Affinity DataIC50: 0.110nMAssay Description:Binding affinity to human HCK using KVEKIGEGTYGVVYK as substrate by radiometric hotspot kinase assayMore data for this Ligand-Target Pair
Affinity DataIC50: 0.160nMAssay Description:Binding affinity to LYN (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 0.280nMAssay Description:Binding affinity to human LCK using poly[Glu:Tyr] (4:1) as substrate by radiometric hotspot kinase assayMore data for this Ligand-Target Pair
Affinity DataIC50: 0.360nMAssay Description:Binding affinity to human FYN using poly[Glu:Tyr] (4:1) as substrate by radiometric hotspot kinase assayMore data for this Ligand-Target Pair
Affinity DataIC50: 0.370nMAssay Description:Binding affinity to human ABL1 using EAIYAAPFAKKK as substrate by radiometric hotspot kinase assayMore data for this Ligand-Target Pair
Affinity DataIC50: 0.890nMAssay Description:Binding affinity to human YES using poly[Glu:Tyr] (4:1) as substrate by radiometric hotspot kinase assayMore data for this Ligand-Target Pair
Affinity DataIC50: 1nMAssay Description:Inhibition of LTA4 hydrolase (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 1.10nMAssay Description:Binding affinity to human PDGFRalpha using poly[Glu:Tyr] (4:1) as substrate by radiometric hotspot kinase assayMore data for this Ligand-Target Pair
Affinity DataIC50: 1.30nMAssay Description:Binding affinity to human FRK using poly[Glu:Tyr] (4:1) as substrate by radiometric hotspot kinase assayMore data for this Ligand-Target Pair
Affinity DataIC50: 1.80nMAssay Description:LTB4 formed was quantified with the HTRF assay in which free LTB4 competes with LTB4-XL665 conjugate (acceptor) for anti-LTB4 monoclonal antibody lab...More data for this Ligand-Target Pair
Affinity DataIC50: 2nMAssay Description:Inhibition of LTA4 hydrolase (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 2.10nMAssay Description:LTB4 formed was quantified with the HTRF assay in which free LTB4 competes with LTB4-XL665 conjugate (acceptor) for anti-LTB4 monoclonal antibody lab...More data for this Ligand-Target Pair
Affinity DataIC50: 2.20nMAssay Description:Binding affinity to human FGFR1 using poly[Glu:Tyr] (4:1) as substrate by radiometric hotspot kinase assayMore data for this Ligand-Target Pair
Affinity DataIC50: 3nMAssay Description:Inhibition of LTA4 hydrolase (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 3nMAssay Description:Inhibition of LTA4 hydrolase (unknown origin) by hydrolase assayMore data for this Ligand-Target Pair
Affinity DataIC50: 3nMAssay Description:Inhibition of LTA4 hydrolase (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 3nMAssay Description:Inhibition of LTA4 hydrolase (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 3nMAssay Description:Inhibition of LTA4 hydrolase (unknown origin) by hydrolase assayMore data for this Ligand-Target Pair
Affinity DataIC50: 3.70nMAssay Description:Binding affinity to FLT1 (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 4nMAssay Description:Inhibition of LTA4 hydrolase (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 4nMAssay Description:Inhibition of LTA4 hydrolase (unknown origin) by hydrolase assayMore data for this Ligand-Target Pair
Affinity DataIC50: 5nMAssay Description:Inhibition of LTA4 hydrolase (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 5nMAssay Description:Inhibition of LTA4 hydrolase (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 5nMAssay Description:Inhibition of LTA4 hydrolase (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 5nMAssay Description:Inhibition of LTA4 hydrolase (unknown origin) by hydrolase assayMore data for this Ligand-Target Pair
Affinity DataIC50: 5.40nMAssay Description:Binding affinity to human SRC using poly[Glu:Tyr] (4:1) as substrate by radiometric hotspot kinase assayMore data for this Ligand-Target Pair
Affinity DataIC50: 6nMAssay Description:Compound potency against the peptidase activity of LTA4 hydrolase was measured by inhibition of the hydrolysis of L-alanine-p-nitroanilide to L-alani...More data for this Ligand-Target Pair
Affinity DataIC50: 6nMAssay Description:Inhibition of LTA4 hydrolase (unknown origin) by hydrolase assayMore data for this Ligand-Target Pair
Affinity DataIC50: 6nMAssay Description:Inhibition of LTA4 hydrolase (unknown origin) by hydrolase assayMore data for this Ligand-Target Pair
Affinity DataIC50: 6nMAssay Description:Inhibition of LTA4 hydrolase (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 6nMAssay Description:Inhibition of LTA4 hydrolase (unknown origin) by hydrolase assayMore data for this Ligand-Target Pair
Affinity DataIC50: 6nMAssay Description:Inhibition of LTA4 hydrolase (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 7nMAssay Description:Inhibition of LTA4 hydrolase (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 7nMAssay Description:Inhibition of LTA4 hydrolase (unknown origin) by hydrolase assayMore data for this Ligand-Target Pair
Affinity DataIC50: 7nMAssay Description:Inhibition of LTA4 hydrolase (unknown origin) by hydrolase assayMore data for this Ligand-Target Pair
Affinity DataIC50: 7nMAssay Description:Inhibition of LTA4 hydrolase (unknown origin) by hydrolase assayMore data for this Ligand-Target Pair
Affinity DataIC50: 7.10nMAssay Description:In brief, the enzyme (29 nM) was incubated with L-alanine-p-nitroanilide (1 mM) in 50 mM HEPES (pH 7.5), 100 mM KCL, 1% DMSO in the absence or presen...More data for this Ligand-Target Pair
Affinity DataIC50: 8nMAssay Description:Inhibition of LTA4 hydrolase (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 9nMAssay Description:Inhibition of LTA4 hydrolase (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 9nMAssay Description:Inhibition of LTA4 hydrolase (unknown origin)More data for this Ligand-Target Pair
TargetEpithelial discoidin domain-containing receptor 1(Homo sapiens (Human))
Promega
Curated by ChEMBL
Promega
Curated by ChEMBL
Affinity DataIC50: 9.40nMAssay Description:Binding affinity to DDR1 (unknown origin) at 5 uMMore data for this Ligand-Target Pair
Affinity DataIC50: <10nMAssay Description:Binding affinity to MAPK14 (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 10nMAssay Description:Inhibition of LTA4 hydrolase (unknown origin) by hydrolase assayMore data for this Ligand-Target Pair
Affinity DataIC50: 11nMAssay Description:Inhibition of LTA4 hydrolase (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 13nMAssay Description:Inhibition of LTA4 hydrolase (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 13nMAssay Description:Binding affinity to human CSK using poly[Glu:Tyr] (4:1) as substrate by radiometric hotspot kinase assayMore data for this Ligand-Target Pair
Affinity DataIC50: 13nMAssay Description:Compound potency against the peptidase activity of LTA4 hydrolase was measured by inhibition of the hydrolysis of L-alanine-p-nitroanilide to L-alani...More data for this Ligand-Target Pair
Affinity DataIC50: 14nMAssay Description:Compound potency against the peptidase activity of LTA4 hydrolase was measured by inhibition of the hydrolysis of L-alanine-p-nitroanilide to L-alani...More data for this Ligand-Target Pair
Affinity DataIC50: 14nMAssay Description:Inhibition of LTA4 hydrolase (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 15nMAssay Description:Inhibition of LTA4 hydrolase (unknown origin)More data for this Ligand-Target Pair