Affinity DataKi: 0.100nMAssay Description:Inhibition of I-iodocyanopindolol binding to human beta 2 adrenergic receptorsMore data for this Ligand-Target Pair
Affinity DataKi: 0.25nMAssay Description:Inhibition of I-iodocyanopindolol binding to human beta 1 adrenergic receptorsMore data for this Ligand-Target Pair
Affinity DataKi: 3.80nMAssay Description:Inhibition of 125 I-Iodocyanopindolol binding to Beta-1 adrenergic receptorMore data for this Ligand-Target Pair
Affinity DataKi: 7.20nMAssay Description:Inhibition of 125 I-Iodocyanopindolol binding to Beta-2 adrenergic receptorMore data for this Ligand-Target Pair
Affinity DataKi: 140nMAssay Description:Binding affinity of compound against Beta-2 adrenergic receptor was determinedMore data for this Ligand-Target Pair
Affinity DataKi: 160nMAssay Description:Inhibition of I-iodocyanopindolol binding to human beta 2 adrenergic receptorsMore data for this Ligand-Target Pair
Affinity DataKi: 180nMAssay Description:Binding affinity of compound against Beta-2 adrenergic receptor was determinedMore data for this Ligand-Target Pair
Affinity DataKi: 240nMAssay Description:Binding affinity of compound against Beta-1 adrenergic receptor was determinedMore data for this Ligand-Target Pair
Affinity DataKi: 480nMAssay Description:Inhibition of I-iodocyanopindolol binding to human beta 2 adrenergic receptorsMore data for this Ligand-Target Pair
Affinity DataKi: 570nMAssay Description:Inhibition of I-iodocyanopindolol binding to human beta 1 adrenergic receptorsMore data for this Ligand-Target Pair
Affinity DataKi: 2.10E+3nMAssay Description:Inhibition of 125 I-Iodocyanopindolol binding to Beta-2 adrenergic receptorMore data for this Ligand-Target Pair
Affinity DataKi: 3.40E+3nMAssay Description:Inhibition of I-iodocyanopindolol binding to human beta 2 adrenergic receptorsMore data for this Ligand-Target Pair
Affinity DataKi: 3.60E+3nMAssay Description:Inhibition of I-iodocyanopindolol binding to human beta 2 adrenergic receptorsMore data for this Ligand-Target Pair
Affinity DataKi: 6.60E+3nMAssay Description:Binding affinity of compound against Beta-1 adrenergic receptor was determinedMore data for this Ligand-Target Pair
Affinity DataKi: 9.10E+3nMAssay Description:Inhibition of 125 I-Iodocyanopindolol binding to Beta-1 adrenergic receptorMore data for this Ligand-Target Pair
Affinity DataKi: 9.49E+3nMAssay Description:Inhibition of 125 I-Iodocyanopindolol binding to Beta-1 adrenergic receptorMore data for this Ligand-Target Pair
Affinity DataKi: 1.16E+4nMAssay Description:Inhibition of I-iodocyanopindolol binding to human beta 2 adrenergic receptorsMore data for this Ligand-Target Pair
Affinity DataKi: 7.40E+4nMAssay Description:Inhibition of 125 I-Iodocyanopindolol binding to Beta-2 adrenergic receptorMore data for this Ligand-Target Pair
Affinity DataKi: 7.92E+4nMAssay Description:Inhibition of I-iodocyanopindolol binding to human beta 2 adrenergic receptorsMore data for this Ligand-Target Pair
Affinity DataKi: >1.00E+5nMAssay Description:Inhibition of I-iodocyanopindolol binding to human beta 1 adrenergic receptorsMore data for this Ligand-Target Pair
Affinity DataKi: >1.00E+5nMAssay Description:Inhibition of I-iodocyanopindolol binding to human beta 1 adrenergic receptorsMore data for this Ligand-Target Pair
Affinity DataKi: >1.00E+5nMAssay Description:Inhibition of I-iodocyanopindolol binding to human beta 1 adrenergic receptorsMore data for this Ligand-Target Pair
Affinity DataKi: >1.00E+5nMAssay Description:Inhibition of I-iodocyanopindolol binding to human beta 1 adrenergic receptorsMore data for this Ligand-Target Pair
Affinity DataKi: >1.00E+5nMAssay Description:Inhibition of I-iodocyanopindolol binding to human beta 1 adrenergic receptorsMore data for this Ligand-Target Pair
Affinity DataKi: >1.00E+5nMAssay Description:Inhibition of I-iodocyanopindolol binding to human beta 1 adrenergic receptorsMore data for this Ligand-Target Pair
Affinity DataKi: >1.00E+5nMAssay Description:Inhibition of I-iodocyanopindolol binding to human beta 2 adrenergic receptorsMore data for this Ligand-Target Pair
Affinity DataIC50: 4nMAssay Description:Compound was tested for the antagonistic activity against Beta-2 adrenergic receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 5.30nMAssay Description:Compound was evaluated in vitro for beta-adrenergic activity against beta-1 adrenergic receptor by the inhibition of insulin stimulated [14C]- glucos...More data for this Ligand-Target Pair
Affinity DataIC50: 27nMAssay Description:Compound was tested for the antagonistic activity against Beta-1 adrenergic receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 30nMAssay Description:Compound was evaluated for its binding affinity towards Beta-2 adrenergic receptor in rat soleus membrane by displacing (-)-isoproterenol (50 microM)More data for this Ligand-Target Pair
Affinity DataIC50: 59nMAssay Description:Compound was evaluated for its binding affinity towards Beta-1 adrenergic receptor in rat heart membrane by displacing [125I]- iodocyanopindololMore data for this Ligand-Target Pair
Affinity DataIC50: 140nMAssay Description:Inhibition of smooth muscle cell ACAT activity for cells stimulated by cationized LDL.More data for this Ligand-Target Pair
Affinity DataIC50: 140nMAssay Description:In vitro inhibitory concentration against Muscarinic acetylcholine receptor derived from smooth muscle cells from thoracic aorta of monkeysMore data for this Ligand-Target Pair
Affinity DataIC50: 190nMAssay Description:Compound was evaluated in vitro for beta-adrenergic activity against beta-1 adrenergic receptor by the inhibition of insulin stimulated [14C]- glucos...More data for this Ligand-Target Pair
Affinity DataIC50: 268nMAssay Description:Compound was tested for the antagonistic activity against Beta-2 adrenergic receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 311nMAssay Description:In vitro inhibitory concentration against Acyl coenzyme A:cholesterol acyltransferase derived from smooth muscle cells from thoracic aorta of monkeysMore data for this Ligand-Target Pair
Affinity DataIC50: 330nMAssay Description:In vitro inhibitory concentration against Acyl coenzyme A:cholesterol acyltransferase derived from rat adrenalsMore data for this Ligand-Target Pair
Affinity DataIC50: 406nMAssay Description:In vitro inhibitory concentration against Acyl coenzyme A:cholesterol acyltransferase derived from rat adrenalsMore data for this Ligand-Target Pair
Affinity DataIC50: 431nMAssay Description:In vitro inhibitory concentration against Acyl coenzyme A:cholesterol acyltransferase derived from smooth muscle cells from thoracic aorta of monkeysMore data for this Ligand-Target Pair
Affinity DataIC50: 446nMAssay Description:In vitro inhibitory concentration against Acyl coenzyme A:cholesterol acyltransferase derived from rat adrenalsMore data for this Ligand-Target Pair
Affinity DataIC50: 484nMAssay Description:In vitro inhibitory concentration against Acyl coenzyme A:cholesterol acyltransferase derived from rat adrenalsMore data for this Ligand-Target Pair
Affinity DataIC50: 500nMAssay Description:Compound was evaluated in vitro for beta-adrenergic activity against beta-1 adrenergic receptor by the inhibition of insulin stimulated [14C]- glucos...More data for this Ligand-Target Pair
Affinity DataIC50: 600nMAssay Description:Compound was evaluated for its binding affinity towards beta-1 adrenergic receptor in rat heart membrane by displacing [125I]- iodocyanopindololMore data for this Ligand-Target Pair
Affinity DataIC50: 629nMAssay Description:In vitro inhibitory concentration against Acyl coenzyme A:cholesterol acyltransferase derived from rat adrenalsMore data for this Ligand-Target Pair
Affinity DataIC50: 721nMAssay Description:In vitro inhibitory concentration against Acyl coenzyme A:cholesterol acyltransferase derived from rat adrenalsMore data for this Ligand-Target Pair
Affinity DataIC50: 740nMAssay Description:Compound was evaluated for the effect on Cholesterol O-Acyltransferase (ACAT) in Liver microsomesMore data for this Ligand-Target Pair
Affinity DataIC50: 810nMAssay Description:Compound was evaluated for the effect on Cholesterol O-Acyltransferase (ACAT) in intestinal microsomesMore data for this Ligand-Target Pair
Affinity DataIC50: 952nMAssay Description:In vitro inhibitory concentration against ACAT derived from rat adrenalsMore data for this Ligand-Target Pair
Affinity DataIC50: 976nMAssay Description:In vitro inhibitory concentration against acyl coenzyme A:cholesterol acyltransferase derived from rat adrenalsMore data for this Ligand-Target Pair
Affinity DataIC50: 1.00E+3nMAssay Description:Compound was evaluated for its binding affinity towards beta-2 adrenergic receptor in rat soleus membrane by displacing(-)-isoproterenol (50 microM)More data for this Ligand-Target Pair