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Found 282 with Last Name = 'koyama' and Initial = 's'
TargetOxytocin receptor(Homo sapiens (Human))
Tohoku University And Department Of Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM50523555(CHEMBL4474284)
Affinity DataKi:  0.510nMAssay Description:Displacement of [3H]OT from recombinant human OTR expressed in HEK293 cell membranes measured after 1 hrMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetOxytocin receptor(Homo sapiens (Human))
Tohoku University And Department Of Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM50205990(CHEMBL395429 | OXYTOCIN)
Affinity DataKi:  0.580nMAssay Description:Displacement of [3H]OT from recombinant human OTR expressed in HEK293 cell membranes measured after 1 hrMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxytocin receptor(Homo sapiens (Human))
Tohoku University And Department Of Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM50523556(CHEMBL4458988)
Affinity DataKi:  0.900nMAssay Description:Displacement of [3H]OT from recombinant human OTR expressed in HEK293 cell membranes measured after 1 hrMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetOxytocin receptor(Homo sapiens (Human))
Tohoku University And Department Of Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM50044686(CHEMBL3354594)
Affinity DataKi:  1.10nMAssay Description:Displacement of [3H]OT from recombinant human OTR expressed in HEK293 cell membranes measured after 1 hrMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxytocin receptor(Homo sapiens (Human))
Tohoku University And Department Of Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM50523557(CHEMBL4583231)
Affinity DataKi:  1.40nMAssay Description:Displacement of [3H]OT from recombinant human OTR expressed in HEK293 cell membranes measured after 1 hrMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetOxytocin receptor(Homo sapiens (Human))
Tohoku University And Department Of Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM50044742(CHEMBL3354579)
Affinity DataKi:  1.40nMAssay Description:Displacement of [3H]OT from recombinant human OTR expressed in HEK293 cell membranes measured after 1 hrMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxytocin receptor(Homo sapiens (Human))
Tohoku University And Department Of Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM50044677(CHEBI:59204 | Carbetocin)
Affinity DataKi:  1.80nMAssay Description:Displacement of [3H]OT from recombinant human OTR expressed in HEK293 cell membranes measured after 1 hrMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMedDrugBank

TargetOxytocin receptor(Homo sapiens (Human))
Tohoku University And Department Of Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM50044777(Arginine Vasopressin | Beta-Hypophamine | CHEBI:34...)
Affinity DataKi:  2nMAssay Description:Displacement of [3H]OT from recombinant human OTR expressed in HEK293 cell membranes measured after 1 hrMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxytocin receptor(Homo sapiens (Human))
Tohoku University And Department Of Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM50523554(CHEMBL4467042)
Affinity DataKi:  3nMAssay Description:Displacement of [3H]OT from recombinant human OTR expressed in HEK293 cell membranes measured after 1 hrMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProstacyclin receptor(Homo sapiens (Human))
Fujisawa Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50168287(CHEMBL363800 | Sodium; {3-[(1R,2S,6S)-1-(4,5-diphe...)
Affinity DataKi:  6.10nMAssay Description:Inhibition of [3H]-Iloprost binding to human Prostanoid IP receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstacyclin receptor(Homo sapiens (Human))
Fujisawa Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM23954(5-[(2E,3aS,4R,5R,6aS)-5-hydroxy-4-[(1E,3S)-3-hydro...)
Affinity DataKi:  6.5nMAssay Description:Ability to inhibit binding of [3H]iloprost to cloned human prostaglandin I2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstacyclin receptor(Homo sapiens (Human))
Fujisawa Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50167887((R)-2-(6-((diphenylcarbamoyloxy)methyl)-6-hydroxy-...)
Affinity DataKi:  8.90nMAssay Description:Displacement of [3H]iloprost from human Prostanoid IP receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstacyclin receptor(Homo sapiens (Human))
Fujisawa Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50167890(CHEMBL190497 | FR-193262 | Sodium; {(R)-5-[(R)-2-(...)
Affinity DataKi:  12nMAssay Description:Displacement of [3H]iloprost from human Prostanoid IP receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstacyclin receptor(Homo sapiens (Human))
Fujisawa Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50167890(CHEMBL190497 | FR-193262 | Sodium; {(R)-5-[(R)-2-(...)
Affinity DataKi:  12nMAssay Description:Ability to inhibit binding of [3H]iloprost to cloned human prostaglandin I2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLysine-specific histone demethylase 1A(Homo sapiens (Human))
Nagoya City University

Curated by ChEMBL
LigandPNGBDBM50240130(CHEMBL4060961)
Affinity DataKi:  30nMAssay Description:Inhibition of human LSD1 (172 to 833 residues) assessed as reduction in H2O2 production using H3K4me2 (1 to 20 residues) peptide as substrate preincu...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLysine-specific histone demethylase 1A(Homo sapiens (Human))
Nagoya City University

Curated by ChEMBL
LigandPNGBDBM50240124(CHEMBL4090728)
Affinity DataKi:  40nMAssay Description:Inhibition of human LSD1 assessed as reduction in H2O2 production using pLys4Met H3 peptide as substrate by peroxidase coupled UV-visible spectrophot...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstacyclin receptor(Homo sapiens (Human))
Fujisawa Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50168291(CHEMBL363350 | Sodium; {3-[(S)-2-(4,5-diphenyl-oxa...)
Affinity DataKi:  41nMAssay Description:Inhibition of [3H]-Iloprost binding to human Prostanoid IP receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstacyclin receptor(Homo sapiens (Human))
Fujisawa Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50370452(CHEMBL132589 | FR-181157)
Affinity DataKi:  54nMAssay Description:Ability to inhibit binding of [3H]iloprost to cloned human prostaglandin I2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstacyclin receptor(Homo sapiens (Human))
Fujisawa Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50136234(CHEMBL132589 | FR-181157 | Sodium; {3-[(R)-2-(4,5-...)
Affinity DataKi:  54nMAssay Description:Inhibition of [3H]-Iloprost binding to human Prostanoid IP receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstacyclin receptor(Homo sapiens (Human))
Fujisawa Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50370452(CHEMBL132589 | FR-181157)
Affinity DataKi:  54nMAssay Description:Displacement of [3H]iloprost from human Prostanoid IP receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLysine-specific histone demethylase 1A(Homo sapiens (Human))
Nagoya City University

Curated by ChEMBL
LigandPNGBDBM50240122(CHEMBL4103690)
Affinity DataKi:  60nMAssay Description:Inhibition of human LSD1 (172 to 833 residues) assessed as reduction in H2O2 production using H3K4me2 (1 to 20 residues) peptide as substrate preincu...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLysine-specific histone demethylase 1A(Homo sapiens (Human))
Nagoya City University

Curated by ChEMBL
LigandPNGBDBM50240126(CHEMBL4105288)
Affinity DataKi:  98nMAssay Description:Inhibition of human LSD1 (172 to 833 residues) assessed as reduction in H2O2 production using H3K4me2 (1 to 20 residues) peptide as substrate preincu...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstacyclin receptor(Homo sapiens (Human))
Fujisawa Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50167892(CHEMBL195456 | {(S)-6-[(Diphenylcarbamoyloxy)-meth...)
Affinity DataKi:  110nMAssay Description:Displacement of [3H]iloprost from human Prostanoid IP receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstacyclin receptor(Homo sapiens (Human))
Fujisawa Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50167891(CHEMBL197319 | {6-[(Diphenylcarbamoyloxy)-methyl]-...)
Affinity DataKi:  140nMAssay Description:Displacement of [3H]iloprost from human Prostanoid IP receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLysine-specific histone demethylase 1A(Homo sapiens (Human))
Nagoya City University

Curated by ChEMBL
LigandPNGBDBM50240123(CHEMBL4085763)
Affinity DataKi:  290nMAssay Description:Inhibition of human LSD1 (172 to 833 residues) assessed as reduction in H2O2 production using H3K4me2 (1 to 20 residues) peptide as substrate preincu...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLysine-specific histone demethylase 1A(Homo sapiens (Human))
Nagoya City University

Curated by ChEMBL
LigandPNGBDBM50240121(CHEMBL4089148)
Affinity DataKi:  380nMAssay Description:Inhibition of human LSD1 (172 to 833 residues) assessed as reduction in H2O2 production using H3K4me2 (1 to 20 residues) peptide as substrate preincu...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThromboxane A2 receptor(Homo sapiens (Human))
Fujisawa Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50168287(CHEMBL363800 | Sodium; {3-[(1R,2S,6S)-1-(4,5-diphe...)
Affinity DataKi:  930nMAssay Description:Inhibition of [3H]-SQ-29,548 binding to human Prostanoid TP receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThromboxane A2 receptor(Homo sapiens (Human))
Fujisawa Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50136234(CHEMBL132589 | FR-181157 | Sodium; {3-[(R)-2-(4,5-...)
Affinity DataKi: >1.00E+3nMAssay Description:Inhibition of [3H]-SQ-29,548 binding to human Prostanoid TP receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin E2 receptor EP2 subtype(Homo sapiens (Human))
Fujisawa Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50136234(CHEMBL132589 | FR-181157 | Sodium; {3-[(R)-2-(4,5-...)
Affinity DataKi: >1.00E+3nMAssay Description:Inhibition of [3H]-PGE-2 binding to Prostanoid EP2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin D2 receptor(Homo sapiens (Human))
Fujisawa Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50136234(CHEMBL132589 | FR-181157 | Sodium; {3-[(R)-2-(4,5-...)
Affinity DataKi: >1.00E+3nMAssay Description:Inhibition of [3H]-PGD-2 binding to human Prostanoid DP receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin F2-alpha receptor(Homo sapiens (Human))
Fujisawa Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50136234(CHEMBL132589 | FR-181157 | Sodium; {3-[(R)-2-(4,5-...)
Affinity DataKi: >1.00E+3nMAssay Description:Inhibition of [3H]-PGF-2 binding to human Prostanoid FP receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin E2 receptor EP1 subtype(Homo sapiens (Human))
Fujisawa Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50136234(CHEMBL132589 | FR-181157 | Sodium; {3-[(R)-2-(4,5-...)
Affinity DataKi: >1.00E+3nMAssay Description:Inhibition of [3H]-PGE-2 binding to Prostanoid EP1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin D2 receptor(Homo sapiens (Human))
Fujisawa Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50167890(CHEMBL190497 | FR-193262 | Sodium; {(R)-5-[(R)-2-(...)
Affinity DataKi: >1.00E+3nMAssay Description:Displacement of [3H]PGD-2 from human Prostanoid DP receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThromboxane A2 receptor(Homo sapiens (Human))
Fujisawa Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50370452(CHEMBL132589 | FR-181157)
Affinity DataKi: >1.00E+3nMAssay Description:Displacement of [3H]SQ-29,548 from human Prostanoid TP receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin E2 receptor EP1 subtype(Homo sapiens (Human))
Fujisawa Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50167891(CHEMBL197319 | {6-[(Diphenylcarbamoyloxy)-methyl]-...)
Affinity DataKi: >1.00E+3nMAssay Description:Displacement of [3H]PGE-2 from human Prostanoid EP1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin D2 receptor(Homo sapiens (Human))
Fujisawa Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50370452(CHEMBL132589 | FR-181157)
Affinity DataKi: >1.00E+3nMAssay Description:Displacement of [3H]PGD-2 from human Prostanoid DP receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin E2 receptor EP2 subtype(Homo sapiens (Human))
Fujisawa Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50167891(CHEMBL197319 | {6-[(Diphenylcarbamoyloxy)-methyl]-...)
Affinity DataKi: >1.00E+3nMAssay Description:Displacement of [3H]-PGE-2 from human Prostanoid EP2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin F2-alpha receptor(Homo sapiens (Human))
Fujisawa Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50167890(CHEMBL190497 | FR-193262 | Sodium; {(R)-5-[(R)-2-(...)
Affinity DataKi: >1.00E+3nMAssay Description:Displacement of [3H]PGF-2 from human Prostanoid FP receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin E2 receptor EP1 subtype(Homo sapiens (Human))
Fujisawa Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50167890(CHEMBL190497 | FR-193262 | Sodium; {(R)-5-[(R)-2-(...)
Affinity DataKi: >1.00E+3nMAssay Description:Displacement of [3H]PGE-2 from human Prostanoid EP1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin E2 receptor EP1 subtype(Homo sapiens (Human))
Fujisawa Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50167892(CHEMBL195456 | {(S)-6-[(Diphenylcarbamoyloxy)-meth...)
Affinity DataKi: >1.00E+3nMAssay Description:Displacement of [3H]PGE-2 from human Prostanoid EP1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin E2 receptor EP2 subtype(Homo sapiens (Human))
Fujisawa Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50167892(CHEMBL195456 | {(S)-6-[(Diphenylcarbamoyloxy)-meth...)
Affinity DataKi: >1.00E+3nMAssay Description:Displacement of [3H]-PGE-2 from human Prostanoid EP2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin E2 receptor EP1 subtype(Homo sapiens (Human))
Fujisawa Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50370452(CHEMBL132589 | FR-181157)
Affinity DataKi: >1.00E+3nMAssay Description:Displacement of [3H]PGE-2 from human Prostanoid EP1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin E2 receptor EP2 subtype(Homo sapiens (Human))
Fujisawa Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50167890(CHEMBL190497 | FR-193262 | Sodium; {(R)-5-[(R)-2-(...)
Affinity DataKi: >1.00E+3nMAssay Description:Displacement of [3H]-PGE-2 from human Prostanoid EP2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin E2 receptor EP2 subtype(Homo sapiens (Human))
Fujisawa Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50370452(CHEMBL132589 | FR-181157)
Affinity DataKi: >1.00E+3nMAssay Description:Displacement of [3H]-PGE-2 from human Prostanoid EP2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin F2-alpha receptor(Homo sapiens (Human))
Fujisawa Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50370452(CHEMBL132589 | FR-181157)
Affinity DataKi: >1.00E+3nMAssay Description:Displacement of [3H]PGF-2 from human Prostanoid FP receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThromboxane A2 receptor(Homo sapiens (Human))
Fujisawa Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50167890(CHEMBL190497 | FR-193262 | Sodium; {(R)-5-[(R)-2-(...)
Affinity DataKi: >1.00E+3nMAssay Description:Displacement of [3H]SQ-29,548 from human Prostanoid TP receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin E2 receptor EP4 subtype(Homo sapiens (Human))
Fujisawa Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50136234(CHEMBL132589 | FR-181157 | Sodium; {3-[(R)-2-(4,5-...)
Affinity DataKi:  1.02E+3nMAssay Description:Inhibition of [3H]-PGE-2 binding to Prostanoid EP4 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin E2 receptor EP4 subtype(Homo sapiens (Human))
Fujisawa Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50370452(CHEMBL132589 | FR-181157)
Affinity DataKi:  1.02E+3nMAssay Description:Displacement of [3H]PGE-2 from human Prostanoid EP4 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLysine-specific histone demethylase 1A(Homo sapiens (Human))
Nagoya City University

Curated by ChEMBL
LigandPNGBDBM50240129(CHEMBL4080345)
Affinity DataKi:  1.40E+3nMAssay Description:Inhibition of human LSD1 (172 to 833 residues) assessed as reduction in H2O2 production using H3K4me2 (1 to 20 residues) peptide as substrate preincu...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin E2 receptor EP2 subtype(Homo sapiens (Human))
Fujisawa Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50168287(CHEMBL363800 | Sodium; {3-[(1R,2S,6S)-1-(4,5-diphe...)
Affinity DataKi:  1.40E+3nMAssay Description:Inhibition of [3H]-PGE-2 binding to Prostanoid EP2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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