TargetD(2) dopamine receptor(Rattus norvegicus (rat))
University of North Texas
Curated by PDSP Ki Database
University of North Texas
Curated by PDSP Ki Database
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
University of North Texas
Curated by PDSP Ki Database
University of North Texas
Curated by PDSP Ki Database
Affinity DataKi: 0.0170nMAssay Description:Inhibition of [125I]- NCQ 298 binding to D2 receptor of rat striatal tissueMore data for this Ligand-Target Pair
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
University of North Texas
Curated by PDSP Ki Database
University of North Texas
Curated by PDSP Ki Database
Affinity DataKi: 0.0200nMAssay Description:Inhibition of [125I]- NCQ 298 binding to D2 receptor of rat striatal tissueMore data for this Ligand-Target Pair
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
University of North Texas
Curated by PDSP Ki Database
University of North Texas
Curated by PDSP Ki Database
Affinity DataKi: 0.0230nMAssay Description:Displacement of [3H]-spiperone from dopamine receptor D2More data for this Ligand-Target Pair
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
University of North Texas
Curated by PDSP Ki Database
University of North Texas
Curated by PDSP Ki Database
Affinity DataKi: 0.0230nMAssay Description:Displacement of [3H]-spiperone from dopamine receptor D2More data for this Ligand-Target Pair
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
University of North Texas
Curated by PDSP Ki Database
University of North Texas
Curated by PDSP Ki Database
Affinity DataKi: 0.0280nMAssay Description:Inhibition of [125I]- NCQ 298 binding to D2 receptor of rat striatal tissueMore data for this Ligand-Target Pair
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
University of North Texas
Curated by PDSP Ki Database
University of North Texas
Curated by PDSP Ki Database
Affinity DataKi: 0.0290nMAssay Description:Displacement of [3H]-spiperone from dopamine receptor D2More data for this Ligand-Target Pair
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
University of North Texas
Curated by PDSP Ki Database
University of North Texas
Curated by PDSP Ki Database
Affinity DataKi: 0.0330nMAssay Description:Displacement of [3H]-spiperone from dopamine receptor D2More data for this Ligand-Target Pair
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
University of North Texas
Curated by PDSP Ki Database
University of North Texas
Curated by PDSP Ki Database
Affinity DataKi: 0.0330nMAssay Description:Inhibition of [125I]- NCQ 298 binding to D2 receptor of rat striatal tissueMore data for this Ligand-Target Pair
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
University of North Texas
Curated by PDSP Ki Database
University of North Texas
Curated by PDSP Ki Database
Affinity DataKi: 0.0350nMAssay Description:Displacement of [3H]-spiperone from dopamine receptor D2More data for this Ligand-Target Pair
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
University of North Texas
Curated by PDSP Ki Database
University of North Texas
Curated by PDSP Ki Database
Affinity DataKi: 0.0360nMAssay Description:Inhibition of [125I]- NCQ 298 binding to D2 receptor of rat striatal tissueMore data for this Ligand-Target Pair
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
University of North Texas
Curated by PDSP Ki Database
University of North Texas
Curated by PDSP Ki Database
Affinity DataKi: 0.0360nMAssay Description:Displacement of [3H]-spiperone from dopamine receptor D2More data for this Ligand-Target Pair
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
University of North Texas
Curated by PDSP Ki Database
University of North Texas
Curated by PDSP Ki Database
Affinity DataKi: 0.0380nMAssay Description:Inhibition of [125I]- NCQ 298 binding to D2 receptor of rat striatal tissueMore data for this Ligand-Target Pair
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
University of North Texas
Curated by PDSP Ki Database
University of North Texas
Curated by PDSP Ki Database
Affinity DataKi: 0.0390nMAssay Description:Displacement of [3H]-spiperone from dopamine receptor D2More data for this Ligand-Target Pair
TargetD(3) dopamine receptor(Rattus norvegicus (Rat))
Wake Forest University School Of Medicine
Curated by ChEMBL
Wake Forest University School Of Medicine
Curated by ChEMBL
Affinity DataKi: 0.0400nMAssay Description:Binding affinity for dopamine receptor D3 expressed in Sf9 cells using [125I]-IABN the radioligand.More data for this Ligand-Target Pair
TargetD(3) dopamine receptor(Rattus norvegicus (Rat))
Wake Forest University School Of Medicine
Curated by ChEMBL
Wake Forest University School Of Medicine
Curated by ChEMBL
Affinity DataKi: 0.0400nMAssay Description:Binding affinity for dopamine receptor D3 expressed in Sf9 cells using [125I]-IABN the radioligand.More data for this Ligand-Target Pair
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
University of North Texas
Curated by PDSP Ki Database
University of North Texas
Curated by PDSP Ki Database
Affinity DataKi: 0.0430nMAssay Description:Displacement of [3H]-spiperone from dopamine receptor D2More data for this Ligand-Target Pair
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
University of North Texas
Curated by PDSP Ki Database
University of North Texas
Curated by PDSP Ki Database
Affinity DataKi: 0.0470nMAssay Description:Binding affinity towards Dopamine receptor D2 by displacing [3H]-spiperoneMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
The University Of Sydney
Curated by ChEMBL
The University Of Sydney
Curated by ChEMBL
Affinity DataKi: 0.0500nMAssay Description:Displacement of [3H](+)-pentazocine from sigma1 receptor in guinea pig brain homogenateMore data for this Ligand-Target Pair
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
University of North Texas
Curated by PDSP Ki Database
University of North Texas
Curated by PDSP Ki Database
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
University of North Texas
Curated by PDSP Ki Database
University of North Texas
Curated by PDSP Ki Database
Affinity DataKi: 0.0500nMAssay Description:Binding affinity for dopamine receptor D2 long expressed in Sf9 cells using [125I]-IABN radioligand.More data for this Ligand-Target Pair
TargetVesicular acetylcholine transporter(Torpedo californica)
University Of Minnesota
Curated by ChEMBL
University Of Minnesota
Curated by ChEMBL
Affinity DataKi: 0.0550nMAssay Description:Displacement of [3H]vesamicol from VAChT in Torpedo californica cholinergic synaptic vesiclesMore data for this Ligand-Target Pair
TargetVesicular acetylcholine transporter(Homo sapiens (Human))
University Of Minnesota
Curated by ChEMBL
University Of Minnesota
Curated by ChEMBL
Affinity DataKi: 0.0550nMAssay Description:Binding to vesicular acetylcholine transporter of torpedo synaptic vesiclesMore data for this Ligand-Target Pair
TargetVesicular acetylcholine transporter(Homo sapiens (Human))
University Of Minnesota
Curated by ChEMBL
University Of Minnesota
Curated by ChEMBL
Affinity DataKi: 0.0550nMAssay Description:Displacement of [3H]vesamicol from human vesicular acetylcholine transporter expressed in rat PC12 cells by liquid scintillation spectrometryMore data for this Ligand-Target Pair
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
University of North Texas
Curated by PDSP Ki Database
University of North Texas
Curated by PDSP Ki Database
Affinity DataKi: 0.0570nMAssay Description:Binding affinity towards Dopamine receptor D2 by displacing [3H]-spiperoneMore data for this Ligand-Target Pair
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
University of North Texas
Curated by PDSP Ki Database
University of North Texas
Curated by PDSP Ki Database
Affinity DataKi: 0.0580nMAssay Description:Displacement of [3H]-spiperone from dopamine receptor D2More data for this Ligand-Target Pair
Affinity DataKi: 0.0600nMAssay Description:Displacement of [125I]IABN from recombinant human D2 long receptor stably expressed in HEK293 cell membranes measured after 60 mins by scintillation ...More data for this Ligand-Target Pair
Affinity DataKi: 0.0600nMAssay Description:Displacement of [125I]ABN from human dopamine D2 long receptor expressed in HEK293 cell membranes after 60 mins by scintillation counting methodMore data for this Ligand-Target Pair
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
University of North Texas
Curated by PDSP Ki Database
University of North Texas
Curated by PDSP Ki Database
Affinity DataKi: 0.0620nMAssay Description:Displacement of [3H]-spiperone from dopamine receptor D2More data for this Ligand-Target Pair
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
University of North Texas
Curated by PDSP Ki Database
University of North Texas
Curated by PDSP Ki Database
Affinity DataKi: 0.0630nMAssay Description:Displacement of [3H]-spiperone from dopamine receptor D2More data for this Ligand-Target Pair
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
University of North Texas
Curated by PDSP Ki Database
University of North Texas
Curated by PDSP Ki Database
Affinity DataKi: 0.0630nMAssay Description:Binding affinity towards Dopamine receptor D2 by displacing [3H]-spiperoneMore data for this Ligand-Target Pair
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
University of North Texas
Curated by PDSP Ki Database
University of North Texas
Curated by PDSP Ki Database
Affinity DataKi: 0.0670nMAssay Description:Binding affinity towards Dopamine receptor D2 by displacing [3H]-spiperoneMore data for this Ligand-Target Pair
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
University of North Texas
Curated by PDSP Ki Database
University of North Texas
Curated by PDSP Ki Database
Affinity DataKi: 0.0690nMAssay Description:Displacement of [3H]-spiperone from dopamine receptor D2More data for this Ligand-Target Pair
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
University of North Texas
Curated by PDSP Ki Database
University of North Texas
Curated by PDSP Ki Database
Affinity DataKi: 0.0700nMAssay Description:Inhibition of [125I]- NCQ 298 binding to D2 receptor of rat striatal tissueMore data for this Ligand-Target Pair
Affinity DataKi: 0.0700nMAssay Description:Displacement of [125I]ABN from human recombinant D2L receptor expressed in HEK cells after 60 mins by gamma counterMore data for this Ligand-Target Pair
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
University of North Texas
Curated by PDSP Ki Database
University of North Texas
Curated by PDSP Ki Database
Affinity DataKi: 0.0870nMAssay Description:Binding affinity towards Dopamine receptor D2 by displacing [3H]-spiperoneMore data for this Ligand-Target Pair
Affinity DataKi: 0.0960nMAssay Description:The compound was tested in vitro for binding affinity towards 5-hydroxytryptamine 2 receptor by displacing [125]I-LSD radioligandMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
The University Of Sydney
Curated by ChEMBL
The University Of Sydney
Curated by ChEMBL
Affinity DataKi: 0.100nMAssay Description:Displacement of [3H](+)-pentazocine from sigma1 receptor in guinea pig brain homogenateMore data for this Ligand-Target Pair
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
University of North Texas
Curated by PDSP Ki Database
University of North Texas
Curated by PDSP Ki Database
Affinity DataKi: 0.118nMAssay Description:Binding affinity towards Dopamine receptor D2 by displacing [3H]-spiperoneMore data for this Ligand-Target Pair
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
University of North Texas
Curated by PDSP Ki Database
University of North Texas
Curated by PDSP Ki Database
Affinity DataKi: 0.119nMAssay Description:Binding affinity towards Dopamine receptor D2 by displacing [3H]-spiperoneMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
The University Of Sydney
Curated by ChEMBL
The University Of Sydney
Curated by ChEMBL
Affinity DataKi: 0.120nMAssay Description:Displacement of [3H](+)-pentazocine from sigma1 receptor in guinea pig brain homogenateMore data for this Ligand-Target Pair
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
University of North Texas
Curated by PDSP Ki Database
University of North Texas
Curated by PDSP Ki Database
Affinity DataKi: 0.120nMAssay Description:Binding affinity towards Dopamine receptor D2 by displacing [3H]-spiperoneMore data for this Ligand-Target Pair
TargetSigma intracellular receptor 2(Homo sapiens (Human))
Guangdong Medical University
Curated by ChEMBL
Guangdong Medical University
Curated by ChEMBL
Affinity DataKi: 0.120nMAssay Description:Binding affinity to sigma-2 receptor (unknown origin)More data for this Ligand-Target Pair
Affinity DataKi: 0.130nMAssay Description:The compound was tested in vitro for binding affinity towards 5-hydroxytryptamine 2 receptor by displacing [125]I-LSD radioligandMore data for this Ligand-Target Pair
TargetVesicular acetylcholine transporter(Homo sapiens (Human))
University Of Minnesota
Curated by ChEMBL
University Of Minnesota
Curated by ChEMBL
Affinity DataKi: 0.130nMAssay Description:Displacement of [3H]vesamicol from Vesicular Acetylcholine Transporter (VAChT)More data for this Ligand-Target Pair
TargetVesicular acetylcholine transporter(Homo sapiens (Human))
University Of Minnesota
Curated by ChEMBL
University Of Minnesota
Curated by ChEMBL
Affinity DataKi: 0.130nMAssay Description:Binding to vesicular acetylcholine transporter of torpedo synaptic vesiclesMore data for this Ligand-Target Pair
Affinity DataKi: 0.140nMAssay Description:Displacement of [125I]ABN from human recombinant D2L receptor expressed in HEK cells after 60 mins by gamma counterMore data for this Ligand-Target Pair
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
University of North Texas
Curated by PDSP Ki Database
University of North Texas
Curated by PDSP Ki Database
Affinity DataKi: 0.149nMAssay Description:Inhibitory constant against binding of [125I]- IBZM to rat striatal membraneMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
The University Of Sydney
Curated by ChEMBL
The University Of Sydney
Curated by ChEMBL
Affinity DataKi: 0.152nMAssay Description:Displacement of [3H](+)-pentazocine from sigma1 receptor in guinea pig brain homogenateMore data for this Ligand-Target Pair
Affinity DataKi: 0.160nMAssay Description:In vitro binding affinity on D3 receptor is inhibition of binding of [125I]- NCQ 298 to Sf9 cells infected with recombinant baculovirusMore data for this Ligand-Target Pair