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Found 14 with Last Name = 'marler' and Initial = 'le'
TargetAromatase(Homo sapiens (Human))
Central Institute of Medicinal and Aromatic Plants

LigandPNGBDBM19461(α-CA inhibitor, 5 | 5,7-dihydroxy-2-(4-hydrox...)
Affinity DataKi:  0.00110nM IC50:  1.00E+3nMAssay Description:Inhibition assay using aromatase enzyme.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
Central Institute of Medicinal and Aromatic Plants

LigandPNGBDBM92556(Neoflavonoid, 8)
Affinity DataKi:  0.00182nM IC50:  1.21E+4nMAssay Description:Inhibition assay using aromatase enzyme.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
Central Institute of Medicinal and Aromatic Plants

LigandPNGBDBM92555(Neoflavonoid, 7)
Affinity DataKi:  0.00216nMAssay Description:Inhibition assay using aromatase enzyme.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
Central Institute of Medicinal and Aromatic Plants

LigandPNGBDBM92557(Neoflavonoid, 9)
Affinity DataKi:  0.00256nMAssay Description:Inhibition assay using aromatase enzyme.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
Central Institute of Medicinal and Aromatic Plants

LigandPNGBDBM92559(Neoflavonoid, 11)
Affinity DataKi:  0.00425nMAssay Description:Inhibition assay using aromatase enzyme.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
Central Institute of Medicinal and Aromatic Plants

LigandPNGBDBM92560(Neoflavonoid, 19)
Affinity DataKi:  0.00597nMAssay Description:Inhibition assay using aromatase enzyme.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
Central Institute of Medicinal and Aromatic Plants

LigandPNGBDBM92558(Neoflavonoid, 10)
Affinity DataKi:  0.00838nMAssay Description:Inhibition assay using aromatase enzyme.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
Central Institute of Medicinal and Aromatic Plants

LigandPNGBDBM92561(Neoflavonoid, 20)
Affinity DataKi:  0.0118nMAssay Description:Inhibition assay using aromatase enzyme.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRibosyldihydronicotinamide dehydrogenase [quinone](Homo sapiens (Human))
Yunnan Normal University

Curated by ChEMBL
LigandPNGBDBM23926((E)-resveratrol | 5-[(E)-2-(4-hydroxyphenyl)etheny...)
Affinity DataIC50:  960nMAssay Description:Inhibition of human quinone reductase 2 expressed in Escherichia coli BL21(DE3) assessed as N-methyldihydronicotinamide oxidation per mg of protein a...More data for this Ligand-Target Pair
TargetRibosyldihydronicotinamide dehydrogenase [quinone](Homo sapiens (Human))
Yunnan Normal University

Curated by ChEMBL
LigandPNGBDBM50339150(5,7-dihydroxy-2-(4-hydroxyphenyl)-3-((2R,3S,4S,5S,...)
Affinity DataIC50:  3.84E+3nMAssay Description:Inhibition of human quinone reductase 2 expressed in Escherichia coli BL21(DE3) assessed as N-methyldihydronicotinamide oxidation per mg of protein a...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
Central Institute of Medicinal and Aromatic Plants

LigandPNGBDBM50339149(CHEMBL1689259 | beta-(3,4-dihydroxyphenyl)ethyl-3-...)
Affinity DataIC50:  2.68E+4nMAssay Description:Inhibition of aromatase preincubated with 2.6 mM NADP+ for 10 mins before substrate addition measured after 30 mins by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
Central Institute of Medicinal and Aromatic Plants

LigandPNGBDBM50339147(CHEMBL1689257 | beta-(4-hydroxyphenyl)ethyl-4-O-E-...)
Affinity DataIC50:  3.07E+4nMAssay Description:Inhibition of aromatase preincubated with 2.6 mM NADP+ for 10 mins before substrate addition measured after 30 mins by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
Central Institute of Medicinal and Aromatic Plants

LigandPNGBDBM50339148(CHEMBL1689258 | beta-(3,4-dihydroxyphenyl)ethyl-6-...)
Affinity DataIC50:  3.23E+4nMAssay Description:Inhibition of aromatase preincubated with 2.6 mM NADP+ for 10 mins before substrate addition measured after 30 mins by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
Central Institute of Medicinal and Aromatic Plants

LigandPNGBDBM50269516(CHEMBL518414 | Calceolarioside B)
Affinity DataIC50:  3.53E+4nMAssay Description:Inhibition of aromatase preincubated with 2.6 mM NADP+ for 10 mins before substrate addition measured after 30 mins by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed