Compile Data Set for Download or QSAR
maximum 50k data
Found 87 with Last Name = 'martins' and Initial = 'ma'
TargetAmine oxidase [flavin-containing] B(Rattus norvegicus (rat))
Universidade Federal De Santa Maria

Curated by ChEMBL
LigandPNGBDBM50265993(CHEMBL451230 | phenyl 4-(4,5-dihydro-1H-imidazol-2...)
Affinity DataKi:  1.38E+3nMAssay Description:Binding affinity to MAOB imidazoline binding site in rat brain mitochondrial homogenate assessed as 4-hydroxyquinoline production by spectrophotometr...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] B(Rattus norvegicus (rat))
Universidade Federal De Santa Maria

Curated by ChEMBL
LigandPNGBDBM50240366(2-(naphthalen-2-yl)-4,5-dihydro-1H-imidazole | 2-N...)
Affinity DataKi:  1.49E+3nMAssay Description:Binding affinity to MAOB imidazoline binding site in rat brain mitochondrial homogenate assessed as 4-hydroxyquinoline production by spectrophotometr...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] B(Rattus norvegicus (rat))
Universidade Federal De Santa Maria

Curated by ChEMBL
LigandPNGBDBM50086502(2-BFi | 2-Benzofuran-2-yl-4,5-dihydro-1H-imidazole...)
Affinity DataKi:  3.63E+3nMAssay Description:Binding affinity to MAOB imidazoline binding site in rat brain mitochondrial homogenate assessed as 4-hydroxyquinoline production by spectrophotometr...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] B(Rattus norvegicus (rat))
Universidade Federal De Santa Maria

Curated by ChEMBL
LigandPNGBDBM50266030(2-(2,4-dichlorophenyl)-4,5-dihydro-1H-imidazole | ...)
Affinity DataKi:  3.98E+3nMAssay Description:Binding affinity to MAOB imidazoline binding site in rat brain mitochondrial homogenate assessed as 4-hydroxyquinoline production by spectrophotometr...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] A(Rattus norvegicus (rat))
Universidade Federal De Santa Maria

Curated by ChEMBL
LigandPNGBDBM50240365(2-(4,5-Dihydro-1H-imidazol-2-yl)-quinoline | 2-(4,...)
Affinity DataKi:  4.86E+3nMAssay Description:Binding affinity to MAOA imidazoline binding site in rat brain mitochondrial homogenate assessed as 4-hydroxyquinoline production by spectrophotometr...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] B(Rattus norvegicus (rat))
Universidade Federal De Santa Maria

Curated by ChEMBL
LigandPNGBDBM50240365(2-(4,5-Dihydro-1H-imidazol-2-yl)-quinoline | 2-(4,...)
Affinity DataKi:  5.32E+3nMAssay Description:Binding affinity to MAOB imidazoline binding site in rat brain mitochondrial homogenate assessed as 4-hydroxyquinoline production by spectrophotometr...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] B(Rattus norvegicus (rat))
Universidade Federal De Santa Maria

Curated by ChEMBL
LigandPNGBDBM50266028(2-(4-chlorophenyl)-4,5-dihydro-1H-imidazole | CHEM...)
Affinity DataKi:  5.35E+3nMAssay Description:Binding affinity to MAOB imidazoline binding site in rat brain mitochondrial homogenate assessed as 4-hydroxyquinoline production by spectrophotometr...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] A(Rattus norvegicus (rat))
Universidade Federal De Santa Maria

Curated by ChEMBL
LigandPNGBDBM50265993(CHEMBL451230 | phenyl 4-(4,5-dihydro-1H-imidazol-2...)
Affinity DataKi:  1.28E+4nMAssay Description:Binding affinity to MAOA imidazoline binding site in rat brain mitochondrial homogenate assessed as 4-hydroxyquinoline production by spectrophotometr...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] B(Rattus norvegicus (rat))
Universidade Federal De Santa Maria

Curated by ChEMBL
LigandPNGBDBM50240362(2-p-tolyl-4,5-dihydro-1H-imidazole | CHEMBL269197)
Affinity DataKi:  1.31E+4nMAssay Description:Binding affinity to MAOB imidazoline binding site in rat brain mitochondrial homogenate assessed as 4-hydroxyquinoline production by spectrophotometr...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] A(Rattus norvegicus (rat))
Universidade Federal De Santa Maria

Curated by ChEMBL
LigandPNGBDBM50265991(2-(3,4-dimethoxyphenyl)-4,5-dihydro-1H-imidazole |...)
Affinity DataKi:  1.36E+4nMAssay Description:Binding affinity to MAOA imidazoline binding site in rat brain mitochondrial homogenate assessed as 4-hydroxyquinoline production by spectrophotometr...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] A(Rattus norvegicus (rat))
Universidade Federal De Santa Maria

Curated by ChEMBL
LigandPNGBDBM50240366(2-(naphthalen-2-yl)-4,5-dihydro-1H-imidazole | 2-N...)
Affinity DataKi:  1.39E+4nMAssay Description:Binding affinity to MAOA imidazoline binding site in rat brain mitochondrial homogenate assessed as 4-hydroxyquinoline production by spectrophotometr...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] A(Rattus norvegicus (rat))
Universidade Federal De Santa Maria

Curated by ChEMBL
LigandPNGBDBM50240364(2-(4-Methoxy-phenyl)-4,5-dihydro-1H-imidazole | 2-...)
Affinity DataKi:  1.58E+4nMAssay Description:Binding affinity to MAOA imidazoline binding site in rat brain mitochondrial homogenate assessed as 4-hydroxyquinoline production by spectrophotometr...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] B(Rattus norvegicus (rat))
Universidade Federal De Santa Maria

Curated by ChEMBL
LigandPNGBDBM50266032(2-(3-nitrophenyl)-4,5-dihydro-1H-imidazole | CHEMB...)
Affinity DataKi:  1.93E+4nMAssay Description:Binding affinity to MAOB imidazoline binding site in rat brain mitochondrial homogenate assessed as 4-hydroxyquinoline production by spectrophotometr...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] B(Rattus norvegicus (rat))
Universidade Federal De Santa Maria

Curated by ChEMBL
LigandPNGBDBM50240363(2-Phenyl-4,5-dihydro-1H-imidazole | CHEMBL274548)
Affinity DataKi:  2.13E+4nMAssay Description:Binding affinity to MAOB imidazoline binding site in rat brain mitochondrial homogenate assessed as 4-hydroxyquinoline production by spectrophotometr...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] B(Rattus norvegicus (rat))
Universidade Federal De Santa Maria

Curated by ChEMBL
LigandPNGBDBM50266029(2-(2-chlorophenyl)-4,5-dihydro-1H-imidazole | CHEM...)
Affinity DataKi:  2.46E+4nMAssay Description:Binding affinity to MAOB imidazoline binding site in rat brain mitochondrial homogenate assessed as 4-hydroxyquinoline production by spectrophotometr...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] A(Rattus norvegicus (rat))
Universidade Federal De Santa Maria

Curated by ChEMBL
LigandPNGBDBM50086502(2-BFi | 2-Benzofuran-2-yl-4,5-dihydro-1H-imidazole...)
Affinity DataKi:  2.49E+4nMAssay Description:Binding affinity to MAOA imidazoline binding site in rat brain mitochondrial homogenate assessed as 4-hydroxyquinoline production by spectrophotometr...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] B(Rattus norvegicus (rat))
Universidade Federal De Santa Maria

Curated by ChEMBL
LigandPNGBDBM50240368(2-(4,5-Dihydro-1H-imidazol-2-yl)-pyridine | 2-(4,5...)
Affinity DataKi:  2.53E+4nMAssay Description:Binding affinity to MAOB imidazoline binding site in rat brain mitochondrial homogenate assessed as 4-hydroxyquinoline production by spectrophotometr...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
Universidade Federal De Santa Maria

Curated by ChEMBL
LigandPNGBDBM50086502(2-BFi | 2-Benzofuran-2-yl-4,5-dihydro-1H-imidazole...)
Affinity DataKi:  2.60E+4nMAssay Description:Binding affinity to human MAOB imidazoline binding siteMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] A(Rattus norvegicus (rat))
Universidade Federal De Santa Maria

Curated by ChEMBL
LigandPNGBDBM50266030(2-(2,4-dichlorophenyl)-4,5-dihydro-1H-imidazole | ...)
Affinity DataKi:  2.88E+4nMAssay Description:Binding affinity to MAOA imidazoline binding site in rat brain mitochondrial homogenate assessed as 4-hydroxyquinoline production by spectrophotometr...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] A(Rattus norvegicus (rat))
Universidade Federal De Santa Maria

Curated by ChEMBL
LigandPNGBDBM50240363(2-Phenyl-4,5-dihydro-1H-imidazole | CHEMBL274548)
Affinity DataKi:  2.88E+4nMAssay Description:Binding affinity to MAOA imidazoline binding site in rat brain mitochondrial homogenate assessed as 4-hydroxyquinoline production by spectrophotometr...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] B(Rattus norvegicus (rat))
Universidade Federal De Santa Maria

Curated by ChEMBL
LigandPNGBDBM50240364(2-(4-Methoxy-phenyl)-4,5-dihydro-1H-imidazole | 2-...)
Affinity DataKi:  3.27E+4nMAssay Description:Binding affinity to MAOB imidazoline binding site in rat brain mitochondrial homogenate assessed as 4-hydroxyquinoline production by spectrophotometr...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] A(Rattus norvegicus (rat))
Universidade Federal De Santa Maria

Curated by ChEMBL
LigandPNGBDBM50240362(2-p-tolyl-4,5-dihydro-1H-imidazole | CHEMBL269197)
Affinity DataKi:  1.02E+5nMAssay Description:Binding affinity to MAOA imidazoline binding site in rat brain mitochondrial homogenate assessed as 4-hydroxyquinoline production by spectrophotometr...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] A(Rattus norvegicus (rat))
Universidade Federal De Santa Maria

Curated by ChEMBL
LigandPNGBDBM50265992(2-(3,4,5-trimethoxyphenyl)-4,5-dihydro-1H-imidazol...)
Affinity DataKi:  1.14E+5nMAssay Description:Binding affinity to MAOA imidazoline binding site in rat brain mitochondrial homogenate assessed as 4-hydroxyquinoline production by spectrophotometr...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] A(Rattus norvegicus (rat))
Universidade Federal De Santa Maria

Curated by ChEMBL
LigandPNGBDBM50266028(2-(4-chlorophenyl)-4,5-dihydro-1H-imidazole | CHEM...)
Affinity DataKi:  1.66E+5nMAssay Description:Binding affinity to MAOA imidazoline binding site in rat brain mitochondrial homogenate assessed as 4-hydroxyquinoline production by spectrophotometr...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] A(Rattus norvegicus (rat))
Universidade Federal De Santa Maria

Curated by ChEMBL
LigandPNGBDBM50266031(2-(4-nitrophenyl)-4,5-dihydro-1H-imidazole | CHEMB...)
Affinity DataKi:  1.81E+5nMAssay Description:Binding affinity to MAOA imidazoline binding site in rat brain mitochondrial homogenate assessed as 4-hydroxyquinoline production by spectrophotometr...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] B(Rattus norvegicus (rat))
Universidade Federal De Santa Maria

Curated by ChEMBL
LigandPNGBDBM50266031(2-(4-nitrophenyl)-4,5-dihydro-1H-imidazole | CHEMB...)
Affinity DataKi: >1.00E+6nMAssay Description:Binding affinity to MAOB imidazoline binding site in rat brain mitochondrial homogenate assessed as 4-hydroxyquinoline production by spectrophotometr...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] A(Rattus norvegicus (rat))
Universidade Federal De Santa Maria

Curated by ChEMBL
LigandPNGBDBM50240368(2-(4,5-Dihydro-1H-imidazol-2-yl)-pyridine | 2-(4,5...)
Affinity DataKi: >1.00E+6nMAssay Description:Binding affinity to MAOA imidazoline binding site in rat brain mitochondrial homogenate assessed as 4-hydroxyquinoline production by spectrophotometr...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] B(Rattus norvegicus (rat))
Universidade Federal De Santa Maria

Curated by ChEMBL
LigandPNGBDBM50138501(2-(furan-2-yl)-4,5-dihydro-1H-imidazole | 2-Furan-...)
Affinity DataKi: >1.00E+6nMAssay Description:Binding affinity to MAOB imidazoline binding site in rat brain mitochondrial homogenate assessed as 4-hydroxyquinoline production by spectrophotometr...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] A(Rattus norvegicus (rat))
Universidade Federal De Santa Maria

Curated by ChEMBL
LigandPNGBDBM50138501(2-(furan-2-yl)-4,5-dihydro-1H-imidazole | 2-Furan-...)
Affinity DataKi: >1.00E+6nMAssay Description:Binding affinity to MAOA imidazoline binding site in rat brain mitochondrial homogenate assessed as 4-hydroxyquinoline production by spectrophotometr...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] B(Rattus norvegicus (rat))
Universidade Federal De Santa Maria

Curated by ChEMBL
LigandPNGBDBM50265991(2-(3,4-dimethoxyphenyl)-4,5-dihydro-1H-imidazole |...)
Affinity DataKi:  1.00E+6nMAssay Description:Binding affinity to MAOB imidazoline binding site in rat brain mitochondrial homogenate assessed as 4-hydroxyquinoline production by spectrophotometr...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] A(Rattus norvegicus (rat))
Universidade Federal De Santa Maria

Curated by ChEMBL
LigandPNGBDBM50266032(2-(3-nitrophenyl)-4,5-dihydro-1H-imidazole | CHEMB...)
Affinity DataKi: >1.00E+6nMAssay Description:Binding affinity to MAOA imidazoline binding site in rat brain mitochondrial homogenate assessed as 4-hydroxyquinoline production by spectrophotometr...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] A(Rattus norvegicus (rat))
Universidade Federal De Santa Maria

Curated by ChEMBL
LigandPNGBDBM50266029(2-(2-chlorophenyl)-4,5-dihydro-1H-imidazole | CHEM...)
Affinity DataKi: >1.00E+6nMAssay Description:Binding affinity to MAOA imidazoline binding site in rat brain mitochondrial homogenate assessed as 4-hydroxyquinoline production by spectrophotometr...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] B(Rattus norvegicus (rat))
Universidade Federal De Santa Maria

Curated by ChEMBL
LigandPNGBDBM50265992(2-(3,4,5-trimethoxyphenyl)-4,5-dihydro-1H-imidazol...)
Affinity DataKi:  1.00E+6nMAssay Description:Binding affinity to MAOB imidazoline binding site in rat brain mitochondrial homogenate assessed as 4-hydroxyquinoline production by spectrophotometr...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4D(Homo sapiens (Human))
Universidade Federal Do Rio De Janeiro

Curated by ChEMBL
LigandPNGBDBM14774(3-(cyclopropylmethoxy)-N-(3,5-dichloropyridin-4-yl...)
Affinity DataIC50:  0.130nMAssay Description:Inhibition of human recombinant PDE4D using [3H]cAMP as substrate preincubated with enzyme for 10 mins followed by substrate addition and measured af...More data for this Ligand-Target Pair
TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4B(Homo sapiens (Human))
Universidade Federal Do Rio De Janeiro

Curated by ChEMBL
LigandPNGBDBM14774(3-(cyclopropylmethoxy)-N-(3,5-dichloropyridin-4-yl...)
Affinity DataIC50:  0.150nMAssay Description:Inhibition of human recombinant PDE4B using [3H]cAMP as substrate preincubated with enzyme for 10 mins followed by substrate addition and measured af...More data for this Ligand-Target Pair
TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4A(Homo sapiens (Human))
Universidade Federal Do Rio De Janeiro

Curated by ChEMBL
LigandPNGBDBM14774(3-(cyclopropylmethoxy)-N-(3,5-dichloropyridin-4-yl...)
Affinity DataIC50:  0.210nMAssay Description:Inhibition of human recombinant PDE4A using [3H]cAMP as substrate preincubated with enzyme for 10 mins followed by substrate addition and measured af...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMedDrugBank

TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4C(Homo sapiens (Human))
Universidade Federal Do Rio De Janeiro

Curated by ChEMBL
LigandPNGBDBM14774(3-(cyclopropylmethoxy)-N-(3,5-dichloropyridin-4-yl...)
Affinity DataIC50:  1.70nMAssay Description:Inhibition of human recombinant PDE4C using [3H]cAMP as substrate preincubated with enzyme for 10 mins followed by substrate addition and measured af...More data for this Ligand-Target Pair
TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4D(Homo sapiens (Human))
Universidade Federal Do Rio De Janeiro

Curated by ChEMBL
LigandPNGBDBM50555898(CHEMBL3182164)
Affinity DataIC50:  3nMAssay Description:Inhibition of PDE4D (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4D(Homo sapiens (Human))
Universidade Federal Do Rio De Janeiro

Curated by ChEMBL
LigandPNGBDBM50346088((1r,4r)-4-cyano-4-(3-(cyclopentyloxy)-4-methoxyphe...)
Affinity DataIC50:  13nMAssay Description:Inhibition of PDE4D (unknown origin)More data for this Ligand-Target Pair
TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4D(Homo sapiens (Human))
Universidade Federal Do Rio De Janeiro

Curated by ChEMBL
LigandPNGBDBM50396783(CHEMBL2172710)
Affinity DataIC50:  31nMAssay Description:Inhibition of human recombinant PDE4DMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4B(Homo sapiens (Human))
Universidade Federal Do Rio De Janeiro

Curated by ChEMBL
LigandPNGBDBM50396783(CHEMBL2172710)
Affinity DataIC50:  47nMAssay Description:Inhibition of human recombinant PDE4BMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4B(Homo sapiens (Human))
Universidade Federal Do Rio De Janeiro

Curated by ChEMBL
LigandPNGBDBM50396784(CHEMBL2172734)
Affinity DataIC50:  53nMAssay Description:Inhibition of human recombinant PDE4BMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4A(Homo sapiens (Human))
Universidade Federal Do Rio De Janeiro

Curated by ChEMBL
LigandPNGBDBM50396783(CHEMBL2172710)
Affinity DataIC50:  64nMAssay Description:Inhibition of human recombinant PDE4AMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4A(Homo sapiens (Human))
Universidade Federal Do Rio De Janeiro

Curated by ChEMBL
LigandPNGBDBM14361((R,S)-Rolipram | 4-(3-cyclopentyloxy-4-methoxy-phe...)
Affinity DataIC50:  67nMAssay Description:Inhibition of PDE4A (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4D(Homo sapiens (Human))
Universidade Federal Do Rio De Janeiro

Curated by ChEMBL
LigandPNGBDBM50396784(CHEMBL2172734)
Affinity DataIC50:  74nMAssay Description:Inhibition of human recombinant PDE4DMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4D(Homo sapiens (Human))
Universidade Federal Do Rio De Janeiro

Curated by ChEMBL
LigandPNGBDBM14361((R,S)-Rolipram | 4-(3-cyclopentyloxy-4-methoxy-phe...)
Affinity DataIC50:  79nMAssay Description:Inhibition of PDE4D (unknown origin)More data for this Ligand-Target Pair
TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4B(Homo sapiens (Human))
Universidade Federal Do Rio De Janeiro

Curated by ChEMBL
LigandPNGBDBM50346088((1r,4r)-4-cyano-4-(3-(cyclopentyloxy)-4-methoxyphe...)
Affinity DataIC50:  120nMAssay Description:Inhibition of PDE4B (unknown origin)More data for this Ligand-Target Pair
TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4D(Homo sapiens (Human))
Universidade Federal Do Rio De Janeiro

Curated by ChEMBL
LigandPNGBDBM50396782(CHEMBL2172731)
Affinity DataIC50:  140nMAssay Description:Inhibition of human recombinant PDE4DMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4A(Homo sapiens (Human))
Universidade Federal Do Rio De Janeiro

Curated by ChEMBL
LigandPNGBDBM50396784(CHEMBL2172734)
Affinity DataIC50:  159nMAssay Description:Inhibition of human recombinant PDE4AMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4A(Homo sapiens (Human))
Universidade Federal Do Rio De Janeiro

Curated by ChEMBL
LigandPNGBDBM50346088((1r,4r)-4-cyano-4-(3-(cyclopentyloxy)-4-methoxyphe...)
Affinity DataIC50:  160nMAssay Description:Inhibition of PDE4A (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Displayed 1 to 50 (of 87 total ) | Next | Last >>
Jump to: