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Found 73 with Last Name = 'margathe' and Initial = 'jf'
TargetApelin(Homo sapiens (Human))
University Of Strasburg

Curated by ChEMBL
LigandPNGBDBM50009575(CHEMBL3234446)
Affinity DataKi:  0.0400nMAssay Description:Displacement of [125I]-pE13F from human apelin receptor expressed in CHO cell membranes after 1 hr by gamma counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxytocin receptor(Homo sapiens (Human))
University Of Strasburg

Curated by ChEMBL
LigandPNGBDBM50077141(CHEMBL3416758)
Affinity DataKi:  0.210nMAssay Description:Competitive binding to human oxytocin receptor by radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxytocin receptor(Homo sapiens (Human))
University Of Strasburg

Curated by ChEMBL
LigandPNGBDBM50077141(CHEMBL3416758)
Affinity DataKi:  0.450nMAssay Description:Competitive binding to SNAP-tagged oxytocin receptor (unknown origin) expressed in HEK293 cells incubated for 1 hr at RT followed by 4 hrs at 4 degC ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxytocin receptor(Homo sapiens (Human))
University Of Strasburg

Curated by ChEMBL
LigandPNGBDBM50077141(CHEMBL3416758)
Affinity DataKi:  0.670nMAssay Description:Competitive binding to SNAP-tagged oxytocin receptor (unknown origin) expressed in HEK293 cells incubated for 1 hr at RT followed by 4 hrs at 4 degC ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxytocin receptor(Homo sapiens (Human))
University Of Strasburg

Curated by ChEMBL
LigandPNGBDBM50205990(CHEMBL395429 | OXYTOCIN)
Affinity DataKi:  0.790nMAssay Description:Binding affinity to OTR (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxytocin receptor(Homo sapiens (Human))
University Of Strasburg

Curated by ChEMBL
LigandPNGBDBM50205990(CHEMBL395429 | OXYTOCIN)
Affinity DataKi:  0.790nMAssay Description:Competitive binding to oxytocin receptor (unknown origin) by radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxytocin receptor(Homo sapiens (Human))
University Of Strasburg

Curated by ChEMBL
LigandPNGBDBM50077140(CHEMBL3416757)
Affinity DataKi:  6.20nMAssay Description:Competitive binding to SNAP-tagged oxytocin receptor (unknown origin) expressed in HEK293 cells incubated for 1 hr at RT followed by 4 hrs at 4 degC ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxytocin receptor(Homo sapiens (Human))
University Of Strasburg

Curated by ChEMBL
LigandPNGBDBM50077140(CHEMBL3416757)
Affinity DataKi:  6.60nMAssay Description:Competitive binding to SNAP-tagged oxytocin receptor (unknown origin) expressed in HEK293 cells incubated for 1 hr at RT followed by 4 hrs at 4 degC ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxytocin receptor(Homo sapiens (Human))
University Of Strasburg

Curated by ChEMBL
LigandPNGBDBM50205990(CHEMBL395429 | OXYTOCIN)
Affinity DataKi:  6.60nMAssay Description:Competitive binding to SNAP-tagged oxytocin receptor (unknown origin) expressed in HEK293 cells incubated for 1 hr at RT followed by 4 hrs at 4 degC ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxytocin receptor(Homo sapiens (Human))
University Of Strasburg

Curated by ChEMBL
LigandPNGBDBM50205990(CHEMBL395429 | OXYTOCIN)
Affinity DataKi:  9.5nMAssay Description:Competitive binding to SNAP-tagged oxytocin receptor (unknown origin) expressed in HEK293 cells incubated for 1 hr at RT followed by 4 hrs at 4 degC ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1a receptor(Homo sapiens (Human))
University Of Strasburg

Curated by ChEMBL
LigandPNGBDBM50077140(CHEMBL3416757)
Affinity DataKi:  18nMAssay Description:Binding affinity to V1aR (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxytocin receptor(Homo sapiens (Human))
University Of Strasburg

Curated by ChEMBL
LigandPNGBDBM50077140(CHEMBL3416757)
Affinity DataKi:  28nMAssay Description:Binding affinity to OTR (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetApelin(Homo sapiens (Human))
University Of Strasburg

Curated by ChEMBL
LigandPNGBDBM50009560(CHEMBL3234454)
Affinity DataKi:  89nMAssay Description:Displacement of [125I]-pE13F from human apelin receptor expressed in CHO cell membranes after 1 hr by gamma counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1a receptor(Homo sapiens (Human))
University Of Strasburg

Curated by ChEMBL
LigandPNGBDBM50205990(CHEMBL395429 | OXYTOCIN)
Affinity DataKi:  120nMAssay Description:Binding affinity to V1aR (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetApelin(Homo sapiens (Human))
University Of Strasburg

Curated by ChEMBL
LigandPNGBDBM50009571(CHEMBL3234461)
Affinity DataKi:  180nMAssay Description:Displacement of [125I]-pE13F from human apelin receptor expressed in CHO cell membranes after 1 hr by gamma counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetApelin(Homo sapiens (Human))
University Of Strasburg

Curated by ChEMBL
LigandPNGBDBM50009572(CHEMBL3234462)
Affinity DataKi:  270nMAssay Description:Displacement of [125I]-pE13F from human apelin receptor expressed in CHO cell membranes after 1 hr by gamma counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetApelin(Homo sapiens (Human))
University Of Strasburg

Curated by ChEMBL
LigandPNGBDBM50009558(CHEMBL3234452)
Affinity DataKi:  310nMAssay Description:Displacement of [125I]-pE13F from human apelin receptor expressed in CHO cell membranes after 1 hr by gamma counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetApelin(Homo sapiens (Human))
University Of Strasburg

Curated by ChEMBL
LigandPNGBDBM50009559(CHEMBL3234453)
Affinity DataKi:  400nMAssay Description:Displacement of [125I]-pE13F from human apelin receptor expressed in CHO cell membranes after 1 hr by gamma counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetApelin(Homo sapiens (Human))
University Of Strasburg

Curated by ChEMBL
LigandPNGBDBM50009580(CHEMBL3234445)
Affinity DataKi:  430nMAssay Description:Displacement of [125I]-pE13F from human apelin receptor expressed in CHO cell membranes after 1 hr by gamma counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetApelin(Homo sapiens (Human))
University Of Strasburg

Curated by ChEMBL
LigandPNGBDBM50009567(CHEMBL3234458)
Affinity DataKi:  450nMAssay Description:Displacement of [125I]-pE13F from human apelin receptor expressed in CHO cell membranes after 1 hr by gamma counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetApelin(Homo sapiens (Human))
University Of Strasburg

Curated by ChEMBL
LigandPNGBDBM50009576(CHEMBL3234447)
Affinity DataKi:  690nMAssay Description:Displacement of [125I]-pE13F from human apelin receptor expressed in CHO cell membranes after 1 hr by gamma counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetApelin(Homo sapiens (Human))
University Of Strasburg

Curated by ChEMBL
LigandPNGBDBM50009574(CHEMBL3234464)
Affinity DataKi:  850nMAssay Description:Displacement of [125I]-pE13F from human apelin receptor expressed in CHO cell membranes after 1 hr by gamma counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V2 receptor(Homo sapiens (Human))
University Of Strasburg

Curated by ChEMBL
LigandPNGBDBM50077140(CHEMBL3416757)
Affinity DataKi:  913nMAssay Description:Binding affinity to V2R (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetApelin(Homo sapiens (Human))
University Of Strasburg

Curated by ChEMBL
LigandPNGBDBM50009573(CHEMBL3234463)
Affinity DataKi:  960nMAssay Description:Displacement of [125I]-pE13F from human apelin receptor expressed in CHO cell membranes after 1 hr by gamma counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetApelin(Homo sapiens (Human))
University Of Strasburg

Curated by ChEMBL
LigandPNGBDBM50009566(CHEMBL3234457)
Affinity DataKi:  970nMAssay Description:Displacement of [125I]-pE13F from human apelin receptor expressed in CHO cell membranes after 1 hr by gamma counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetApelin(Homo sapiens (Human))
University Of Strasburg

Curated by ChEMBL
LigandPNGBDBM50009570(CHEMBL3234460)
Affinity DataKi:  980nMAssay Description:Displacement of [125I]-pE13F from human apelin receptor expressed in CHO cell membranes after 1 hr by gamma counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetApelin(Homo sapiens (Human))
University Of Strasburg

Curated by ChEMBL
LigandPNGBDBM50009569(CHEMBL3234459)
Affinity DataKi:  1.20E+3nMAssay Description:Displacement of [125I]-pE13F from human apelin receptor expressed in CHO cell membranes after 1 hr by gamma counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetApelin(Homo sapiens (Human))
University Of Strasburg

Curated by ChEMBL
LigandPNGBDBM50009579(CHEMBL3234448)
Affinity DataKi:  1.40E+3nMAssay Description:Displacement of [125I]-pE13F from human apelin receptor expressed in CHO cell membranes after 1 hr by gamma counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetApelin(Homo sapiens (Human))
University Of Strasburg

Curated by ChEMBL
LigandPNGBDBM50009577(CHEMBL3234450)
Affinity DataKi:  1.50E+3nMAssay Description:Displacement of [125I]-pE13F from human apelin receptor expressed in CHO cell membranes after 1 hr by gamma counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V2 receptor(Homo sapiens (Human))
University Of Strasburg

Curated by ChEMBL
LigandPNGBDBM50205990(CHEMBL395429 | OXYTOCIN)
Affinity DataKi:  1.54E+3nMAssay Description:Binding affinity to V2R (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1b receptor(Homo sapiens (Human))
University Of Strasburg

Curated by ChEMBL
LigandPNGBDBM50205990(CHEMBL395429 | OXYTOCIN)
Affinity DataKi:  1.78E+3nMAssay Description:Binding affinity to V1bR (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor(Homo sapiens (Human))
University Of Strasburg

Curated by ChEMBL
LigandPNGBDBM50009576(CHEMBL3234447)
Affinity DataKi:  2.23E+3nMAssay Description:Displacement of [125I]-angiotensin 2 from human angiotensin 2 type-1 receptor expressed in CHO cell membranes after 1 hr by gamma counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetApelin(Homo sapiens (Human))
University Of Strasburg

Curated by ChEMBL
LigandPNGBDBM50009578(CHEMBL3234449)
Affinity DataKi:  3.00E+3nMAssay Description:Displacement of [125I]-pE13F from human apelin receptor expressed in CHO cell membranes after 1 hr by gamma counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetApelin(Homo sapiens (Human))
University Of Strasburg

Curated by ChEMBL
LigandPNGBDBM50009557(CHEMBL3234451)
Affinity DataKi:  9.00E+3nMAssay Description:Displacement of [125I]-pE13F from human apelin receptor expressed in CHO cell membranes after 1 hr by gamma counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor(Homo sapiens (Human))
University Of Strasburg

Curated by ChEMBL
LigandPNGBDBM50009560(CHEMBL3234454)
Affinity DataKi:  9.80E+4nMAssay Description:Displacement of [125I]-angiotensin 2 from human angiotensin 2 type-1 receptor expressed in CHO cell membranes after 1 hr by gamma counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetApelin(Homo sapiens (Human))
University Of Strasburg

Curated by ChEMBL
LigandPNGBDBM50009564(CHEMBL3234456)
Affinity DataKi: >1.00E+5nMAssay Description:Displacement of [125I]-pE13F from human apelin receptor expressed in CHO cell membranes after 1 hr by gamma counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetApelin(Homo sapiens (Human))
University Of Strasburg

Curated by ChEMBL
LigandPNGBDBM50009563(CHEMBL3234455)
Affinity DataKi: >1.00E+5nMAssay Description:Displacement of [125I]-pE13F from human apelin receptor expressed in CHO cell membranes after 1 hr by gamma counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor(Homo sapiens (Human))
University Of Strasburg

Curated by ChEMBL
LigandPNGBDBM50009575(CHEMBL3234446)
Affinity DataKi: >1.00E+5nMAssay Description:Displacement of [125I]-angiotensin 2 from human angiotensin 2 type-1 receptor expressed in CHO cell membranes after 1 hr by gamma counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor(Homo sapiens (Human))
University Of Strasburg

Curated by ChEMBL
LigandPNGBDBM50009559(CHEMBL3234453)
Affinity DataKi: >1.00E+6nMAssay Description:Displacement of [125I]-angiotensin 2 from human angiotensin 2 type-1 receptor expressed in CHO cell membranes after 1 hr by gamma counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetApelin(Rattus norvegicus)
University Of Strasburg

Curated by ChEMBL
LigandPNGBDBM50009575(CHEMBL3234446)
Affinity DataIC50:  1.40nMAssay Description:Agonist activity at rat apelin receptor expressed in CHO cell membranes coexpressing EGFP assessed as inhibition of forskolin-induced cAMP production...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetApelin(Rattus norvegicus)
University Of Strasburg

Curated by ChEMBL
LigandPNGBDBM50009560(CHEMBL3234454)
Affinity DataIC50:  1.70E+3nMAssay Description:Agonist activity at rat apelin receptor expressed in CHO cell membranes coexpressing EGFP assessed as inhibition of forskolin-induced cAMP production...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetApelin(Rattus norvegicus)
University Of Strasburg

Curated by ChEMBL
LigandPNGBDBM50009559(CHEMBL3234453)
Affinity DataIC50:  3.00E+3nMAssay Description:Agonist activity at rat apelin receptor expressed in CHO cell membranes coexpressing EGFP assessed as inhibition of forskolin-induced cAMP production...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetApelin(Rattus norvegicus)
University Of Strasburg

Curated by ChEMBL
LigandPNGBDBM50009576(CHEMBL3234447)
Affinity DataIC50:  4.30E+3nMAssay Description:Agonist activity at rat apelin receptor expressed in CHO cell membranes coexpressing EGFP assessed as inhibition of forskolin-induced cAMP production...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxytocin receptor(Homo sapiens (Human))
University Of Strasburg

Curated by ChEMBL
LigandPNGBDBM50077134(CHEMBL3416751)
Affinity DataKon:  0.000315M-1s-1Assay Description:Binding affinity to SNAP-tagged oxytocin receptor (unknown origin) expressed in HEK293 cells assessed as dissociation constant after 5 to 120 mins by...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1b receptor(Homo sapiens (Human))
University Of Strasburg

Curated by ChEMBL
LigandPNGBDBM50077135(CHEMBL3416750)
Affinity DataKd: >1.00E+3nMAssay Description:Binding affinity to V1bR (unknown origin) expressed in HEK293 cells by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1b receptor(Homo sapiens (Human))
University Of Strasburg

Curated by ChEMBL
LigandPNGBDBM50077136(CHEMBL3416749)
Affinity DataKd: >1.00E+3nMAssay Description:Binding affinity to V1bR (unknown origin) expressed in HEK293 cells by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1a receptor(Homo sapiens (Human))
University Of Strasburg

Curated by ChEMBL
LigandPNGBDBM50077137(CHEMBL3416754)
Affinity DataKd: >1.00E+3nMAssay Description:Binding affinity to V1aR (unknown origin) expressed in HEK293 cells by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1a receptor(Homo sapiens (Human))
University Of Strasburg

Curated by ChEMBL
LigandPNGBDBM50077138(CHEMBL3416753)
Affinity DataKd: >1.00E+3nMAssay Description:Binding affinity to V1aR (unknown origin) expressed in HEK293 cells by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1a receptor(Homo sapiens (Human))
University Of Strasburg

Curated by ChEMBL
LigandPNGBDBM50077139(CHEMBL3416752)
Affinity DataKd: >1.00E+3nMAssay Description:Binding affinity to V1aR (unknown origin) expressed in HEK293 cells by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1a receptor(Homo sapiens (Human))
University Of Strasburg

Curated by ChEMBL
LigandPNGBDBM50077134(CHEMBL3416751)
Affinity DataKd: >1.00E+3nMAssay Description:Binding affinity to V1aR (unknown origin) expressed in HEK293 cells by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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