Affinity DataKi: 0.00250nMAssay Description:Binding affinity towards thrombinMore data for this Ligand-Target Pair
Affinity DataKi: 0.0560nMAssay Description:Inhibitory activity against human thrombinMore data for this Ligand-Target Pair
Affinity DataKi: 0.0900nMAssay Description:Binding affinity towards thrombinMore data for this Ligand-Target Pair
Affinity DataKi: 0.0900nMAssay Description:Binding affinity towards thrombin was determinedMore data for this Ligand-Target Pair
Affinity DataKi: 0.100nMAssay Description:Inhibitory activity against human thrombinMore data for this Ligand-Target Pair
Affinity DataKi: 0.100nMAssay Description:Binding affinity towards thrombin was determinedMore data for this Ligand-Target Pair
Affinity DataKi: 0.100nMAssay Description:Inhibitory activity against human thrombinMore data for this Ligand-Target Pair
Affinity DataKi: 0.100nMAssay Description:Binding affinity towards thrombinMore data for this Ligand-Target Pair
Affinity DataKi: 0.100nMAssay Description:Binding affinity towards thrombinMore data for this Ligand-Target Pair
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Merck Research Laboratories
Curated by ChEMBL
Merck Research Laboratories
Curated by ChEMBL
Affinity DataKi: 0.240nMAssay Description:Compound was evaluated in vitro for the inhibition of HIV-Protease, using a peptide hydrolysis assayMore data for this Ligand-Target Pair
Affinity DataKi: 0.280nM Koff: 2.51E+3s-1Assay Description:Inhibition of ThrombinMore data for this Ligand-Target Pair
Affinity DataKi: 0.310nMAssay Description:Binding affinity of the compound was evaluated on serine protease thrombin.More data for this Ligand-Target Pair
Affinity DataKi: 0.400nMAssay Description:Binding affinity towards thrombinMore data for this Ligand-Target Pair
Affinity DataKi: 0.450nMAssay Description:Binding affinity of the compound was evaluated on serine protease thrombin.More data for this Ligand-Target Pair
Affinity DataKi: 0.5nMAssay Description:Binding affinity of the compound was evaluated on serine protease thrombin.More data for this Ligand-Target Pair
Affinity DataKi: 0.610nMAssay Description:Binding affinity of the compound was evaluated on serine protease thrombin.More data for this Ligand-Target Pair
Affinity DataKi: 0.740nMAssay Description:Binding affinity of the compound was evaluated on serine protease thrombin.More data for this Ligand-Target Pair
Affinity DataKi: 1.5nMAssay Description:Binding affinity towards thrombin was determinedMore data for this Ligand-Target Pair
Affinity DataKi: 2nM Koff: 2.10E+3s-1Assay Description:Inhibition of ThrombinMore data for this Ligand-Target Pair
Affinity DataKi: 2.5nMAssay Description:Binding affinity towards thrombin was determinedMore data for this Ligand-Target Pair
Affinity DataKi: 2.5nMAssay Description:Binding affinity towards thrombin was determinedMore data for this Ligand-Target Pair
Affinity DataKi: 2.5nMAssay Description:Binding affinity of the compound was evaluated on serine protease thrombin.More data for this Ligand-Target Pair
Affinity DataKi: 3nMAssay Description:Binding affinity towards thrombinMore data for this Ligand-Target Pair
Affinity DataKi: 3nMAssay Description:Binding affinity towards thrombin was determinedMore data for this Ligand-Target Pair
Affinity DataKi: 3nMAssay Description:Binding affinity towards thrombinMore data for this Ligand-Target Pair
Affinity DataKi: 3nMAssay Description:Binding affinity of the compound was evaluated on serine protease thrombin.More data for this Ligand-Target Pair
Affinity DataKi: 3nM Koff: 1.80E+3s-1Assay Description:Inhibition of ThrombinMore data for this Ligand-Target Pair
Affinity DataKi: 3.40nM Koff: 1.55E+3s-1Assay Description:Inhibition of ThrombinMore data for this Ligand-Target Pair
Affinity DataKi: 4nMAssay Description:Binding affinity towards trypsinMore data for this Ligand-Target Pair
Affinity DataKi: 4nMAssay Description:In vitro inhibition of Histamine H2 receptor by measuring its ability to block the histamine-stimulated adenylate cyclase of guinea pig hippocampal h...More data for this Ligand-Target Pair
Affinity DataKi: 4.90nMAssay Description:Binding affinity towards thrombin was determinedMore data for this Ligand-Target Pair
Affinity DataKi: 5nMAssay Description:Binding affinity towards thrombinMore data for this Ligand-Target Pair
Affinity DataKi: 5nMAssay Description:Binding affinity of the compound was evaluated on serine protease thrombin.More data for this Ligand-Target Pair
Affinity DataKi: 6.30nMAssay Description:In vitro inhibition of Histamine H2 receptor by measuring its ability to block the histamine-stimulated adenylate cyclase of guinea pig hippocampal h...More data for this Ligand-Target Pair
Affinity DataKi: 6.30nMAssay Description:In vitro inhibition of Histamine H2 receptor by measuring its ability to block the histamine-stimulated adenylate cyclase of guinea pig hippocampal h...More data for this Ligand-Target Pair
Affinity DataKi: 10nM Koff: 2.10E+3s-1Assay Description:Inhibition of ThrombinMore data for this Ligand-Target Pair
Affinity DataKi: 12nM Koff: 1.80E+3s-1Assay Description:Inhibition of ThrombinMore data for this Ligand-Target Pair
Affinity DataKi: 14nM Koff: 2.30E+3s-1Assay Description:Inhibition of ThrombinMore data for this Ligand-Target Pair
Affinity DataKi: 18nMAssay Description:Binding affinity of the compound was evaluated on serine protease thrombin.More data for this Ligand-Target Pair
Affinity DataKi: 20nMAssay Description:Binding affinity of the compound was evaluated on serine protease thrombin.More data for this Ligand-Target Pair
Affinity DataKi: 32nMAssay Description:Evaluated in vitro for Histamine H2 receptor inhibition using the dimaprit stimulated chronotropic response of the guinea pig atriumMore data for this Ligand-Target Pair
Affinity DataKi: 40nMAssay Description:Binding affinity towards thrombinMore data for this Ligand-Target Pair
Affinity DataKi: 60nMAssay Description:Binding affinity of the compound was evaluated on serine protease thrombin.More data for this Ligand-Target Pair
Affinity DataKi: 70nMAssay Description:Binding affinity towards thrombinMore data for this Ligand-Target Pair
Affinity DataKi: 75nMAssay Description:Binding affinity towards thrombin was determinedMore data for this Ligand-Target Pair
Affinity DataKi: 94nMAssay Description:Inhibitory activity against human trypsinMore data for this Ligand-Target Pair
Affinity DataKi: 110nMAssay Description:Binding affinity towards thrombinMore data for this Ligand-Target Pair