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Found 244 with Last Name = 'lee' and Initial = 'bj'
TargetReceptor-type tyrosine-protein kinase FLT3(Homo sapiens (Human))
Korea University

Curated by ChEMBL
LigandPNGBDBM50300690(1-(5-Tert-Butyl-1,2-Oxazol-3-Yl)-3-(4-{7-[2-(Morph...)
Affinity DataIC50: <0.510nMAssay Description:Inhibition of human FLT3 using EAIYAAPFAKKK substrate and [gamma-33P]-ATP by radiometric biochemical kinase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 3(Homo sapiens (Human))
Korea University

Curated by ChEMBL
LigandPNGBDBM50413752(CHEMBL2012519 | L-783277)
Affinity DataIC50:  0.730nMAssay Description:Inhibition of human VEGFR3 using poly[Glu:Tyr] (4:1) substrate and [gamma-33P]-ATP by radiometric biochemical kinase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Dong-A Pharm.

Curated by ChEMBL
LigandPNGBDBM50344779((R)-4-((R)-3-amino-4-(2,4,5-trifluorophenyl)butano...)
Affinity DataIC50:  0.900nMAssay Description:Inhibition of recombinant human DPP-4 assessed as H-Gly-Pro-AMC cleavage after 1 hr by fluorescence assayMore data for this Ligand-Target Pair
TargetBone morphogenetic protein receptor type-1B(Homo sapiens (Human))
Korea University

Curated by ChEMBL
LigandPNGBDBM50262079(4-(6-(4-(piperazin-1-yl)phenyl)pyrazolo[1,5-a]pyri...)
Affinity DataIC50:  0.940nMAssay Description:Inhibition of human ALK6 using casein as substrate in presence of 10 uM ATP by radiometric kinase assayMore data for this Ligand-Target Pair
TargetVascular endothelial growth factor receptor 3(Homo sapiens (Human))
Korea University

Curated by ChEMBL
LigandPNGBDBM50413752(CHEMBL2012519 | L-783277)
Affinity DataIC50:  1.10nMAssay Description:Inhibition of human FLT4 using poly[Glu:Tyr] (4:1) as substrate in presence of [gamma-33P]-ATP by scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 3(Homo sapiens (Human))
Korea University

Curated by ChEMBL
LigandPNGBDBM50509140(CHEMBL4453304)
Affinity DataIC50:  1.10nMAssay Description:Inhibition of human VEGFR3 using poly[Glu:Tyr] (4:1) substrate and [gamma-33P]-ATP by radiometric biochemical kinase assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 3(Homo sapiens (Human))
Korea University

Curated by ChEMBL
LigandPNGBDBM50509146(CHEMBL4303275)
Affinity DataIC50:  1.20nMAssay Description:Inhibition of human VEGFR3 using poly[Glu:Tyr] (4:1) substrate and [gamma-33P]-ATP by radiometric biochemical kinase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Dong-A Pharm.

Curated by ChEMBL
LigandPNGBDBM50344783((S)-4-((R)-3-amino-4-(2,4,5-trifluorophenyl)butano...)
Affinity DataIC50:  1.30nMAssay Description:Inhibition of recombinant human DPP-4 assessed as H-Gly-Pro-AMC cleavage after 1 hr by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReceptor-type tyrosine-protein kinase FLT3(Homo sapiens (Human))
Korea University

Curated by ChEMBL
LigandPNGBDBM50413752(CHEMBL2012519 | L-783277)
Affinity DataIC50:  1.60nMAssay Description:Inhibition of human FLT3 using EAIYAAPFAKKK peptide as substrate in presence of [gamma-33P]-ATP by scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Dong-A Pharm.

Curated by ChEMBL
LigandPNGBDBM50344777((R)-4-((R)-3-amino-4-(2,4,5-trifluorophenyl)butano...)
Affinity DataIC50:  1.70nMAssay Description:Inhibition of recombinant human DPP-4 assessed as H-Gly-Pro-AMC cleavage after 1 hr by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReceptor-type tyrosine-protein kinase FLT3(Homo sapiens (Human))
Korea University

Curated by ChEMBL
LigandPNGBDBM50413752(CHEMBL2012519 | L-783277)
Affinity DataIC50:  1.80nMAssay Description:Inhibition of human FLT3 using EAIYAAPFAKKK substrate and [gamma-33P]-ATP by radiometric biochemical kinase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBone morphogenetic protein receptor type-1A(Homo sapiens (Human))
Korea University

Curated by ChEMBL
LigandPNGBDBM50262079(4-(6-(4-(piperazin-1-yl)phenyl)pyrazolo[1,5-a]pyri...)
Affinity DataIC50:  2.20nMAssay Description:Inhibition of human ALK3 using casein as substrate in presence of 10 uM ATP by radiometric kinase assayMore data for this Ligand-Target Pair
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Dong-A Pharm.

Curated by ChEMBL
LigandPNGBDBM50344778((R)-4-((R)-3-amino-4-(2,4,5-trifluorophenyl)butano...)
Affinity DataIC50:  2.20nMAssay Description:Inhibition of recombinant human DPP-4 assessed as H-Gly-Pro-AMC cleavage after 1 hr by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Korea University

Curated by ChEMBL
LigandPNGBDBM50413752(CHEMBL2012519 | L-783277)
Affinity DataIC50:  2.90nMAssay Description:Inhibition of human VEGFR2 using poly[Glu:Tyr] (4:1) substrate and [gamma-33P]-ATP by radiometric biochemical kinase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetActivin receptor type-1(Homo sapiens (Human))
Korea University

Curated by ChEMBL
LigandPNGBDBM50262079(4-(6-(4-(piperazin-1-yl)phenyl)pyrazolo[1,5-a]pyri...)
Affinity DataIC50:  3.30nMAssay Description:Inhibition of human ALK2 using casein as substrate in presence of 10 uM ATP by radiometric kinase assayMore data for this Ligand-Target Pair
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Korea University

Curated by ChEMBL
LigandPNGBDBM50509140(CHEMBL4453304)
Affinity DataIC50:  3.60nMAssay Description:Inhibition of human VEGFR2 using poly[Glu:Tyr] (4:1) substrate and [gamma-33P]-ATP by radiometric biochemical kinase assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Dong-A Pharm.

Curated by ChEMBL
LigandPNGBDBM50344776((R)-4-((R)-3-amino-4-(2,4,5-trifluorophenyl)butano...)
Affinity DataIC50:  4.30nMAssay Description:Inhibition of recombinant human DPP-4 assessed as H-Gly-Pro-AMC cleavage after 1 hr by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReceptor-type tyrosine-protein kinase FLT3(Homo sapiens (Human))
Korea University

Curated by ChEMBL
LigandPNGBDBM50509140(CHEMBL4453304)
Affinity DataIC50:  4.40nMAssay Description:Inhibition of human FLT3 using EAIYAAPFAKKK substrate and [gamma-33P]-ATP by radiometric biochemical kinase assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPeptide deformylase(Pseudomonas aeruginosa)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50334431(CHEMBL1643873 | N-((3S,5R)-5-((N-hydroxyformamido)...)
Affinity DataIC50:  5nMAssay Description:Inhibition of Pseudomonas aeruginosa peptide deformylase after 10 mins by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Dong-A Pharm.

Curated by ChEMBL
LigandPNGBDBM50344782((R)-4-((R)-3-amino-4-(2,4,5-trifluorophenyl)butano...)
Affinity DataIC50:  5.20nMAssay Description:Inhibition of recombinant human DPP-4 assessed as H-Gly-Pro-AMC cleavage after 1 hr by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Korea University

Curated by ChEMBL
LigandPNGBDBM50413752(CHEMBL2012519 | L-783277)
Affinity DataIC50:  6.30nMAssay Description:Inhibition of human KDR using poly[Glu:Tyr] (4:1) as substrate in presence of [gamma-33P]-ATP by scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Dong-A Pharm.

Curated by ChEMBL
LigandPNGBDBM50344788((R)-4-(3-amino-4-(2,4,5-trifluorophenyl)butanoyl)-...)
Affinity DataIC50:  7.40nMAssay Description:Inhibition of recombinant human DPP-4 assessed as H-Gly-Pro-AMC cleavage after 1 hr by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Dong-A Pharm.

Curated by ChEMBL
LigandPNGBDBM50344775((R)-4-((R)-3-amino-4-(2,4,5-trifluorophenyl)butano...)
Affinity DataIC50:  7.40nMAssay Description:Inhibition of recombinant human DPP-4 assessed as H-Gly-Pro-AMC cleavage after 1 hr by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeptide deformylase(Pseudomonas aeruginosa)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50334430(CHEMBL1643872 | N-((3S,5R)-5-((N-hydroxyformamido)...)
Affinity DataIC50:  8nMAssay Description:Inhibition of Pseudomonas aeruginosa peptide deformylase after 10 mins by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDual specificity mitogen-activated protein kinase kinase 2(Homo sapiens (Human))
Korea University

Curated by ChEMBL
LigandPNGBDBM50413752(CHEMBL2012519 | L-783277)
Affinity DataIC50:  8.20nMAssay Description:Inhibition of human MEK2 using ERK2 as substrate in presence of [gamma-33P]-ATP by scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 3(Homo sapiens (Human))
Korea University

Curated by ChEMBL
LigandPNGBDBM50509148(CHEMBL4452766)
Affinity DataIC50:  9.20nMAssay Description:Inhibition of human VEGFR3 using poly[Glu:Tyr] (4:1) substrate and [gamma-33P]-ATP by radiometric biochemical kinase assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 3(Homo sapiens (Human))
Korea University

Curated by ChEMBL
LigandPNGBDBM50509144(CHEMBL4530473)
Affinity DataIC50:  9.90nMAssay Description:Inhibition of human VEGFR3 using poly[Glu:Tyr] (4:1) substrate and [gamma-33P]-ATP by radiometric biochemical kinase assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPeptide deformylase(Pseudomonas aeruginosa)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50334433(CHEMBL1643875 | N-((2R,4S)-2-butyl-4-(3-cyclopenty...)
Affinity DataIC50:  10nMAssay Description:Inhibition of Pseudomonas aeruginosa peptide deformylase after 10 mins by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeptide deformylase(Pseudomonas aeruginosa)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50416424(CHEMBL1208984)
Affinity DataIC50:  11nMAssay Description:Inhibition of Pseudomonas aeruginosa Peptide deformylase by fluorescence analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Dong-A Pharm.

Curated by ChEMBL
LigandPNGBDBM50344781((R)-4-((R)-3-amino-4-(2,4,5-trifluorophenyl)butano...)
Affinity DataIC50:  11nMAssay Description:Inhibition of recombinant human DPP-4 assessed as H-Gly-Pro-AMC cleavage after 1 hr by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase receptor R3(Homo sapiens (Human))
Korea University

Curated by ChEMBL
LigandPNGBDBM50262079(4-(6-(4-(piperazin-1-yl)phenyl)pyrazolo[1,5-a]pyri...)
Affinity DataIC50:  11nMAssay Description:Inhibition of human ALK1 using casein as substrate in presence of 10 uM ATP by radiometric kinase assayMore data for this Ligand-Target Pair
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Dong-A Pharm.

Curated by ChEMBL
LigandPNGBDBM50344774((R)-4-((R)-3-amino-4-(2,4,5-trifluorophenyl)butano...)
Affinity DataIC50:  12nMAssay Description:Inhibition of recombinant human DPP-4 assessed as H-Gly-Pro-AMC cleavage after 1 hr by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeptide deformylase(Pseudomonas aeruginosa)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50416414(CHEMBL1208855)
Affinity DataIC50:  13nMAssay Description:Inhibition of Pseudomonas aeruginosa Peptide deformylase by fluorescence analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeptide deformylase(Pseudomonas aeruginosa)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50416415(CHEMBL1208856)
Affinity DataIC50:  13nMAssay Description:Inhibition of Pseudomonas aeruginosa Peptide deformylase by fluorescence analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Dong-A Pharm.

Curated by ChEMBL
LigandPNGBDBM50344769((R)-4-(3-amino-4-(2,4,5-trifluorophenyl)butanoyl)-...)
Affinity DataIC50:  13.7nMAssay Description:Inhibition of recombinant human DPP-4 assessed as H-Gly-Pro-AMC cleavage after 1 hr by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Korea University

Curated by ChEMBL
LigandPNGBDBM50509144(CHEMBL4530473)
Affinity DataIC50:  14nMAssay Description:Inhibition of human VEGFR2 using poly[Glu:Tyr] (4:1) substrate and [gamma-33P]-ATP by radiometric biochemical kinase assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPeptide deformylase(Pseudomonas aeruginosa)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50416413(CHEMBL1208854)
Affinity DataIC50:  15nMAssay Description:Inhibition of Pseudomonas aeruginosa Peptide deformylase by fluorescence analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeptide deformylase(Pseudomonas aeruginosa)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50334432(CHEMBL1643874 | N-((2R,4S)-2-butyl-4-(3-isopropylu...)
Affinity DataIC50:  16nMAssay Description:Inhibition of Pseudomonas aeruginosa peptide deformylase after 10 mins by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeptide deformylase(Pseudomonas aeruginosa)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50416425(CHEMBL1208985)
Affinity DataIC50:  17nMAssay Description:Inhibition of Pseudomonas aeruginosa Peptide deformylase by fluorescence analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Dong-A Pharm.

Curated by ChEMBL
LigandPNGBDBM50344780((R)-4-((R)-3-amino-4-(2,4,5-trifluorophenyl)butano...)
Affinity DataIC50:  17nMAssay Description:Inhibition of recombinant human DPP-4 assessed as H-Gly-Pro-AMC cleavage after 1 hr by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReceptor-type tyrosine-protein kinase FLT3(Homo sapiens (Human))
Korea University

Curated by ChEMBL
LigandPNGBDBM50509142(CHEMBL4515000)
Affinity DataIC50:  17nMAssay Description:Inhibition of human FLT3 using EAIYAAPFAKKK substrate and [gamma-33P]-ATP by radiometric biochemical kinase assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPeptide deformylase(Pseudomonas aeruginosa)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50416423(CHEMBL1208983)
Affinity DataIC50:  19nMAssay Description:Inhibition of Pseudomonas aeruginosa Peptide deformylase by fluorescence analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeptide deformylase(Pseudomonas aeruginosa)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50416412(CHEMBL1209868)
Affinity DataIC50:  21nMAssay Description:Inhibition of Pseudomonas aeruginosa Peptide deformylase by fluorescence analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeptide deformylase(Pseudomonas aeruginosa)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50334426(CHEMBL1643868 | N-((3S,5R)-5-((N-hydroxyformamido)...)
Affinity DataIC50:  22nMAssay Description:Inhibition of Pseudomonas aeruginosa peptide deformylase after 10 mins by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 3(Homo sapiens (Human))
Korea University

Curated by ChEMBL
LigandPNGBDBM50509139(CHEMBL4533447)
Affinity DataIC50:  23nMAssay Description:Inhibition of human VEGFR3 using poly[Glu:Tyr] (4:1) substrate and [gamma-33P]-ATP by radiometric biochemical kinase assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Dong-A Pharm.

Curated by ChEMBL
LigandPNGBDBM50390170(CHEMBL2069848)
Affinity DataIC50:  24.9nMAssay Description:Inhibition of recombinant human DPP4 after 1 hr by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Dong-A Pharm.

Curated by ChEMBL
LigandPNGBDBM50344786((R)-4-(3-amino-4-(2,4,5-trifluorophenyl)butanoyl)-...)
Affinity DataIC50:  26.7nMAssay Description:Inhibition of recombinant human DPP-4 assessed as H-Gly-Pro-AMC cleavage after 1 hr by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 3(Homo sapiens (Human))
Korea University

Curated by ChEMBL
LigandPNGBDBM50509142(CHEMBL4515000)
Affinity DataIC50:  27nMAssay Description:Inhibition of human VEGFR3 using poly[Glu:Tyr] (4:1) substrate and [gamma-33P]-ATP by radiometric biochemical kinase assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTGF-beta receptor type-1(Homo sapiens (Human))
Korea University

Curated by ChEMBL
LigandPNGBDBM50262079(4-(6-(4-(piperazin-1-yl)phenyl)pyrazolo[1,5-a]pyri...)
Affinity DataIC50:  27nMAssay Description:Inhibition of human ALK5 using casein as substrate in presence of 10 uM ATP by radiometric kinase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeptide deformylase(Pseudomonas aeruginosa)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50416428(CHEMBL1209044)
Affinity DataIC50:  28nMAssay Description:Inhibition of Pseudomonas aeruginosa Peptide deformylase by fluorescence analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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