Found 36 Enz. Inhib. hit(s) with Target = 'Oxytocin receptor' and Ligand = 'BDBM50205990' 
Affinity DataKi: 0.440nMAssay Description:Displacement of [3H]8-arginine-vasopressin from human oxytocin receptor expressed in CHO cell membrane incubated for 1 hr by liquid scintillation cou...More data for this Ligand-Target Pair
Affinity DataKi: 0.580nMAssay Description:Displacement of [3H]OT from recombinant human OTR expressed in HEK293 cell membranes measured after 1 hrMore data for this Ligand-Target Pair
Affinity DataKi: 0.790nMAssay Description:Displacement of [3H]OT from oxytocin receptor expressed in COS1 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 0.790nMAssay Description:Competitive binding to oxytocin receptor (unknown origin) by radioligand binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 0.790nMAssay Description:Binding affinity to OTR (unknown origin)More data for this Ligand-Target Pair
Affinity DataKi: 0.800nMAssay Description:Binding affinity for human oxytocin receptorMore data for this Ligand-Target Pair
Affinity DataKi: 0.800nMAssay Description:Agonist activity at human oxytocin receptor expressed in HEK293 cells assessed as increase in IP1 accumulation preincubated for 1 hr followed by addi...More data for this Ligand-Target Pair
Affinity DataKi: 0.890nMAssay Description:Binding affinity against oxytocin receptor in rat uterusMore data for this Ligand-Target Pair
Affinity DataKi: 1.20nMAssay Description:Displacement of [3H]OT from human mammary gland oxytocin receptor expressed in HEK293 cell membrane after 1 hr by scintillation counting methodMore data for this Ligand-Target Pair
Affinity DataKi: 1.70nMAssay Description:Binding affinity against Oxytocin receptor was determined in rat uterine membrane using radioligand [3H]-oxytocinMore data for this Ligand-Target Pair
Affinity DataKi: 6.60nMAssay Description:Competitive binding to SNAP-tagged oxytocin receptor (unknown origin) expressed in HEK293 cells incubated for 1 hr at RT followed by 4 hrs at 4 degC ...More data for this Ligand-Target Pair
Affinity DataKi: 6.80nMAssay Description:Binding affinity to oxytocin receptorMore data for this Ligand-Target Pair
Affinity DataKi: 9.5nMAssay Description:Competitive binding to SNAP-tagged oxytocin receptor (unknown origin) expressed in HEK293 cells incubated for 1 hr at RT followed by 4 hrs at 4 degC ...More data for this Ligand-Target Pair
Affinity DataIC50: 2.70nMAssay Description:Displacement of [3H]OT from human OT receptor expressed in HEK cellsMore data for this Ligand-Target Pair
Affinity DataEC50: 26nMAssay Description:Agonist activity at human OTR receptor expressed in HEK293FT cells incubated for 30 mins by beta-arrestin recruitment assayMore data for this Ligand-Target Pair
Affinity DataEC50: 0.0400nMAssay Description:Agonist activity at human OTR expressed in CHO cells assessed as increase in calcium flux after 60 to 120 mins by fluo-4 dye based FLIPR assayMore data for this Ligand-Target Pair
Affinity DataEC50: 0.00460nMAssay Description:Agonist activity at human OTR receptor expressed in HEK293 cells assessed as intracellular calcium level measured at 3 secs interval for 5 mins by fu...More data for this Ligand-Target Pair
Affinity DataEC50: 2.30nMAssay Description:Agonist activity at recombinant human Gi/Go-coupled OTR expressed in CHOK1 cells assessed as induction of beta-arrestin recruitment measured after 90...More data for this Ligand-Target Pair
Affinity DataEC50: 1.30nMAssay Description:Agonist activity at recombinant human Gi/Go-coupled OTR expressed in CHOK1 cells assessed as induction of beta-arrestin recruitment measured after 90...More data for this Ligand-Target Pair
Affinity DataEC50: 2.10nMAssay Description:Agonist activity at human oxytocin receptor expressed in HEK293 cells coexpressing Rluc8-tagged Galphaq, N-terminal GFP-tagged Ggamma2 and Gbeta1 pro...More data for this Ligand-Target Pair
Affinity DataEC50: 0.0100nMAssay Description:Agonist activity at recombinant human OTR expressed in HEK293 cells assessed as increase in intracellular calcium level measured at 3 secs interval f...More data for this Ligand-Target Pair
Affinity DataEC50: 0.700nMAssay Description:Agonist activity at human OTR receptor expressed in HEK293FT cells assessed as stimulation of calcium release by Aequorin based assayMore data for this Ligand-Target Pair
Affinity DataEC50: 2nMAssay Description:Agonist activity at mouse OTR receptor expressed in HEK293FT cells assessed as stimulation of calcium release by Aequorin based assayMore data for this Ligand-Target Pair
Affinity DataEC50: 0.300nMAssay Description:Agonist activity at human mammary gland oxytocin receptor expressed in CHO cells assessed as increase in intracellular calcium flux measured for 5 mi...More data for this Ligand-Target Pair
Affinity DataEC50: 9nMAssay Description:Binding affinity against Vasopressin receptor in rat liverMore data for this Ligand-Target Pair
Affinity DataEC50: 0.00800nMAssay Description:Agonist activity at human OTR expressed in CHO cells assessed as calcium mobilization measured after 30 mins by Fluo-4-AM dye based FLIPR assayMore data for this Ligand-Target Pair
Affinity DataEC50: 2.30nMAssay Description:Biological activity against Oxytocin receptor in ratMore data for this Ligand-Target Pair
Affinity DataEC50: 3nMAssay Description:Agonist activity at recombinant human oxytocin receptor expressed in CHO-DUKX-A2 cells assessed as change in intracellular calcium level by FLIPR ass...More data for this Ligand-Target Pair
Affinity DataEC50: 8nMAssay Description:Agonist activity at SNAP-tagged oxytocin receptor (unknown origin) expressed in HEK293 cells assessed as intracellular calcium flux after 3 mins by f...More data for this Ligand-Target Pair
Affinity DataEC50: 5nMAssay Description:Agonist activity at wild type OTR (unknown origin) expressed in HEK293 cells assessed as intracellular calcium flux after 3 mins by fluorescence assa...More data for this Ligand-Target Pair
Affinity DataEC50: 2.30nMAssay Description:Agonist activity at human oxytocin receptor expressed in CHO-K1 cells after 5 hrs by firefly luciferase reporter gene assayMore data for this Ligand-Target Pair
Affinity DataKd: 6.70nMAssay Description:Inhibition of radioligand [3H]OT binding to oxytocin receptor (OT) in guinea pig myometrium membraneMore data for this Ligand-Target Pair
Affinity DataKd: 6.70nMAssay Description:Compound was evaluated for its dissociation constant (Kd) to guinea pig myometrial Oxytocin receptorMore data for this Ligand-Target Pair
Affinity DataEC50: 15nMAssay Description:Activity at oxytocin receptor expressed in COS1 cells assessed as IP-one generation by HTRF assayMore data for this Ligand-Target Pair
Affinity DataEC50: 10.8nMAssay Description:Agonist activity at human oxytocin receptor expressed CHO cells assessed as induction of phospholipase C activity after 15 mins by inositol phosphate...More data for this Ligand-Target Pair
Affinity DataEC50: 0.0400nMAssay Description:Agonist activity at human oxytocin receptor expressed in CHO cells assessed as increase in intracellular calcium flux measured for 90 sec by fluo-4 d...More data for this Ligand-Target Pair
