBA248 binding to recombinant human N-terminal His6-tagged BRD4 bromodomain 1 (44 to 168 residues) expressed in Rosetta2 DE...More data for this Ligand-Target Pair
Affinity DataKi: <0.5nMAssay Description:Inhibition of FAM-labeled ZBA248 binding to recombinant human N-terminal His6-tagged BRD4 bromodomain 1 (44 to 168 residues) expressed in Rosetta2 DE...More data for this Ligand-Target Pair
Affinity DataKi: 0.5nMAssay Description:Inhibition of FAM-labeled ZBA248 binding to recombinant human BRD4 bromodomain 1 (44 to 168 residues) expressed in Rosetta2 Escherichia coli DE3 cell...More data for this Ligand-Target Pair
Affinity DataKi: <0.5nMAssay Description:Inhibition of FAM-labeled ZBA248 binding to recombinant human N-terminal His6-tagged BRD4 bromodomain 1 (44 to 168 residues) expressed in Rosetta2 DE...More data for this Ligand-Target Pair
TargetMelatonin receptor type 1A(Homo sapiens (Human))
Glaxo Wellcome Research and Development
Curated by PDSP Ki Database
Glaxo Wellcome Research and Development
Curated by PDSP Ki Database
Affinity DataKi: 0.590nMAssay Description:Inhibition of human bradykinin B1 receptorMore data for this Ligand-Target Pair
TargetMelatonin receptor type 1A(GUINEA PIG)
Glaxo Wellcome Research and Development
Curated by PDSP Ki Database
Glaxo Wellcome Research and Development
Curated by PDSP Ki Database
TargetBromodomain-containing protein 3 [326-398](Homo sapiens (Human))
The Regents of The University of Michigan
US Patent
The Regents of The University of Michigan
US Patent
Affinity DataKi: 0.650nM ΔG°: -52.4kJ/moleT: 2°CAssay Description:Fluorescence Polarization (FP) competitive binding studies (see above) were carried out using the FAM labeled fluorescent probe Cpd. No. 350 to deter...More data for this Ligand-Target Pair
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Nida Addiction Research Center
Curated by PDSP Ki Database
Nida Addiction Research Center
Curated by PDSP Ki Database
TargetMelatonin receptor type 1A(Homo sapiens (Human))
Glaxo Wellcome Research and Development
Curated by PDSP Ki Database
Glaxo Wellcome Research and Development
Curated by PDSP Ki Database
Affinity DataKi: 0.700nMAssay Description:Inhibition of FAM-labeled ZBA248 binding to recombinant human N-terminal His6-tagged BRD4 bromodomain 2 (333 to 460 residues) expressed in Rosetta2 D...More data for this Ligand-Target Pair
Affinity DataKi: 0.700nMAssay Description:Inhibition of FAM-labeled ZBA248 binding to recombinant human BRD4 bromodomain 1 (44 to 168 residues) expressed in Rosetta2 Escherichia coli DE3 cell...More data for this Ligand-Target Pair
TargetMelatonin receptor type 1A(GUINEA PIG)
Glaxo Wellcome Research and Development
Curated by PDSP Ki Database
Glaxo Wellcome Research and Development
Curated by PDSP Ki Database
Affinity DataKi: 0.800nMAssay Description:Binding affinity to N-terminus 6X His-tagged human Bcl2 expressed in Escherichia coli BL21 (DE3) cells after 2 hrs by fluorescence polarization assayMore data for this Ligand-Target Pair
Affinity DataKi: 0.800nMAssay Description:Binding affinity to N-terminal 6xHis-tagged human Bcl-2 expressed in Escherichia coli BL21 (DE3) after 2 hrs by fluorescence polarization assayMore data for this Ligand-Target Pair
Affinity DataKi: 0.800nMAssay Description:Inhibition of FAM-labeled ZBA248 binding to recombinant human BRD4 bromodomain 1 (44 to 168 residues) expressed in Rosetta2 Escherichia coli DE3 cell...More data for this Ligand-Target Pair
Affinity DataKi: 0.800nMAssay Description:Inhibition of FAM-labeled ZBA248 binding to recombinant human BRD4 bromodomain 1 (44 to 168 residues) expressed in Rosetta2 Escherichia coli DE3 cell...More data for this Ligand-Target Pair
Affinity DataKi: 0.800nMAssay Description:Inhibition of FAM-labeled ZBA248 binding to recombinant human N-terminal His6-tagged BRD4 bromodomain 1 (44 to 168 residues) expressed in Rosetta2 DE...More data for this Ligand-Target Pair
TargetBromodomain-containing protein 3 [326-398](Homo sapiens (Human))
The Regents of The University of Michigan
US Patent
The Regents of The University of Michigan
US Patent
Affinity DataKi: 0.820nM ΔG°: -51.9kJ/moleT: 2°CAssay Description:Fluorescence Polarization (FP) competitive binding studies (see above) were carried out using the FAM labeled fluorescent probe Cpd. No. 350 to deter...More data for this Ligand-Target Pair
Affinity DataKi: 0.900nMAssay Description:Inhibition of FAM-labeled ZBA248 binding to recombinant human N-terminal His6-tagged BRD4 bromodomain 2 (333 to 460 residues) expressed in Rosetta2 D...More data for this Ligand-Target Pair
Affinity DataKi: 0.920nMAssay Description:Compound was tested for inhibition against rat Bradykinin receptor B1More data for this Ligand-Target Pair
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Nida Addiction Research Center
Curated by PDSP Ki Database
Nida Addiction Research Center
Curated by PDSP Ki Database
TargetBromodomain-containing protein 3 [326-398](Homo sapiens (Human))
The Regents of The University of Michigan
US Patent
The Regents of The University of Michigan
US Patent
Affinity DataKi: 1nM ΔG°: -51.4kJ/moleT: 2°CAssay Description:Fluorescence Polarization (FP) competitive binding studies (see above) were carried out using the FAM labeled fluorescent probe Cpd. No. 350 to deter...More data for this Ligand-Target Pair
Affinity DataKi: 1nMAssay Description:Inhibition of FAM-probe binding to Menin (unknown origin) after 60 mins by fluorescence polarization competitive binding assayMore data for this Ligand-Target Pair