Affinity DataKi: 0.110nM ΔG°: -56.3kJ/molepH: 7.5 T: 2°CAssay Description:The enzyme activities were determined kinetically as the initial rate of cleavage of a peptide p-nitroanilide. Km for enzyme and substrate was determ...More data for this Ligand-Target Pair
Affinity DataKi: 0.200nMAssay Description:In vitro inhibition of human Coagulation factor X.More data for this Ligand-Target Pair
Affinity DataKi: 0.270nM ΔG°: -54.1kJ/molepH: 7.5 T: 2°CAssay Description:The enzyme activities were determined kinetically as the initial rate of cleavage of a peptide p-nitroanilide. Km for enzyme and substrate was determ...More data for this Ligand-Target Pair
Affinity DataKi: 0.600nMAssay Description:In vitro inhibition of human Coagulation factor X.More data for this Ligand-Target Pair
Affinity DataKi: 0.660nMAssay Description:Inhibitory activity against human Coagulation factor XMore data for this Ligand-Target Pair
Affinity DataKi: 0.660nM ΔG°: -51.9kJ/molepH: 7.5 T: 2°CAssay Description:The enzyme activities were determined kinetically as the initial rate of cleavage of a peptide p-nitroanilide. Km for enzyme and substrate was determ...More data for this Ligand-Target Pair
Affinity DataKi: 0.660nMAssay Description:Compound was tested for inhibition activity against Coagulation factor XMore data for this Ligand-Target Pair
Affinity DataKi: 0.900nMAssay Description:In vitro inhibition of human Coagulation factor X.More data for this Ligand-Target Pair
Affinity DataKi: 1.60nMAssay Description:In vitro inhibition of human Coagulation factor X.More data for this Ligand-Target Pair
Affinity DataKi: 1.60nM ΔG°: -49.7kJ/molepH: 7.5 T: 2°CAssay Description:The enzyme activities were determined kinetically as the initial rate of cleavage of a peptide p-nitroanilide. Km for enzyme and substrate was determ...More data for this Ligand-Target Pair
Affinity DataKi: 3.5nMAssay Description:In vitro inhibition of human Coagulation factor X.More data for this Ligand-Target Pair
Affinity DataKi: 4nMAssay Description:In vitro inhibition of human Coagulation factor X.More data for this Ligand-Target Pair
Affinity DataKi: 4.60nMAssay Description:In vitro inhibition of human Coagulation factor X.More data for this Ligand-Target Pair
Affinity DataKi: 5nMAssay Description:In vitro inhibition of human Coagulation factor X.More data for this Ligand-Target Pair
Affinity DataKi: 6nMAssay Description:In vitro inhibition of human Coagulation factor X.More data for this Ligand-Target Pair
Affinity DataKi: 12nMAssay Description:Compound was tested for inhibition activity against Coagulation factor XMore data for this Ligand-Target Pair
Affinity DataKi: 13nMAssay Description:Compound was tested for inhibition activity against Coagulation factor XMore data for this Ligand-Target Pair
Affinity DataKi: 14nM ΔG°: -44.4kJ/molepH: 7.5 T: 2°CAssay Description:The enzyme activities were determined kinetically as the initial rate of cleavage of a peptide p-nitroanilide. Km for enzyme and substrate was determ...More data for this Ligand-Target Pair
Affinity DataKi: 18nM ΔG°: -43.8kJ/molepH: 7.5 T: 2°CAssay Description:The enzyme activities were determined kinetically as the initial rate of cleavage of a peptide p-nitroanilide. Km for enzyme and substrate was determ...More data for this Ligand-Target Pair
Affinity DataKi: 20nM ΔG°: -43.5kJ/molepH: 7.5 T: 2°CAssay Description:The enzyme activities were determined kinetically as the initial rate of cleavage of a peptide p-nitroanilide. Km for enzyme and substrate was determ...More data for this Ligand-Target Pair
Affinity DataKi: 20nMAssay Description:In vitro inhibition of human Coagulation factor X.More data for this Ligand-Target Pair
Affinity DataKi: 20nMAssay Description:In vitro inhibition of bovine trypsin.More data for this Ligand-Target Pair
Affinity DataKi: 22nMAssay Description:Compound was tested for inhibition activity against factor Xa (FXa)More data for this Ligand-Target Pair
Affinity DataKi: 23nMAssay Description:Compound was tested for inhibition activity against Coagulation factor XMore data for this Ligand-Target Pair
Affinity DataKi: 24nMAssay Description:Compound was tested for inhibition activity against Coagulation factor XMore data for this Ligand-Target Pair
Affinity DataKi: 30nMAssay Description:In vitro inhibition of bovine trypsin.More data for this Ligand-Target Pair
Affinity DataKi: 30nMAssay Description:In vitro inhibition of human Coagulation factor X.More data for this Ligand-Target Pair
Affinity DataKi: 30nMAssay Description:In vitro inhibition of bovine trypsin.More data for this Ligand-Target Pair
Affinity DataKi: 32nMAssay Description:Compound was tested for inhibition activity against Coagulation factor XMore data for this Ligand-Target Pair
Affinity DataKi: 33nM ΔG°: -42.3kJ/molepH: 7.5 T: 2°CAssay Description:The enzyme activities were determined kinetically as the initial rate of cleavage of a peptide p-nitroanilide. Km for enzyme and substrate was determ...More data for this Ligand-Target Pair
Affinity DataKi: 33nMAssay Description:Compound was tested for inhibition activity against bovine trypsin.More data for this Ligand-Target Pair
Affinity DataKi: 34nMAssay Description:Compound was tested for inhibition activity against Coagulation factor XMore data for this Ligand-Target Pair
Affinity DataKi: 36nM ΔG°: -42.1kJ/molepH: 7.5 T: 2°CAssay Description:The enzyme activities were determined kinetically as the initial rate of cleavage of a peptide p-nitroanilide. Km for enzyme and substrate was determ...More data for this Ligand-Target Pair
Affinity DataKi: 40nMAssay Description:In vitro inhibition of human Coagulation factor II.More data for this Ligand-Target Pair
Affinity DataKi: 40nMAssay Description:In vitro inhibition of bovine trypsin.More data for this Ligand-Target Pair
Affinity DataKi: 42nMAssay Description:Compound was tested for inhibition activity against Coagulation factor XMore data for this Ligand-Target Pair
Affinity DataKi: 50nMAssay Description:In vitro inhibition of human Coagulation factor II.More data for this Ligand-Target Pair
Affinity DataKi: 51nMAssay Description:Compound was tested for inhibition activity against Coagulation factor XMore data for this Ligand-Target Pair
Affinity DataKi: 52nMAssay Description:Compound was tested for inhibition activity against Coagulation factor XMore data for this Ligand-Target Pair
Affinity DataKi: 53nMAssay Description:Compound was tested for inhibition activity against Coagulation factor XMore data for this Ligand-Target Pair
Affinity DataKi: 53nMAssay Description:Compound was tested for inhibition activity against Coagulation factor XMore data for this Ligand-Target Pair
Affinity DataKi: 59nMAssay Description:Compound was tested for inhibition activity against Coagulation factor XMore data for this Ligand-Target Pair
Affinity DataKi: 59nMAssay Description:Compound was tested for inhibition activity against Coagulation factor XMore data for this Ligand-Target Pair
Affinity DataKi: 60nMAssay Description:In vitro inhibition of human Coagulation factor X.More data for this Ligand-Target Pair
Affinity DataKi: 60nMAssay Description:Compound was tested for inhibition activity against Coagulation factor XMore data for this Ligand-Target Pair
Affinity DataKi: 60nMAssay Description:In vitro inhibition of bovine trypsin.More data for this Ligand-Target Pair
Affinity DataKi: 62nMAssay Description:Compound was tested for inhibition activity against Coagulation factor XMore data for this Ligand-Target Pair
Affinity DataKi: 80nMAssay Description:In vitro inhibition of bovine trypsin.More data for this Ligand-Target Pair
Affinity DataKi: 85nM ΔG°: -40.0kJ/molepH: 7.5 T: 2°CAssay Description:The enzyme activities were determined kinetically as the initial rate of cleavage of a peptide p-nitroanilide. Km for enzyme and substrate was determ...More data for this Ligand-Target Pair
Affinity DataKi: 90nMAssay Description:In vitro inhibition of bovine trypsin.More data for this Ligand-Target Pair