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Found 24 with Last Name = 'madan' and Initial = 'm'
TargetProstaglandin G/H synthase 2(Homo sapiens (Human))
Dr. Reddy'S Laboratories

Curated by ChEMBL
LigandPNGBDBM50133024(3-Fluoro-4-[5-(4-methylsulfanyl-phenyl)-3-trifluor...)
Affinity DataIC50:  34nMAssay Description:In vitro inhibition of the compound against human Prostaglandin G/H synthase 2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Al-Azhar University

Curated by ChEMBL
LigandPNGBDBM5446(CHEMBL553 | ERLOTINIB HYDROCHLORIDE | Erlotinib | ...)
Affinity DataIC50:  60nMAssay Description:Inhibition of His6-tagged EGFR cytoplasmic domain (645 to 1186 residues) (unknown origin) expressed in baculovirus infected Sf9 insect cells after 10...More data for this Ligand-Target Pair
TargetProstaglandin G/H synthase 1(Ovis aries (Sheep))
Dr. Reddy'S Laboratories

Curated by ChEMBL
LigandPNGBDBM17638(2-{1-[(4-chlorophenyl)carbonyl]-5-methoxy-2-methyl...)
Affinity DataIC50:  67nMAssay Description:In vitro inhibition of the compound against Prostaglandin G/H synthase 1 from ram seminal vesiclesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 2(Homo sapiens (Human))
Dr. Reddy'S Laboratories

Curated by ChEMBL
LigandPNGBDBM11639(4-[5-(4-methylphenyl)-3-(trifluoromethyl)-1H-pyraz...)
Affinity DataIC50:  70nMAssay Description:In vitro inhibition of the compound against human Prostaglandin G/H synthase 2More data for this Ligand-Target Pair
TargetProstaglandin G/H synthase 2(Homo sapiens (Human))
Dr. Reddy'S Laboratories

Curated by ChEMBL
LigandPNGBDBM50133025(3-Fluoro-4-[5-(4-methoxy-phenyl)-3-trifluoromethyl...)
Affinity DataIC50:  150nMAssay Description:In vitro inhibition of the compound against human Prostaglandin G/H synthase 2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Al-Azhar University

Curated by ChEMBL
LigandPNGBDBM50517778(CHEMBL4447196)
Affinity DataIC50:  500nMAssay Description:Inhibition of His6-tagged EGFR cytoplasmic domain (645 to 1186 residues) (unknown origin) expressed in baculovirus infected Sf9 insect cells after 10...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 1(Homo sapiens (Human))
Al-Azhar University

Curated by ChEMBL
LigandPNGBDBM50517776(CHEMBL4449599)
Affinity DataIC50:  540nMAssay Description:Inhibition of VEGFR1 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetDNA gyrase subunit A/B(Escherichia coli (strain K12))
Al-Azhar University

Curated by ChEMBL
LigandPNGBDBM21690(1-cyclopropyl-6-fluoro-4-oxo-7-(piperazin-1-yl)-1,...)
Affinity DataIC50:  661nMAssay Description:Inhibition of Escherichia coli DNA gyrase supercoiling activity using topoisomerase II treated decatenated kDNA as substrate incubated for 15 to 30 m...More data for this Ligand-Target Pair
In DepthDetails PubMedDrugBank

TargetEpidermal growth factor receptor(Homo sapiens (Human))
Al-Azhar University

Curated by ChEMBL
LigandPNGBDBM50517774(CHEMBL4462971)
Affinity DataIC50:  700nMAssay Description:Inhibition of His6-tagged EGFR cytoplasmic domain (645 to 1186 residues) (unknown origin) expressed in baculovirus infected Sf9 insect cells after 10...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Al-Azhar University

Curated by ChEMBL
LigandPNGBDBM50517771(CHEMBL4585048)
Affinity DataIC50:  1.20E+3nMAssay Description:Inhibition of His6-tagged EGFR cytoplasmic domain (645 to 1186 residues) (unknown origin) expressed in baculovirus infected Sf9 insect cells after 10...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Al-Azhar University

Curated by ChEMBL
LigandPNGBDBM50517773(CHEMBL4588486)
Affinity DataIC50:  1.40E+3nMAssay Description:Inhibition of His6-tagged EGFR cytoplasmic domain (645 to 1186 residues) (unknown origin) expressed in baculovirus infected Sf9 insect cells after 10...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Al-Azhar University

Curated by ChEMBL
LigandPNGBDBM50517777(CHEMBL4464785)
Affinity DataIC50:  1.60E+3nMAssay Description:Inhibition of His6-tagged EGFR cytoplasmic domain (645 to 1186 residues) (unknown origin) expressed in baculovirus infected Sf9 insect cells after 10...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase Chk2(Homo sapiens (Human))
Al-Azhar University

Curated by ChEMBL
LigandPNGBDBM50517776(CHEMBL4449599)
Affinity DataIC50:  1.70E+3nMAssay Description:Inhibition of CHK2 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetDNA gyrase subunit A/B(Escherichia coli (strain K12))
Al-Azhar University

Curated by ChEMBL
LigandPNGBDBM50606969(CHEMBL5221057)
Affinity DataIC50:  1.72E+3nMAssay Description:Inhibition of Escherichia coli DNA gyrase supercoiling activity using topoisomerase II treated decatenated kDNA as substrate incubated for 15 to 30 m...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Al-Azhar University

Curated by ChEMBL
LigandPNGBDBM50517770(CHEMBL4474429)
Affinity DataIC50:  2.80E+3nMAssay Description:Inhibition of His6-tagged EGFR cytoplasmic domain (645 to 1186 residues) (unknown origin) expressed in baculovirus infected Sf9 insect cells after 10...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Al-Azhar University

Curated by ChEMBL
LigandPNGBDBM50517775(CHEMBL4540070)
Affinity DataIC50:  2.90E+3nMAssay Description:Inhibition of His6-tagged EGFR cytoplasmic domain (645 to 1186 residues) (unknown origin) expressed in baculovirus infected Sf9 insect cells after 10...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Al-Azhar University

Curated by ChEMBL
LigandPNGBDBM50517772(CHEMBL4568408)
Affinity DataIC50:  3.20E+3nMAssay Description:Inhibition of His6-tagged EGFR cytoplasmic domain (645 to 1186 residues) (unknown origin) expressed in baculovirus infected Sf9 insect cells after 10...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetDNA gyrase subunit A/B(Escherichia coli (strain K12))
Al-Azhar University

Curated by ChEMBL
LigandPNGBDBM50606970(CHEMBL5220268)
Affinity DataIC50:  5.72E+3nMAssay Description:Inhibition of Escherichia coli DNA gyrase supercoiling activity using topoisomerase II treated decatenated kDNA as substrate incubated for 15 to 30 m...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetProstaglandin G/H synthase 2(Homo sapiens (Human))
Dr. Reddy'S Laboratories

Curated by ChEMBL
LigandPNGBDBM17638(2-{1-[(4-chlorophenyl)carbonyl]-5-methoxy-2-methyl...)
Affinity DataIC50:  7.80E+3nMAssay Description:In vitro inhibition of the compound against human Prostaglandin G/H synthase 2More data for this Ligand-Target Pair
TargetProstaglandin G/H synthase 2(Homo sapiens (Human))
Dr. Reddy'S Laboratories

Curated by ChEMBL
LigandPNGBDBM50133026(2-Fluoro-4-[5-(4-methoxy-phenyl)-3-trifluoromethyl...)
Affinity DataIC50:  1.35E+4nMAssay Description:In vitro inhibition of the compound against human Prostaglandin G/H synthase 2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 1(Ovis aries (Sheep))
Dr. Reddy'S Laboratories

Curated by ChEMBL
LigandPNGBDBM11639(4-[5-(4-methylphenyl)-3-(trifluoromethyl)-1H-pyraz...)
Affinity DataIC50:  1.53E+4nMAssay Description:In vitro inhibition of the compound against Prostaglandin G/H synthase 1 from ram seminal vesiclesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 1(Ovis aries (Sheep))
Dr. Reddy'S Laboratories

Curated by ChEMBL
LigandPNGBDBM50133024(3-Fluoro-4-[5-(4-methylsulfanyl-phenyl)-3-trifluor...)
Affinity DataIC50:  2.43E+4nMAssay Description:In vitro inhibition of the compound against Prostaglandin G/H synthase 1 from ram seminal vesiclesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 1(Ovis aries (Sheep))
Dr. Reddy'S Laboratories

Curated by ChEMBL
LigandPNGBDBM50133025(3-Fluoro-4-[5-(4-methoxy-phenyl)-3-trifluoromethyl...)
Affinity DataIC50: >3.00E+4nMAssay Description:In vitro inhibition of the compound against Prostaglandin G/H synthase 1 from ram seminal vesiclesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 1(Ovis aries (Sheep))
Dr. Reddy'S Laboratories

Curated by ChEMBL
LigandPNGBDBM50133026(2-Fluoro-4-[5-(4-methoxy-phenyl)-3-trifluoromethyl...)
Affinity DataIC50: >1.70E+5nMAssay Description:In vitro inhibition of the compound against Prostaglandin G/H synthase 1 from ram seminal vesiclesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed