Affinity DataKi: 0.00110nM IC50: 1.00E+3nMAssay Description:Inhibition assay using aromatase enzyme.More data for this Ligand-Target Pair
Affinity DataKi: 0.00182nM IC50: 1.21E+4nMAssay Description:Inhibition assay using aromatase enzyme.More data for this Ligand-Target Pair
Affinity DataKi: 0.00216nMAssay Description:Inhibition assay using aromatase enzyme.More data for this Ligand-Target Pair
Affinity DataKi: 0.00256nMAssay Description:Inhibition assay using aromatase enzyme.More data for this Ligand-Target Pair
Affinity DataKi: 0.00425nMAssay Description:Inhibition assay using aromatase enzyme.More data for this Ligand-Target Pair
Affinity DataKi: 0.00597nMAssay Description:Inhibition assay using aromatase enzyme.More data for this Ligand-Target Pair
Affinity DataKi: 0.00838nMAssay Description:Inhibition assay using aromatase enzyme.More data for this Ligand-Target Pair
Affinity DataKi: 0.0118nMAssay Description:Inhibition assay using aromatase enzyme.More data for this Ligand-Target Pair
TargetRibosyldihydronicotinamide dehydrogenase [quinone](Homo sapiens (Human))
Yunnan Normal University
Curated by ChEMBL
Yunnan Normal University
Curated by ChEMBL
Affinity DataIC50: 960nMAssay Description:Inhibition of human quinone reductase 2 expressed in Escherichia coli BL21(DE3) assessed as N-methyldihydronicotinamide oxidation per mg of protein a...More data for this Ligand-Target Pair
TargetRibosyldihydronicotinamide dehydrogenase [quinone](Homo sapiens (Human))
Yunnan Normal University
Curated by ChEMBL
Yunnan Normal University
Curated by ChEMBL
Affinity DataIC50: 3.84E+3nMAssay Description:Inhibition of human quinone reductase 2 expressed in Escherichia coli BL21(DE3) assessed as N-methyldihydronicotinamide oxidation per mg of protein a...More data for this Ligand-Target Pair
Affinity DataIC50: 2.68E+4nMAssay Description:Inhibition of aromatase preincubated with 2.6 mM NADP+ for 10 mins before substrate addition measured after 30 mins by fluorescence assayMore data for this Ligand-Target Pair
Affinity DataIC50: 3.07E+4nMAssay Description:Inhibition of aromatase preincubated with 2.6 mM NADP+ for 10 mins before substrate addition measured after 30 mins by fluorescence assayMore data for this Ligand-Target Pair
Affinity DataIC50: 3.23E+4nMAssay Description:Inhibition of aromatase preincubated with 2.6 mM NADP+ for 10 mins before substrate addition measured after 30 mins by fluorescence assayMore data for this Ligand-Target Pair
Affinity DataIC50: 3.53E+4nMAssay Description:Inhibition of aromatase preincubated with 2.6 mM NADP+ for 10 mins before substrate addition measured after 30 mins by fluorescence assayMore data for this Ligand-Target Pair