Affinity DataKi: 0.00110nM IC50: 1.00E+3nMAssay Description:Inhibition assay using aromatase enzyme.More data for this Ligand-Target Pair
Affinity DataKi: 0.00182nM IC50: 1.21E+4nMAssay Description:Inhibition assay using aromatase enzyme.More data for this Ligand-Target Pair
Affinity DataKi: 0.00216nMAssay Description:Inhibition assay using aromatase enzyme.More data for this Ligand-Target Pair
Affinity DataKi: 0.00256nMAssay Description:Inhibition assay using aromatase enzyme.More data for this Ligand-Target Pair
Affinity DataKi: 0.00425nMAssay Description:Inhibition assay using aromatase enzyme.More data for this Ligand-Target Pair
Affinity DataKi: 0.00597nMAssay Description:Inhibition assay using aromatase enzyme.More data for this Ligand-Target Pair
Affinity DataKi: 0.00838nMAssay Description:Inhibition assay using aromatase enzyme.More data for this Ligand-Target Pair
Affinity DataKi: 0.0118nMAssay Description:Inhibition assay using aromatase enzyme.More data for this Ligand-Target Pair
TargetTryptase beta-2/delta/gamma(Homo sapiens (Human))
Yoshitomi Pharmaceutical Industries
Curated by ChEMBL
Yoshitomi Pharmaceutical Industries
Curated by ChEMBL
Affinity DataKi: 0.0190nMAssay Description:Inhibition of tryptase activityMore data for this Ligand-Target Pair
Affinity DataKi: 0.0200nMAssay Description:Displacement of [3H]-NMS from Sprague-Dawley rat muscarinic M1 receptor in cortex membraneMore data for this Ligand-Target Pair
Affinity DataKi: 0.0200nMAssay Description:Displacement of [3H]-NMS from Sprague-Dawley rat muscarinic M3 receptor in submandibular glandMore data for this Ligand-Target Pair
Affinity DataKi: 0.0200nMAssay Description:Competitive inhibition of human aromatase using dibenzylfluorescein substrate after 10 mins preincubation measured every 10 sec for 5 mins by Michael...More data for this Ligand-Target Pair
Affinity DataKi: 0.0270nMAssay Description:Displacement of [3H]-NMS from Sprague-Dawley rat muscarinic M2 receptor in heartMore data for this Ligand-Target Pair
TargetTryptase beta-2/delta/gamma(Homo sapiens (Human))
Yoshitomi Pharmaceutical Industries
Curated by ChEMBL
Yoshitomi Pharmaceutical Industries
Curated by ChEMBL
Affinity DataKi: 0.0280nMAssay Description:Inhibition of tryptase activityMore data for this Ligand-Target Pair
TargetTryptase beta-2/delta/gamma(Homo sapiens (Human))
Yoshitomi Pharmaceutical Industries
Curated by ChEMBL
Yoshitomi Pharmaceutical Industries
Curated by ChEMBL
Affinity DataKi: 0.0290nMAssay Description:Inhibition of tryptase activityMore data for this Ligand-Target Pair
Affinity DataKi: 0.0410nMAssay Description:Displacement of [3H]-NMS from Sprague-Dawley rat muscarinic M1 receptor in cortex membraneMore data for this Ligand-Target Pair
TargetTryptase beta-2/delta/gamma(Homo sapiens (Human))
Yoshitomi Pharmaceutical Industries
Curated by ChEMBL
Yoshitomi Pharmaceutical Industries
Curated by ChEMBL
Affinity DataKi: 0.0460nMAssay Description:Inhibition of tryptase activityMore data for this Ligand-Target Pair
Affinity DataKi: 0.0490nMAssay Description:Displacement of [3H]-NMS from Sprague-Dawley rat muscarinic M3 receptor in submandibular glandMore data for this Ligand-Target Pair
Affinity DataKi: 0.0500nMAssay Description:Competitive inhibition of human aromatase using dibenzylfluorescein substrate after 10 mins preincubation measured every 10 sec for 5 mins by Michael...More data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Yamanouchi Pharmaceutical
Curated by ChEMBL
Yamanouchi Pharmaceutical
Curated by ChEMBL
Affinity DataKi: 0.0500nMAssay Description:Displacement of [3H]8-OH-DPAT from rat hippocampal 5-hydroxytryptamine 1A receptorMore data for this Ligand-Target Pair
Affinity DataKi: 0.0530nMAssay Description:Displacement of [3H]-NMS from Sprague-Dawley rat muscarinic M2 receptor in heartMore data for this Ligand-Target Pair
Affinity DataKi: 0.0550nMAssay Description:Displacement of [3H]-NMS from Sprague-Dawley rat muscarinic M1 receptor in cortex membraneMore data for this Ligand-Target Pair
Affinity DataKi: 0.0560nMAssay Description:Displacement of [3H]-NMS from Sprague-Dawley rat muscarinic M3 receptor in submandibular glandMore data for this Ligand-Target Pair
TargetTryptase beta-2/delta/gamma(Homo sapiens (Human))
Yoshitomi Pharmaceutical Industries
Curated by ChEMBL
Yoshitomi Pharmaceutical Industries
Curated by ChEMBL
Affinity DataKi: 0.0570nMAssay Description:Inhibition of tryptase activityMore data for this Ligand-Target Pair
Affinity DataKi: 0.0600nMAssay Description:Competitive inhibition of human aromatase using dibenzylfluorescein substrate after 10 mins preincubation measured every 10 sec for 5 mins by Michael...More data for this Ligand-Target Pair
Affinity DataKi: 0.0640nMAssay Description:Displacement of [3H]-NMS from Sprague-Dawley rat muscarinic M3 receptor in submandibular glandMore data for this Ligand-Target Pair
Affinity DataKi: 0.0730nMAssay Description:Displacement of [3H]-NMS from Sprague-Dawley rat muscarinic M1 receptor in cortex membraneMore data for this Ligand-Target Pair
TargetSuppressor of tumorigenicity 14 protein(Homo sapiens (Human))
Aurigene Discovery Technologies
Curated by ChEMBL
Aurigene Discovery Technologies
Curated by ChEMBL
Affinity DataKi: 0.0800nMAssay Description:Inhibition of recombinant matriptase (unknown origin) using Boc-Gln-Ala-Arg-7-amido-4-methyl coumarin hydrobromideMore data for this Ligand-Target Pair
Affinity DataKi: 0.0950nMAssay Description:Displacement of [3H]-NMS from Sprague-Dawley rat muscarinic M1 receptor in cortex membraneMore data for this Ligand-Target Pair
Affinity DataKi: 0.100nMAssay Description:Displacement of [3H]-NMS from Sprague-Dawley rat muscarinic M3 receptor in submandibular glandMore data for this Ligand-Target Pair
Affinity DataKi: 0.120nMAssay Description:Displacement of [3H]-NMS from Sprague-Dawley rat muscarinic M1 receptor in cortex membraneMore data for this Ligand-Target Pair
Affinity DataKi: 0.120nMAssay Description:Displacement of [3H]-NMS from Sprague-Dawley rat muscarinic M3 receptor in submandibular glandMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Yamanouchi Pharmaceutical
Curated by ChEMBL
Yamanouchi Pharmaceutical
Curated by ChEMBL
Affinity DataKi: 0.120nMAssay Description:Displacement of [3H]8-OH-DPAT from rat hippocampal 5-hydroxytryptamine 1A receptorMore data for this Ligand-Target Pair
Affinity DataKi: 0.120nMAssay Description:Displacement of [3H]-NMS from Sprague-Dawley rat muscarinic M3 receptor in submandibular glandMore data for this Ligand-Target Pair
TargetTryptase beta-2/delta/gamma(Homo sapiens (Human))
Yoshitomi Pharmaceutical Industries
Curated by ChEMBL
Yoshitomi Pharmaceutical Industries
Curated by ChEMBL
Affinity DataKi: 0.120nMAssay Description:Inhibition of tryptase activityMore data for this Ligand-Target Pair
Affinity DataKi: 0.120nMAssay Description:Displacement of [3H]-NMS from Sprague-Dawley rat muscarinic M2 receptor in heartMore data for this Ligand-Target Pair
Affinity DataKi: 0.130nMAssay Description:Competitive inhibition of human aromatase using dibenzylfluorescein substrate after 10 mins preincubation measured every 10 sec for 5 mins by Michael...More data for this Ligand-Target Pair
Affinity DataKi: 0.140nMAssay Description:Displacement of [3H]-NMS from Sprague-Dawley rat muscarinic M3 receptor in submandibular glandMore data for this Ligand-Target Pair
Affinity DataKi: 0.149nMAssay Description:Binding affinity against dopamine receptor D2 on rat striatum using [3H]-spiperone as radioligand.More data for this Ligand-Target Pair
Affinity DataKi: 0.150nMAssay Description:Displacement of [3H]-NMS from Sprague-Dawley rat muscarinic M2 receptor in heartMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Yamanouchi Pharmaceutical
Curated by ChEMBL
Yamanouchi Pharmaceutical
Curated by ChEMBL
Affinity DataKi: 0.159nMAssay Description:Binding affinity against 5-hydroxytryptamine 1A receptor on rat hippocampus using [3H]-8-OH-DPAT as radioligand.More data for this Ligand-Target Pair
Affinity DataKi: 0.160nMAssay Description:Displacement of [3H]-NMS from Sprague-Dawley rat muscarinic M1 receptor in cortex membraneMore data for this Ligand-Target Pair
Affinity DataKi: 0.180nMAssay Description:Displacement of [3H]-NMS from Sprague-Dawley rat muscarinic M3 receptor in submandibular glandMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Yamanouchi Pharmaceutical
Curated by ChEMBL
Yamanouchi Pharmaceutical
Curated by ChEMBL
Affinity DataKi: 0.188nMAssay Description:Binding affinity against 5-hydroxytryptamine 1A receptor on rat hippocampus using [3H]-8-OH-DPAT as radioligand.More data for this Ligand-Target Pair
Affinity DataKi: 0.190nMAssay Description:Displacement of [3H]-NMS from Sprague-Dawley rat muscarinic M3 receptor in submandibular glandMore data for this Ligand-Target Pair
Affinity DataKi: 0.190nMAssay Description:Displacement of [3H]-NMS from Sprague-Dawley rat muscarinic M1 receptor in cortex membraneMore data for this Ligand-Target Pair
Affinity DataKi: 0.200nMAssay Description:Displacement of [3H]-NMS from Sprague-Dawley rat muscarinic M3 receptor in submandibular glandMore data for this Ligand-Target Pair
Affinity DataKi: 0.210nMAssay Description:Displacement of [3H]-NMS from Sprague-Dawley rat muscarinic M3 receptor in submandibular glandMore data for this Ligand-Target Pair
Affinity DataKi: 0.210nMAssay Description:Displacement of [3H]-NMS from Sprague-Dawley rat muscarinic M2 receptor in heartMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Yamanouchi Pharmaceutical
Curated by ChEMBL
Yamanouchi Pharmaceutical
Curated by ChEMBL
Affinity DataKi: 0.220nMAssay Description:Displacement of [3H]8-OH-DPAT from rat hippocampal 5-hydroxytryptamine 1A receptorMore data for this Ligand-Target Pair